Hypervalent iodine(iii) catalyzed oxidative C–N bond formation in water: synthesis of benzimidazole-fused heterocycles

Base-Catalyzed Synthesis of Substituted Indazoles under Mild, Transition-Metal-Free Conditions

(2013) Isabelle Thomé et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

C–H cycloamination of N-aryl-2-aminopyridines and N-arylamidines catalyzed by an in situ generated hypervalent iodine(iii) reagent

(2013) Yimiao He et al.   CHEMICAL COMMUNICATIONS

C–N bond forming cross-coupling reactions: an overview

(2013) Jitender Bariwal et al.   CHEMICAL SOCIETY REVIEWS

sp2 C–H bond activation in water and catalytic cross-coupling reactions

(2013) Bin Li et al.   CHEMICAL SOCIETY REVIEWS

Oxidative C–H amination reactions

(2013) Marie-Laure Louillat et al.   CHEMICAL SOCIETY REVIEWS

Metal-Free Oxidative Carbon-Heteroatom Bond Formation Through C-H Bond Functionalization

(2013) Rajarshi Samanta et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of imidazo and benzimidazo[2,1-a]isoquinolines by rhodium-catalyzed intramolecular double C–H bond activation

(2013) Vutukuri Prakash Reddy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Novel Strategy for Synthesis of Substituted Benzimidazo[1,2-a]quinolines

(2013) Jun-ya Kato et al.   ORGANIC LETTERS

A Metal-Free Tandem Demethylenation/C(sp2)–H Cycloamination Process of N-Benzyl-2-aminopyridines via C–C and C–N Bond Cleavage

(2013) Dongdong Liang et al.   ORGANIC LETTERS

Synthesis of Indolines via Pd(II)-Catalyzed Amination of C–H Bonds Using PhI(OAc)2 as the Bystanding Oxidant

(2013) Tian-Sheng Mei et al.   ORGANIC LETTERS

Oxidative Diamination Promoted by Dinuclear Iodine(III) Reagents

(2013) Caren Röben et al.   ORGANIC LETTERS

Mild Metal-Free Sequential Dual Oxidative Amination of C(sp3)–H bonds: Efficient Synthesis of Imidazo[1,5-a]pyridines

(2013) Yizhe Yan et al.   ORGANIC LETTERS

Iodobenzene Catalyzed C–H Amination of N-Substituted Amidines Using m-Chloroperbenzoic Acid

(2013) Santhosh Kumar Alla et al.   ORGANIC LETTERS

Ruthenium-catalyzed benzimidazoisoquinoline synthesis via oxidative coupling of 2-arylbenzimidazoles with alkynes

(2013) Nerella Kavitha et al.   TETRAHEDRON LETTERS

Base and ligand free copper-catalyzed N-arylation of 2-amino-N-heterocycles with boronic acids in air

(2013) D. Nageswar Rao et al.   RSC Advances

Selective Iodine-Catalyzed Intermolecular Oxidative Amination of C(sp3)H Bonds with ortho-Carbonyl-Substituted Anilines to Give Quinazolines

(2012) Yizhe Yan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-free direct amination/aromatization of 2-cyclohexenones to iodo-N-arylanilines and N-arylanilines promoted by iodine

(2012) M. Teresa Barros et al.   CHEMICAL COMMUNICATIONS

Synthesis of Benzimidazoles by PIDA-Promoted Direct C(sp2)H Imidation ofN-Arylamidines

(2012) Jinbo Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

AgI-Catalyzed Cascade Strategy: Regioselective Access to Diversely Substituted Fused Benzimidazo[2,1-a]isoquinolines, Naphthyridines, Thienopyridines, and Quinoxalines in Water

(2012) Vineeta Rustagi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

TBHP/I2-promoted oxidative coupling of acetophenones with amines at room temperature under metal-free and solvent-free conditions for the synthesis of α-ketoamides

(2012) Xiaobin Zhang et al.   GREEN CHEMISTRY

Elusive Metal-Free Primary Amination of Arylboronic Acids: Synthetic Studies and Mechanism by Density Functional Theory

(2012) Chen Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transition-Metal-Free Intramolecular N-Arylations

(2012) Isabelle Thomé et al.   ORGANIC LETTERS

Copper-Catalyzed Synthesis of Purine-Fused Polycyclics

(2012) Gui-Rong Qu et al.   ORGANIC LETTERS

Copper-Catalyzed Sequential Ullmann N-Arylation and Aerobic Oxidative C–H Amination: A Convenient Route to Indolo[1,2-c]quinazoline Derivatives

(2012) Peng Sang et al.   ORGANIC LETTERS

Copper-Catalyzed Aliphatic C–H Amination with an Amidine Moiety

(2012) Hui Chen et al.   ORGANIC LETTERS

Highly Regioselective C–N Bond Formation through C–H Azolation of Indoles Promoted by Iodine in Aqueous Media

(2012) Wen-Bin Wu et al.   ORGANIC LETTERS

The Complementary Competitors: Palladium and Copper in C–N Cross-Coupling Reactions

(2012) Irina P. Beletskaya et al.   ORGANOMETALLICS

Synthesis of annulated benzimidazoles via amidine cyclization

(2012) Kostiantyn Liubchak et al.   TETRAHEDRON

Organocatalytic, Oxidative, Intramolecular CH Bond Amination and Metal-free Cross-Amination of Unactivated Arenes at Ambient Temperature

(2011) Andrey P. Antonchick et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Novel biologically active nitro and amino substituted benzimidazo[1,2-a]quinolines

(2011) Nataša Perin et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Copper-catalyzed cascade synthesis of benzimidazoquinazoline derivatives under mild condition

(2011) Shan Xu et al.   CHEMICAL COMMUNICATIONS

Green chemistry oriented organic synthesis in water

(2011) Marc-Olivier Simon et al.   CHEMICAL SOCIETY REVIEWS

On the Importance of an Acid Additive in the Synthesis of Pyrido[1,2-a]benzimidazoles by Direct Copper-Catalyzed Amination

(2011) Kye-Simeon Masters et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Pyrido[1,2-a]benzimidazoles through a Copper-Catalyzed Cascade C-N Coupling Process

(2011) Zhiqing Wu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Antimalarial Pyrido[1,2-a]benzimidazoles

(2011) Albert J. Ndakala et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Mediated Synthesis of Substituted 2-Aryl-N-benzylbenzimidazoles and 2-Arylbenzoxazoles via C–H Functionalization/C–N/C–O Bond Formation

(2011) Murali Mohan Guru et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Oxidative C−N Bond Formation for the Synthesis of Carbazoles: Comparison of Reactivity between the Copper-Catalyzed and Metal-Free Conditions

(2011) Seung Hwan Cho et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Intermolecular Oxidative C–N Bond Formation under Metal-Free Conditions: Control of Chemoselectivity between Aryl sp2and Benzylic sp3C–H Bond Imidation

(2011) Hyun Jin Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Free Intermolecular Oxidative C–N Bond Formation via Tandem C–H and N–H Bond Functionalization

(2011) Abhishek A. Kantak et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd-Catalyzed C−H Activation/C−N Bond Formation: A New Route to 1-Aryl-1H-benzotriazoles

(2011) Rapolu Kiran Kumar et al.   ORGANIC LETTERS

Potassium Hydroxide/Dimethyl Sulfoxide Promoted Intramolecular Cyclization for the Synthesis of Benzimidazol-2-ones

(2011) Astrid Beyer et al.   ORGANIC LETTERS

Pd-Catalyzed Intramolecular Oxidative C–H Amination: Synthesis of Carbazoles

(2011) So Won Youn et al.   ORGANIC LETTERS

Copper-Catalyzed Aerobic Oxidative Intramolecular C–H Amination Leading to Imidazobenzimidazole Derivatives

(2011) Xiaoqiang Wang et al.   ORGANIC LETTERS

Non-Cyclizing Direct Transformation of Arene Carbon-Hydrogen Bonds into Carbon-Nitrogen Bonds

(2011) Ming Zhang et al.   SYNTHESIS-STUTTGART

Synthesis of Benzimidazole-Fused Heterocycles by Intramolecular Oxidative C-N Bond Formation Using Hypervalent Iodine Reagents

(2011) Noriki Kutsumura et al.   SYNTHESIS-STUTTGART

Novel pyridobenzimidazole derivatives exhibiting antifungal activity by the inhibition of β-1,6-glucan synthesis

(2010) Hiroshi Takeshita et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Facile Synthesis of Koser’s Reagent and Derivatives from Iodine or Aryl Iodides

(2010) Eleanor A. Merritt et al.   JOURNAL OF ORGANIC CHEMISTRY

A Direct Intramolecular C−H Amination Reaction Cocatalyzed by Copper(II) and Iron(III) as Part of an Efficient Route for the Synthesis of Pyrido[1,2-a]benzimidazoles fromN-Aryl-2-aminopyridines

(2010) Honggen Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Amination of Aromatic C−H Bonds with Oxime Esters

(2010) Yichen Tan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enhanced Reactivity of [Hydroxy(tosyloxy)iodo]benzene in Fluoroalcohol Media. Efficient Direct Synthesis of Thienyl(aryl)iodonium Salts

(2010) Motoki Ito et al.   MOLECULES

Hypervalent iodine reagents as a new entrance to organocatalysts

(2009) Toshifumi Dohi et al.   CHEMICAL COMMUNICATIONS

A Convenient Approach to Fused Indeno-1,4-diazepinones through Hypervalent Iodine Chemistry

(2009) Elizabeth Malamidou-Xenikaki et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd(II)-Catalyzed Amination of C−H Bonds Using Single-Electron or Two-electron Oxidants

(2009) Tian-Sheng Mei et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

CH Functionalization/CN Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

(2008) Gordon Brasche et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Novel Amidino-Substituted Thienyl- and Furylvinylbenzimidazole: Derivatives and Their Photochemical Conversion into Corresponding Diazacyclopenta[c]fluorenes. Synthesis, Interactions with DNA and RNA, and Antitumor Evaluation. 4

(2008) Marijana Hranjec et al.   JOURNAL OF MEDICINAL CHEMISTRY

Clean and Efficient Benzylic C−H Oxidation in Water Using a Hypervalent Iodine Reagent: Activation of Polymeric Iodosobenzene with KBr in the Presence of Montmorillonite-K10

(2008) Toshifumi Dohi et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Method for the Synthesis of Carbazoles via Tandem C−H Functionalization and C−N Bond Formation

(2008) W. C. Peter Tsang et al.   JOURNAL OF ORGANIC CHEMISTRY

Oxidative Pd(II)-Catalyzed C−H Bond Amination to Carbazole at Ambient Temperature

(2008) James A. Jordan-Hore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY