A Facile Synthesis of Pyrazoles through Metal-Free Oxidative C(sp2)H Cycloamination of Vinyl Hydrazones

Indole Synthesis Based On A Modified Koser Reagent

(2014) Laura Fra et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium nanomaterials in catalytic intramolecular C–H amination reactions

(2014) Leng Leng Chng et al.   CHEMICAL COMMUNICATIONS

Synthesis of Indazoles and Azaindazoles by Intramolecular Aerobic Oxidative CN Coupling under Transition-Metal-Free Conditions

(2014) Jiantao Hu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Hypervalent Iodine(III) Promoted Direct Synthesis of Imidazo[1,2-a]pyrimidines

(2014) Guangyin Qian et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Facile Access to 1H-Indazoles through Iodobenzene-Catalyzed C-H Amination under Mild, Transition-Metal-Free Conditions

(2014) Mitsuhiro Kashiwa et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Alkene Diamination Using Electron-Rich Amines: Hypervalent Iodine-Promoted Inter-/Intramolecular C–N Bond Formation

(2014) Ki Bum Hong et al.   ORGANIC LETTERS

Solvent/Oxidant-Switchable Synthesis of Multisubstituted Quinazolines and Benzimidazoles via Metal-Free Selective Oxidative Annulation of Arylamidines

(2014) Jian-Ping Lin et al.   ORGANIC LETTERS

Hypervalent iodine(iii) catalyzed oxidative C–N bond formation in water: synthesis of benzimidazole-fused heterocycles

(2014) D. Nageswar Rao et al.   RSC Advances

C–H cycloamination of N-aryl-2-aminopyridines and N-arylamidines catalyzed by an in situ generated hypervalent iodine(iii) reagent

(2013) Yimiao He et al.   CHEMICAL COMMUNICATIONS

Theoretical studies of iron(iii)-catalyzed intramolecular C–H amination of azides

(2013) Juan Li et al.   DALTON TRANSACTIONS

Pyrazole scaffold: A remarkable tool in the development of anticancer agents

(2013) Harish Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal-Free Oxidative Carbon-Heteroatom Bond Formation Through C-H Bond Functionalization

(2013) Rajarshi Samanta et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Aerobic C(sp2)–H Functionalization for C–N Bond Formation: Synthesis of Pyrazoles and Indazoles

(2013) Xianwei Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 1H-Indazoles and 1H-Pyrazoles via FeBr3/O2 Mediated Intramolecular C–H Amination

(2013) Tianshui Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Development of Intramolecular Vicinal Diamination of Alkenes: From Palladium to Bromine Catalysis

(2013) Kilian Muñiz et al.   JOURNAL OF ORGANIC CHEMISTRY

Pyrazolines: A Biological Review

(2013) Akranth Marella et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

A Metal-Free Tandem Demethylenation/C(sp2)–H Cycloamination Process of N-Benzyl-2-aminopyridines via C–C and C–N Bond Cleavage

(2013) Dongdong Liang et al.   ORGANIC LETTERS

Synthesis of Indolines via Pd(II)-Catalyzed Amination of C–H Bonds Using PhI(OAc)2 as the Bystanding Oxidant

(2013) Tian-Sheng Mei et al.   ORGANIC LETTERS

Oxidative Diamination Promoted by Dinuclear Iodine(III) Reagents

(2013) Caren Röben et al.   ORGANIC LETTERS

Iodobenzene Catalyzed C–H Amination of N-Substituted Amidines Using m-Chloroperbenzoic Acid

(2013) Santhosh Kumar Alla et al.   ORGANIC LETTERS

The applications of hypervalent iodine(III) reagents in the constructions of heterocyclic compounds through oxidative coupling reactions

(2013) ZiSheng Zheng et al.   Science China-Chemistry

Copper-Catalyzed Aerobic Oxidative Synthesis of 5-Substituted Imidazo/Benzimidazoquinazolinones through Intramolecular CH Amination

(2012) Lujun Chen et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly Stereoselective Metal-Free Oxyaminations Using Chiral Hypervalent Iodine Reagents

(2012) Umar Farid et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Preparation and Chemistry of 3/5-Halogenopyrazoles

(2012) Yves L. Janin   CHEMICAL REVIEWS

Synthesis of Benzimidazoles by PIDA-Promoted Direct C(sp2)H Imidation ofN-Arylamidines

(2012) Jinbo Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Catalyzed Intramolecular Oxidative CH Functionalization and CN Formation of 2-Aminobenzophenones: Unusual Pseudo-1,2-Shift of the Substituent on the Aryl Ring

(2012) Pang-Chi Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Iodine(III)-Promoted Intermolecular Diamination of Alkenes

(2012) José A. Souto et al.   Chemistry-An Asian Journal

Synthesis of carbazolones and 3-acetylindoles via oxidative C–N bond formation through PIFA-mediated annulation of 2-aryl enaminones

(2012) Xu Ban et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient Synthesis of Chiral 2,2′-Bipyrrolidines by an anti-Selective Alkene Diamination

(2012) Christian H. Müller et al.   ORGANIC LETTERS

Intramolecular Oxidative Diamination and Aminohydroxylation of Olefins under Metal-Free Conditions

(2012) Hyun Jin Kim et al.   ORGANIC LETTERS

Copper-Catalyzed Synthesis of Purine-Fused Polycyclics

(2012) Gui-Rong Qu et al.   ORGANIC LETTERS

Copper-Catalyzed Sequential Ullmann N-Arylation and Aerobic Oxidative C–H Amination: A Convenient Route to Indolo[1,2-c]quinazoline Derivatives

(2012) Peng Sang et al.   ORGANIC LETTERS

Copper-Catalyzed Aliphatic C–H Amination with an Amidine Moiety

(2012) Hui Chen et al.   ORGANIC LETTERS

Synthesis of Tri- and Tetrasubstituted Pyrazoles via Ru(II) Catalysis: Intramolecular Aerobic Oxidative C–N Coupling

(2012) Jiantao Hu et al.   ORGANIC LETTERS

Metal-Free Oxidative C-H Bond Amination at Ambient Temperature

(2012) Andrey Antonchick et al.   SYNLETT

The Application of [Bis(trifluoroacetoxy)iodo]benzene (PIFA) in the Synthesis of Nitrogen-Containing Heterocycles

(2012) Imanol Tellitu et al.   SYNLETT

Intramolecular Olefin Diamination for the Stereoselective Synthesis of 3-Aminopiperidines

(2012) Simon Blakey et al.   SYNTHESIS-STUTTGART

Organocatalytic, Oxidative, Intramolecular CH Bond Amination and Metal-free Cross-Amination of Unactivated Arenes at Ambient Temperature

(2011) Andrey P. Antonchick et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Metal-Free Diamination of Styrenes

(2011) Caren Röben et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles

(2011) Santos Fustero et al.   CHEMICAL REVIEWS

o-Alkoxyphenyliminoiodanes: Highly Efficient Reagents for the Catalytic Aziridination of Alkenes and the Metal-Free Amination of Organic Substrates

(2011) Akira Yoshimura et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Mediated Synthesis of Substituted 2-Aryl-N-benzylbenzimidazoles and 2-Arylbenzoxazoles via C–H Functionalization/C–N/C–O Bond Formation

(2011) Murali Mohan Guru et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Oxidative C−N Bond Formation for the Synthesis of Carbazoles: Comparison of Reactivity between the Copper-Catalyzed and Metal-Free Conditions

(2011) Seung Hwan Cho et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Heterocycle Synthesis via Direct C–H/N–H Coupling

(2011) Enrico T. Nadres et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Efficient Syntheses of Azetidines, Pyrrolidines, and Indolines via Palladium Catalyzed Intramolecular Amination of C(sp3)–H and C(sp2)–H Bonds at γ and δ Positions

(2011) Gang He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxidative aromatic C–N bond formation: convenient synthesis of N-amino-3-nitrile-indoles via FeBr3-mediated intramolecular cyclization

(2011) Zisheng Zheng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Pd-Catalyzed C−H Activation/C−N Bond Formation: A New Route to 1-Aryl-1H-benzotriazoles

(2011) Rapolu Kiran Kumar et al.   ORGANIC LETTERS

Pd-Catalyzed Intramolecular Oxidative C–H Amination: Synthesis of Carbazoles

(2011) So Won Youn et al.   ORGANIC LETTERS

Copper-Catalyzed Aerobic Oxidative Intramolecular C–H Amination Leading to Imidazobenzimidazole Derivatives

(2011) Xiaoqiang Wang et al.   ORGANIC LETTERS

Synthesis of Benzimidazole-Fused Heterocycles by Intramolecular Oxidative C-N Bond Formation Using Hypervalent Iodine Reagents

(2011) Noriki Kutsumura et al.   SYNTHESIS-STUTTGART

Facile Synthesis of Koser’s Reagent and Derivatives from Iodine or Aryl Iodides

(2010) Eleanor A. Merritt et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Intramolecular Amidation of C(sp2)−H Bonds: Synthesis of 4-Aryl-2-quinolinones

(2010) Kiyofumi Inamoto et al.   JOURNAL OF ORGANIC CHEMISTRY

A Direct Intramolecular C−H Amination Reaction Cocatalyzed by Copper(II) and Iron(III) as Part of an Efficient Route for the Synthesis of Pyrido[1,2-a]benzimidazoles fromN-Aryl-2-aminopyridines

(2010) Honggen Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Free Highly Regioselective Aminotrifluoroacetoxylation of Alkenes

(2010) Helena M. Lovick et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Amination of Aromatic C−H Bonds with Oxime Esters

(2010) Yichen Tan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Intramolecular diamination and alkoxyamination of alkenes with N-sulfonyl ureas employing N-iodosuccinimide

(2010) Hao Li et al.   TETRAHEDRON

Amine directed Pd(ii)-catalyzed C–H bond functionalization under ambient conditions

(2010) Benjamin Haffemayer et al.   Chemical Science

Hypervalent iodine reagents as a new entrance to organocatalysts

(2009) Toshifumi Dohi et al.   CHEMICAL COMMUNICATIONS

Hypervalent iodine-mediated oxidation of alcohols

(2009) Muhammet Uyanik et al.   CHEMICAL COMMUNICATIONS

Asymmetric 1,3-dipolar cycloadditions of acrylamides

(2009) Marie Kissane et al.   CHEMICAL SOCIETY REVIEWS

A Convenient Approach to Fused Indeno-1,4-diazepinones through Hypervalent Iodine Chemistry

(2009) Elizabeth Malamidou-Xenikaki et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd(II)-Catalyzed Amination of C−H Bonds Using Single-Electron or Two-electron Oxidants

(2009) Tian-Sheng Mei et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Intramolecular Oxamidation of UnsaturatedO-Alkyl Hydroxamates: A Remarkably Versatile Entry to Hydroxy Lactams

(2009) Duncan J. Wardrop et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Free Intramolecular Aziridination of Alkenes Using Hypervalent Iodine Based Sulfonyliminoiodanes

(2009) Robert M. Moriarty et al.   ORGANIC LETTERS

Iodobenzene Diacetate Mediated Oxidation of N-Substituted Hydrazones of Chalcones: An Efficient Regioselective Synthesis of 1,3,5-Trisubstituted Pyrazoles

(2009) Ranjana Aggarwal et al.   SYNTHETIC COMMUNICATIONS

CH Functionalization/CN Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

(2008) Gordon Brasche et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chemistry of Polyvalent Iodine

(2008) Viktor V. Zhdankin et al.   CHEMICAL REVIEWS

Intramolecular Diamination of Alkenes with Palladium(II)/Copper(II) Bromide and IPy2BF4: The Role of Halogenated Intermediates

(2008) Kilian Muñiz et al.   Chemistry-An Asian Journal

Catalytic Version of and Reuse in Hypervalent Organo-λ3- and -λ5-iodane Oxidation

(2008) Masahito Ochiai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Method for the Synthesis of Carbazoles via Tandem C−H Functionalization and C−N Bond Formation

(2008) W. C. Peter Tsang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of β-, γ-, and δ-Lactams via Pd(II)-Catalyzed C−H Activation Reactions

(2008) Masayuki Wasa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxidative Pd(II)-Catalyzed C−H Bond Amination to Carbazole at Ambient Temperature

(2008) James A. Jordan-Hore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Free Oxidative Cyclization of Urea-Tethered Alkenes with Hypervalent Iodine

(2008) Brian M. Cochran et al.   ORGANIC LETTERS