标题
A gold mine for drug discovery: Strategies to develop cyclic peptides into therapies
作者
关键词
-
出版物
MEDICINAL RESEARCH REVIEWS
Volume -, Issue -, Pages -
出版商
Wiley
发表日期
2019-10-10
DOI
10.1002/med.21639
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注意：仅列出部分参考文献，下载原文获取全部文献信息。- Multicomponent Reaction Toolbox for Peptide Macrocyclization and Stapling
- (2019) Leslie Reguera et al. CHEMICAL REVIEWS
- Understanding Cell Penetration of Cyclic Peptides
- (2019) Patrick G. Dougherty et al. CHEMICAL REVIEWS
- The identification and chromatographic separation of a new highly analogous impurity of the active pharmaceutical ingredient icatibant
- (2019) Bassam Lajin et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Amphiphilic Peptides for Efficient siRNA Delivery
- (2019) Saghar Mozaffari et al. Polymers
- Ligation Technologies for the Synthesis of Cyclic Peptides
- (2019) Hoi Yee Chow et al. CHEMICAL REVIEWS
- Cyclic Cell-Penetrating Peptides As Efficient Intracellular Drug Delivery Tools
- (2019) Shang Eun Park et al. MOLECULAR PHARMACEUTICS
- De novo macrocyclic peptides that specifically modulate Lys48-linked ubiquitin chains
- (2019) Mickal Nawatha et al. Nature Chemistry
- Permeability of Cyclic Peptide Macrocycles and Cyclotides and Their Potential as Therapeutics
- (2019) Spiros Liras et al. ACS Medicinal Chemistry Letters
- Development of a high-throughput strategy for discovery of potent analogues of antibiotic lysocin E
- (2019) Hiroaki Itoh et al. Nature Communications
- Establishing the structure-activity relationship of teixobactin
- (2019) Eilidh Matheson et al. CHINESE CHEMICAL LETTERS
- Correlation of DOTATOC Uptake and Pathologic Grade in Neuroendocrine Tumors
- (2019) Hilary Chan et al. PANCREAS
- Endosomal Size and Membrane Leakiness Influence Proton Sponge-Based Rupture of Endosomal Vesicles
- (2018) Lotte M. P. Vermeulen et al. ACS Nano
- Synthesis and antibacterial studies of teixobactin analogues with non-isostere substitution of enduracididine
- (2018) Kang Jin et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Pasireotide in the treatment of neuroendocrine tumors: a review of the literature
- (2018) Giovanni Vitale et al. ENDOCRINE-RELATED CANCER
- The proton sponge hypothesis: Fable or fact?
- (2018) Lotte M.P. Vermeulen et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Cell penetrating peptides in ocular drug delivery: State of the art
- (2018) S. Pescina et al. JOURNAL OF CONTROLLED RELEASE
- Study of forced degradation behavior of pramlintide acetate by HPLC and LC–MS
- (2018) Yu Yuan et al. JOURNAL OF FOOD AND DRUG ANALYSIS
- Developing Equipotent Teixobactin Analogues against Drug-Resistant Bacteria and Discovering a Hydrophobic Interaction between Lipid II and Teixobactin
- (2018) Yu Zong et al. JOURNAL OF MEDICINAL CHEMISTRY
- Pentaminomycins A and B, Hydroxyarginine-Containing Cyclic Pentapeptides from Streptomyces sp. RK88-1441
- (2018) Jun-Pil Jang et al. JOURNAL OF NATURAL PRODUCTS
- Synthesis and evaluation of analogues of the glycinocin family of calcium-dependent antibiotics
- (2018) Leo Corcilius et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Efficient cell delivery mediated by lipid-specific endosomal escape of supercharged branched peptides
- (2018) Dakota J. Brock et al. TRAFFIC
- Accelerated microfluidic native chemical ligation at difficult amino acids toward cyclic peptides
- (2018) Nathalie Ollivier et al. Nature Communications
- Culture-independent discovery of the malacidins as calcium-dependent antibiotics with activity against multidrug-resistant Gram-positive pathogens
- (2018) Bradley M. Hover et al. Nature Microbiology
- Isolation and identification of four major impurities in capreomycin sulfate
- (2018) Guozhu Liu et al. JOURNAL OF CHROMATOGRAPHY A
- Direct Peptide Cyclization and One-Pot Modification Using the MeDbz Linker
- (2018) Bengt H. Gless et al. JOURNAL OF ORGANIC CHEMISTRY
- An amphipathic cyclic tetrapeptide scaffold containing halogenated β2,2 -amino acids with activity against multiresistant bacteria
- (2018) Marianne H. Paulsen et al. JOURNAL OF PEPTIDE SCIENCE
- Natural Cyclic Peptides as an Attractive Modality for Therapeutics: A Mini Review
- (2018) Muna Abdalla et al. MOLECULES
- Plecanatide for Treatment of Chronic Constipation and Irritable Bowel Syndrome
- (2018) Bryan L. Love AMERICAN JOURNAL OF MEDICINE
- Introducing the Petasis Reaction for the Late-Stage Multicomponent Diversification, Labeling and Stapling of Peptides
- (2018) Daniel G. Rivera et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- RNA Display Methods for the Discovery of Bioactive Macrocycles
- (2018) Yichao Huang et al. CHEMICAL REVIEWS
- Enzymatic On-Resin Peptide Cleavage and in Situ Cyclization One-Pot Strategy for the Synthesis of Cyclopeptide and Cyclotide
- (2018) Xiaozhong Cheng et al. JOURNAL OF ORGANIC CHEMISTRY
- Design and Biosynthesis of Dimeric Alboflavusins with Biaryl Linkages via Regiospecific C–C Bond Coupling
- (2018) Zhengyan Guo et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Somatostatin analogs in the treatment of neuroendocrine tumors: current and emerging aspects
- (2017) Gherardo Mazziotti et al. EXPERT OPINION ON PHARMACOTHERAPY
- Outpatient treatment of osteomyelitis with telavancin
- (2017) Claudia P. Schroeder et al. INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS
- Antifungal and Antiviral Cyclic Peptides from the Deep-Sea-Derived Fungus Simplicillium obclavatum EIODSF 020
- (2017) Xiao Liang et al. JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
- Diabetes insipidus after discontinuation of vasopressin infusion for septic shock
- (2017) H. Rana et al. JOURNAL OF CLINICAL PHARMACY AND THERAPEUTICS
- Converting Teixobactin into a Cationic Antimicrobial Peptide (AMP)
- (2017) Shimaa A. H. Abdel Monaim et al. JOURNAL OF MEDICINAL CHEMISTRY
- ENETS Consensus Guidelines for the Standards of Care in Neuroendocrine Neoplasms: Systemic Therapy - Biotherapy and Novel Targeted Agents
- (2017) Marianne Pavel et al. NEUROENDOCRINOLOGY
- Total Synthesis and Stereochemical Assignment of Gymnopeptides A and B
- (2017) Zhengyin Pan et al. ORGANIC LETTERS
- Comprehensive computational design of ordered peptide macrocycles
- (2017) Parisa Hosseinzadeh et al. SCIENCE
- Antiviral peptides from marine gorgonian-derived fungus Aspergillus sp. SCSIO 41501
- (2017) Xuan Ma et al. TETRAHEDRON LETTERS
- Chemical synthesis of a homoserine-mutant of the antibacterial, head-to-tail cyclized protein AS-48 by α-ketoacid–hydroxylamine (KAHA) ligation
- (2017) Florian Rohrbacher et al. Chemical Science
- Highly selective inhibition of histone demethylases by de novo macrocyclic peptides
- (2017) Akane Kawamura et al. Nature Communications
- Synthesis and structure–activity relationship studies of teixobactin analogues
- (2017) Chunlei Wu et al. RSC Advances
- Dual Targeting of Cell Wall Precursors by Teixobactin Leads to Cell Lysis
- (2016) Tomoyuki Homma et al. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
- Discovery and Mechanism of Highly Efficient Cyclic Cell-Penetrating Peptides
- (2016) Ziqing Qian et al. BIOCHEMISTRY
- Application of constrained aza-valine analogs for Smac mimicry
- (2016) Ramesh Chingle et al. BIOPOLYMERS
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- (2016) M. Horn et al. CHEMICAL COMMUNICATIONS
- Synthesis of Natural and Unnatural Cyclooligomeric Depsipeptides Enabled by Flow Chemistry
- (2016) Daniel Lücke et al. CHEMISTRY-A EUROPEAN JOURNAL
- Pharmacokinetics and Pharmacodynamics of Follicle-Stimulating Hormone in Healthy Women Receiving Single and Multiple Doses of Highly Purified Human Menotrophin and Urofollitrophin
- (2016) Andrea F. D. Di Stefano et al. CLINICAL DRUG INVESTIGATION
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- (2016) Terhi Hermanson et al. Expert Opinion On Drug Safety
- ASP2397: a novel antifungal agent produced by Acremonium persicinum MF-347833
- (2016) Ikuko Nakamura et al. JOURNAL OF ANTIBIOTICS
- Evolution of phage display technology: from discovery to application
- (2016) Leila Rahbarnia et al. JOURNAL OF DRUG TARGETING
- Recent Progress in Histone Demethylase Inhibitors
- (2016) Tom E. McAllister et al. JOURNAL OF MEDICINAL CHEMISTRY
- Wewakazole B, a Cytotoxic Cyanobactin from the Cyanobacterium Moorea producens Collected in the Red Sea
- (2016) Julius Adam V. Lopez et al. JOURNAL OF NATURAL PRODUCTS
- Subvisible Particle Content, Formulation, and Dose of an Erythropoietin Peptide Mimetic Product Are Associated With Severe Adverse Postmarketing Events
- (2016) Joseph Kotarek et al. JOURNAL OF PHARMACEUTICAL SCIENCES
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- (2016) Xinya Hemu et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Total Synthesis of Mannopeptimycins α and β
- (2016) Bo Wang et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Gymnopeptides A and B, Cyclic Octadecapeptides from the Mushroom Gymnopus fusipes
- (2016) Attila Ványolós et al. ORGANIC LETTERS
- 5-Methylisoxazole-3-carboxamide-Directed Palladium-Catalyzed γ-C(sp3)–H Acetoxylation and Application to the Synthesis of γ-Mercapto Amino Acids for Native Chemical Ligation
- (2016) Kalyan Kumar Pasunooti et al. ORGANIC LETTERS
- Solution- and Solid-Phase Macrocyclization of Peptides by the Ugi–Smiles Multicomponent Reaction: Synthesis of N-Aryl-Bridged Cyclic Lipopeptides
- (2016) Micjel C. Morejón et al. ORGANIC LETTERS
- Endolides A and B, Vasopressin and Serotonin-Receptor Interacting N-Methylated Peptides from the Sponge-Derived Fungus Stachylidium sp.
- (2016) Celso Almeida et al. ORGANIC LETTERS
- Total Synthesis of Teixobactin
- (2016) Andrew M. Giltrap et al. ORGANIC LETTERS
- Fusion of Enveloped Viruses in Endosomes
- (2016) Judith M. White et al. TRAFFIC
- Total synthesis of teixobactin
- (2016) Kang Jin et al. Nature Communications
- Dynamic Docking of Conformationally Constrained Macrocycles: Methods and Applications
- (2015) Scott E. Allen et al. ACS Chemical Biology
- Evaluation of Effectiveness and Safety of High-Dose Daptomycin: Results from Patients Included in the European Cubicin® Outcomes Registry and Experience
- (2015) R. Andrew Seaton et al. ADVANCES IN THERAPY
- A Thiol-Ene Coupling Approach to Native Peptide Stapling and Macrocyclization
- (2015) Yuanxiang Wang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Intracellular Delivery of Peptidyl Ligands by Reversible Cyclization: Discovery of a PDZ Domain Inhibitor that Rescues CFTR Activity
- (2015) Ziqing Qian et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Site-Specific N-Terminal Labeling of Peptides and Proteins using Butelase 1 and Thiodepsipeptide
- (2015) Giang K. T. Nguyen et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Sortase-mediated backbone cyclization of proteins and peptides
- (2015) Wim van ’t Hof et al. BIOLOGICAL CHEMISTRY
- Butelase-mediated synthesis of protein thioesters and its application for tandem chemoenzymatic ligation
- (2015) Yuan Cao et al. CHEMICAL COMMUNICATIONS
- Modified Regulatory Pathways to Approve Generic Drugs in the US and a Systematic Review of Their Outcomes
- (2015) Aaron S. Kesselheim et al. DRUGS
- PURE mRNA display forin vitroselection of single-chain antibodies
- (2015) Yu Nagumo et al. JOURNAL OF BIOCHEMISTRY
- Cyclic Colisporifungin and Linear Cavinafungins, Antifungal Lipopeptides Isolated from Colispora cavincola
- (2015) Francisco Javier Ortíz-López et al. JOURNAL OF NATURAL PRODUCTS
- A Sequential Ugi Multicomponent/Cu-Catalyzed Azide–Alkyne Cycloaddition Approach for the Continuous Flow Generation of Cyclic Peptoids
- (2015) Carlos Eduardo M. Salvador et al. JOURNAL OF ORGANIC CHEMISTRY
- Macrocyclization of Peptide Side Chains by the Ugi Reaction: Achieving Peptide Folding and Exocyclic N-Functionalization in One Shot
- (2015) Aldrin V. Vasco et al. JOURNAL OF ORGANIC CHEMISTRY
- Chemical Protein Synthesis Using a Second-Generation N-Acylurea Linker for the Preparation of Peptide-Thioester Precursors
- (2015) Juan B. Blanco-Canosa et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Efficient Synthesis and Stereochemical Revision of Coibamide A
- (2015) Guiyang Yao et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Structures and Activity of New Anabaenopeptins Produced by Baltic Sea Cyanobacteria
- (2015) Lisa Spoof et al. Marine Drugs
- A new antibiotic kills pathogens without detectable resistance
- (2015) Losee L. Ling et al. NATURE
- Bidirectional macrocyclization of peptides by double multicomponent reactions
- (2015) Manuel G. Ricardo et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Thiazolidine-Protected β-Thiol Asparagine: Applications in One-Pot Ligation–Desulfurization Chemistry
- (2015) Jessica Sayers et al. ORGANIC LETTERS
- A new strategy for total solid-phase synthesis of polymyxins
- (2015) Wei-Liang Xu et al. TETRAHEDRON LETTERS
- Nonclinical evaluation of the potential for mast cell activation by an erythropoietin analog
- (2015) James L. Weaver et al. TOXICOLOGY AND APPLIED PHARMACOLOGY
- Solid-phase total synthesis of cyclic peptide brachystemin A and its immunomodulating activity
- (2015) Zafar Ali SHAH et al. TURKISH JOURNAL OF CHEMISTRY
- mRNA expression of somatostatin receptor subtypes SSTR-2, SSTR-3, and SSTR-5 and its significance in pancreatic cancer
- (2015) Muhammad Shahbaz et al. World Journal of Surgical Oncology
- Efficient backbone cyclization of linear peptides by a recombinant asparaginyl endopeptidase
- (2015) Karen S. Harris et al. Nature Communications
- Linaclotide: A novel agent for chronic constipation and irritable bowel syndrome
- (2014) B. L. Love et al. AMERICAN JOURNAL OF HEALTH-SYSTEM PHARMACY
- Design and synthesis of novel azapeptide activators of apoptosis mediated by caspase-9 in cancer cells
- (2014) Carine B. Bourguet et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Peptide inhibitors of C3 activation as a novel strategy of complement inhibition for the treatment of paroxysmal nocturnal hemoglobinuria
- (2014) Antonio M. Risitano et al. BLOOD
- Peptide Macrocyclization Catalyzed by a Prolyl Oligopeptidase Involved in α-Amanitin Biosynthesis
- (2014) Hong Luo et al. CHEMISTRY & BIOLOGY
- A Phase I Trial of LY2510924, a CXCR4 Peptide Antagonist, in Patients with Advanced Cancer
- (2014) M. D. Galsky et al. CLINICAL CANCER RESEARCH
- Structural parameters modulating the cellular uptake of disulfide-rich cyclic cell-penetrating peptides: MCoTI-II and SFTI-1
- (2014) Charlotte D’Souza et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Peptides Containing β-Amino Acid Patterns: Challenges and Successes in Medicinal Chemistry
- (2014) Chiara Cabrele et al. JOURNAL OF MEDICINAL CHEMISTRY
- Psychrophilins E–H and Versicotide C, Cyclic Peptides from the Marine-Derived Fungus Aspergillus versicolor ZLN-60
- (2014) Jixing Peng et al. JOURNAL OF NATURAL PRODUCTS
- Reniochalistatins A–E, Cyclic Peptides from the Marine Sponge Reniochalina stalagmitis
- (2014) Kai-Xuan Zhan et al. JOURNAL OF NATURAL PRODUCTS
- Cell penetration: scope and limitations by the application of cell-penetrating peptides
- (2014) Siegmund Reissmann JOURNAL OF PEPTIDE SCIENCE
- Total Synthesis and Stereochemistry Revision of Mannopeptimycin Aglycone
- (2014) Shinichiro Fuse et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Theonellamide G, a Potent Antifungal and Cytotoxic Bicyclic Glycopeptide from the Red Sea Marine Sponge Theonella swinhoei
- (2014) Diaa Youssef et al. Marine Drugs
- Cyclic Peptide-Capped Gold Nanoparticles for Enhanced siRNA Delivery
- (2014) Amir Shirazi et al. MOLECULES
- Psychrophilin E, a new cyclotripeptide, from co-fermentation of two marine alga-derived fungi of the genusAspergillus
- (2014) Sherif S. Ebada et al. NATURAL PRODUCT RESEARCH
- Butelase 1 is an Asx-specific ligase enabling peptide macrocyclization and synthesis
- (2014) Giang K T Nguyen et al. Nature Chemical Biology
- Incidence of erythropoietin antibody-mediated pure red cell aplasia: the Prospective Immunogenicity Surveillance Registry (PRIMS)
- (2014) Iain C. Macdougall et al. NEPHROLOGY DIALYSIS TRANSPLANTATION
- Investigating peptide sequence variations for ‘double-click’ stapled p53 peptides
- (2014) Yu Heng Lau et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Enzyme-Catalyzed Macrocyclization of Long Unprotected Peptides
- (2014) Chi Zhang et al. ORGANIC LETTERS
- In Vitro Evolution and Affinity-Maturation with Coliphage Qβ Display
- (2014) Claudia Skamel et al. PLoS One
- Evaluation of genotoxicity testing of FDA approved large molecule therapeutics
- (2014) Satin G. Sawant et al. REGULATORY TOXICOLOGY AND PHARMACOLOGY
- Functionalised staple linkages for modulating the cellular activity of stapled peptides
- (2014) Yu Heng Lau et al. Chemical Science
- Effect of an oxytocin receptor antagonist (atosiban) on uterine electrical activity
- (2013) Eran Hadar et al. AMERICAN JOURNAL OF OBSTETRICS AND GYNECOLOGY
- Chemoselective Peptide Ligation-Desulfurization at Aspartate
- (2013) Robert E. Thompson et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Synthesis of Constrained Head-to-Tail Cyclic Tetrapeptides by an Imine-Induced Ring-Closing/Contraction Strategy
- (2013) Clarence T. T. Wong et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Wall Teichoic Acids of Gram-Positive Bacteria
- (2013) Stephanie Brown et al. Annual Review of Microbiology
- Peptide Ligation-Desulfurization Chemistry at Arginine
- (2013) Lara R. Malins et al. CHEMBIOCHEM
- NW-G12, a Novel Nonchlorinated Cyclohexapeptide from Streptomyces alboflavus 313
- (2013) Lixia Fan et al. CHEMISTRY OF NATURAL COMPOUNDS
- Cyclization enhances function of linear anti-arthritic peptides
- (2013) Marina Ali et al. CLINICAL IMMUNOLOGY
- mRNA display: from basic principles to macrocycle drug discovery
- (2013) Kristopher Josephson et al. DRUG DISCOVERY TODAY
- Managing dialysis patients who develop anemia caused by chronic kidney disease: focus on peginesatide
- (2013) Michael Hofmann et al. International Journal of Nanomedicine
- High-affinity Cyclic Peptide Matriptase Inhibitors
- (2013) Pedro Quimbar et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Total Synthesis of Daptomycin by Cyclization via a Chemoselective Serine Ligation
- (2013) Hiu Yung Lam et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Drugs derived from phage display
- (2013) Andrew E Nixon et al. mAbs
- Surface Decorated Gold Nanoparticles by Linear and Cyclic Peptides as Molecular Transporters
- (2013) Amir Nasrolahi Shirazi et al. MOLECULAR PHARMACEUTICS
- Discovery and development of first in class antifungal caspofungin (CANCIDAS®)—A case study
- (2013) James M. Balkovec et al. NATURAL PRODUCT REPORTS
- Peginesatide for Anemia in Patients with Chronic Kidney Disease Not Receiving Dialysis
- (2013) Iain C. Macdougall et al. NEW ENGLAND JOURNAL OF MEDICINE
- Peginesatide in Patients with Anemia Undergoing Hemodialysis
- (2013) Steven Fishbane et al. NEW ENGLAND JOURNAL OF MEDICINE
- Total Synthesis of Human Galanin-Like Peptide through an Aspartic Acid Ligation
- (2013) Xiaoyang Guan et al. ORGANIC LETTERS
- A Thioethylalkylamido (TEA) Thioester Surrogate in the Synthesis of a Cyclic Peptide via a Tandem Acyl Shift
- (2013) Misako Taichi et al. ORGANIC LETTERS
- Stapled α−helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy
- (2013) Yong S. Chang et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Chemoselective sulfenylation and peptide ligation at tryptophan
- (2013) Lara R. Malins et al. Chemical Science
- In Vitro Selection of Anti-Akt2 Thioether-Macrocyclic Peptides Leading to Isoform-Selective Inhibitors
- (2012) Yuuki Hayashi et al. ACS Chemical Biology
- Redesign of Glycopeptide Antibiotics: Back to the Future
- (2012) Robert C. James et al. ACS Chemical Biology
- Discovery of Macrocyclic Peptides Armed with a Mechanism-Based Warhead: Isoform-Selective Inhibition of Human Deacetylase SIRT2
- (2012) Jumpei Morimoto et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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- (2012) David J. Craik et al. Chemical Biology & Drug Design
- Micafungin
- (2012) Lesley J. Scott DRUGS
- Three novel cyclic hexapeptides from Streptomyces alboflavus 313 and their antibacterial activity
- (2012) Zhiqin Ji et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
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- (2012) E. Prakoso et al. INTERNAL MEDICINE JOURNAL
- Daptomycin-Mediated Reorganization of Membrane Architecture Causes Mislocalization of Essential Cell Division Proteins
- (2012) J. Pogliano et al. JOURNAL OF BACTERIOLOGY
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- (2012) James P. Tam et al. JOURNAL OF BIOLOGICAL CHEMISTRY
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- (2012) Teshome L. Aboye et al. JOURNAL OF MEDICINAL CHEMISTRY
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- (2012) Farzana Shaheen et al. JOURNAL OF NATURAL PRODUCTS
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- (2012) Jochen Spiegel et al. JOURNAL OF ORGANIC CHEMISTRY
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- (2012) Steven D. Townsend et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
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- (2012) Jisun Lee et al. NATURAL PRODUCT REPORTS
- Chemoselective cyclization of unprotected linear peptides by α-ketoacid–hydroxylamine amide-ligation
- (2012) Takeo Fukuzumi et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Native Chemical Ligation at Glutamine
- (2012) Peter Siman et al. ORGANIC LETTERS
- Cell-Penetrating Homochiral Cyclic Peptides as Nuclear-Targeting Molecular Transporters
- (2011) Deendayal Mandal et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Synthesis of cell-permeable stapled peptide dual inhibitors of the p53-Mdm2/Mdmx interactions via photoinduced cycloaddition
- (2011) Michael M. Madden et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Engineering pro-angiogenic peptides using stable, disulfide-rich cyclic scaffolds
- (2011) L. Y. Chan et al. BLOOD
- Synthesis of Cyclic Peptides through an Intramolecular Amide Bond Rearrangement
- (2011) Derek Macmillan et al. CHEMBIOCHEM
- Promoting peptide α-helix formation with dynamic covalent oxime side-chain cross-links
- (2011) Conor M. Haney et al. CHEMICAL COMMUNICATIONS
- Natural Product-Like Macrocyclic N-Methyl-Peptide Inhibitors against a Ubiquitin Ligase Uncovered from a Ribosome-Expressed De Novo Library
- (2011) Yusuke Yamagishi et al. CHEMISTRY & BIOLOGY
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- (2011) Catherine Liu et al. CLINICAL INFECTIOUS DISEASES
- Sortase A as a tool for high-yield histatin cyclization
- (2011) Jan G. M. Bolscher et al. FASEB JOURNAL
- Azapeptides and their therapeutic potential
- (2011) Caroline Proulx et al. Future Medicinal Chemistry
- Identification and Characterization of a New Family of Cell-penetrating Peptides
- (2011) Laura Cascales et al. JOURNAL OF BIOLOGICAL CHEMISTRY
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- (2011) Keith K. Khoo et al. JOURNAL OF MEDICINAL CHEMISTRY
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- (2011) Steven A. Kawamoto et al. JOURNAL OF MEDICINAL CHEMISTRY
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- (2011) Nathan S. Trookman et al. JOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY
- An Advance in Proline Ligation
- (2011) Shiying Shang et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Rethinking amide bond synthesis
- (2011) Vijaya R. Pattabiraman et al. NATURE
- On-resin N-methylation of cyclic peptides for discovery of orally bioavailable scaffolds
- (2011) Tina R White et al. Nature Chemical Biology
- Contemporary strategies for peptide macrocyclization
- (2011) Christopher J. White et al. Nature Chemistry
- Chemical synthesis of a cyclotide via intramolecular cyclization of peptide O-esters
- (2011) Ji-Shen Zheng et al. Science China-Chemistry
- Use of Ichip for High-Throughput In Situ Cultivation of "Uncultivable" Microbial Species
- (2010) D. Nichols et al. APPLIED AND ENVIRONMENTAL MICROBIOLOGY
- Cell-Penetrating Peptide Induces Leaky Fusion of Liposomes Containing Late Endosome-Specific Anionic Lipid
- (2010) Sung-Tae Yang et al. BIOPHYSICAL JOURNAL
- Protein Synthesis Assisted by Native Chemical Ligation at Leucine
- (2010) Ziv Harpaz et al. CHEMBIOCHEM
- Enzymatic Cyclisation of Peptides with a Transglutaminase
- (2010) Jeremy Touati et al. CHEMBIOCHEM
- NW-G01, a novel cyclic hexapeptide antibiotic, produced by Streptomyces alboflavus 313: II. Structural elucidation
- (2010) Zhengyan Guo et al. JOURNAL OF ANTIBIOTICS
- Macrolactonization of Peptide Thioesters Catalyzed by Imidazole and Its Application in the Synthesis of Kahalalide B and Analogues
- (2010) Yangmei Li et al. ORGANIC LETTERS
- Synthesis of All-lCyclic Tetrapeptides Using Pseudoprolines as Removable Turn Inducers
- (2010) Kelly A. Fairweather et al. ORGANIC LETTERS
- Cyclic Peptide Synthesis with Thioacids
- (2010) Kaname Sasaki et al. ORGANIC LETTERS
- Salicylaldehyde Ester-Induced Chemoselective Peptide Ligations: Enabling Generation of Natural Peptidic Linkages at the Serine/Threonine Sites
- (2010) Xuechen Li et al. ORGANIC LETTERS
- Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency
- (2010) R. S. Harrison et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
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- (2010) B. Wu et al. SCIENCE
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- (2009) David Crich et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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- (2009) David Crich et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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- (2009) Jaeheon Lee et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
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- (2008) Edward J. Hayes et al. AMERICAN JOURNAL OF OBSTETRICS AND GYNECOLOGY
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- (2008) Rolf Kleineweischede et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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- (2008) Jin Chen et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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