Design and synthesis of glycomimetics: Recent advances

Phostine 3.1a as a pharmacological compound with antiangiogenic properties against diseases with excess vascularization

(2019) Simon Bousseau et al.   FASEB JOURNAL

Stereoretentive Reactions at the Anomeric Position: Synthesis of Selenoglycosides

(2018) Feng Zhu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct N -Glycofunctionalization of Amides with Glycosyl Trichloroacetimidate by Thiourea/Halogen Bond Donor Co-Catalysis

(2018) Yusuke Kobayashi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Non-Classical Arylated C-Saccharides through Nickel/Photoredox Dual Catalysis

(2018) Audrey Dumoulin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Reversed C -Acyl Glycosides through Ni/Photoredox Dual Catalysis

(2018) Shorouk O. Badir et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The sugar code: Why glycans are so important

(2018) Hans-Joachim Gabius   BIOSYSTEMS

Synthesis and glycosidase inhibition potency of all- trans substituted 1- C -perfluoroalkyl iminosugars

(2018) Fabien Massicot et al.   CARBOHYDRATE RESEARCH

On-chip screening of a glycomimetic library with C-type lectins reveals structural features responsible for preferential binding of dectin-2 over DC-SIGN/R and langerin

(2018) Laura Medve et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Carba-Cyclophellitols: a New Class of Carbohydrate Mimetics

(2018) Thomas J. M. Beenakker et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

The conformation of the mannopyranosyl phosphate repeating unit of the capsular polysaccharide of Neisseria meningitidis serogroup A and its carba-mimetic

(2018) Jesus Jimenez-Barbero et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Stereocontrolled Synthesis of 2-Fluorinated C -Glycosides

(2018) Anna Sadurní et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Fluorinated Leishmania Cap Trisaccharides for Diagnostic Tool and Vaccine Development

(2018) Andreas Baumann et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Back to (non-)Basics: An Update on Neutral and Charge-Balanced Glycosidase Inhibitors

(2018) Michela I. Simone et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Convergent Synthesis of N,S-bis Glycosylquinolin-2-ones via a Pd-G3-XantPhos Precatalyst Catalysis

(2018) Wafa Redjdal et al.   MOLECULES

Probing the Inhibitor versus Chaperone Properties of sp2-Iminosugars towards Human β-Glucocerebrosidase: A Picomolar Chaperone for Gaucher Disease

(2018) Teresa Mena-Barragán et al.   MOLECULES

Recent Advances in the Synthesis of Glycoconjugates for Vaccine Development

(2018) Cinzia Colombo et al.   MOLECULES

Glycosyl Cross-Coupling with Diaryliodonium Salts: Access to Aryl C-Glycosides of Biomedical Relevance

(2018) Duk Yi et al.   ORGANIC LETTERS

One-Pot Assembly of Unsymmetrical Biaryl Thioglycosides through Chemoselective Palladium-Catalyzed Three-Component Tandem Reaction

(2018) Sara Benmahdjoub et al.   ORGANIC LETTERS

Design and synthesis of constrained bicyclic molecules as candidate inhibitors of influenza A neuraminidase

(2018) Cinzia Colombo et al.   PLoS One

Recent Advances in Transition-Metal-Catalyzed Functionalization of 1-Thiosugars

(2018) Nada Ibrahim et al.   Asian Journal of Organic Chemistry

Allosteric Inhibition of a Mammalian Lectin

(2018) Jonas Aretz et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Acyl Glycosides through Stereospecific Glycosyl Cross-Coupling: Rapid Access to C(sp3)-Linked Glycomimetics

(2018) Feng Zhu et al.   ACS Central Science

Synthesis of Oxaphosphinane-Based Pseudodisaccharides

(2017) Rachida Babouri et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Observation of a Tricyclic[4.1.0.02,4]heptane During a Michael Addition-Ring Closure Reaction and a Computational Study on Its Mechanism of Formation

(2017) Marco Farren-Dai et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of (1 → 2)-S-Linked Saccharides and S-Linked Glycoconjugates via a Palladium-G3-XantPhos Precatalyst Catalysis

(2017) Riyadh Ahmed Atto AL-Shuaeeb et al.   JOURNAL OF ORGANIC CHEMISTRY

Carba-cyclophellitols Are Neutral Retaining-Glucosidase Inhibitors

(2017) Thomas J. M. Beenakker et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Glycosyl Cross-Coupling of Anomeric Nucleophiles: Scope, Mechanism, and Applications in the Synthesis of Aryl C-Glycosides

(2017) Feng Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Phostine PST3.1a Targets MGAT5 and Inhibits Glioblastoma-Initiating Cell Invasiveness and Proliferation

(2017) Zahra Hassani et al.   MOLECULAR CANCER RESEARCH

Glycosyl Stille Cross-Coupling with Anomeric Nucleophiles – A General Solution to a Long-Standing Problem of Stereocontrolled Synthesis of C-Glycosides

(2017) Maciej Walczak et al.   SYNLETT

Carbohydrate-active enzymes: sequences, shapes, contortions and cells

(2016) G. J. Davies et al.   BIOCHEMICAL SOCIETY TRANSACTIONS

Hydrophobic substituents increase the potency of salacinol, a potent α-glucosidase inhibitor from Ayurvedic traditional medicine ‘Salacia’

(2016) Genzoh Tanabe et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The Staudinger/aza-Wittig/Grignard reaction as key step for the concise synthesis of 1-C-Alkyl-iminoalditol glycomimetics

(2016) Manuel Zoidl et al.   CARBOHYDRATE RESEARCH

A building block approach to the synthesis of a family of S-linked α-1,6-oligomannosides

(2016) Tyson Belz et al.   CARBOHYDRATE RESEARCH

Influence of the configurational pattern of sp2-iminosugar pseudo N-, S-, O- and C-glycosides on their glycoside inhibitory and antitumor properties

(2016) Elena M. Sánchez-Fernández et al.   CARBOHYDRATE RESEARCH

Glycomimetic-based pharmacological chaperones for lysosomal storage disorders: lessons from Gaucher, GM1-gangliosidosis and Fabry diseases

(2016) Elena M. Sánchez-Fernández et al.   CHEMICAL COMMUNICATIONS

Migalastat: First Global Approval

(2016) Anthony Markham   DRUGS

Design, synthesis and biological evaluation of 3′-benzylated analogs of 3′-epi-neoponkoranol as potent α-glucosidase inhibitors

(2016) Dan Liu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Reaction of Glyconitriles with Organometallic Reagents: Access to Acyl β-C-Glycosides

(2016) Nicolas E. S. Guisot et al.   JOURNAL OF ORGANIC CHEMISTRY

Stereoselective Chirality Extension of syn,anti- and syn,syn-Oxazine and Stereochemical Analysis of Chiral 1,3-Oxazines: Stereoselective Total Syntheses of (+)-1-Deoxygalactonojirimycin and (−)-1-Deoxygulonojirimycin

(2016) Jin-Seok Kim et al.   JOURNAL OF ORGANIC CHEMISTRY

A Chiron Approach to Diversity-Oriented Synthesis of Aminocyclitols, (−)-Conduramine F-4 and Polyhydroxyaminoazepanes from a Common Precursor

(2016) Vimal Kant Harit et al.   JOURNAL OF ORGANIC CHEMISTRY

Resistance to Mutant Group 2 Influenza Virus Neuraminidases of an Oseltamivir-Zanamivir Hybrid Inhibitor

(2016) Yan Wu et al.   JOURNAL OF VIROLOGY

Advancement of Sialyltransferase Inhibitors: Therapeutic Challenges and Opportunities

(2016) Rémi Szabo et al.   MEDICINAL RESEARCH REVIEWS

Synthesis of 28a-homoselenolupanes and 28a-homoselenolupane saponins

(2016) Katarzyna Sidoryk et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis and evaluation of influenza A viral neuraminidase candidate inhibitors based on a bicyclo[3.1.0]hexane scaffold

(2016) Cinzia Colombo et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Lewis Acid Induced Anomerization of Se-Glycosides. Application to Synthesis of α-Se-GalCer

(2016) Anthony W. McDonagh et al.   ORGANIC LETTERS

Glycosylation, an effective synthetic strategy to improve the bioavailability of therapeutic peptides

(2016) Shayli Varasteh Moradi et al.   Chemical Science

Stereoselective innovative synthesis and biological evaluation of new real carba analogues of minimal epitope Manα(1,2)Man as DC-SIGN inhibitors

(2016) Vittorio Bordoni et al.   RSC Advances

A Convenient Approach to Stereoisomeric Iminocyclitols: Generation of Potent Brain-Permeable OGA Inhibitors

(2015) Milan Bergeron-Brlek et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Thio- and selenoglycosides as ligands for biomedically relevant lectins: Valency–activity correlations for benzene-based dithiogalactoside clusters and first assessment for (di)selenodigalactosides

(2015) Sabine André et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The cancer glycome: Carbohydrates as mediators of metastasis

(2015) Siobhan V. Glavey et al.   BLOOD REVIEWS

Thioglycosides in Carbohydrate Research

(2015) Gaoyan Lian et al.   CARBOHYDRATE RESEARCH

Glycosyldiselenides as lectin ligands detectable by NMR in biofluids

(2015) Ignacio Pérez-Victoria et al.   CHEMICAL COMMUNICATIONS

Intramolecular thiol–yne cyclisation as a novel strategy for thioglycal synthesis

(2015) Vincent Corcé et al.   CHEMICAL COMMUNICATIONS

Glycosylated Porphyrins, Phthalocyanines, and Other Porphyrinoids for Diagnostics and Therapeutics

(2015) Sunaina Singh et al.   CHEMICAL REVIEWS

Conformational Plasticity in Glycomimetics: Fluorocarbamethyl-L-idopyranosides Mimic the Intrinsic Dynamic Behaviour of Natural Idose Rings

(2015) Luca Unione et al.   CHEMISTRY-A EUROPEAN JOURNAL

α-Halogenated oxaphosphinanes: Synthesis, unexpected reactions and evaluation as inhibitors of cancer cell proliferation

(2015) Rachida Babouri et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Perfluoroalkylation of Nitrones for the Synthesis of a Series of Fucosidase Inhibitors

(2015) Jadwiga Paszkowska et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Selective S-deacetylation inspired by native chemical ligation: practical syntheses of glycosyl thiols and drug mercapto-analogues

(2015) Penghua Shu et al.   GREEN CHEMISTRY

Ruthenium Catalyzed Stereo/Chemo/Regioselective One-Pot Synthesis of C(2)–C(3) Unsaturated and α-d-Mannopyranosyl Sulfones

(2015) Sravanthi Chittela et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Evaluation of Hydroxymethylaminocyclitols as Glycosidase Inhibitors

(2015) Ana Trapero et al.   JOURNAL OF ORGANIC CHEMISTRY

Pharmacological Chaperone Therapy: Preclinical Development, Clinical Translation, and Prospects for the Treatment of Lysosomal Storage Disorders

(2015) Giancarlo Parenti et al.   MOLECULAR THERAPY

Synthesis and biological properties of multivalent iminosugars

(2015) Renaud Zelli et al.   NEW JOURNAL OF CHEMISTRY

Novel Multiple Type Molecular Targeted Antitumor Agents: Preparation and Preclinical Evaluation of Low-Molecular-Weight Phospha Sugar Derivatives

(2015) Reiko Makita et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

Alditol thiacrowns via a ring-closing metathesis of carbohydrate-derived α,ω-dithioallylethers

(2015) Mohammed Benazza et al.   TETRAHEDRON

Synthesis and binding affinity analysis of positional thiol analogs of mannopyranose for the elucidation of sulfur in different position

(2015) Bin Wu et al.   TETRAHEDRON

Direct synthesis of imino-C-nucleoside analogues and other biologically active iminosugars

(2015) Milan Bergeron-Brlek et al.   Nature Communications

gem-Difluorocarbadisaccharides: Restoring theexo-Anomeric Effect

(2014) Bixue Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Protecting-Group-Free One-Pot Synthesis of Glycoconjugates Directly from Reducing Sugars

(2014) David Lim et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Expanded potential of seleno-carbohydrates as a molecular tool for X-ray structural determination of a carbohydrate–protein complex with single/multi-wavelength anomalous dispersion phasing

(2014) Tatsuya Suzuki et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A potential CARB-pharmacophore for antineoplastic activity: Part 1

(2014) Zbigniew J. Witczak et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Thio-sugar motif of functional CARB-pharmacophore for antineoplastic activity. Part 2

(2014) Zbigniew J. Witczak et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The synthesis of gemcitabine

(2014) Kylie Brown et al.   CARBOHYDRATE RESEARCH

The Multivalent Effect in Glycosidase Inhibition: A New, Rapidly Emerging Topic in Glycoscience

(2014) Philippe Compain et al.   CHEMBIOCHEM

Glycomimetics versus Multivalent Glycoconjugates for the Design of High Affinity Lectin Ligands

(2014) Samy Cecioni et al.   CHEMICAL REVIEWS

Multivalent Inhibitors for Carbohydrate-Processing Enzymes: Beyond the “Lock-and-Key” Concept

(2014) Sébastien G. Gouin   CHEMISTRY-A EUROPEAN JOURNAL

Dissecting conformational contributions to glycosidase catalysis and inhibition

(2014) Gaetano Speciale et al.   CURRENT OPINION IN STRUCTURAL BIOLOGY

Synthesis of Cyclophellitol, Cyclophellitol Aziridine, and Their Tagged Derivatives

(2014) Kah-Yee Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Medicinal applications of perfluoroalkylated chain-containing compounds

(2014) Eva Prchalová et al.   Future Medicinal Chemistry

C-Glycoside Mimetics Inhibit Glioma Stem Cell Proliferation, Migration, and Invasion

(2014) Ludovic Clarion et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Evaluation of Di- and Trimeric Hydroxylamine-Based β-(1→3)-Glucan Mimetics

(2014) Angélique Ferry et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ni-Catalyzed Reductive Coupling of Alkyl Acids with Unactivated Tertiary Alkyl and Glycosyl Halides

(2014) Chenglong Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthetic Applications of Intramolecular Thiol-Ene “Click” Reactions

(2014) Eoin Scanlan et al.   MOLECULES

Sulfonium ions as inhibitors of the mycobacterial galactofuranosyltransferase GlfT2

(2014) Jing Li et al.   MedChemComm

A mechanism-based inactivator of glycoside hydrolases involving formation of a transient non-classical carbocation

(2014) Saswati Chakladar et al.   Nature Communications

Computational and Experimental Prediction of Human C-Type Lectin Receptor Druggability

(2014) Jonas Aretz et al.   Frontiers in Immunology

Naturally Occurring Sulfonium-Ion Glucosidase Inhibitors and Their Derivatives: A Promising Class of Potential Antidiabetic Agents

(2013) Sankar Mohan et al.   ACCOUNTS OF CHEMICAL RESEARCH

C-(α-d-Glucopyranosyl)-phenyldiazomethanes—irreversible inhibitors of α-glucosidase

(2013) Yiqun Geng et al.   BIOORGANIC & MEDICINAL CHEMISTRY

An α-selective, visible light photocatalytic glycosylation of alcohols with selenoglycosides

(2013) Mark Spell et al.   CARBOHYDRATE RESEARCH

De novo synthesis of 1-deoxythiosugars

(2013) Thanikachalam Gunasundari et al.   CARBOHYDRATE RESEARCH

Recent developments in design and synthesis of bicyclic azasugars, carbasugars and related molecules as glycosidase inhibitors

(2013) Rima Lahiri et al.   CHEMICAL SOCIETY REVIEWS

Glycotherapy: New Advances Inspire a Reemergence of Glycans in Medicine

(2013) Jason E. Hudak et al.   CHEMISTRY & BIOLOGY

Selective Targeting of Dendritic Cell-Specific Intercellular Adhesion Molecule-3-Grabbing Nonintegrin (DC-SIGN) with Mannose-Based Glycomimetics: Synthesis and Interaction Studies of Bis(benzylamide) Derivatives of a Pseudomannobioside

(2013) Norbert Varga et al.   CHEMISTRY-A EUROPEAN JOURNAL

Applications of 5-exo-trig Thiyl Radical Cyclizations for the Synthesis of Thiosugars

(2013) Aoife Malone et al.   JOURNAL OF ORGANIC CHEMISTRY

Determination of Proton Affinities and Acidity Constants of Sugars

(2013) Shuting Feng et al.   JOURNAL OF PHYSICAL CHEMISTRY A

Chemical Insight into the Emergence of Influenza Virus Strains That Are Resistant to Relenza

(2013) Fahimeh S. Shidmoossavee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The carbohydrate-active enzymes database (CAZy) in 2013

(2013) Vincent Lombard et al.   NUCLEIC ACIDS RESEARCH

Stereoselective Ribosylation of Amino Acids

(2013) Hans A. V. Kistemaker et al.   ORGANIC LETTERS

Applications of Thiyl Radical Cyclizations for the Synthesis of Thiosugars

(2013) Aoife Malone et al.   ORGANIC LETTERS

Realizing the promise of chemical glycobiology

(2013) Lai-Xi Wang et al.   Chemical Science

Structural basis for a class of nanomolar influenza A neuraminidase inhibitors

(2013) Philip S. Kerry et al.   Scientific Reports

Transition States, Analogues, and Drug Development

(2012) Vern L. Schramm   ACS Chemical Biology

Click and Pick: Identification of Sialoside Analogues for Siglec-Based Cell Targeting

(2012) Cory D. Rillahan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Carbohydrate derivatives from the roots of Brassica rapa ssp. campestris and their effects on ROS production and glutamate-induced cell death in HT-22 cells

(2012) Qian Wu et al.   CARBOHYDRATE RESEARCH

Stereoselective Synthesis of α- and β-Glycofuranosyl Amides by Traceless Ligation of Glycofuranosyl Azides

(2012) Filippo Nisic et al.   CHEMISTRY-A EUROPEAN JOURNAL

NO Bond as a Glycosidic-Bond Surrogate: Synthetic Studies Toward PolyhydroxylatedN-Alkoxypiperidines

(2012) Gaëlle Malik et al.   CHEMISTRY-A EUROPEAN JOURNAL

Research and Development of Phospha Sugar Anti-cancer Agents with Anti-leukemic Activity

(2012) Junko Yamashita et al.   HETEROCYCLIC COMMUNICATIONS

Oxaphosphinanes: New Therapeutic Perspectives for Glioblastoma

(2012) Ludovic Clarion et al.   JOURNAL OF MEDICINAL CHEMISTRY

Target Selectivity of FimH Antagonists

(2012) Meike Scharenberg et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Characterization, and Coupling Reactions of Six-Membered Cyclic P-Chiral Ammonium Phosphonite–Boranes; Reactive H-Phosphinate Equivalents for the Stereoselective Synthesis of Glycomimetics

(2012) Angélique Ferry et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Increasing O-GlcNAc slows neurodegeneration and stabilizes tau against aggregation

(2012) Scott A Yuzwa et al.   Nature Chemical Biology

Developing inhibitors of glycan processing enzymes as tools for enabling glycobiology

(2012) Tracey M Gloster et al.   Nature Chemical Biology

Synthesis and preliminary biological evaluation of carba analogues from Neisseria meningitidis A capsular polysaccharide

(2012) Qi Gao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Access to l- and d-Iminosugar C-Glycosides from a d-gluco-Derived 6-Azidolactol Exploiting a Ring Isomerization/Alkylation Strategy

(2012) Martine Mondon et al.   ORGANIC LETTERS

Convenient one-pot synthesis of thiosugars and their efficient conversion to polyoxygenated cycloalkenes

(2012) Jingjing Zhang et al.   TETRAHEDRON

The first synthesis of 7-(hydroxymethyl)thiepane-3,4,5-triols from d-(−)-quinic acid

(2012) Tzenge-Lien Shih et al.   TETRAHEDRON

Isolation, structure identification and SAR studies on thiosugar sulfonium salts, neosalaprinol and neoponkoranol, as potent α-glucosidase inhibitors

(2011) Weijia Xie et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Biological evaluation of 3′-O-alkylated analogs of salacinol, the role of hydrophobic alkyl group at 3′ position in the side chain on the α-glucosidase inhibitory activity

(2011) Genzoh Tanabe et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Stereochemical Differentiation in the Simmons-Smith Reaction for Cyclopropanated Glucopyranose Derivatives as Molecular Probes for Glycosidases

(2011) Nanako AKIYAMA et al.   BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY

Iridium-catalysed condensation of alcohols and amines as a method for aminosugar synthesis

(2011) Ian Cumpstey et al.   CHEMICAL COMMUNICATIONS

Antibody recognition of fluorinated MUC1 glycopeptide antigens

(2011) Thomas Oberbillig et al.   CHEMICAL COMMUNICATIONS

Recent applications of thiol–ene coupling as a click process for glycoconjugation

(2011) Alessandro Dondoni et al.   CHEMICAL SOCIETY REVIEWS

The role of Dectin-1 in the host defence against fungal infections

(2011) Rebecca A Drummond et al.   CURRENT OPINION IN MICROBIOLOGY

Synthesis and biological activity of novel organoselenium derivatives targeting multiple kinases and capable of inhibiting cancer progression to metastases

(2011) Krikor Bijian et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of α-N-Linked Glycopeptides

(2011) Cinzia Colombo et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Photoinitiated Glycosylation at 350 nm

(2011) Ian Cumpstey et al.   JOURNAL OF CARBOHYDRATE CHEMISTRY

Unprecedented furan-2-carbonyl C-glycosides and phenolic diglycosides from Scleropyrum pentandrum

(2011) Wannaporn Disadee et al.   PHYTOCHEMISTRY

Targeted drugs by olefin metathesis: piperidine-based iminosugars

(2011) Ileana Dragutan et al.   RSC Advances

Dramatic effect of modified boranes in diastereoselective reduction of chiral cyclic α-ketophosphinates

(2011) Damien Filippini et al.   RSC Advances

Inhibition of DC-SIGN-Mediated HIV Infection by a Linear Trimannoside Mimic in a Tetravalent Presentation

(2010) Sara Sattin et al.   ACS Chemical Biology

Thiol-Ene Click Chemistry

(2010) Charles E. Hoyle et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of a biologically active isomer of kotalanol, a naturally occurring glucosidase inhibitor

(2010) Razieh Eskandari et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Preparation and characterization of novel 4-bromo-3,4-dimethyl-1-phenyl-2-phospholene 1-oxide and the analogous phosphorus heterocycles or phospha sugars

(2010) Manabu Yamada et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Iminosugars past, present and future: medicines for tomorrow

(2010) Graeme Horne et al.   DRUG DISCOVERY TODAY

Carbohydrate mimetics and scaffolds: sweet spots in medicinal chemistry

(2010) Laura Cipolla et al.   Future Medicinal Chemistry

Enantioselective and Protecting Group-Free Synthesis of 1-Deoxythionojirimycin, 1-Deoxythiomannojirimycin, and 1-Deoxythiotalonojirimycin

(2010) Thanikachalam Gunasundari et al.   JOURNAL OF ORGANIC CHEMISTRY

pH-Dependent Mutarotation of 1-Thioaldoses in Water. Unexpected Behavior of (2S)-d-Aldopyranoses

(2010) Rémi Caraballo et al.   JOURNAL OF ORGANIC CHEMISTRY

Design, synthesis and activity evaluation of mannose-based DC-SIGN antagonists

(2010) Nataša Obermajer et al.   MOLECULAR DIVERSITY

Permissive Secondary Mutations Enable the Evolution of Influenza Oseltamivir Resistance

(2010) J. D. Bloom et al.   SCIENCE

Synthesis and discovery of pyrazole-5-carbohydrazide N-glycosides as inducer of autophagy in A549 lung cancer cells

(2009) Song Lian et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Metal-Catalyzed Olefin Cyclopropanation with Ethyl Diazoacetate: Control of the Diastereoselectivity

(2009) Ana Caballero et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Palladium-Controlled β-Selective Glycosylation in the Absence of the C(2)-Ester Participatory Group

(2009) Enoch A. Mensah et al.   JOURNAL OF ORGANIC CHEMISTRY

Modeling of synthetic phosphono and carba analogues of N-acetyl-α-d-mannosamine 1-phosphate, the repeating unit of the capsular polysaccharide from Neisseria meningitidis serovar A

(2009) Lucio Toma et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Glycosidase inhibition: assessing mimicry of the transition state

(2009) Tracey M. Gloster et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The First N-Glycosylated Indoxyls and Their Application to the Synthesis of Indirubin-N-glycosides (Purple Sugars)

(2009) Peter Langer et al.   SYNLETT

Covalent inhibitors of glycosidases and their applications in biochemistry and biology

(2008) B. P Rempel et al.   GLYCOBIOLOGY

Synthesis of 6H-indolo[2,3-b]quinoxaline-N-glycosides and their cytotoxic activity against human ceratinocytes (HaCaT)

(2008) Katrin Marie Driller et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Hemicarbasucrose: Turning off the Exoanomeric Effect Induces Less Flexibility

(2007) Blanca López-Méndez et al.   Chemistry-An Asian Journal