The applications of hypervalent iodine(III) reagents in the constructions of heterocyclic compounds through oxidative coupling reactions

Metal-Free Radical Azidoarylation of Alkenes: Rapid Access to Oxindoles by Cascade CN and CC Bond-Forming Reactions

(2013) Kiran Matcha et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

C–H cycloamination of N-aryl-2-aminopyridines and N-arylamidines catalyzed by an in situ generated hypervalent iodine(iii) reagent

(2013) Yimiao He et al.   CHEMICAL COMMUNICATIONS

One-Pot Synthesis of 3-Hydroxyquinolin-2(1H)-ones from N-Phenylacetoacetamide via PhI(OCOCF3)2-Mediated α-Hydroxylation and H2SO4-Promoted Intramolecular Cyclization

(2013) Yucheng Yuan et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine(III)-Mediated [3 + 2] Cyclization for One-Pot Synthesis of Benzo[d]isoxazole-4,7-diols in Aqueous Medium

(2013) Yingwei Hou et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Dearomatizing Spirolactonization of Naphthols Catalyzed by Spirobiindane-Based Chiral Hypervalent Iodine Species

(2013) Toshifumi Dohi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hypervalent Iodine Catalyzed Generation of Nitrile Oxides from Oximes and their Cycloaddition with Alkenes or Alkynes

(2013) Akira Yoshimura et al.   ORGANIC LETTERS

PhI(OCOCF3)2-Mediated C–C Bond Formation Concomitant with a 1,2-Aryl Shift in a Metal-Free Synthesis of 3-Arylquinolin-2-ones

(2013) Le Liu et al.   ORGANIC LETTERS

Iodobenzene Catalyzed C–H Amination of N-Substituted Amidines Using m-Chloroperbenzoic Acid

(2013) Santhosh Kumar Alla et al.   ORGANIC LETTERS

One-Step Synthesis of 5-Substituted 1H-Tetrazoles from an Aldehyde by Reaction with Acetohydroxamic Acid and Sodium Azide under Bi(OTf)3 Catalysis

(2013) Madabhushi Sridhar et al.   SYNTHESIS-STUTTGART

Oxidative cycloaddition and cross-coupling processes on unactivated benzene derivatives

(2013) Guillaume Jacquemot et al.   Chemical Science

Synthesis of coumarins via PIDA/I2-mediated oxidative cyclization of substituted phenylacrylic acids

(2013) Jinming Li et al.   RSC Advances

Highly Stereoselective Metal-Free Oxyaminations Using Chiral Hypervalent Iodine Reagents

(2012) Umar Farid et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Benzimidazoles by PIDA-Promoted Direct C(sp2)H Imidation ofN-Arylamidines

(2012) Jinbo Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organoiodine(III) Mediated Synthesis of Novel SymmetricalBis([1,2,4]triazolo)[3,4-a:4′,3′-c]phthalazines as Antibacterial and Antifungal Agents

(2012) Om Prakash et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Synthesis of Oxazoles from Enamides via Phenyliodine Diacetate-Mediated Intramolecular Oxidative Cyclization

(2012) Yunhui Zheng et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine(III)-Mediated Tandem Oxidative Cyclization for Construction of 2-Nitrobenzo[b]furans

(2012) Shi-Chao Lu et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Tetramic Acid Derivatives via Intramolecular sp3 C–H Amination Mediated by Hypervalent Iodine(III) Reagents/Brønsted Acids

(2012) Lujia Mao et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Iodine(III)-Promoted Direct Intermolecular C–H Amination Reactions of Acetylenes

(2012) José A. Souto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of carbazolones and 3-acetylindoles via oxidative C–N bond formation through PIFA-mediated annulation of 2-aryl enaminones

(2012) Xu Ban et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Intramolecular Oxidative Diamination and Aminohydroxylation of Olefins under Metal-Free Conditions

(2012) Hyun Jin Kim et al.   ORGANIC LETTERS

Application of Dearomatization Strategy on the Synthesis of Furoquinolinone and Angelicin Derivatives

(2012) Yang Ye et al.   ORGANIC LETTERS

Phenyliodine Bis(trifluoroacetate)-Mediated Oxidative C–C Bond Formation: Synthesis of 3-Hydroxy-2-oxindoles and Spirooxindoles from Anilides

(2012) Junwei Wang et al.   ORGANIC LETTERS

Direct β-Acyloxylation of Enamines via PhIO-Mediated Intermolecular Oxidative C–O Bond Formation and Its Application to the Synthesis of Oxazoles

(2012) Xin Liu et al.   ORGANIC LETTERS

Enantioselective Total Synthesis of (+)-Lithospermic Acid

(2012) Arun K. Ghosh et al.   ORGANIC LETTERS

Phenyliodine Bis(trifluoroacetate) Mediated Intramolecular Oxidative Coupling of Electron-Rich N-Phenyl Benzamides

(2012) Wei Yu et al.   SYNLETT

Metal-Free Oxidative C-H Bond Amination at Ambient Temperature

(2012) Andrey Antonchick et al.   SYNLETT

Facile Oxidative Rearrangements Using Hypervalent Iodine Reagents

(2012) Fateh V. Singh et al.   ChemistryOpen

Facile Construction of Oxa-Aza Spirobicycles via a Tandem Carbon-Hydrogen Bond Oxidation

(2011) Yi Sun et al.   ADVANCED SYNTHESIS & CATALYSIS

Organocatalytic, Oxidative, Intramolecular CH Bond Amination and Metal-free Cross-Amination of Unactivated Arenes at Ambient Temperature

(2011) Andrey P. Antonchick et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of Stabilized Bisiodonium Salts as Intermediates in the Carbon-Carbon Bond Formation of Alkynes

(2011) Toshifumi Dohi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

In Situ Generated (Hypo)Iodite Catalysts for the Direct α-Oxyacylation of Carbonyl Compounds with Carboxylic Acids

(2011) Muhammet Uyanik et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Divergent Synthesis of Benzo[d]thiazoles by PIFA-Mediated Cyclization of β-Oxo Thioamides

(2011) Peng Huang et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

Iodobenzene catalysed synthesis of spirofurans and benzopyrans by oxidative cyclisation of vinylogous esters

(2011) Marsewi Ngatimin et al.   CHEMICAL COMMUNICATIONS

Synthesis of isoxazoles by hypervalent iodine-induced cycloaddition of nitrile oxides to alkynes

(2011) Anup M. Jawalekar et al.   CHEMICAL COMMUNICATIONS

A Metal-Free Route to 2-Aminooxazoles by Taking Advantage of the Unique Ring Opening of Benzoxazoles and Oxadiazoles with Secondary Amines

(2011) Jomy Joseph et al.   CHEMISTRY-A EUROPEAN JOURNAL

Potent, Selective, and Orally Available Benzoisothiazolone Phosphomannose Isomerase Inhibitors as Probes for Congenital Disorder of Glycosylation Ia

(2011) Russell Dahl et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of 2-(Trifluoromethyl)oxazoles from β-Monosubstituted Enamines via PhI(OCOCF3)2-Mediated Trifluoroacetoxylation and Cyclization

(2011) Feifei Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

Forming Spirocyclohexadienone-Oxocarbenium Cation Species in the Biomimetic Synthesis of Amomols

(2011) Mariam Traoré et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Oxidative C−N Bond Formation for the Synthesis of Carbazoles: Comparison of Reactivity between the Copper-Catalyzed and Metal-Free Conditions

(2011) Seung Hwan Cho et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

New synthesis of spirocycles by utilizing in situ forming hypervalent iodine species

(2011) Toshifumi Dohi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Benzimidazole-Fused Heterocycles by Intramolecular Oxidative C-N Bond Formation Using Hypervalent Iodine Reagents

(2011) Noriki Kutsumura et al.   SYNTHESIS-STUTTGART

Enantioselective Kita Oxidative Spirolactonization Catalyzed by In Situ Generated Chiral Hypervalent Iodine(III) Species

(2010) Muhammet Uyanik et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantiodifferentiating endo-Selective Oxylactonization of ortho-Alk-1-enylbenzoate with a Lactate-Derived Aryl-λ3-Iodane

(2010) Morifumi Fujita et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Construction of 3-oxyindoles via hypervalent iodine mediated tandem cyclization–acetoxylation of o-acyl anilines

(2010) Yi Sun et al.   CHEMICAL COMMUNICATIONS

Designer μ-oxo-bridged hypervalent iodine(iii) organocatalysts for greener oxidations

(2010) Toshifumi Dohi et al.   CHEMICAL COMMUNICATIONS

Organic synthesis using a hypervalent iodine reagent: unexpected and novel domino reaction leading to spiro cyclohexadienone lactones

(2010) Hiromichi Fujioka et al.   CHEMICAL COMMUNICATIONS

Revisiting the Kinnel–Scheuer hypothesis for the biosynthesis of palau'amine

(2010) Zhiqiang Ma et al.   CHEMICAL COMMUNICATIONS

Oxidative Spirocyclization of Phenolic Sulfonamides: Scope and Applications

(2010) Huan Liang et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Facile One-pot Synthesis of2,5-Disubstituted Oxazoles Using Poly[styrene(iodosodiacetate)]

(2010) Xian Huang et al.   CHINESE JOURNAL OF CHEMISTRY

‘On-water’ synthesis of chromeno-isoxazoles mediated by [hydroxy(tosyloxy)iodo]benzene (HTIB)

(2010) Mustafa J. Raihan et al.   GREEN CHEMISTRY

Exploring the Structural Requirements for Inhibition of the Ubiquitin E3 Ligase Breast Cancer Associated Protein 2 (BCA2) as a Treatment for Breast Cancer

(2010) Ghali Brahemi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Aqueous Iodine(III)-Mediated Stereoselective Oxidative Cyclization for the Synthesis of Functionalized Fused Dihydrofuran Derivatives

(2010) Yang Ye et al.   JOURNAL OF ORGANIC CHEMISTRY

Oxidation of α-Oxo-Oximes to Nitrile Oxides with Hypervalent Iodine Reagents

(2010) Tim Jen et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Highly Regioselective Aminotrifluoroacetoxylation of Alkenes

(2010) Helena M. Lovick et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Stereoselective Construction of Highly Functionalized Azetidines via a [2 + 2]-Cycloaddition

(2010) Yang Ye et al.   ORGANIC LETTERS

Tandem Phenolic Oxidative Amidation−Intramolecular Diels−Alder Reaction: An Approach to the Himandrine Core

(2010) Huan Liang et al.   ORGANIC LETTERS

Hypervalent iodine(III)-mediated tandem oxidative reactions: application for the synthesis of bioactive polyspirocyclohexa-2,5-dienones

(2010) Mariam Traoré et al.   TETRAHEDRON

‘Aromatic ring umpolung’, a rapid access to the main core of several natural products

(2010) Kimiaka C. Guérard et al.   TETRAHEDRON

A versatile PIFA-mediated approach to structurally diverse pyrrolo(benzo)diazepines from linear alkynylamides

(2010) Leticia M. Pardo et al.   TETRAHEDRON

Chiral hypervalent iodine-catalyzed enantioselective oxidative Kita spirolactonization of 1-naphthol derivatives and one-pot diastereo-selective oxidation to epoxyspirolactones

(2010) Muhammet Uyanik et al.   TETRAHEDRON

Hypervalent iodine-mediated oxygenative phenol dearomatization reactions

(2010) Laurent Pouységu et al.   TETRAHEDRON

Synthetic aspects of the oxidative amidation of phenols

(2010) Huan Liang et al.   TETRAHEDRON

Hypervalent iodine-mediated phenol dearomatization in natural product synthesis

(2010) Laurent Pouységu et al.   TETRAHEDRON

Dearomatization applications of I(III) reagents and some unusual reactivity amongst resorcinol derived cyclohexadienones

(2010) Todd A. Wenderski et al.   TETRAHEDRON

PIDA-mediated synthesis of oxazoles through oxidative cycloisomerization of propargylamides

(2010) Akio Saito et al.   TETRAHEDRON LETTERS

Synthesis of Cyclopamine Using a Biomimetic and Diastereoselective Approach

(2009) Athanassios Giannis et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organoiodine-Catalyzed Oxidative Spirocyclization of Phenols using Peracetic Acid as a Green and Economic Terminal Oxidant

(2009) Yutaka Minamitsuji et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

Hypervalent iodine-catalyzed oxylactonization of ketocarboxylic acids to ketolactones

(2009) Muhammet Uyanik et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

An Oxidative Dearomatization Cyclization Model for Cortistatin A

(2009) Samuel J. Danishefsky et al.   HETEROCYCLES

Diversity Oriented Synthesis of Benzimidazole and Benzoxa/(thia)zole Libraries through Polymer-Supported Hypervalent Iodine Reagent

(2009) Atul Kumar et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

A Convenient Approach to Fused Indeno-1,4-diazepinones through Hypervalent Iodine Chemistry

(2009) Elizabeth Malamidou-Xenikaki et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Total Synthesis of All of the Known Chiral Cleroindicins (C−F): Clarification Among Optical Rotations and Assignments

(2009) Todd A. Wenderski et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Oxamidation of UnsaturatedO-Alkyl Hydroxamates: A Remarkably Versatile Entry to Hydroxy Lactams

(2009) Duncan J. Wardrop et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iodine(III)-Mediated Tandem Acetoxylation−Cyclization ofo-Acyl Phenols for the Facile Construction of α-Acetoxy Benzofuranones

(2009) Renhua Fan et al.   ORGANIC LETTERS

Oxidation of Oximes to Nitrile Oxides with Hypervalent Iodine Reagents

(2009) Brian A. Mendelsohn et al.   ORGANIC LETTERS

Solvent-Controlled Oxidative Cyclization for Divergent Synthesis of Highly Functionalized Oxetanes and Cyclopropanes

(2009) Yang Ye et al.   ORGANIC LETTERS

A Hypervalent Iodine-Induced Double Annulation Enables a Concise Synthesis of the Pentacyclic Core Structure of the Cortistatins

(2009) Jessica L. Frie et al.   ORGANIC LETTERS

PIFA-Mediated Oxidative Cyclization of 1-Carbamoyl-1-oximylcycloalkanes: Synthesis of Spiro-Fused Pyrazolin-5-oneN-Oxides

(2009) Kewei Wang et al.   ORGANIC LETTERS

PIDA-Mediated Oxidative C−C Bond Formation: Novel Synthesis of Indoles fromN-Aryl Enamines

(2009) Wenquan Yu et al.   ORGANIC LETTERS

Simple Conversion of Enamines to 2H-Azirines and Their Rearrangements under Thermal Conditions

(2009) Xiaoxun Li et al.   ORGANIC LETTERS

Metal-Free Intramolecular Aziridination of Alkenes Using Hypervalent Iodine Based Sulfonyliminoiodanes

(2009) Robert M. Moriarty et al.   ORGANIC LETTERS

An Efficient Catalytic Sulfonyloxylactonization of Alkenoic Acids Using Hypervalent Iodine(III) Reagent

(2009) Jie Yan et al.   SYNLETT

Iodoarene-catalyzed one-pot preparation of 2,4,5-trisubstituted oxazoles from alkyl aryl ketones with mCPBA in nitriles

(2009) Yuhta Kawano et al.   TETRAHEDRON

Facile iodine(III)-induced oxidative cycloaddition of N-sulfonyl imines with methylene compounds under neutral conditions

(2009) Renhua Fan et al.   TETRAHEDRON LETTERS

Ion-supported PhI-catalyzed cyclization of N-methoxy-2-arylethanesulfonamides with mCPBA

(2009) Yoshihide Ishiwata et al.   TETRAHEDRON LETTERS

PhIO/Bu4NI mediated oxidative cyclization of amidoalkylation adducts for the synthesis of N-benzoyl aziridines and oxazolines

(2009) Renhua Fan et al.   TETRAHEDRON LETTERS

Direct oxidative cyclization of 3-arylpropionic acids using PIFA or Oxone: synthesis of 3,4-dihydrocoumarins

(2009) Yonghong Gu et al.   TETRAHEDRON LETTERS

One‐Pot Oxidative Heteroannulations ofN‐Sulfonylanilines with Styrenes for the Construction of 5‐Aminocoumaran Derivatives

(2008) Renhua Fan et al.   ADVANCED SYNTHESIS & CATALYSIS

Iodobenzene Diacetate/Tetrabutylammonium Iodide‐Induced Aziridination ofN‐Tosylimines with Activated Methylene Compounds under Mild Conditions

(2008) Renhua Fan et al.   ADVANCED SYNTHESIS & CATALYSIS

A Chiral Hypervalent Iodine(III) Reagent for Enantioselective Dearomatization of Phenols

(2008) Toshifumi Dohi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rapid Construction of the Cortistatin Pentacyclic Core

(2008) Eric M. Simmons et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Diastereoselective Synthesis of Orthoquinone Monoketals through λ3-Iodane-Mediated Oxidative Dearomatization of Phenols

(2008) Laurent Pouységu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chemistry of Polyvalent Iodine

(2008) Viktor V. Zhdankin et al.   CHEMICAL REVIEWS

Organoiodine (III)-mediated synthesis of 3-aryl/heteroaryl-5,7-dimethyl-1,2,4-triazolo[4,3-c]pyrimidines as antibacterial agents

(2008) Ravi Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Enhanced Antimalarial Activity of Novel Synthetic Aculeatin Derivatives

(2008) Marine Peuchmaur et al.   JOURNAL OF MEDICINAL CHEMISTRY

Generation of Nitrile Oxides under Nanometer Micelles Built in Neutral Aqueous Media: Synthesis of Novel Glycal-Based Chiral Synthons and Optically Pure 2,8-Dioxabicyclo[4.4.0]decene Core

(2008) Nirbhik Chatterjee et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Oxidative Cyclization of Urea-Tethered Alkenes with Hypervalent Iodine

(2008) Brian M. Cochran et al.   ORGANIC LETTERS

A New H2O2/Acid Anhydride System for the Iodoarene-Catalyzed C−C Bond-Forming Reactions of Phenols

(2008) Toshifumi Dohi et al.   ORGANIC LETTERS

Oxidative Dearomatization of Phenols: Why, How and What For?

(2008) Stéphane Quideau et al.   SYNLETT

Intriguing formal [2+3] cycloaddition promoted by a hypervalent iodine reagent

(2008) Didier Bérard et al.   TETRAHEDRON

Conversion of thiobenzamides to benzothiazoles via intramolecular cyclization of the aryl radical cation

(2008) Nadale K. Downer-Riley et al.   TETRAHEDRON

Synthesis of seco-psymberin/irciniastatin A: the discovery of a novel PhI(OAc)2 mediated cascade cyclization reaction

(2008) Xianhai Huang et al.   TETRAHEDRON LETTERS