Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors
Published 2015 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors
Authors
Keywords
-
Journal
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Volume 31, Issue 2, Pages 205-211
Publisher
Informa UK Limited
Online
2015-03-20
DOI
10.3109/14756366.2015.1014477
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- New series of sulfonamides containing amino acid moiety act as effective and selective inhibitors of tumor-associated carbonic anhydrase XII
- (2014) Mariangela Ceruso et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Sulfonamides with Potent Inhibitory Action and Selectivity against the α-Carbonic Anhydrase from Vibrio cholerae
- (2014) Mariangela Ceruso et al. ACS Medicinal Chemistry Letters
- Carbonic anhydrases
- (2013) Claudiu T. Supuran BIOORGANIC & MEDICINAL CHEMISTRY
- Hypoxia induced CA9 inhibitory targeting by two different sulfonamide derivatives including Acetazolamide in human Glioblastoma
- (2013) Harun M. Said et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Exploiting the hydrophobic and hydrophilic binding sites for designing carbonic anhydrase inhibitors
- (2013) Giuseppina De Simone et al. Expert Opinion on Drug Discovery
- Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
- (2012) Vincenzo Alterio et al. CHEMICAL REVIEWS
- Carbonic Anhydrase IX Promotes Tumor Growth and Necrosis In Vivo and Inhibition Enhances Anti-VEGF Therapy
- (2012) A. McIntyre et al. CLINICAL CANCER RESEARCH
- Sulfonamides: a patent review (2008 – 2012)
- (2012) Fabrizio Carta et al. EXPERT OPINION ON THERAPEUTIC PATENTS
- Structure-based drug discovery of carbonic anhydrase inhibitors
- (2012) Claudiu T. Supuran JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Function of carbonic anhydrase IX in glioblastoma multiforme
- (2012) M. A. Proescholdt et al. NEURO-ONCOLOGY
- Carbonic anhydrase inhibitors and activators for novel therapeutic applications
- (2011) Claudiu T Supuran Future Medicinal Chemistry
- Ureido-Substituted Benzenesulfonamides Potently Inhibit Carbonic Anhydrase IX and Show Antimetastatic Activity in a Model of Breast Cancer Metastasis
- (2011) Fabio Pacchiano et al. JOURNAL OF MEDICINAL CHEMISTRY
- Interfering with pH regulation in tumours as a therapeutic strategy
- (2011) Dario Neri et al. NATURE REVIEWS DRUG DISCOVERY
- Carbonic anhydrase inhibitors
- (2010) Claudiu T. Supuran BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Carbonic anhydrase IX: Biochemical and crystallographic characterization of a novel antitumor target
- (2009) Giuseppina De Simone et al. BIOCHIMICA ET BIOPHYSICA ACTA-PROTEINS AND PROTEOMICS
- Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX
- (2009) V. Alterio et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Imaging of CA IX with fluorescent labelled sulfonamides distinguishes hypoxic and (re)-oxygenated cells in a xenograft tumour model
- (2009) Ludwig Dubois et al. RADIOTHERAPY AND ONCOLOGY
- Estrogen Receptor Regulation of Carbonic Anhydrase XII through a Distal Enhancer in Breast Cancer
- (2008) D. H. Barnett et al. CANCER RESEARCH
- Carbonic anhydrases: novel therapeutic applications for inhibitors and activators
- (2008) Claudiu T. Supuran NATURE REVIEWS DRUG DISCOVERY
- Identification of an alternatively spliced isoform of carbonic anhydrase XII in diffusely infiltrating astrocytic gliomas
- (2008) Joonas Haapasalo et al. NEURO-ONCOLOGY
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreAdd your recorded webinar
Do you already have a recorded webinar? Grow your audience and get more views by easily listing your recording on Peeref.
Upload Now