Novel hypervalent iodine catalyzed synthesis of α-sulfonoxy ketones: Biological activity and molecular docking studies

Design, synthesis, molecular docking, and some metabolic enzyme inhibition properties of novel quinazolinone derivatives

(2021) Feyzi S. Tokalı et al.   ARCHIV DER PHARMAZIE

Potent Acetylcholinesterase Inhibitors: Potential Drugs for Alzheimer’s Disease

(2020) Hulya Akıncıoğlu et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

N ‐Substituted pyrimidinethione and acetophenone derivatives as a new therapeutic approach in diabetes

(2020) Parham Taslimi et al.   ARCHIV DER PHARMAZIE

Quinoline‐based promising anticancer and antibacterial agents, and some metabolic enzyme inhibitors

(2020) Salih Ökten et al.   ARCHIV DER PHARMAZIE

Synthesis, characterization, biological evaluation, and in silico studies of novel 1,3‐diaryltriazene‐substituted sulfathiazole derivatives

(2020) Mesut Işık et al.   ARCHIV DER PHARMAZIE

Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds – Determination of their carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibition properties

(2020) İlhami Gülçin et al.   BIOORGANIC CHEMISTRY

Synthesis, characterization, biological activity and molecular docking studies of novel schiff bases derived from thiosemicarbazide: Biochemical and computational approach

(2020) Feyzi Sinan Tokalı et al.   JOURNAL OF MOLECULAR STRUCTURE

Synthesis, crystal structure, and biological evaluation of optically active 2-amino-4-aryl-7,7-dimethyl-5-oxo-5,6,7,8-tetrahydro-4H -chromen-3-carbonitriles: Antiepileptic, antidiabetic, and anticholinergics potentials

(2019) Abel Maharramov et al.   ARCHIV DER PHARMAZIE

Phytochemical content, antioxidant activity, and enzyme inhibition effect of Salvia eriophora Boiss. & Kotschy against acetylcholinesterase, α-amylase, butyrylcholinesterase, and α-glycosidase enzymes

(2019) Ercan Bursal et al.   JOURNAL OF FOOD BIOCHEMISTRY

Synthesis, characterization, molecular docking and biological activities of novel pyrazoline derivatives

(2019) Fikret Turkan et al.   ARCHIV DER PHARMAZIE

Synthesis of Oxazolidinone from Enantiomerically Enriched Allylic Alcohols and Determination of Their Molecular Docking and Biologic Activities

(2019) Ufuk Atmaca et al.   BIOORGANIC CHEMISTRY

Mono- or di-substituted imidazole derivatives for inhibition of acetylcholine and butyrylcholine esterases

(2019) Burak Kuzu et al.   BIOORGANIC CHEMISTRY

Synthesis, biological evaluation and molecular docking of novel pyrazole derivatives as potent carbonic anhydrase and acetylcholinesterase inhibitors

(2019) Fikret Turkan et al.   BIOORGANIC CHEMISTRY

Synthesis and biological evaluation of bromophenol derivatives with cyclopropyl moiety: Ring opening of cyclopropane with monoester

(2019) Murat Boztas et al.   BIOORGANIC CHEMISTRY

Synthesis and biological evaluation of novel tris-chalcones as potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibitors

(2019) Serdar Burmaoglu et al.   BIOORGANIC CHEMISTRY

Investigation of inhibitory properties of some hydrazone compounds on hCA I, hCA II and AChE enzymes

(2019) Kaan Kucukoglu et al.   BIOORGANIC CHEMISTRY

Sage (Salvia pilifera): determination of its polyphenol contents, anticholinergic, antidiabetic and antioxidant activities

(2019) İlhami Gülçin et al.   Journal of Food Measurement and Characterization

Novel eugenol bearing oxypropanolamines: Synthesis, characterization, antibacterial, antidiabetic, and anticholinergic potentials

(2019) Hayriye Genç Bilgiçli et al.   BIOORGANIC CHEMISTRY

The green synthesis and molecular docking of novel N-substituted rhodanines as effective inhibitors for carbonic anhydrase and acetylcholinesterase enzymes

(2019) Sinan Bayindir et al.   BIOORGANIC CHEMISTRY

5-Arylisothiazol-3(2H)-one-1,(1)-(di)oxides: A new class of selective tumor-associated carbonic anhydrases (hCA IX and XII) inhibitors

(2019) Benedetta Cornelio et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pyrazole[3,4-d]pyridazine derivatives: Molecular docking and explore of acetylcholinesterase and carbonic anhydrase enzymes inhibitors as anticholinergics potentials

(2019) Parham Taslimi et al.   BIOORGANIC CHEMISTRY

Novel 2-methylimidazolium salts: Synthesis, characterization, molecular docking, and carbonic anhydrase and acetylcholinesterase inhibitory properties

(2019) Selma Bal et al.   BIOORGANIC CHEMISTRY

Novel 2-aminopyridine liganded Pd(II) N-heterocyclic carbene complexes: Synthesis, characterization, crystal structure and bioactivity properties

(2019) Fatoş Erdemir et al.   BIOORGANIC CHEMISTRY

Novel tribenzylaminobenzolsulphonylimine based on their pyrazine and pyridazines: Synthesis, characterization, antidiabetic, anticancer, anticholinergic, and molecular docking studies

(2019) Gulnar Mamedova et al.   BIOORGANIC CHEMISTRY

meta -Cyanobenzyl substituted benzimidazolium salts: Synthesis, characterization, crystal structure and carbonic anhydrase, α-glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties

(2018) Ferhat Türker et al.   ARCHIV DER PHARMAZIE

The in vivo effects of cefazolin, cefuroxime, and cefoperazon on the carbonic anhydrase in different rat tissues

(2018) Fikret Türkan et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Antioxidant and anticholinergic properties of olivetol

(2018) Parham Taslimi et al.   JOURNAL OF FOOD BIOCHEMISTRY

Synthesis, characterization and crystal structure of 2-(4-hydroxyphenyl)ethyl and 2-(4-nitrophenyl)ethyl Substituted Benzimidazole Bromide Salts: Their inhibitory properties against carbonic anhydrase and acetylcholinesterase

(2018) Ayten Behçet et al.   JOURNAL OF MOLECULAR STRUCTURE

2-Hydroxyethyl substituted NHC precursors: Synthesis, characterization, crystal structure and carbonic anhydrase, α-glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties

(2018) Fatoş Erdemir et al.   JOURNAL OF MOLECULAR STRUCTURE

The effects of some antibiotics from cephalosporin groups on the acetylcholinesterase and butyrylcholinesterase enzymes activities in different tissues of rats

(2018) Fikret Türkan et al.   ARCHIVES OF PHYSIOLOGY AND BIOCHEMISTRY

Combined in Vitro and in Silico Studies for the Anticholinesterase Activity and Pharmacokinetics of Coumarinyl Thiazoles and Oxadiazoles

(2018) Aliya Ibrar et al.   Frontiers in Chemistry

Novel Benzylic Substituted Imidazolinium, Tetrahydropyrimidinium and Tetrahydrodiazepinium Salts: Potent Carbonic Anhydrase and Acetylcholinesterase Inhibitors

(2018) Beyhan Yiğit et al.   ChemistrySelect

Novel thymol bearing oxypropanolamine derivatives as potent some metabolic enzyme inhibitors – Their antidiabetic, anticholinergic and antibacterial potentials

(2018) Mustafa Zengin et al.   BIOORGANIC CHEMISTRY

Antidiabetic and antiparasitic potentials: Inhibition effects of some natural antioxidant compounds on α-glycosidase, α-amylase and human glutathione S-transferase enzymes

(2018) İlhami Gulçin et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Synthesis, characterization, crystal structure, electrochemical studies and biological evaluation of metal complexes with thiosemicarbazone of glyoxylic acid

(2018) Mansura Huseynova et al.   POLYHEDRON

Screening the in vitro antioxidant, antimicrobial, anticholinesterase, antidiabetic activities of endemic Achillea cucullata (Asteraceae) ethanol extract

(2018) N. Eruygur et al.   SOUTH AFRICAN JOURNAL OF BOTANY

The effects of hesperidin on sodium arsenite-induced different organ toxicity in rats on metabolic enzymes as antidiabetic and anticholinergics potentials: A biochemical approach

(2018) Cuneyt Caglayan et al.   JOURNAL OF FOOD BIOCHEMISTRY

Synthesis, characterization, crystal structures, theoretical calculations and biological evaluations of novel substituted tacrine derivatives as cholinesterase and carbonic anhydrase enzymes inhibitors

(2018) Salih Ökten et al.   JOURNAL OF MOLECULAR STRUCTURE

Novel morpholine liganded Pd-based N-heterocyclic carbene complexes: Synthesis, characterization, crystal structure, antidiabetic and anticholinergic properties

(2018) Aydın Aktaş et al.   POLYHEDRON

One-pot four-component synthesis of thiazolidin-2-imines using CuI/ZnII dual catalysis: A new class of acetylcholinesterase inhibitors

(2018) Syeda Aaliya Shehzadi et al.   BIOORGANIC CHEMISTRY

Synthesis, characterization, crystal structure of novel bis-thiomethylcyclohexanone derivatives and their inhibitory properties against some metabolic enzymes

(2018) Abdullah Biçer et al.   BIOORGANIC CHEMISTRY

The first synthesis, carbonic anhydrase inhibition and anticholinergic activities of some bromophenol derivatives with S including natural products

(2018) Cetin Bayrak et al.   BIOORGANIC CHEMISTRY

The toxicological effects of some avermectins on goat liver carbonic anhydrase enzyme

(2017) Cuneyt Caglayan et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Synephrine and phenylephrine act as α-amylase, α-glycosidase, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase enzymes inhibitors

(2017) Parham Taslimi et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Inhibition properties of some flavonoids on carbonic anhydrase I and II isoenzymes purified from human erythrocytes

(2017) Zübeyir Huyut et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Synthesis and investigation of the conversion reactions of pyrimidine-thiones with nucleophilic reagent and evaluation of their acetylcholinesterase, carbonic anhydrase inhibition, and antioxidant activities

(2017) Parham Taslimi et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Inhibition Effects of Some Lignans on Carbonic Anhydrase, Acetylcholinesterase and Butyrylcholinesterase Enzymes Leyla Polat Köse and İlhami Gülçin

(2017) Leyla Polat Köse et al.   Records of Natural Products

Synthesis and investigation of antibacterial activities and carbonic anhydrase and acetyl cholinesterase inhibition profiles of novel 4,5-dihydropyrazol and pyrazolyl-thiazole derivatives containing methanoisoindol-1,3-dion unit

(2017) Yakup Budak et al.   SYNTHETIC COMMUNICATIONS

Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles

(2017) Umit Muhammet Kocyigit et al.   ARCHIVES OF PHYSIOLOGY AND BIOCHEMISTRY

Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds

(2016) Bünyamin Özgeriş et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of diaryl ethers with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions

(2016) Fadime Özbey et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of 4,5-disubstituted-2-thioxo-1,2,3,4-tetrahydropyrimidines and investigation of their acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase I/II inhibitory and antioxidant activities

(2016) Emin Garibov et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of some tetrahydropyrimidine-5-carboxylates, determination of their metal chelating effects and inhibition profiles against acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase

(2016) Afsun Sujayev et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Perspectives for the structure-based design of acetylcholinesterase reactivators

(2016) Rodrigo Ochoa et al.   JOURNAL OF MOLECULAR GRAPHICS & MODELLING

X-ray crystallography-promoted drug design of carbonic anhydrase inhibitors

(2015) Jekaterina Ivanova et al.   CHEMICAL COMMUNICATIONS

LC–MS/MS analysis, antioxidant and anticholinergic properties of galanga (Alpinia officinarum Hance) rhizomes

(2015) Leyla Polat Köse et al.   INDUSTRIAL CROPS AND PRODUCTS

The effects of some bromophenols on human carbonic anhydrase isoenzymes

(2015) Parham Taslimi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Exploration of a library of triazolothiadiazole and triazolothiadiazine compounds as a highly potent and selective family of cholinesterase and monoamine oxidase inhibitors: design, synthesis, X-ray diffraction analysis and molecular docking studies

(2015) Imtiaz Khan et al.   RSC Advances

Synthesis and Carbonic Anhydrase Inhibitory Effects of Novel Sulfamides Derived from 1-Aminoindanes and Anilines

(2014) Yusuf Akbaba et al.   ARCHIV DER PHARMAZIE

Active compounds from a diverse library of triazolothiadiazole and triazolothiadiazine scaffolds: Synthesis, crystal structure determination, cytotoxicity, cholinesterase inhibitory activity, and binding mode analysis

(2014) Imtiaz Khan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitory properties of novel benzylsulfamides using molecular modeling and experimental studies

(2014) Süleyman Göksu et al.   BIOORGANIC CHEMISTRY

Synthesis, crystal structure and biological evaluation of some novel 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazines

(2014) Imtiaz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Oxidative Coupling of Terminal Alkyne with α-Hydroxy Ketone: An Expedient Approach toward Ynediones

(2014) Zeguang Zhang et al.   ORGANIC LETTERS

Oxidations of alkenes with hypervalent iodine reagents: an alternative ozonolysis of phenyl substituted alkenes and allylic oxidation of unsubstituted cyclic alkenes

(2014) Ufuk Atmaca et al.   TETRAHEDRON LETTERS

Novel Sulphamides and Sulphonamides Incorporating the Tetralin Scaffold as Carbonic Anhydrase and Acetylcholine Esterase Inhibitors

(2013) Akın Akıncıoğlu et al.   ARCHIV DER PHARMAZIE

Synthesis, Antioxidant, and Antiacetylcholinesterase Activities of Sulfonamide Derivatives of Dopamine-Related Compounds

(2013) Hülya Göçer et al.   ARCHIV DER PHARMAZIE

Novel sulfamides as potential carbonic anhydrase isoenzymes inhibitors

(2013) Akın Akıncıoğlu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine

(2013) Kadir Aksu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Structure-Based Search for New Inhibitors of Cholinesterases

(2013) Marek Bajda et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Structures of Human Acetylcholinesterase Bound to Dihydrotanshinone I and Territrem B Show Peripheral Site Flexibility

(2013) Jonah Cheung et al.   ACS Medicinal Chemistry Letters

Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

(2012) Vincenzo Alterio et al.   CHEMICAL REVIEWS

A step toward the reactivation of aged cholinesterases – Crystal structure of ligands binding to aged human butyrylcholinesterase

(2012) Marielle Wandhammer et al.   CHEMICO-BIOLOGICAL INTERACTIONS

One-step purification of lactoperoxidase from bovine milk by affinity chromatography

(2012) Ali Atasever et al.   FOOD CHEMISTRY

(3,4-Dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and its derivatives as carbonic anhydrase isoenzymes inhibitors

(2012) Meryem Nar et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

In Vitro Inhibition of Human Carbonic Anhydrase I and II Isozymes with Natural Phenolic Compounds

(2011) Murat Şentürk et al.   Chemical Biology & Drug Design

The Inhibitory Effects of L-Adrenaline on Lactoperoxidase Enzyme Purified from Bovine Milk

(2011) Melda Şisecioglu et al.   INTERNATIONAL JOURNAL OF FOOD PROPERTIES

Effects of Ceftazidime Pentahydrate, Prednisolone, Amikacin Sulfate, Ceftriaxone Sodium and Teicoplanin on Bovine Milk Lactoperoxidase Activity

(2011) M. Sisecioglu et al.   International Journal of Pharmacology

Oxidation reactions using polymer-supported 2-benzenesulfonyl-3-(4-nitrophenyl)oxaziridine

(2011) Woen Susanto et al.   TETRAHEDRON

Carbonic Anhydrase Inhibitors: Inhibition of Human Erythrocyte Isozymes I and II with a Series of Phenolic Acids

(2010) S. Beyza Öztürk Sarıkaya et al.   Chemical Biology & Drug Design

Pyrazine Biosynthesis in Corynebacterium glutamicum

(2010) Jeroen S. Dickschat et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols

(2009) Murat Şentürk et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Sildenafil is a strong activator of mammalian carbonic anhydrase isoforms I–XIV

(2009) T. Abdülkadir Coban et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Efficient one-pot synthesis of quinoxalines in the presence of zinc iodide as catalyst

(2009) J. N. Sangshetti et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

m-Iodosylbenzoic Acid: Recyclable Hypervalent Iodine Reagent for α-Tosyloxylation and α-Mesyloxylation of Ketones

(2009) Mekhman S. Yusubov et al.   SYNTHETIC COMMUNICATIONS

Chemistry of Polyvalent Iodine

(2008) Viktor V. Zhdankin et al.   CHEMICAL REVIEWS

Reductions of Benzene Derivatives Whose Benzylic Positions Bear Oxygen Atoms under Mild Conditions

(2008) Abdullah Menzek et al.   HELVETICA CHIMICA ACTA