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Title
Molecular Imaging of Hydrolytic Enzymes Using PET and SPECT
Authors
Keywords
-
Journal
Molecular Imaging
Volume 16, Issue -, Pages 153601211771785
Publisher
SAGE Publications
Online
2017-09-20
DOI
10.1177/1536012117717852
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Note: Only part of the references are listed.- [18F]-Organotrifluoroborates as Radioprosthetic Groups for PET Imaging: From Design Principles to Preclinical Applications
- (2016) David M. Perrin ACCOUNTS OF CHEMICAL RESEARCH
- Metal-dependent Deacetylases: Cancer and Epigenetic Regulators
- (2016) Jeffrey E. López et al. ACS Chemical Biology
- A Novel Radiotracer for Imaging Monoacylglycerol Lipase in the Brain Using Positron Emission Tomography
- (2016) Changning Wang et al. ACS Chemical Neuroscience
- Cathepsin S-cleavable, multi-block HPMA copolymers for improved SPECT/CT imaging of pancreatic cancer
- (2016) Wei Fan et al. BIOMATERIALS
- N-(3,4-Dimethylisoxazol-5-yl)piperazine-4-[4-(2-fluoro-4-[11C]methylphenyl)thiazol-2-yl]-1-carboxamide: A promising positron emission tomography ligand for fatty acid amide hydrolase
- (2016) Yoko Shimoda et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Fluorinated matrix metalloproteinases inhibitors—Phosphonate based potential probes for positron emission tomography
- (2016) Bernd Beutel et al. BIOORGANIC & MEDICINAL CHEMISTRY
- A Novel Way To Radiolabel Human Butyrylcholinesterase for Positron Emission Tomography through Irreversible Transfer of the Radiolabeled Moiety
- (2016) Edgar Sawatzky et al. ChemMedChem
- Prostate-specific membrane antigen positron emission tomography in prostate cancer
- (2016) Kirsten Bouchelouche et al. CURRENT OPINION IN ONCOLOGY
- Dual-Modality Activity-Based Probes as Molecular Imaging Agents for Vascular Inflammation
- (2016) N. P. Withana et al. JOURNAL OF NUCLEAR MEDICINE
- 18F-FNDP for PET Imaging of Soluble Epoxide Hydrolase
- (2016) A. G. Horti et al. JOURNAL OF NUCLEAR MEDICINE
- Novel Radioligands for Cyclic Nucleotide Phosphodiesterase Imaging with Positron Emission Tomography: An Update on Developments Since 2012
- (2016) Susann Schröder et al. MOLECULES
- Concerted nucleophilic aromatic substitution with 19F− and 18F−
- (2016) Constanze N. Neumann et al. NATURE
- Current use of PSMA–PET in prostate cancer management
- (2016) Tobias Maurer et al. Nature Reviews Urology
- Radiolabeled hydroxamate-based matrix metalloproteinase inhibitors: How chemical modifications affect pharmacokinetics and metabolic stability
- (2016) Verena Hugenberg et al. NUCLEAR MEDICINE AND BIOLOGY
- Molecular imaging using PET and SPECT for identification of breast cancer subtypes
- (2016) Hao Liu et al. NUCLEAR MEDICINE COMMUNICATIONS
- PET imaging of prostate-specific membrane antigen in prostate cancer: current state of the art and future challenges
- (2016) S P Rowe et al. PROSTATE CANCER AND PROSTATIC DISEASES
- Insights into neuroepigenetics through human histone deacetylase PET imaging
- (2016) Hsiao-Ying Wey et al. Science Translational Medicine
- Synthesis and Preclinical Evaluation of Sulfonamido-based [11C-Carbonyl]-Carbamates and Ureas for Imaging Monoacylglycerol Lipase
- (2016) Lu Wang et al. Theranostics
- Non-invasive Imaging of Idiopathic Pulmonary Fibrosis Using Cathepsin Protease Probes
- (2016) Nimali P. Withana et al. Scientific Reports
- Synthesis and Preliminary PET Imaging Studies of a FAAH Radiotracer ([11C]MPPO) Based on α-Ketoheterocyclic Scaffold
- (2015) Lu Wang et al. ACS Chemical Neuroscience
- Kinetic Analysis and Quantification of [11C]Martinostat for in Vivo HDAC Imaging of the Brain
- (2015) Hsiao-Ying Wey et al. ACS Chemical Neuroscience
- Development of a Fluorinated Class-I HDAC Radiotracer Reveals Key Chemical Determinants of Brain Penetrance
- (2015) Martin G. Strebl et al. ACS Chemical Neuroscience
- Lysosomal Storage Diseases: From Pathophysiology to Therapy
- (2015) Giancarlo Parenti et al. Annual Review of Medicine
- From Unorthodox to Established: The Current Status of 18F-Trifluoroborate- and 18F-SiFA-Based Radiopharmaceuticals in PET Nuclear Imaging
- (2015) Vadim Bernard-Gauthier et al. BIOCONJUGATE CHEMISTRY
- Next Generation of SiFAlin-Based TATE Derivatives for PET Imaging of SSTR-Positive Tumors: Influence of Molecular Design on In Vitro SSTR Binding and In Vivo Pharmacokinetics
- (2015) S. Litau et al. BIOCONJUGATE CHEMISTRY
- A dual inhibitor of matrix metalloproteinases and a disintegrin and metalloproteinases, [18F]FB-ML5, as a molecular probe for non-invasive MMP/ADAM-targeted imaging
- (2015) Nathalie Matusiak et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Novel fluorine-18 labeled 5-(1-pyrrolidinylsulfonyl)-7-azaisatin derivatives as potential PET tracers for in vivo imaging of activated caspases in apoptosis
- (2015) Christopher M. Waldmann et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Small Molecule Active Site Directed Tools for Studying Human Caspases
- (2015) Marcin Poreba et al. CHEMICAL REVIEWS
- Noninvasive Molecular Imaging of Apoptosis in a Mouse Model of Anthracycline-Induced Cardiotoxicity
- (2015) H. Su et al. Circulation-Cardiovascular Imaging
- A Systematic Comparison of 18F-C-SNAT to Established Radiotracer Imaging Agents for the Detection of Tumor Response to Treatment
- (2015) T. H. Witney et al. CLINICAL CANCER RESEARCH
- Bioresponsive probes for molecular imaging: concepts andin vivoapplications
- (2015) Sander M. J. van Duijnhoven et al. Contrast Media & Molecular Imaging
- Isatin sulfonamides: potent caspases-3 and -7 inhibitors, and promising PET and SPECT radiotracers for apoptosis imaging
- (2015) Panupun Limpachayaporn et al. Future Medicinal Chemistry
- Blocking of Fatty Acid Amide Hydrolase Activity with PF-04457845 in Human Brain: A Positron Emission Tomography Study with the Novel Radioligand [11C]CURB
- (2015) Isabelle Boileau et al. JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM
- The Fatty Acid Amide Hydrolase C385A Variant Affects Brain Binding of the Positron Emission Tomography Tracer [11C]CURB
- (2015) Isabelle Boileau et al. JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM
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- (2014) Sander M. J. van Duijnhoven et al. Contrast Media & Molecular Imaging
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- (2014) Changning Wang et al. JOURNAL OF MEDICINAL CHEMISTRY
- In Vivo Imaging of Human Acetylcholinesterase Density in Peripheral Organs Using 11C-Donepezil: Dosimetry, Biodistribution, and Kinetic Analyses
- (2014) T. Gjerloff et al. JOURNAL OF NUCLEAR MEDICINE
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- (2014) D. Dick JOURNAL OF NUCLEAR MEDICINE
- Whole-Body Radiation Dosimetry of 11C-Carbonyl-URB694: A PET Tracer for Fatty Acid Amide Hydrolase
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- (2014) Timothy M. Shoup et al. MOLECULAR IMAGING AND BIOLOGY
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- PET Imaging of Fatty Acid Amide Hydrolase with [18F]DOPP in Nonhuman Primates
- (2014) Benjamin H. Rotstein et al. MOLECULAR PHARMACEUTICS
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- (2014) Justin W. Hicks et al. NUCLEAR MEDICINE AND BIOLOGY
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- (2014) Tadashi Watabe et al. PLoS One
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- (2014) Benjamin H. Rotstein et al. Nature Communications
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- (2013) Zhibo Liu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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- (2013) Oleg Sadovski et al. BIOORGANIC & MEDICINAL CHEMISTRY
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- (2013) Hiroyuki Kimura et al. BIOORGANIC & MEDICINAL CHEMISTRY
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- (2013) Balasubramanian Gopalan et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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- (2013) Young Jun Seo et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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- (2013) Eric W. Price et al. CHEMICAL SOCIETY REVIEWS
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- (2008) Aleksey G. Kazantsev et al. NATURE REVIEWS DRUG DISCOVERY
- Targeting the endocannabinoid system: to enhance or reduce?
- (2008) Vincenzo Di Marzo NATURE REVIEWS DRUG DISCOVERY
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