Synthesis of 4,5-disubstituted-2-thioxo-1,2,3,4-tetrahydropyrimidines and investigation of their acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase I/II inhibitory and antioxidant activities

Isatin analogs as novel inhibitors of Candida spp. β-carbonic anhydrase enzymes

(2016) Atilla Akdemir et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds

(2016) Bünyamin Özgeriş et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Comparison of the sulfonamide inhibition profiles of the α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae

(2016) Sonia Del Prete et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Acetylcholinesterase Inhibitory and Antioxidant Activities of Novel Symmetric Sulfamides Derived from Phenethylamines

(2015) Kadir Aksu et al.   ARCHIV DER PHARMAZIE

Discovery of potent carbonic anhydrase and acetylcholine esterase inhibitors: Novel sulfamoylcarbamates and sulfamides derived from acetophenones

(2015) Akın Akıncıoğlu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II

(2015) Alper Yıldırım et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Antioxidant and acetylcholinesterase inhibition properties of novel bromophenol derivatives

(2015) Necla Öztaşkın et al.   BIOORGANIC CHEMISTRY

Synthesis of 4-[2-(3,4-dimethoxybenzyl)cyclopentyl]-1,2-dimethoxybenzene Derivatives and Evaluations of Their Carbonic Anhydrase Isoenzymes Inhibitory Effects

(2015) Tekin Artunç et al.   Chemical Biology & Drug Design

LC–MS/MS analysis, antioxidant and anticholinergic properties of galanga (Alpinia officinarum Hance) rhizomes

(2015) Leyla Polat Köse et al.   INDUSTRIAL CROPS AND PRODUCTS

Purification and Characterization of Polyphenol Oxidase from Hemşin Apple (Malus communisL.)

(2015) Bahar Aydin et al.   INTERNATIONAL JOURNAL OF FOOD PROPERTIES

Determination of Antioxidant Properties of Gypsophila bitlisensis Bark.

(2015) Hatice Tohma et al.   International Journal of Pharmacology

Dithiocarbamates with potent inhibitory activity against theSaccharomyces cerevisiaeβ-carbonic anhydrase

(2015) Murat Bozdag et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Tacrine–propargylamine derivatives with improved acetylcholinesterase inhibitory activity and lower hepatotoxicity as a potential lead compound for the treatment of Alzheimer’s disease

(2015) Fei Mao et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors

(2015) Mariangela Ceruso et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Protonography, a technique applicable for the analysis ofη-carbonic anhydrase activity

(2015) Sonia Del Prete et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII)

(2015) Andrea Scozzafava et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Antioxidant, antiradical, and anticholinergic properties of cynarin purified from the Illyrian thistle (Onopordum illyricumL.)

(2015) Meryem Topal et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Antioxidant activity of taxifolin: an activity–structure relationship

(2015) Fevzi Topal et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of 4-(2-substituted hydrazinyl)benzenesulfonamides and their carbonic anhydrase inhibitory effects

(2015) Halise Inci Gul et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The effects of some bromophenols on human carbonic anhydrase isoenzymes

(2015) Parham Taslimi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The human carbonic anhydrase isoenzymes I and II (hCA I and II) inhibition effects of trimethoxyindane derivatives

(2015) Parham Taslimi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

How many carbonic anhydrase inhibition mechanisms exist?

(2015) Claudiu T. Supuran   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and Carbonic Anhydrase Inhibitory Effects of Novel Sulfamides Derived from 1-Aminoindanes and Anilines

(2014) Yusuf Akbaba et al.   ARCHIV DER PHARMAZIE

Synthesis and Carbonic Anhydrase Isoenzymes Inhibitory Effects of Brominated Diphenylmethanone and Its Derivatives

(2014) Yasin Çetinkaya et al.   ARCHIV DER PHARMAZIE

Oxidation of cyanobenzocycloheptatrienes: Synthesis, photooxygenation reaction and carbonic anhydrase isoenzymes inhibition properties of some new benzotropone derivatives

(2014) Murat Güney et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum —The η-carbonic anhydrases

(2014) Sonia Del Prete et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Carbonic anhydrase inhibitory properties of novel benzylsulfamides using molecular modeling and experimental studies

(2014) Süleyman Göksu et al.   BIOORGANIC CHEMISTRY

The η-class carbonic anhydrases as drug targets for antimalarial agents

(2014) Claudiu T Supuran et al.   EXPERT OPINION ON THERAPEUTIC TARGETS

Antioxidant capacity and functionality of oleaster (Elaeagnus angustifoliaL.) flour and crust in a new kind of fruity ice cream

(2014) Songül Çakmakçı et al.   INTERNATIONAL JOURNAL OF FOOD SCIENCE AND TECHNOLOGY

Inhibition profile of a series of phenolic acids on bovine lactoperoxidase enzyme

(2014) S. Beyza Ozturk Sarikaya et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Pistachio (Pistacia veraL.) Gum: a potent inhibitor of reactive oxygen species

(2014) M. Hilal Sehitoglu et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Carbonic anhydrase and acetylcholinesterase inhibitory effects of carbamates and sulfamoylcarbamates

(2014) Hülya Göçer et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitors: guaiacol and catechol derivatives effectively inhibit certain human carbonic anhydrase isoenzymes (hCA I, II, IX and XII)

(2014) Andrea Scozzafava et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties

(2014) Murat Boztaş et al.   JOURNAL OF MEDICINAL CHEMISTRY

Capsaicin: A Potent Inhibitor of Carbonic Anhydrase Isoenzymes

(2014) Betul Arabaci et al.   MOLECULES

Rosmarinic acid: a potent carbonic anhydrase isoenzymes inhibitor

(2014) Meryem TOPAL et al.   TURKISH JOURNAL OF CHEMISTRY

Colorimetric and Fluorometric Assays Based on Conjugated Polydiacetylene Supramolecules for Screening Acetylcholinesterase and Its Inhibitors

(2013) Guodong Zhou et al.   ACS Applied Materials & Interfaces

Novel Sulphamides and Sulphonamides Incorporating the Tetralin Scaffold as Carbonic Anhydrase and Acetylcholine Esterase Inhibitors

(2013) Akın Akıncıoğlu et al.   ARCHIV DER PHARMAZIE

Synthesis, Antioxidant, and Antiacetylcholinesterase Activities of Sulfonamide Derivatives of Dopamine-Related Compounds

(2013) Hülya Göçer et al.   ARCHIV DER PHARMAZIE

Carbonic anhydrases

(2013) Claudiu T. Supuran   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine

(2013) Kadir Aksu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Exploiting the hydrophobic and hydrophilic binding sites for designing carbonic anhydrase inhibitors

(2013) Giuseppina De Simone et al.   Expert Opinion on Drug Discovery

Anti-infective carbonic anhydrase inhibitors: a patent and literature review

(2013) Clemente Capasso et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Diuretics with carbonic anhydrase inhibitory action: a patent and literature review (2005 – 2013)

(2013) Fabrizio Carta et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins

(2013) Yusuf Akbaba et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and carbonic anhydrase isoenzymes I and II inhibitory effects of novel benzylamine derivatives

(2013) Yasin Çetinkaya et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and Kinetic Testing of Tetrahydropyrimidine-2-thione and Pyrrole Derivatives as Inhibitors of the Metallo-β-lactamase fromKlebsiella pneumoniaandPseudomonas aeruginosa

(2012) Waleed M. Hussein et al.   Chemical Biology & Drug Design

Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1H)-ones as Sodium Iodide Symporter Inhibitors

(2012) Pierre Lacotte et al.   ChemMedChem

One-step purification of lactoperoxidase from bovine milk by affinity chromatography

(2012) Ali Atasever et al.   FOOD CHEMISTRY

Antioxidant activity and polyphenol content of cherry stem (Cerasus avium L.) determined by LC–MS/MS

(2012) Ercan Bursal et al.   FOOD RESEARCH INTERNATIONAL

(3,4-Dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and its derivatives as carbonic anhydrase isoenzymes inhibitors

(2012) Meryem Nar et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and Antioxidant Properties of (3,4-Dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and Its Derivatives

(2011) Yasin Çetinkaya et al.   ARCHIV DER PHARMAZIE

Antioxidant activity of food constituents: an overview

(2011) İlhami Gülçin   ARCHIVES OF TOXICOLOGY

Evaluation of dihydropyrimidin-(2H)-one analogues and rhodanine derivatives as tyrosinase inhibitors

(2011) Jinbing Liu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compounds

(2011) Sevim Beyza Öztürk Sarikaya et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

In Vitro Inhibition of Human Carbonic Anhydrase I and II Isozymes with Natural Phenolic Compounds

(2011) Murat Şentürk et al.   Chemical Biology & Drug Design

Polyphenol contents and in vitro antioxidant activities of lyophilised aqueous extract of kiwifruit (Actinidia deliciosa)

(2011) Ercan Bursal et al.   FOOD RESEARCH INTERNATIONAL

Caffeic acid phenethyl ester (CAPE): correlation of structure and antioxidant properties

(2011) Hülya Göçer et al.   INTERNATIONAL JOURNAL OF FOOD SCIENCES AND NUTRITION

Apoptotic, antioxidant and antiradical effects of majdine and isomajdine fromVinca herbaceaWaldst. and kit

(2011) I˙lhami Gülçi˙n et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Pomological Features, Nutritional Quality, Polyphenol Content Analysis, and Antioxidant Properties of Domesticated and 3 Wild Ecotype Forms of Raspberries (Rubus idaeus L.)

(2011) İlhami Gülçin et al.   JOURNAL OF FOOD SCIENCE

Antioxidant Activity of Eugenol: A Structure–Activity Relationship Study

(2011) İlhami Gülçin   JOURNAL OF MEDICINAL FOOD

Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I–XIV with a series of natural product polyphenols and phenolic acids

(2010) Alessio Innocenti et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitors. Antioxidant polyphenols effectively inhibit mammalian isoforms I–XV

(2010) Alessio Innocenti et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Carbonic Anhydrase Inhibitors: Inhibition of Human Erythrocyte Isozymes I and II with a Series of Phenolic Acids

(2010) S. Beyza Öztürk Sarıkaya et al.   Chemical Biology & Drug Design

Polyphenol contents and antioxidant activity of lyophilized aqueous extract of propolis from Erzurum, Turkey

(2010) İlhami Gülçin et al.   FOOD AND CHEMICAL TOXICOLOGY

Antioxidant, Antimicrobial, Antifungal, and Antiradical Activities ofCyclotrichium Niveum(BOISS.) Manden and Scheng

(2010) Ilhami Gulcin et al.   INTERNATIONAL JOURNAL OF FOOD PROPERTIES

Antioxidant and Radical Scavenging Activity of Aerial Parts and Roots of Turkish Liquorice (Glycyrrhiza Glabra L.)

(2010) Hatice Serbetci Tohma et al.   INTERNATIONAL JOURNAL OF FOOD PROPERTIES

Synthesis and antioxidant properties of diphenylmethane derivative bromophenols including a natural product

(2010) Halis Türker Balaydın et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Efficient, Green, Solvent-Free Synthesis of 3,4-Dihydropyrimidin-2(1H)-ones via Biginelli Reaction Catalyzed by Cu(NO3)2·3H2O

(2010) Dong-Chao Wang et al.   SYNTHETIC COMMUNICATIONS

Antioxidant activity of clove oil – A powerful antioxidant source

(2010) İlhami Gülçin et al.   Arabian Journal of Chemistry

Antioxidant activity of 5,10-dihydroindeno[1,2-b]indoles containing substituents on dihydroindeno part

(2009) Oktay Talaz et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols

(2009) Murat Şentürk et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Antioxidant properties of resveratrol: A structure–activity insight

(2009) İlhami Gülçin   Innovative Food Science & Emerging Technologies

The effect of ethanol on erythrocyte carbonic anhydrase isoenzymes activity: An in vitro and in vivo study

(2009) T. Abdulkadir Çoban et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Antioxidant activity of bisbenzylisoquinoline alkaloids from Stephania rotunda: cepharanthine and fangchinoline

(2009) İlhami Gülçin et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Highly Enantioselective Organocatalytic Biginelli and Biginelli-Like Condensations: Reversal of the Stereochemistry by Tuning the 3,3′-Disubstituents of Phosphoric Acids

(2009) Nan Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An improved synthesis of Biginelli-type compounds via phase-transfer catalysis

(2009) Bahar Ahmed et al.   TETRAHEDRON LETTERS

Radical scavenging and antioxidant activity of tannic acid

(2009) İlhami Gülçin et al.   Arabian Journal of Chemistry

Antioxidant and radical scavenging properties of curcumin

(2008) Tuba Ak et al.   CHEMICO-BIOLOGICAL INTERACTIONS

Antioxidant activity of l-adrenaline: A structure–activity insight

(2008) İlhami Gülçin   CHEMICO-BIOLOGICAL INTERACTIONS

Measurement of antioxidant ability of melatonin and serotonin by the DMPD and CUPRAC methods as trolox equivalent

(2008) Ilhami Gülçin   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

In vitroantioxidant activity of silymarin

(2008) Ekrem KÖksal et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Carbamates with Differential Mechanism of Inhibition Toward Acetylcholinesterase and Butyrylcholinesterase

(2008) Sultan Darvesh et al.   JOURNAL OF MEDICINAL CHEMISTRY

Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

(2008) Claudiu T. Supuran   NATURE REVIEWS DRUG DISCOVERY

Antioxidant secoiridoids from fringe tree (Chionanthus virginicus L.)

(2008) İlhami Gülçin et al.   WOOD SCIENCE AND TECHNOLOGY