Quinazoline-Directed C-H Bond Functionalization Catalyzed by Ruthenium(II) Carboxylate - Construction of Polyconjugated Aryl-Heteroaryl Systems

Half-sandwich cycloruthenated complexes from aryloxazolines: synthesis, structures, and catalytic activities

(2016) Wei-Guo Jia et al.   DALTON TRANSACTIONS

Synthesis of 8-heteroaryl nitroxoline analogues via one-pot sequential Pd-catalyzed coupling reactions

(2016) Helena Brodnik et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rhodium-catalyzed C–C coupling reactions via double C–H activation

(2016) Shuai-Shuai Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Advances in the development of catalytic tethering directing groups for C–H functionalization reactions

(2016) Huan Sun et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Ru-catalysed C–H functionalisations as a tool for selective organic synthesis

(2016) Sara Ruiz et al.   TETRAHEDRON LETTERS

Undirected, Homogeneous C–H Bond Functionalization: Challenges and Opportunities

(2016) John F. Hartwig et al.   ACS Central Science

Substrate Activation Strategies in Rhodium(III)-Catalyzed Selective Functionalization of Arenes

(2015) Guoyong Song et al.   ACCOUNTS OF CHEMICAL RESEARCH

The cascade synthesis of quinazolinones and quinazolines using an α-MnO2 catalyst and tert-butyl hydroperoxide (TBHP) as an oxidant

(2015) Zhe Zhang et al.   CHEMICAL COMMUNICATIONS

Transition metal-catalyzed ketone-directed or mediated C–H functionalization

(2015) Zhongxing Huang et al.   CHEMICAL SOCIETY REVIEWS

Single-Component Phosphinous Acid Ruthenium(II) Catalysts for Versatile C−H Activation by Metal-Ligand Cooperation

(2015) Daniel Zell et al.   CHEMISTRY-A EUROPEAN JOURNAL

Transition-Metal-Catalyzed π-Bond-Assisted CH Bond Functionalization: An Emerging Trend in Organic Synthesis

(2015) Parthasarathy Gandeepan et al.   Chemistry-An Asian Journal

Ruthenium-Catalyzed C–H Activation and Coupling Reactions in Organic Synthesis

(2015) Arpad Molnar et al.   CURRENT ORGANIC CHEMISTRY

Rhodium-Catalyzed Regioselective Direct C-H Amidation of 2,4-Diarylquinazoline with Sulfonyl Azides: An Example of Steric Hindrance Regulated Mono- and Diamidation Selectivity

(2015) Chunyan Zhang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of quinazolines and quinazolinones via palladium-mediated approach

(2015) Ibrahim M. Abdou et al.   HETEROCYCLIC COMMUNICATIONS

Further Insight into the Lability of MeCN Ligands of Cytotoxic Cycloruthenated Compounds: Evidence for the Antisymbiotic Effect Trans to the Carbon Atom at the Ru Center

(2015) Ana Soraya Lima Barbosa et al.   INORGANIC CHEMISTRY

Cycloruthenation of aryl imines and N-heteroaryl benzenes via C–H bond activation with Ru(II) and acetate partners

(2015) Bin Li et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

A new and facile CuCl2·2H2O-catalyzed one-pot three-component synthesis for quinazolines

(2015) Syed Muhammad Saad et al.   MONATSHEFTE FUR CHEMIE

Following directions

(2015) Lutz Ackermann et al.   Nature Chemistry

Ruthenium-catalyzed oxidative coupling of 2-aryl-4-quinazolinones with olefins: synthesis of pyrrolo[2,1-b]quinazolin-9(1H)-one motifs

(2015) Yong Zheng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition metal catalyzed meta-C–H functionalization of aromatic compounds

(2015) Jiong Yang   ORGANIC & BIOMOLECULAR CHEMISTRY

Advances in Transition-Metal-Catalyzed Direct sp3-Carbon–Hydrogen Bond Functionalization

(2015) Nai-Xing Wang et al.   SYNLETT

Quinazoline-directed regioselective arylation via palladium catalysis: synthesis of 2-(1-biaryl)-4-arylquinazolines

(2015) Yiyuan Peng et al.   TETRAHEDRON

Recent advances in the C–H-functionalization of the distal positions in pyridines and quinolines

(2015) David E. Stephens et al.   TETRAHEDRON

Carbon–hydrogen (C–H) bond activation at PdIV: a Frontier in C–H functionalization catalysis

(2015) Joseph J. Topczewski et al.   Chemical Science

Transition-Metal-Catalyzed Site-Selective C–H Functionalization of Quinolines beyond C2 Selectivity

(2015) Tomohiro Iwai et al.   ACS Catalysis

Cyclometallated ruthenium(ii) complexes with ditopic thienyl–NHC ligands: syntheses and alkyne annulations

(2015) Xiaoke Xie et al.   Organic Chemistry Frontiers

Transition metal-catalyzed C–H bond functionalizations by the use of diverse directing groups

(2015) Zhengkai Chen et al.   Organic Chemistry Frontiers

Potassium Iodide-Catalyzed Three-Component Synthesis of 2-ArylquinazolinesviaAmination of Benzylic CH Bonds of Methylarenes

(2014) Dan Zhao et al.   ADVANCED SYNTHESIS & CATALYSIS

One-Pot Synthesis of 2-Arylquinazolines and Tetracyclic Isoindolo[1,2-a]quinazolinesviaCyanation Followed by Rearrangement ofortho-Substituted 2-Halo-N-arylbenzamides

(2014) Sachin D. Gawande et al.   ADVANCED SYNTHESIS & CATALYSIS

Weakly Coordinating Directing Groups for Ruthenium(II)- Catalyzed CH Activation

(2014) Suman De Sarkar et al.   ADVANCED SYNTHESIS & CATALYSIS

Functionalization of Remote CH Bonds: Expanding the Frontier

(2014) Johannes Schranck et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Unlocking nature’s CH bonds

(2014) Marcus E. Farmer et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Ligands Control Reactivity and Selectivity in Palladium-Catalyzed Functionalization of Unactivated C sp3H Bonds

(2014) M. Ángeles Fernández-Ibáñez   ChemCatChem

Heterocycle Construction via Transition Metal-Catalyzed C-H Functionalization and C-Heteroatom Bond Formation

(2014) Yajun Liu et al.   CURRENT ORGANIC CHEMISTRY

Quinazolines: New horizons in anticonvulsant therapy

(2014) Vinod G. Ugale et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pd-Catalyzed Intramolecular Aerobic Oxidative C–H Amination of 2-Aryl-3-(arylamino)quinazolinones: Synthesis of Fluorescent Indazolo[3,2-b]quinazolinones

(2014) Weiguang Yang et al.   ORGANIC LETTERS

A convenient palladium-catalyzed carbonylative synthesis of quinazolines from 2-aminobenzylamine and aryl bromides

(2014) Jianbin Chen et al.   RSC Advances

Recent advances in directed C–H functionalizations using monodentate nitrogen-based directing groups

(2014) Min Zhang et al.   Organic Chemistry Frontiers

Metalation Dictates Remote Regioselectivity: Ruthenium-Catalyzed Functionalization ofmetaCArH Bonds

(2013) Francisco Juliá-Hernández et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups

(2013) Guy Rouquet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Quinazolines and Tetrahydroquinazolines: Copper-Catalyzed Tandem Reactions of 2-Bromobenzyl Bromides with Aldehydes and Aqueous Ammonia or Amines

(2013) Xuesen Fan et al.   Chemistry-An Asian Journal

Palladium Catalyzed C–H Activation and its Application to Multi-bond Forming Reactions

(2013) Krishnan Ramachandiran et al.   CURRENT ORGANIC CHEMISTRY

Organometallic aspects of transition-metal catalysed regioselective C–H bond functionalisation of arenes and heteroarenes

(2013) Anant R. Kapdi   DALTON TRANSACTIONS

C–H Arylation Reaction: Atom Efficient and Greener Syntheses of π-Conjugated Small Molecules and Macromolecules for Organic Electronic Materials

(2013) Ken Okamoto et al.   MACROMOLECULES

Cross-coupling/annulations of quinazolones with alkynes for access to fused polycyclic heteroarenes under mild conditions

(2013) Hui Lu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals

(2012) Junichiro Yamaguchi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ruthenium(II)-Catalyzed C–H Bond Activation and Functionalization

(2012) Percia Beatrice Arockiam et al.   CHEMICAL REVIEWS

Copper-Catalyzed Synthesis of Quinazolines in Water Starting from o-Bromobenzylbromides and Benzamidines

(2012) Chandi C. Malakar et al.   CHEMISTRY-A EUROPEAN JOURNAL

Cyclometallation of arylimines and nitrogen-containing heterocycles via room-temperature C–H bond activation with arene ruthenium(ii) acetate complexes

(2012) Bin Li et al.   DALTON TRANSACTIONS

Quinazolinone-Directed C-H Activation: A Novel Strategy for the Acetoxylation-Methoxylation of the Arenes

(2012) B. Reddy et al.   SYNLETT

Copper-catalyzed three-component one-pot synthesis of quinazolines

(2012) Jia Ju et al.   TETRAHEDRON

Weak Coordination as a Powerful Means for Developing Broadly Useful C–H Functionalization Reactions

(2011) Keary M. Engle et al.   ACCOUNTS OF CHEMICAL RESEARCH

Carboxylate-Assisted Transition-Metal-Catalyzed C−H Bond Functionalizations: Mechanism and Scope

(2011) Lutz Ackermann   CHEMICAL REVIEWS

The Scope of Ambiphilic Acetate-Assisted Cyclometallation with Half-Sandwich Complexes of Iridium, Rhodium and Ruthenium

(2011) Youcef Boutadla et al.   CHEMISTRY-A EUROPEAN JOURNAL

CuCl/DABCO/4-HO-TEMPO-Catalyzed Aerobic Oxidative Synthesis of 2-Substituted Quinazolines and 4H-3,1-Benzoxazines

(2011) Bing Han et al.   JOURNAL OF ORGANIC CHEMISTRY

Iron-Catalyzed Stereospecific Activation of Olefinic C–H Bonds with Grignard Reagent for Synthesis of Substituted Olefins

(2011) Laurean Ilies et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalysed Direct Arylation of Heteroaromatics Bearing Unprotected Hydroxyalkyl Functions using Aryl Bromides

(2010) Julien Roger et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly Efficient One-Pot Synthesis of 2-Substituted Quinazolines and 4H-Benzo[d][1,3]oxazinesviaCross Dehydrogenative Coupling using Sodium Hypochlorite

(2010) C. Uma Maheswari et al.   ADVANCED SYNTHESIS & CATALYSIS

CH Bond Functionalization in Water Catalyzed by Carboxylato Ruthenium(II) Systems

(2010) Percia B. Arockiam et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

(2010) Thomas W. Lyons et al.   CHEMICAL REVIEWS

Functionalization of Organic Molecules by Transition-Metal-Catalyzed C(sp3)H Activation

(2010) Rodolphe Jazzar et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ruthenium(II) Acetate Catalyst for Direct Functionalisation of sp2-CH Bonds with Aryl Chlorides and Access to Tris- Heterocyclic Molecules

(2009) Franc Požgan et al.   ADVANCED SYNTHESIS & CATALYSIS

Cycloruthenated Compounds - Synthesis and Applications

(2009) Jean-Pierre Djukic et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Investigating Biological Activity Spectrum for Novel Styrylquinazoline Analogues

(2009) Josef Jampilek et al.   MOLECULES

Ligand-Free Palladium-Catalysed Direct Arylation of Heteroaromatics Using Low Catalyst Loadings

(2008) Franc Požgan et al.   ChemSusChem

Syntheses of 4-(indole-3-yl)quinazolines – A new class of epidermal growth factor receptor tyrosine kinase inhibitors

(2007) Anja Lüth et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS