Part II: nitroalkenes in the synthesis of heterocyclic compounds

Synthesis of Optically Active 2H-Thiopyrano[2,3-b]quinolines with Three Contiguous Stereocentersviaan Organocatalytic Asymmetric Tandem Michael-Henry Reaction

(2013) Lulu Wu et al.   ADVANCED SYNTHESIS & CATALYSIS

High analgesic and anti-inflammatory in vivo activities of six new hybrids NSAIAs tetrahydropyran derivatives

(2013) Saulo L. Capim et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Metal-free transannulation reaction of indoles with nitrostyrenes: a simple practical synthesis of 3-substituted 2-quinolones

(2013) Alexander V. Aksenov et al.   CHEMICAL COMMUNICATIONS

N-Heterocyclic Carbene Catalyzed [4+2] Cycloaddition of Nitroalkenes with Oxodienes

(2013) Xiang-Yu Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Efficient Synthesis of Quinoxaline Derivatives by Selective Modification of 3-Chloro-6-fluoroquinoxalin-2(1H)-one 4-Oxide

(2013) Jan Maichrowski et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Stereoselective Synthesis of Hexahydro-1H-pyrano- and thiopyrano[3,4-c]quinoline Derivatives through a Prins Cascade Cyclization

(2013) B.V. Subba Reddy et al.   JOURNAL OF ORGANIC CHEMISTRY

Modular Pyridine Synthesis from Oximes and Enals through Synergistic Copper/Iminium Catalysis

(2013) Ye Wei et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

β-Nitroacrylates as key building blocks for the synthesis of alkyl 3-substituted 5-oxopiperazine-2-carboxylates under fully heterogeneous conditions

(2013) Serena Gabrielli et al.   MONATSHEFTE FUR CHEMIE

Squaramide–Tertiary Amine Catalyzed Asymmetric Cascade Sulfa-Michael/Michael Addition via Dynamic Kinetic Resolution: Access to Highly Functionalized Chromans with Three Contiguous Stereocenters

(2013) Wen Yang et al.   ORGANIC LETTERS

An unexpected one-pot synthesis of multi-substituted quinolines via a cascade reaction of Michael/Staudinger/aza-Wittig/aromatization of ortho-azido-β-nitro-styrenes with various carbonyl compounds

(2013) Zhi-Hua Yu et al.   TETRAHEDRON

Novel thiophosphonodiamides as efficient hydrogen bond donor catalysts in tandem Michael addition–cyclization of malononitrile and 2-(E)-2-nitrovinylphenols

(2013) Keling Hu et al.   TETRAHEDRON

Synthesis of 5-(trifluoromethyl)-5H-chromeno[3,4-b]pyridines from 3-nitro-2-(trifluoromethyl)-2H-chromenes and aminoenones derived from acetylacetone and cyclic amines

(2013) Vladislav Yu. Korotaev et al.   TETRAHEDRON LETTERS

Chiral bifunctional squaramide catalyzed asymmetric tandem Michael-cyclization reaction: efficient synthesis of optically active 2-amino-4H-chromene-3-carbonitrile derivatives

(2013) Keling Hu et al.   TETRAHEDRON-ASYMMETRY

Carbohydrate-auxiliary assisted preparation of enantiopure 1,2-oxazine derivatives and aminopolyols

(2012) Marcin Jasiński et al.   Beilstein Journal of Organic Chemistry

Reactions of salicylaldehyde and enolates or their equivalents: versatile synthetic routes to chromane derivatives

(2012) Ishmael B Masesane et al.   Beilstein Journal of Organic Chemistry

Relay catalysis: combined metal catalyzed oxidation and asymmetric iminium catalysis for the synthesis of Bi- and tricyclic chromenes

(2012) Magnus Rueping et al.   CHEMICAL COMMUNICATIONS

Total Synthesis of Tetrahydropyran-Containing Natural Products Exploiting Intramolecular Oxa-Conjugate Cyclization

(2012) Haruhiko Fuwa   HETEROCYCLES

Construction of Multisubstituted Tetrahydropyrans by a Domino Oxa-Michael/Tsuji–Trost Reaction

(2012) Liang Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

A Hetero Diels–Alder Approach to the Synthesis of Chromans (3,4-Dihydrobenzopyrans) Using Oxonium Ion Chemistry: The Oxa-Povarov Reaction

(2012) Rivka R. R. Taylor et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Efficient Asymmetric Synthesis of Enantiopure Dihydro-1,2-oxazines: Dual-Organocatalyst-Promoted Asymmetric Cascade Reaction

(2012) Hua Lin et al.   ORGANIC LETTERS

Trifluoroacetic Anhydride Promoted Tandem Conjugate Addition of Boronic Acids/Acetal Ring Opening

(2012) Silvia Roscales et al.   ORGANIC LETTERS

Chiral Phosphoric Acid Catalyzed Inverse-Electron-Demand Aza-Diels–Alder Reaction of Isoeugenol Derivatives

(2012) Long He et al.   ORGANIC LETTERS

Asymmetric Synthesis of Polysubstituted 4-Amino- and 3,4-Diaminochromanes with a Chiral Multifunctional Organocatalyst

(2012) Wenduan Hou et al.   ORGANIC LETTERS

Simple synthesis of functionalized 7-aza-2H-chromenes from pyridoxal and nitroalkenes in aqueous medium

(2012) V. Yu. Korotaev et al.   RUSSIAN CHEMICAL BULLETIN

Asymmetric Synthesis of Functionalized Chromans via a One-Pot Organocatalytic Domino Michael-Hemiacetalization or -Lactonization and Dehydration Sequence

(2012) Dieter Enders et al.   SYNTHESIS-STUTTGART

One-Pot, Pseudo Five-Component Synthesis of Spirooxindole Derivatives Containing Fused 1,4-Dihydropyridines in Water

(2012) Abdolali Alizadeh et al.   SYNTHESIS-STUTTGART

Chemistry of biologically important flavones

(2012) Alok K. Verma et al.   TETRAHEDRON

Rapid access of 2,3,4-trisubstituted-2,3,4,9-tetrahydrothiopyrano[2,3-b]indole derivatives via one-pot three component reaction using organocatalysis

(2012) Shivendra Singh et al.   TETRAHEDRON LETTERS

Organocatalyzed stereoselective construction of N-formylpiperidines via a Michael-aza-Henry-hemiaminalization reaction cascade

(2012) Ruchi Chawla et al.   TETRAHEDRON LETTERS

Bismuth nitrate-catalyzed multicomponent reaction for efficient and one-pot synthesis of densely functionalized piperidine scaffolds at room temperature

(2012) Goutam Brahmachari et al.   TETRAHEDRON LETTERS

Cu(II)-catalyzed synthesis of quinoxalines from o-phenylenediamines and nitroolefins

(2012) Yongxin Chen et al.   TETRAHEDRON LETTERS

Efficient organocatalytic asymmetric synthesis of 2-amino-4H-chromene-3-carbonitrile derivatives

(2012) Yu Gao et al.   TETRAHEDRON-ASYMMETRY

Synthesis of Polysubstituted 2-Piperidinones via a Michael Addition/Nitro-Mannich/Lactamization Cascade

(2012) Hui Liu et al.   ACS Combinatorial Science

Design, synthesis and in vitro evaluation of novel chroman-4-one, chroman, and 2H-chromene derivatives as human rhinovirus capsid-binding inhibitors

(2011) Cinzia Conti et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, evaluation and metabolic studies of radiotracers containing a 4-(4-[18F]-fluorobenzyl)piperidin-1-yl moiety for the PET imaging of NR2B NMDA receptors

(2011) Romain Labas et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Stereoselective Synthesis of 2,6-Cis-Substituted Tetrahydropyrans: Brønsted Acid-Catalyzed Intramolecular Oxa-Conjugate Cyclization of α,β-Unsaturated Ester Surrogates

(2011) Haruhiko Fuwa et al.   JOURNAL OF ORGANIC CHEMISTRY

Chiral Phosphoric Acid-Catalyzed Enantioselective Three-Component Povarov Reaction Using Enecarbamates as Dienophiles: Highly Diastereo- and Enantioselective Synthesis of Substituted 4-Aminotetrahydroquinolines

(2011) Guillaume Dagousset et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chromone and Flavonoid Alkaloids: Occurrence and Bioactivity

(2011) Shahriar Khadem et al.   MOLECULES

Flavonoids: chemical properties and analytical methodologies of identification and quantitation in foods and plants

(2011) Eleonora Corradini et al.   NATURAL PRODUCT RESEARCH

Catalytic Asymmetric Aza-Michael−Michael Addition Cascade: Enantioselective Synthesis of Polysubstituted 4-Aminobenzopyrans

(2011) Xu-Fan Wang et al.   ORGANIC LETTERS

Au-Catalyzed Piperidine Synthesis via Tandem Acyloxy Migration/Intramolecular [3 + 2] Cycloaddition of Enynyl Esters

(2011) Huaiji Zheng et al.   ORGANIC LETTERS

Organocatalytic Approach to Polysubstituted Piperidines and Tetrahydropyrans

(2011) You Wang et al.   ORGANIC LETTERS

Practical and Novel One-Pot Protocol for the Synthesis of Highly Functionalized Pyridinols and Pyrido[1,2-a]-Fused 1,3-Diazaheterocycles

(2011) Abdolali Alizadeh et al.   SYNLETT

Organocatalytic Asymmetric Synthesis of Functionalized 4H-Chromenes via a One-Pot Domino Michael-Hemiacetalization and Dehydration Sequence

(2011) Dieter Enders et al.   SYNTHESIS-STUTTGART

Highly enantioselective organocatalytic cascade reaction for the synthesis of piperidines and oxazolidines

(2011) Sylva Číhalová et al.   TETRAHEDRON

Synthesis of heteroannulated 3-nitro- and 3-aminopyridines by cyclocondensation of electron-rich aminoheterocycles with 3-nitrochromone

(2011) Viktor O. Iaroshenko et al.   TETRAHEDRON

Stereoselective cascade reactions for construction of polyfunctionalised octahydroquinolines via [2C+2C+1C,1N] cyclisation

(2011) Ankita Rai et al.   TETRAHEDRON LETTERS

Efficient one-pot synthesis of functionalized piperidine scaffolds via ZrOCl2·8H2O catalyzed tandem reactions of aromatic aldehydes with amines and acetoacetic esters

(2011) Sarita Mishra et al.   TETRAHEDRON LETTERS

Thiophosphoramide catalyzed asymmetric Michael addition of acetone to functionalized nitrostyrenes: a convenient approach to optically active tetrahydropyrans

(2011) Yang Wu et al.   TETRAHEDRON-ASYMMETRY

Enantioselective Synthesis of Chromans with a Quaternary Stereogenic Centre through Catalytic Asymmetric Cascade Reactions

(2011) Qiu-Lin Hua et al.   ACS Catalysis

Concise Synthesis of Tetrahydropyrans by a Tandem Oxa-Michael/Tsuji-Trost Reaction

(2010) Liang Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Multiple-Organocatalyst-Promoted Cascade Reaction: A Fast and Efficient Entry into Fully Substituted Piperidines

(2010) Yao Wang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Strategies for the Synthesis of Pyridine Derivatives

(2010) Matthew D. Hill   CHEMISTRY-A EUROPEAN JOURNAL

Cooperative Catalysis with Metal and Secondary Amine: Synthesis of 2-Substituted Quinolines via Addition/Cycloisomerization Cascade

(2010) Nitin T. Patil et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Stereoselective7-Endo-Trig/Ring Contraction Cascade To Construct Pyrrolo[1,2-a]quinoline Derivatives

(2010) Xinyu Li et al.   ORGANIC LETTERS

Enantio- and Diastereoselective Synthesis of Piperidines by Coupling of Four Components in a “One-Pot” Sequence Involving Diphenylprolinol Silyl Ether Mediated Michael Reaction

(2010) Tatsuya Urushima et al.   ORGANIC LETTERS

One-Pot Enantioselective Syntheses of Iminosugar Derivatives Using Organocatalyticanti-Michael−anti-Aza-Henry Reactions

(2010) Ritsuo Imashiro et al.   ORGANIC LETTERS

Organocatalytic asymmetric assembly reactions for the syntheses of carbohydrate derivatives by intermolecular Michael-Henry reactions

(2010) H. Uehara et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Alkyl 2,3-dibromo-3-nitroacrylates in the reaction with o-phenylenediamine

(2010) K. V. Kovalenko et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Efficient One-Pot Synthesis of Spirooxindole Derivatives Containing 1,4-Dihydropyridine-Fused-1,3-Diazaheterocycle Fragments via Four-Component Reaction

(2010) Abdolali Alizadeh et al.   SYNTHESIS-STUTTGART

A three-component domino protocol for the facile synthesis of highly functionalized tetrahydroisoquinolines by creation of their benzene ring

(2010) Kamaraj Balamurugan et al.   TETRAHEDRON

Domino reaction of arylaldehydes and 1-acetylcyclopropanecarboxamides: one-pot access to highly functionalized spiropiperidine-2,4-diones

(2010) Jing Liu et al.   TETRAHEDRON LETTERS

l-Proline-catalyzed one-pot expeditious synthesis of highly substituted pyridines at room temperature

(2010) Chhanda Mukhopadhyay et al.   TETRAHEDRON LETTERS

Synthesis of (−)-Berkelic Acid

(2009) Xiaoxing Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Phosphine-Catalyzed Enantioselective Synthesis of Oxygen Heterocycles

(2009) Ying Kit Chung et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Tetrahydroisoquinolines as dopaminergic ligands: 1-Butyl-7-chloro-6-hydroxy-tetrahydroisoquinoline, a new compound with antidepressant-like activity in mice

(2009) Inmaculada Berenguer et al.   BIOORGANIC & MEDICINAL CHEMISTRY

2-(3-Aryl-2-propenoyl)-3-methylquinoxaline-1,4-dioxides: A novel cluster of tumor-specific cytotoxins which reverse multidrug resistance

(2009) Umashankar Das et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Amino sugars and their mimetics via 1,2-oxazines

(2009) Fabian Pfrengle et al.   CHEMICAL SOCIETY REVIEWS

An efficient procedure for the synthesis of substituted pyridines using KF·Al2O3

(2009) Biswanath Das et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Reactions of Conjugate Phosphinyl- and Phosphonyl-Nitroso Alkenes with Enamines. Preparation ofN-Hydroxypyrrole Derivatives†

(2009) Jesús M. de los Santos et al.   JOURNAL OF ORGANIC CHEMISTRY

Exploring Catalyst and Solvent Effects in the Multicomponent Synthesis of Pyridine-3,5-dicarbonitriles

(2009) Kai Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Oxazolone Cycloadducts as Heterocyclic Scaffolds for Alkaloid Construction: Synthesis of (±)-2-epi-Pumiliotoxin C

(2009) Stephen Philip Fearnley et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Intramolecular Friedel−Crafts-Type α-Arylation of Aldehydes

(2009) K. C. Nicolaou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chiral Brønsted Acid-Catalyzed Enantioselective Three-Component Povarov Reaction

(2009) Hua Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (+)-Sorangicin A

(2009) Amos B. Smith et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mn(III)-Mediated Reactions of Cyclopropanols with Vinyl Azides: Synthesis of Pyridine and 2-Azabicyclo[3.3.1]non-2-en-1-ol Derivatives

(2009) Yi-Feng Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

One hundred years of Meldrum’s acid: advances in the synthesis of pyridine and pyrimidine derivatives

(2009) Victoria V. Lipson et al.   MOLECULAR DIVERSITY

One-Pot Asymmetric Synthesis of Substituted Piperidines by Exocyclic Chirality Induction

(2009) Yunfeng Chen et al.   ORGANIC LETTERS

A Multicomponent Coupling Sequence for Direct Access to Substituted Quinolines

(2009) Supriyo Majumder et al.   ORGANIC LETTERS

Catalytic Asymmetric oxa-Michael−Michael Cascade for Facile Construction of Chiral Chromans via an Aminal Intermediate

(2009) Liansuo Zu et al.   ORGANIC LETTERS

Synthesis of Chromans via [3 + 3] Cyclocoupling of Phenols with Allylic Alcohols Using a Mo/o-Chloranil Catalyst System

(2009) Yoshihiko Yamamoto et al.   ORGANIC LETTERS

Domino Synthesis of Bridged Bicyclic Tetrahydro-1,2-oxazines: Access to Stereodefined 4-Aminocyclohexanols

(2009) Dwayne A. Dias et al.   ORGANIC LETTERS

Asymmetric synthesis of chiral chromans

(2009) Hong C. Shen   TETRAHEDRON

β-Nitroacrylates and silyl enol ethers as key starting materials for the synthesis of polyfunctionalized β-nitro esters and 1,2-oxazine-2-oxides

(2009) Roberto Ballini et al.   TETRAHEDRON

Rearrangement of 3-alkylidene-2-siloxy-tetrahydro-1,2-oxazines (ASENA). A new approach toward the synthesis of 3-α-hydroxyalkyl-5,6-dihydro-4H-1,2-oxazines

(2009) Andrey A. Tabolin et al.   TETRAHEDRON

Stereoselective hetero-Diels–Alder reaction of 3-nitro-2-trihalomethyl-2H-chromenes with 2,3-dihydrofuran and ethyl vinyl ether under solvent-free conditions

(2009) Vladislav Yu. Korotaev et al.   TETRAHEDRON

Nitroketene acetal chemistry: efficient synthesis of 2-amino-3-nitro-4H-chromenes

(2009) H. Surya Prakash Rao et al.   TETRAHEDRON LETTERS

Evolution of the Petasis−Ferrier Union/Rearrangement Tactic: Construction of Architecturally Complex Natural Products Possessing the Ubiquitouscis-2,6-Substituted Tetrahydropyran Structural Element

(2008) Amos B. Smith et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of 2,3,4-Trisubstituted Thiochromanes using an Organocatalytic Enantioselective Tandem Michael-Henry Reaction

(2008) Rajasekhar Dodda et al.   ADVANCED SYNTHESIS & CATALYSIS

A Novel Enantioselective Catalytic Tandem Oxa-Michael-Henry Reaction: One-Pot Organocatalytic Asymmetric Synthesis of 3-Nitro-2H-chromenes

(2008) Dan-Qian Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

A Short Route to α‐Tocopherol

(2008) Kegang Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Highly Stereoselective Hydrogen-Bond-Mediated Michael–Michael Cascade Process through Dynamic Kinetic Resolution

(2008) Jian Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric α-Aminoxylation/Aza-Michael Reactions for the Synthesis of Functionalized Tetrahydro-1,2-oxazines

(2008) Min Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Novel piperidinylpyrimidine derivatives as inhibitors of HIV-1 LTR activation

(2008) Norio Fujiwara et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and characterization of 5,6,7,8-tetrahydroquinoline C5a receptor antagonists

(2008) J. Kent Barbay et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and bioevaluation of hybrid 4-aminoquinoline triazines as a new class of antimalarial agents

(2008) Ashok Kumar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, in vitro antitrypanosomal and antibacterial activity of phenoxy, phenylthio or benzyloxy substituted quinolones

(2008) Xiang Ma et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Stereocontrolled synthesis of fully functionalized d-glucosamine monosaccharides via a domino nitro-Michael/Henry reaction

(2008) Alexander Adibekian et al.   CHEMICAL COMMUNICATIONS

4-Hydroxy-2-quinolones 144. Alkyl-, arylalkyl-, and arylamides of 2-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxylic acid and their diuretic properties

(2008) I. V. Ukrainets et al.   Chemistry of Heterocyclic Compounds

Synthesis and pharmacological screening of derivatives of isoxazolo[4,5-d]pyrimidine

(2008) Edwin Wagner et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

BINOLate–Magnesium Catalysts for Enantioselective Hetero-Diels–Alder Reaction of Danishefsky's Diene with Aldehydes

(2008) Haifeng Du et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Reactions of nitroxides, part 7: Synthesis of novel nitroxide selenoureas

(2008) Jerzy Zakrzewski et al.   HETEROATOM CHEMISTRY

BF3·Et2O-Mediated Cascade Cyclizations: Synthesis of Schweinfurthins F and G

(2008) Nolan R. Mente et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2H-chromenes and 1,2-dihydroquinolines from aryl aldehydes, amines, and alkenylboron compounds

(2008) Nicos A. Petasis et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

[4 + 2] Cycloadditions ofN-Alkenyl Iminium Ions: Structurally Complex Heterocycles from a Three-Component Diels−Alder Reaction Sequence

(2008) Nihar Sarkar et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Mediated Cyclization of Aryl and Benzyl Glycidyl Ethers: A Complete Scenario

(2008) Rocío Marcos et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ruthenium-Catalyzed Enantioselective Carbon−Carbon Bond Forming Reaction via Allenylidene-Ene Process: Synthetic Approach to Chiral Heterocycles Such As Chromane, Thiochromane, and 1,2,3,4-Tetrahydroquinoline Derivatives

(2008) Koji Fukamizu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Syntheses of Racemic, Natural (−) and Unnatural (+) Glyceollin I

(2008) Rahul S. Khupse et al.   ORGANIC LETTERS

A Highly Stereoselective Organocatalytic Tandem Aminoxylation/Aza-Michael Reaction for the Synthesis of Tetrahydro-1,2-Oxazines

(2008) Di Zhu et al.   ORGANIC LETTERS

Diastereoselective Synthesis of α-Tocopherol: A New Concept for the Formation of Chromanols

(2008) Julien Chapelat et al.   ORGANIC LETTERS

Cyclic Imine Nitro-Mannich/Lactamization Cascades: A Direct Stereoselective Synthesis of Multicyclic Piperidinone Derivatives

(2008) Pavol Jakubec et al.   ORGANIC LETTERS

A New Approach to Neuraminic Acid Analogues via 1,2-Oxazines

(2008) Bettina Bressel et al.   ORGANIC LETTERS

Total Synthesis of Brevetoxin A

(2008) Michael T. Crimmins et al.   ORGANIC LETTERS

A simple and convenient synthesis of 4-methyl-3-nitro-2-trihalomethyl-2H-chromenes from N-unsubstituted imines of 2-hydroxyacetophenones and trichloro(trifluoro)ethylidene nitromethanes

(2008) Vladislav Yu. Korotaev et al.   TETRAHEDRON

Synthesis of pharmaceutically active compounds containing a disubstituted piperidine framework

(2007) Sara Källström et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design, synthesis, and biological activity of piperidine diamine derivatives as factor Xa inhibitor

(2007) Akiyoshi Mochizuki et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Acid-Induced and Reductive Transfor­mations of Enantiopure 3,6-Dihydro-2H-1,2-oxazines – Synthesis of Dideoxyamino Carbohydrate Derivatives

(2007) Bettina Bressel et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Highly Chemoselective Metal-Free Reduction of Tertiary Amides

(2007) Guillaume Barbe et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY