Synthesis of 2,3-Disubstituted Quinazolinone Derivatives through Copper Catalyzed C-H Amidation Reactions

Copper-Catalyzed Synthesis of 2-Arylquinazolinones from 2-Arylindoles with Amines or Ammoniums

(2015) Yadong Feng et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Radical Methylation/C–H Amination/Oxidation Cascade for the Synthesis of Quinazolinones

(2015) Yajie Bao et al.   JOURNAL OF ORGANIC CHEMISTRY

Discovery of Antibiotic (E)-3-(3-Carboxyphenyl)-2-(4-cyanostyryl)quinazolin-4(3H)-one

(2015) Renee Bouley et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ligand-Free Pd-Catalyzed and Copper-Assisted C–H Arylation of Quinazolin-4-ones with Aryl Iodides under Microwave Heating

(2015) Sylvain Laclef et al.   ORGANIC LETTERS

Synthesis of Fused Isoquinolinone and Iminoisoindolinone Derivativesviaa Copper-Catalyzed Regioselective Switching Process

(2014) Veerababurao Kavala et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal-free oxidative synthesis of quinazolinones via dual amination of sp3 C–H bonds

(2014) Dan Zhao et al.   CHEMICAL COMMUNICATIONS

Copper-Catalyzed Arylation of Nitrogen Heterocycles from Anilines under Ligand-Free Conditions

(2014) Dounia Toummini et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent advances in the structural library of functionalized quinazoline and quinazolinone scaffolds: Synthetic approaches and multifarious applications

(2014) Imtiaz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Domino Reaction Involving C-C Bond Cleavage To Construct 2-Aryl Quinazolinones

(2014) Li-Xia Wang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Syntheses of quinazolinones from 2-iodobenzamides and enaminones via copper-catalyzed domino reactions

(2014) Teerawat Songsichan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalyzed Aerobic Oxidative Amination of sp3C–H Bonds: Efficient Synthesis of 2-Hetarylquinazolin-4(3H)-ones

(2014) Qiang Li et al.   ORGANIC LETTERS

Copper-Catalyzed Enantioselective Intramolecular Aryl C–N Coupling: Synthesis of Enantioenriched 2-Oxo-1,2,3,4-tetrahydroquinoline-3-carboxamides via an Asymmetric Desymmetrization Strategy

(2014) Nian He et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Amination of Quinoline N-Oxides via C–H Bond Activation under Mild Conditions

(2014) Chongwei Zhu et al.   ORGANIC LETTERS

Glyoxylic acid in the reaction of isatoic anhydride with amines: a rapid synthesis of 3-(un)substituted quinazolin-4(3H)-ones leading to rutaecarpine and evodiamine

(2014) K. Raghavendra Rao et al.   TETRAHEDRON LETTERS

Synthesis of quinazolinones from anthranilamides and aldehydes via metal-free aerobic oxidation in DMSO

(2014) Na Yeun Kim et al.   TETRAHEDRON LETTERS

Silver decorated multi-walled carbon nanotubes as a heterogeneous catalyst in the sonication of 2-aryl-2,3-dihydroquinazolin-4(1H)-ones

(2014) Javad Safari et al.   RSC Advances

Recent advances in 4(3H)-quinazolinone syntheses

(2014) Lin He et al.   RSC Advances

Copper-catalyzed tandem N-arylation/condensation: synthesis of quinazolin-4(3H)-ones from 2-halobenzonitriles and amides

(2014) Hongxin Chai et al.   RSC Advances

Rapid assembly of quinazolinone scaffold via copper-catalyzed tandem reaction of 2-bromobenzamides with aldehydes and aqueous ammonia: application to the synthesis of the alkaloid tryptanthrin

(2014) Shenghai Guo et al.   RSC Advances

Synthesis of Chiral Amino Acid Anilides by Ligand-Free Copper-Catalyzed SelectiveN-Arylation of Amino Acid Amides

(2013) Junyu Dong et al.   ADVANCED SYNTHESIS & CATALYSIS

Ligandless Copper-Catalyzed Coupling of Heteroaryl Bromides with Gaseous Ammonia

(2013) Serena Fantasia et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly Efficient Four-Component Synthesis of 4(3H)-Quinazolinones: Palladium-Catalyzed Carbonylative Coupling Reactions

(2013) Lin He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Heterogeneous CuII-Catalysed Solvent-Controlled Selective N-Arylation of Cyclic Amides and Amines with Bromo-iodoarenes

(2013) Debasish Kundu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Cascade synthesis of quinazolinones from 2-aminobenzonitriles and aryl bromides via palladium-catalyzed carbonylation reaction

(2013) Haoquan Li et al.   GREEN CHEMISTRY

Synthesis of Quinazolin-4(3H)-ones via Amidine N-Arylation

(2013) Bryan Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Iron-Catalyzed One-Pot 2,3-Diarylquinazolinone Formation from 2-Nitrobenzamides and Alcohols

(2013) Huamin Wang et al.   ORGANIC LETTERS

Palladium-catalyzed carbonylative synthesis of N-(2-cyanoaryl)benzamides and sequential synthesis of quinazolinones

(2013) Xiao-Feng Wu et al.   TETRAHEDRON

A recyclable CuO-catalyzed synthesis of 4(3H)-quinazolinones

(2013) Dan Zhan et al.   RSC Advances

Syntheses of indolo[1,2-a]quinazolinone derivatives via palladium catalyzed intramolecular C–H amidation

(2013) Trimurtulu Kotipalli et al.   RSC Advances

Oxidative synthesis of quinazolinones and benzothiadiazine 1,1-dioxides from 2-aminobenzamide and 2-aminobenzenesulfonamide with benzyl alcohols and aldehydes

(2013) Muhammad Sharif et al.   RSC Advances

One-Pot Tandem Synthesis of 2-Arylbenzoxazole Derivatives via Copper-Catalyzed CN and CO Bond Formation

(2012) Veerababurao Kavala et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Isocoumarin Derivatives via the Copper-Catalyzed Tandem Sequential Cyclization of 2- Halo-N-phenyl Benzamides and Acyclic 1,3-Diketones

(2012) Veerababurao Kavala et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed Benzylic C–H Amidation with Benzyl Alcohols in Water: A Strategy To Construct Quinazolinones

(2012) Hidemasa Hikawa et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-mediated domino synthesis of pyrimido[4,5-b]carbazolones via Ullmann N-arylation and aerobic oxidative C–H amidation

(2012) Devanga K. Sreenivas et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient syntheses of 2,3-disubstituted natural quinazolinones via iridium catalysis

(2012) Jie Fang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of 3-Substituted and 2,3-Disubstituted Quinazolinones via Cu-Catalyzed Aryl Amidation

(2012) Lanting Xu et al.   ORGANIC LETTERS

Quinazolinone-Directed C-H Activation: A Novel Strategy for the Acetoxylation-Methoxylation of the Arenes

(2012) B. Reddy et al.   SYNLETT

One-pot synthesis of 4(3H)-quinazolinones from azides, alkynes, anilines, and carbon monoxide

(2012) Yang Shen et al.   TETRAHEDRON LETTERS

Copper-Catalyzed Domino Synthesis of Quinazolinones via Ullmann-Type Coupling and Aerobic Oxidative C−H Amidation

(2011) Wei Xu et al.   ORGANIC LETTERS

Quinazolinone linked pyrrolo[2,1-c][1,4]benzodiazepine (PBD) conjugates: Design, synthesis and biological evaluation as potential anticancer agents

(2009) Ahmed Kamal et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Circumdatin I, a New Ultraviolet-A Protecting Benzodiazepine Alkaloid from a Marine Isolate of the Fungus Exophiala

(2009) Dahai Zhang et al.   JOURNAL OF ANTIBIOTICS

Environmentally Friendly Iron-Catalyzed Cascade Synthesis of 1,2,4-Benzothiadiazine 1,1-Dioxide and Quinazolinone Derivatives

(2009) Daoshan Yang et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

A Simple and Efficient Approach to Quinazolinones under Mild Copper-Catalyzed Conditions

(2008) Xiaowei Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Sequential Metal-Catalyzed C−N Bond Formation in the Synthesis of 2-Amido-indoles

(2008) Pei-Yuan Yao et al.   ORGANIC LETTERS

N-Amidation by Copper-Mediated Cross-Coupling of Organostannanes or Boronic Acids withO-Acetyl Hydroxamic Acids

(2008) Zhihui Zhang et al.   ORGANIC LETTERS

New Diimine−Copper Complexes: An Efficient and Simple Catalyst System for BuchwaldN-Arylation of Indole

(2008) Mariappan Periasamy et al.   ORGANOMETALLICS

Synthesis and CNS depressant activity of some novel 3-[5-substituted 1,3,4-thiadiazole-2-yl]-2-styryl quinazoline-4(3H)-ones

(2007) Varsha Jatav et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY