Rhodium-Catalyzed Regioselective Direct C-H Amidation of 2,4-Diarylquinazoline with Sulfonyl Azides: An Example of Steric Hindrance Regulated Mono- and Diamidation Selectivity

Iridium-Catalyzed Direct CH Amidation with Weakly Coordinating Carbonyl Directing Groups under Mild Conditions

(2014) Jinwoo Kim et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-free oxidative synthesis of quinazolinones via dual amination of sp3 C–H bonds

(2014) Dan Zhao et al.   CHEMICAL COMMUNICATIONS

n-Bu4NI-catalyzed selective dual amination of sp3 C–H bonds: oxidative domino synthesis of imidazo[1,5-c]quinazolines on a gram-scale

(2014) Dan Zhao et al.   CHEMICAL COMMUNICATIONS

Ruthenium-Catalyzed C7 Amidation of Indoline CH Bonds with Sulfonyl Azides

(2014) Changduo Pan et al.   CHEMISTRY-A EUROPEAN JOURNAL

[RhIII(Cp*)]-Catalyzedortho-Selective Direct C(sp2)H Bond Amidation/Amination of Benzoic Acids byN-Chlorocarbamates andN-Chloromorpholines. A Versatile Synthesis of Functionalized Anthranilic Acids

(2014) Fo-Ning Ng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Rhodium-Catalyzed Direct Amination of Arenes with Nitrosobenzenes: A New Route to Diarylamines

(2014) Juanjuan Du et al.   CHEMISTRY-A EUROPEAN JOURNAL

Rhodium-Catalyzed Direct C–H Amidation of Azobenzenes with Sulfonyl Azides: A Synthetic Route to Sterically Hindered ortho-Substituted Aromatic Azo Compounds

(2014) Xuefeng Jia et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium-Catalyzed Direct ortho C–N Bond Formation of Aromatic Azo Compounds with Azides

(2014) Hao Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Cu-Catalyzed Direct Amidation of Aromatic C–H Bonds: An Access to Arylamines

(2014) Hui Xu et al.   JOURNAL OF ORGANIC CHEMISTRY

Iridium-Catalyzed C–H Amination with Anilines at Room Temperature: Compatibility of Iridacycles with External Oxidants

(2014) Hyunwoo Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Anthranilic Acid Derivatives through Iron-Catalyzed Ortho Amination of Aromatic Carboxamides with N-Chloroamines

(2014) Tatsuaki Matsubara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Non-innocent Additives in a Palladium(II)-Catalyzed C–H Bond Activation Reaction: Insights into Multimetallic Active Catalysts

(2014) Megha Anand et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mechanistic Studies of the Rhodium-Catalyzed Direct C–H Amination Reaction Using Azides as the Nitrogen Source

(2014) Sae Hume Park et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu(II)-Mediated C–H Amidation and Amination of Arenes: Exceptional Compatibility with Heterocycles

(2014) Ming Shang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iridium-Catalyzed Intermolecular Amidation of sp3 C–H Bonds: Late-Stage Functionalization of an Unactivated Methyl Group

(2014) Taek Kang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 4-alkynylquinazolines: Pd–Cu-cocatalyzed coupling of quinazoline-4-tosylates with terminal alkynes using N-heterocyclic carbenes as ligands

(2014) Yiyuan Peng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of 2-Aryl-2H-benzotrizoles from Azobenzenes and N-Sulfonyl Azides through Sequential Rhodium-Catalyzed Amidation and Oxidation in One Pot

(2014) Taekyu Ryu et al.   ORGANIC LETTERS

Copper-Catalyzed C(sp2)–H Amidation with Azides as Amino Sources

(2014) Jiangling Peng et al.   ORGANIC LETTERS

Ruthenium-Catalyzed Direct C–H Amidation of Arenes: A Mechanistic Study

(2014) Lu−Lu Zhang et al.   ORGANOMETALLICS

Ru-catalyzed direct C–H amidation of 2-arylbenzo[d]thiazoles with sulfonyl azides

(2014) Xiaoli Zhou et al.   TETRAHEDRON

Copper-mediated C(sp2)–H amination using TMSN3 as a nitrogen source: redox-neutral access to primary anilines

(2014) Jiangling Peng et al.   Organic Chemistry Frontiers

Rhodium(III)-Catalyzed C(sp2)H Activation and Electrophilic Amidation withN-Fluorobenzenesulfonimide

(2013) Ren-Jin Tang et al.   ADVANCED SYNTHESIS & CATALYSIS

Directed Amination of Non-Acidic Arene CH Bonds by a Copper-Silver Catalytic System

(2013) Ly Dieu Tran et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct CH Amination of Arenes with Alkyl Azides under Rhodium Catalysis

(2013) Kwangmin Shin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ru(ii)-catalyzed intermolecular C–H amidation of weakly coordinating ketones

(2013) Qing-Zhong Zheng et al.   CHEMICAL COMMUNICATIONS

Copper-catalyzed annulation of amidines for quinazoline synthesis

(2013) Yunhe Lv et al.   CHEMICAL COMMUNICATIONS

Ru(ii)-catalyzed intermolecular ortho-C–H amidation of aromatic ketones with sulfonyl azides

(2013) M. Bhanuchandra et al.   CHEMICAL COMMUNICATIONS

[Cp*RhCl2]2-catalyzed ortho-C–H bond amination of acetophenone o-methyloximes with primary N-chloroalkylamines: convenient synthesis of N-alkyl-2-acylanilines

(2013) Ka-Ho Ng et al.   CHEMICAL COMMUNICATIONS

Oxidative C–H amination reactions

(2013) Marie-Laure Louillat et al.   CHEMICAL SOCIETY REVIEWS

Ruthenium-Catalyzed Direct CH Amidation of Arenes Including Weakly Coordinating Aromatic Ketones

(2013) Jiyu Kim et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Quinazolines and Tetrahydroquinazolines: Copper-Catalyzed Tandem Reactions of 2-Bromobenzyl Bromides with Aldehydes and Aqueous Ammonia or Amines

(2013) Xuesen Fan et al.   Chemistry-An Asian Journal

Rh-Catalyzed Diarylamine Synthesis by Intermolecular C-H Amination of Heteroarylarenes

(2013) Conghui Tang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iridium-Catalyzed Direct Arene C–H Bond Amidation with Sulfonyl- and Aryl Azides

(2013) Donggun Lee et al.   JOURNAL OF ORGANIC CHEMISTRY

Unexpected Copper-Catalyzed Cascade Synthesis of Quinazoline Derivatives

(2013) Zhongyan Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Ir(III)-Catalyzed Mild C–H Amidation of Arenes and Alkenes: An Efficient Usage of Acyl Azides as the Nitrogen Source

(2013) Jaeyune Ryu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

RhIII/CuII-Cocatalyzed Synthesis of 1H-Indazoles through C–H Amidation and N–N Bond Formation

(2013) Da-Gang Yu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hydrogen-Bond-Assisted Controlled C–H Functionalization via Adaptive Recognition of a Purine Directing Group

(2013) Hyun Jin Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cross-coupling/annulations of quinazolones with alkynes for access to fused polycyclic heteroarenes under mild conditions

(2013) Hui Lu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rhodium-Catalyzed Direct Addition of Aryl C–H Bonds to Nitrosobenzenes at Room Temperature

(2013) Bing Zhou et al.   ORGANIC LETTERS

Expedient C–H Amidations of Heteroaryl Arenes Catalyzed by Versatile Ruthenium(II) Catalysts

(2013) Vedhagiri S. Thirunavukkarasu et al.   ORGANIC LETTERS

Rh(III)-Catalyzed Intermolecular C–H Amination of 1-Aryl-1H-pyrazol-5(4H)-ones with Alkylamines

(2013) Kui Wu et al.   ORGANIC LETTERS

Sulfoximine Directed Intermolecular o-C–H Amidation of Arenes with Sulfonyl Azides

(2013) M. Ramu Yadav et al.   ORGANIC LETTERS

Ru(II)-Catalyzed ortho-C–H Amination of Arenes and Heteroarenes at Room Temperature

(2013) Ming Shang et al.   ORGANIC LETTERS

Rh[III]-Catalyzed C–H Amidation Using Aroyloxycarbamates To Give N-Boc Protected Arylamines

(2013) Christoph Grohmann et al.   ORGANIC LETTERS

Rhodium(III)-Catalyzed Intermolecular N-Chelator-Directed Aromatic C–H Amidation with Amides

(2013) Huaiqing Zhao et al.   ORGANIC LETTERS

Synthesis of 4-Arylquinazolines by Arylation of Quinazolin-4-ones under Mild Conditions

(2013) Yiyuan Peng et al.   SYNTHESIS-STUTTGART

Palladium-Catalyzed Cyanation of Quinazoline-4-tosylates for Access to 4-CN-Functionalized Quinazolines

(2013) Yiyuan Peng et al.   SYNTHESIS-STUTTGART

Rhodium-Catalyzed Direct CH Amination of Benzamides with Aryl Azides: A Synthetic Route to Diarylamines

(2012) Jaeyune Ryu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selective Iodine-Catalyzed Intermolecular Oxidative Amination of C(sp3)H Bonds with ortho-Carbonyl-Substituted Anilines to Give Quinazolines

(2012) Yizhe Yan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A convenient synthesis of anthranilic acids by Pd-catalyzed direct intermolecular ortho-C–H amidation of benzoic acids

(2012) Ka-Ho Ng et al.   CHEMICAL COMMUNICATIONS

Copper-Catalyzed Synthesis of Quinazolines in Water Starting from o-Bromobenzylbromides and Benzamidines

(2012) Chandi C. Malakar et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalyst-free synthesis of quinazoline derivatives using low melting sugar–urea–salt mixture as a solvent

(2012) Zhan-Hui Zhang et al.   GREEN CHEMISTRY

Rhodium-Catalyzed Intermolecular Amidation of Arenes with Sulfonyl Azides via Chelation-Assisted C–H Bond Activation

(2012) Ji Young Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium-catalyzed regioselective amidation of indoles with sulfonyl azides via C–H bond activation

(2012) Jingjing Shi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Palladium-Catalyzed N-Monoarylation of Amidines and a One-Pot Synthesis of Quinazoline Derivatives

(2012) Meredeth A. McGowan et al.   ORGANIC LETTERS

Direct Sulfanylation of 4-Quinazolinone via C-OH Bond Activation: An Efficient Route to 2-Aryl-4-sulfanylquinazolines

(2012) Yiyuan Peng et al.   SYNTHESIS-STUTTGART

Metal-free intramolecular oxidative decarboxylative amination of primary α-amino acids with product selectivity

(2011) Yizhe Yan et al.   CHEMICAL COMMUNICATIONS

Microwave-promoted efficient synthesis of dihydroquinazolines

(2011) Rupam Sarma et al.   GREEN CHEMISTRY

Palladium-Catalyzed Intermolecular Directed C−H Amidation of Aromatic Ketones

(2011) Bin Xiao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed C−H Aminations of Anilides withN-Fluorobenzenesulfonimide

(2011) Kai Sun et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd-Catalyzed Intermolecular C–H Amination with Alkylamines

(2011) Eun Jeong Yoo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Intramolecular C(sp2)–H Amidination by Isonitrile Insertion Provides Direct Access to 4-Aminoquinazolines fromN-Arylamidines

(2011) Yong Wang et al.   ORGANIC LETTERS

Rhodium(III)-Catalyzed Intermolecular Direct Amination of Aromatic C–H Bonds with N-Chloroamines

(2011) Ka-Ho Ng et al.   ORGANIC LETTERS

Rh[III]-Catalyzed Direct C–H Amination Using N-Chloroamines at Room Temperature

(2011) Christoph Grohmann et al.   ORGANIC LETTERS

Highly Efficient One-Pot Synthesis of 2-Substituted Quinazolines and 4H-Benzo[d][1,3]oxazinesviaCross Dehydrogenative Coupling using Sodium Hypochlorite

(2010) C. Uma Maheswari et al.   ADVANCED SYNTHESIS & CATALYSIS

A convenient one-pot procedure for the synthesis of 2-aryl quinazolines using active MnO2 as oxidant

(2010) Yi-Yuan Peng et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Copper-Catalyzed Synthesis of Quinazoline Derivatives via Ullmann-Type Coupling and Aerobic Oxidation

(2010) Chen Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed Intermolecularortho-C−H Amidation of Anilides byN-Nosyloxycarbamate

(2010) Ka-Ho Ng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent advances in transition metal-catalyzed N-atom transfer reactions of azides

(2010) Tom G. Driver   ORGANIC & BIOMOLECULAR CHEMISTRY

Direct Synthesis of Quinazolines through Copper-Catalyzed Reaction of Aniline-Derived Benzamidines

(2010) Yusuke Ohta et al.   ORGANIC LETTERS

A Simple and Efficient Approach to the Synthesis of 2-Phenylquinazolines via sp3C−H Functionalization

(2010) Jintang Zhang et al.   ORGANIC LETTERS

Catalytic C–H amination: recent progress and future directions

(2009) Florence Collet et al.   CHEMICAL COMMUNICATIONS

2-(Aminoaryl)alkanone O-phenyl oximes: versatile reagents for syntheses of quinazolines

(2008) Fernando Portela-Cubillo et al.   CHEMICAL COMMUNICATIONS

Highly efficient copper-catalyzed cascade synthesis of quinazoline and quinazolinone derivatives

(2008) Cheng Huang et al.   CHEMICAL COMMUNICATIONS