Stoichiometric Leverage: Rapid18F-Aryltrifluoroborate Radiosynthesis at High Specific Activity for Click Conjugation

Efficient Method for Site-Specific 18F-Labeling of Biomolecules Using the Rapid Condensation Reaction between 2-Cyanobenzothiazole and Cysteine

(2012) Jongho Jeon et al.   BIOCONJUGATE CHEMISTRY

A historical perspective on the specific activity of radiopharmaceuticals: what have we learned in the 35 years of the ISRC?

(2012) Suzanne E. Lapi et al.   NUCLEAR MEDICINE AND BIOLOGY

Biomedical Applications of Tetrazine Cycloadditions

(2011) Neal K. Devaraj et al.   ACCOUNTS OF CHEMICAL RESEARCH

18F-PEG-biotin: Precursor (boroaryl-PEG-biotin) synthesis, 18F-labelling and an in-vitro assessment of its binding with Neutravidin™–trastuzumab pre-treated cells

(2011) Tim A.D. Smith et al.   APPLIED RADIATION AND ISOTOPES

Rapid and Simple One-Step F-18 Labeling of Peptides

(2011) Orit Jacobson et al.   BIOCONJUGATE CHEMISTRY

High-Yielding Aqueous18F-Labeling of Peptides via Al18F Chelation

(2011) Christopher A. D’Souza et al.   BIOCONJUGATE CHEMISTRY

New F-18 Prosthetic Group via Oxime Coupling

(2011) Patrick Carberry et al.   BIOCONJUGATE CHEMISTRY

Oxalic Acid Supported Si–18F-Radiofluorination: One-Step Radiosynthesis of N-Succinimidyl 3-(Di-tert-butyl[18F]fluorosilyl)benzoate ([18F]SiFB) for Protein Labeling

(2011) Alexey P. Kostikov et al.   BIOCONJUGATE CHEMISTRY

Rapid aqueous [18F]-labeling of a bodipy dye for positron emission tomography/fluorescence dual modality imaging

(2011) Zibo Li et al.   CHEMICAL COMMUNICATIONS

Inorganic approaches for radiolabelling biomolecules with fluorine-18 for imaging with Positron Emission Tomography

(2011) Gareth E. Smith et al.   DALTON TRANSACTIONS

Chelating Agents and their Use in Radiopharmaceutical Sciences

(2011) B. Wangler et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Development of 18F-fluorinatable dendrons and their application to cancer cell targeting

(2011) Laurent Trembleau et al.   NEW JOURNAL OF CHEMISTRY

A Fluoride-Derived Electrophilic Late-Stage Fluorination Reagent for PET Imaging

(2011) E. Lee et al.   SCIENCE

SiFA Azide: A New Building Block for PET Imaging Using Click Chemistry

(2011) Lutz Tietze et al.   SYNLETT

Towards kit-like 18F-labeling of marimastat, a noncovalent inhibitor drug for in vivo PET imaging cancer associated matrix metalloproteases

(2011) Ying Li et al.   MedChemComm

Peptide-Based Probes for Targeted Molecular Imaging

(2010) Seulki Lee et al.   BIOCHEMISTRY

Radiosynthesis and Biodistribution of a Prosthetic Group (18F-FENMA) Conjugated to Cyclic RGD Peptides

(2010) Dag Erlend Olberg et al.   BIOCONJUGATE CHEMISTRY

Fast18F Labeling of a Near-Infrared Fluorophore Enables Positron Emission Tomography and Optical Imaging of Sentinel Lymph Nodes

(2010) Richard Ting et al.   BIOCONJUGATE CHEMISTRY

Novel Matrix Metalloproteinase Inhibitor [18F]Marimastat-Aryltrifluoroborate as a Probe for In vivo Positron Emission Tomography Imaging in Cancer

(2010) U. auf dem Keller et al.   CANCER RESEARCH

Stabilization of zwitterionic aryltrifluoroborates against hydrolysis

(2010) Casey R. Wade et al.   CHEMICAL COMMUNICATIONS

Peptides and Peptide Hormones for Molecular Imaging and Disease Diagnosis

(2010) Seulki Lee et al.   CHEMICAL REVIEWS

A Novel Facile Method of Labeling Octreotide with 18F-Fluorine

(2010) P. Laverman et al.   JOURNAL OF NUCLEAR MEDICINE

Direct One-Step18F-Labeling of Peptides via Nucleophilic Aromatic Substitution

(2009) Jessica Becaud et al.   BIOCONJUGATE CHEMISTRY

Radiolabeled Cyclic RGD Peptides as Integrin αvβ3-Targeted Radiotracers: Maximizing Binding Affinity via Bivalency

(2009) Shuang Liu   BIOCONJUGATE CHEMISTRY

New Strategy for the Preparation of Clickable Peptides and Labeling with 1-(Azidomethyl)-4-[18F]-fluorobenzene for PET

(2009) David Thonon et al.   BIOCONJUGATE CHEMISTRY

Modular strategies for PET imaging agents

(2009) Jacob M Hooker   CURRENT OPINION IN CHEMICAL BIOLOGY

Teflon radiolysis as the major source of carrier in fluorine-18

(2009) M. S. Berridge et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Single-Step High-Yield Radiosynthesis and Evaluation of a Sensitive18F-Labeled Ligand for Imaging Brain Peripheral Benzodiazepine Receptors with PET

(2009) Emmanuelle Briard et al.   JOURNAL OF MEDICINAL CHEMISTRY

High-throughput in vivo screening of targeted molecular imaging agents

(2009) M. K. J. Gagnon et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Synthesis and Application of [18F]FDG-Maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-Based Prosthetic Group for the Chemoselective18F-Labeling of Peptides and Proteins†

(2008) Frank Wuest et al.   BIOCONJUGATE CHEMISTRY

Chemistry with [18F]Fluoride Ion

(2008) Lisheng Cai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Capturing aqueous [18F]-fluoride with an arylboronic ester for PET: Synthesis and aqueous stability of a fluorescent [18F]-labeled aryltrifluoroborate

(2008) Richard Ting et al.   JOURNAL OF FLUORINE CHEMISTRY

In Vivo Positron Emission Tomography (PET) Imaging with an αvβ6Specific Peptide Radiolabeled using18F-“Click” Chemistry: Evaluation and Comparison with the Corresponding 4-[18F]Fluorobenzoyl- and 2-[18F]Fluoropropionyl-Peptides

(2008) Sven H. Hausner et al.   JOURNAL OF MEDICINAL CHEMISTRY

Substituent Effects on Aryltrifluoroborate Solvolysis in Water: Implications for Suzuki−Miyaura Coupling and the Design of Stable18F-Labeled Aryltrifluoroborates for Use in PET Imaging

(2008) Richard Ting et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of masked haloareneboronic acids via iridium-catalyzed aromatic C–H borylation with 1,8-naphthalenediaminatoborane (danBH)

(2008) Noriyuki Iwadate et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Toward [18F]-Labeled Aryltrifluoroborate Radiotracers: In Vivo Positron Emission Tomography Imaging of Stable Aryltrifluoroborate Clearance in Mice

(2008) Richard Ting et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

True radiotracers: are we approaching theoretical specific activity with Tc-99m and I-123?

(2008) William C. Eckelman et al.   NUCLEAR MEDICINE AND BIOLOGY

Differentially Protected Benzenediboronic Acids:  Divalent Cross-Coupling Modules for the Efficient Synthesis of Boron-Substituted Oligoarenes

(2008) Hiroyoshi Noguchi et al.   ORGANIC LETTERS