Synthesis of diaryl ethers with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions

Application of PEG-400 as a green biodegradable polymeric medium for the catalyst-free synthesis of spiro-dihydropyridines and their use as acetyl and butyrylcholinesterase inhibitors

(2016) Ammar Maryamabadi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, molecular docking and biological evaluation of N,N-disubstituted 2-aminothiazolines as a new class of butyrylcholinesterase and carboxylesterase inhibitors

(2016) Galina F. Makhaeva et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds

(2016) Bünyamin Özgeriş et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and anti-acetylcholinesterase activity of scopoletin derivatives

(2016) Nisachon Khunnawutmanotham et al.   BIOORGANIC CHEMISTRY

Acetylcholinesterase Inhibitory and Antioxidant Activities of Novel Symmetric Sulfamides Derived from Phenethylamines

(2015) Kadir Aksu et al.   ARCHIV DER PHARMAZIE

Design, synthesis, and biological evaluation of a series of alkoxy-3-indolylacetic acids as peroxisome proliferator-activated receptor γ/δ agonists

(2015) Hyo Jin Gim et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of potent carbonic anhydrase and acetylcholine esterase inhibitors: Novel sulfamoylcarbamates and sulfamides derived from acetophenones

(2015) Akın Akıncıoğlu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II

(2015) Alper Yıldırım et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Antioxidant and acetylcholinesterase inhibition properties of novel bromophenol derivatives

(2015) Necla Öztaşkın et al.   BIOORGANIC CHEMISTRY

Synthesis of 4-[2-(3,4-dimethoxybenzyl)cyclopentyl]-1,2-dimethoxybenzene Derivatives and Evaluations of Their Carbonic Anhydrase Isoenzymes Inhibitory Effects

(2015) Tekin Artunç et al.   Chemical Biology & Drug Design

LC–MS/MS analysis, antioxidant and anticholinergic properties of galanga (Alpinia officinarum Hance) rhizomes

(2015) Leyla Polat Köse et al.   INDUSTRIAL CROPS AND PRODUCTS

The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII)

(2015) Andrea Scozzafava et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Antioxidant, antiradical, and anticholinergic properties of cynarin purified from the Illyrian thistle (Onopordum illyricumL.)

(2015) Meryem Topal et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of 4-(2-substituted hydrazinyl)benzenesulfonamides and their carbonic anhydrase inhibitory effects

(2015) Halise Inci Gul et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The effects of some bromophenols on human carbonic anhydrase isoenzymes

(2015) Parham Taslimi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The human carbonic anhydrase isoenzymes I and II (hCA I and II) inhibition effects of trimethoxyindane derivatives

(2015) Parham Taslimi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

How many carbonic anhydrase inhibition mechanisms exist?

(2015) Claudiu T. Supuran   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins

(2015) Marta Ferraroni et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Carbonic Anhydrase Inhibitory Effects of Novel Sulfamides Derived from 1-Aminoindanes and Anilines

(2014) Yusuf Akbaba et al.   ARCHIV DER PHARMAZIE

Synthesis and Carbonic Anhydrase Isoenzymes Inhibitory Effects of Brominated Diphenylmethanone and Its Derivatives

(2014) Yasin Çetinkaya et al.   ARCHIV DER PHARMAZIE

Oxidation of cyanobenzocycloheptatrienes: Synthesis, photooxygenation reaction and carbonic anhydrase isoenzymes inhibition properties of some new benzotropone derivatives

(2014) Murat Güney et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitory properties of novel benzylsulfamides using molecular modeling and experimental studies

(2014) Süleyman Göksu et al.   BIOORGANIC CHEMISTRY

An overview of the alpha-, beta- and gamma-carbonic anhydrases fromBacteria: can bacterial carbonic anhydrases shed new light on evolution of bacteria?

(2014) Clemente Capasso et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Carbonic anhydrase and acetylcholinesterase inhibitory effects of carbamates and sulfamoylcarbamates

(2014) Hülya Göçer et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitors: guaiacol and catechol derivatives effectively inhibit certain human carbonic anhydrase isoenzymes (hCA I, II, IX and XII)

(2014) Andrea Scozzafava et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties

(2014) Murat Boztaş et al.   JOURNAL OF MEDICINAL CHEMISTRY

Capsaicin: A Potent Inhibitor of Carbonic Anhydrase Isoenzymes

(2014) Betul Arabaci et al.   MOLECULES

Rosmarinic acid: a potent carbonic anhydrase isoenzymes inhibitor

(2014) Meryem TOPAL et al.   TURKISH JOURNAL OF CHEMISTRY

Synthesis and Biological Evaluation of Novel Bromophenol Derivatives as Carbonic Anhydrase Inhibitors

(2013) Yusuf Akbaba et al.   ARCHIV DER PHARMAZIE

Novel Sulphamides and Sulphonamides Incorporating the Tetralin Scaffold as Carbonic Anhydrase and Acetylcholine Esterase Inhibitors

(2013) Akın Akıncıoğlu et al.   ARCHIV DER PHARMAZIE

Synthesis, Antioxidant, and Antiacetylcholinesterase Activities of Sulfonamide Derivatives of Dopamine-Related Compounds

(2013) Hülya Göçer et al.   ARCHIV DER PHARMAZIE

Novel sulfamides as potential carbonic anhydrase isoenzymes inhibitors

(2013) Akın Akıncıoğlu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine

(2013) Kadir Aksu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitors: an editorial

(2013) Claudiu T Supuran   EXPERT OPINION ON THERAPEUTIC PATENTS

Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins

(2013) Yusuf Akbaba et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and carbonic anhydrase isoenzymes I and II inhibitory effects of novel benzylamine derivatives

(2013) Yasin Çetinkaya et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

(3,4-Dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and its derivatives as carbonic anhydrase isoenzymes inhibitors

(2012) Meryem Nar et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Diaryl ether derivatives as anticancer agents – a review

(2012) Florence Bedos-Belval et al.   MedChemComm

Kinetic and docking studies of phenol-based inhibitors of carbonic anhydrase isoforms I, II, IX and XII evidence a new binding mode within the enzyme active site

(2011) Serdar Durdagi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compounds

(2011) Sevim Beyza Öztürk Sarikaya et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

In Vitro Inhibition of Human Carbonic Anhydrase I and II Isozymes with Natural Phenolic Compounds

(2011) Murat Şentürk et al.   Chemical Biology & Drug Design

Thyronamines—Past, Present, and Future

(2011) S. Piehl et al.   ENDOCRINE REVIEWS

Inhibition of human carbonic anhydrase isozymes I, II and VI with a series of bisphenol, methoxy and bromophenol compounds

(2011) Halis Türker Balaydin et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Interfering with pH regulation in tumours as a therapeutic strategy

(2011) Dario Neri et al.   NATURE REVIEWS DRUG DISCOVERY

Pods of Khejri (Prosopis cineraria) consumed as a vegetable showed functional food properties

(2011) Yunbao Liu et al.   Journal of Functional Foods

Structure-based design, synthesis, and biological evaluation of lipophilic-tailed monocationic inhibitors of neuronal nitric oxide synthase

(2010) Fengtian Xue et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Bromophenols as Candida albicans isocitrate lyase inhibitors

(2010) Ki-Bong Oh et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

7,8-Disubstituted- but not 6,7-disubstituted coumarins selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic ones I and II in the low nanomolar/subnanomolar range

(2010) Alfonso Maresca et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Carbonic Anhydrase Inhibitors: Inhibition of Human Erythrocyte Isozymes I and II with a Series of Phenolic Acids

(2010) S. Beyza Öztürk Sarıkaya et al.   Chemical Biology & Drug Design

Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols

(2009) Murat Şentürk et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The effect of ethanol on erythrocyte carbonic anhydrase isoenzymes activity: An in vitro and in vivo study

(2009) T. Abdulkadir Çoban et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Deciphering the Mechanism of Carbonic Anhydrase Inhibition with Coumarins and Thiocoumarins

(2009) Alfonso Maresca et al.   JOURNAL OF MEDICINAL CHEMISTRY

Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

(2008) Claudiu T. Supuran   NATURE REVIEWS DRUG DISCOVERY