Stereoselective Multiple Bond-Forming Transformations (MBFTs): The Power of 1,2- and 1,3-Dicarbonyl Compounds

Control of Six Contiguous Stereocenters in an Asymmetric Organocatalytic One-Pot Michael/Michael/Aldol Addition Sequence

(2012) Dieter Enders et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric transformations involving 1,2-dicarbonyl compounds as pronucleophiles

(2012) Wilfried Raimondi et al.   CHEMICAL COMMUNICATIONS

Isatins As Privileged Molecules in Design and Synthesis of Spiro-Fused Cyclic Frameworks

(2012) Girija S. Singh et al.   CHEMICAL REVIEWS

Indoles in Multicomponent Processes (MCPs)

(2012) Morteza Shiri   CHEMICAL REVIEWS

Chemistry and Biology Of Multicomponent Reactions

(2012) Alexander Dömling et al.   CHEMICAL REVIEWS

Recent developments in asymmetric multicomponent reactions

(2012) Corien de Graaff et al.   CHEMICAL SOCIETY REVIEWS

Catalyst- and Halogen-Free Regioselective Friedel-Crafts α-Ketoacylations

(2012) Kishor Mohanan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Domino Constructions of Pentacyclic Indeno[2,1-c]quinolines and Pyrano[4,3-b]oxepines by [4+1]/[3+2+1]/[5+1] and [4+3] Multiple Cyclizations

(2012) Bo Jiang et al.   CHEMISTRY-A EUROPEAN JOURNAL

FeCl3⋅6H2O-Catalyzed Intermolecular-Cascade Cyclization of Acetoacetanilide: Aldehyde-Tuned Synthesis to Valuable 2-Pyridone Analogues

(2012) Tista Sengupta et al.   CHEMISTRY-A EUROPEAN JOURNAL

Microwave-Assisted Domino Benzannulation of α-Oxo Ketenes: Preparation of 1,3-Dihydro-2H-1,5-benzodiazepin-2-ones

(2012) Juan-Carlos Castillo et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Recent Advances in Asymmetric Isocyanide-Based Multicomponent Reactions

(2012) Sander S. van Berkel et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Multicomponent reactions in unconventional solvents: state of the art

(2012) Yanlong Gu   GREEN CHEMISTRY

Highly enantioselective Biginelli reaction catalyzed by SPINOL-phosphoric acids

(2012) Fangxi Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Bismuth nitrate-catalyzed multicomponent reaction for efficient and one-pot synthesis of densely functionalized piperidine scaffolds at room temperature

(2012) Goutam Brahmachari et al.   TETRAHEDRON LETTERS

Synthesis and Antiproliferative Activity of Polysubstituted Tetrahydropyridine and Piperidin-4-one-3-carboxylate Derivatives

(2012) Raghunath Aeluri et al.   Asian Journal of Organic Chemistry

Brønsted-Acid-Catalyzed Asymmetric Multicomponent Reactions for the Facile Synthesis of Highly Enantioenriched Structurally Diverse Nitrogenous Heterocycles

(2011) Jie Yu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Enantioselective Organocatalytic Synthesis of Oxazolidine Derivatives through a One-Pot Cascade Reaction

(2011) Zhichao Jin et al.   ADVANCED SYNTHESIS & CATALYSIS

General and Efficient Organocatalytic Synthesis of Indoloquinolizidines, Pyridoquinazolines and Quinazolinones through a One-Pot Domino Michael Addition-Cyclization- Pictet-Spengler or 1,2-Amine Addition Reaction

(2011) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

A Highly Diastereo- and Enantioselective Reaction for Constructing Functionalized Cyclohexanes: Six Contiguous Stereocenters in One Step

(2011) Dengjian Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

1,2-Dicarbonyl Compounds as Pronucleophiles in Organocatalytic Asymmetric Transformations

(2011) Wilfried Raimondi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

PEG-embedded KBr3: A recyclable catalyst for multicomponent coupling reaction for the efficient synthesis of functionalized piperidines

(2011) Sanny Verma et al.   Beilstein Journal of Organic Chemistry

Single-Step Metallocatalyzed and Organocatalyzed Enantioselective Construction of Bicyclo[3.2.1]octanes

(2011) Marc Presset et al.   ChemCatChem

A Stereodivergent Strategy for the Preparation of Corynantheine and Ipecac Alkaloids, Their Epimers, and Analogues: Efficient Total Synthesis of (−)-Dihydrocorynantheol, (−)-Corynantheol, (−)-Protoemetinol, (−)-Corynantheal, (−)-Protoemetine, and Related

(2011) Wei Zhang et al.   CHEMISTRY-A EUROPEAN JOURNAL

N-Heterocyclic Carbene-Catalyzed Michael Additions of 1,3-Dicarbonyl Compounds

(2011) Thomas Boddaert et al.   CHEMISTRY-A EUROPEAN JOURNAL

Combination of Rearrangement with Metallic and Organic Catalyses - a Step- and Atom-Economical Approach to α-Spiroactones and -lactams

(2011) Thomas Boddaert et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Multicomponent reactions in ionic liquids: convenient and ecocompatible access to the 2,6-DABCO core

(2011) Zhor El Asri et al.   GREEN CHEMISTRY

Diastereo- and Enantioselective Synthesis of Oxazine and Oxazolidine Derivatives with a Chiral Quaternary Carbon Center under Multifunctional Catalysis

(2011) Zhichao Jin et al.   ORGANIC LETTERS

1,3-Dipolar Cycloaddition of Hydrazones with α-Oxo-ketenes: A Three-Component Stereoselective Entry to Pyrazolidinones and an Original Class of Spirooxindoles

(2011) Marc Presset et al.   ORGANIC LETTERS

N-Phenacylpyridinium bromides in the one-pot synthesis of 2,3-dihydrofurans

(2011) Che-Ping Chuang et al.   TETRAHEDRON

Lewis acid mediated diastereoselective synthesis of fused fluorinated spiroketal as potential biologically active compounds

(2011) Oluropo C. Agbaje et al.   TETRAHEDRON LETTERS

Diverse Asymmetric Quinolizidine Synthesis: A Stereodivergent One-Pot Approach

(2010) Wei Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Asymmetric Synthesis of Oxindoles Bearing a Tetrasubstituted Stereocenter at the C-3 Position

(2010) Feng Zhou et al.   ADVANCED SYNTHESIS & CATALYSIS

Protecting-Group-Free Total Syntheses: A Challenging Approach

(2010) Emmanuel Roulland   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalyzed enantioselective one-pot three-component access to indoloquinolizidines by a Michael addition–Pictet–Spengler sequence

(2010) Xiaoyu Wu et al.   CHEMICAL COMMUNICATIONS

Multicomponent reactions and ionic liquids: a perfect synergy for eco-compatible heterocyclic synthesis

(2010) Nicolas Isambert et al.   CHEMICAL SOCIETY REVIEWS

Primary Amine Catalyzed Biginelli Reaction for the Enantioselective Synthesis of 3,4-Dihydropyrimidin-2(1H)-ones

(2010) Derong Ding et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

An Investigation of Wall Effects in Microwave-Assisted Ring-Closing Metathesis and Cyclotrimerization Reactions

(2010) Doris Dallinger et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Organocatalytic Biginelli Reaction: Dependence of the Catalyst on Sterics, Hydrogen Bonding, and Reinforced Chirality

(2010) Satyajit Saha et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Diastereo- and Enantioselective Organocatalytic Michael Addition of α-Ketoamides to Nitroalkenes

(2010) Olivier Baslé et al.   ORGANIC LETTERS

Periselectivity Switch of Acylketenes in Cycloadditions with 1-Azadienes: Microwave-Assisted Diastereoselective Domino Three-Component Synthesis of α-Spiro-δ-lactams

(2010) Marc Presset et al.   ORGANIC LETTERS

Synthesis of Dihydropyrimidinones and Thiones by Multicomponent Reactions: Strategies Beyond the Classical Biginelli Reaction

(2010) Jie-Ping Wan et al.   SYNTHESIS-STUTTGART

Regio and diastereoselective synthesis of functionalized 2,3-dihydrofuro[3,2-c]coumarins via a one-pot three-component reaction

(2010) Elisa Altieri et al.   TETRAHEDRON

Synthesis of highly functionalized piperidines by one-pot multicomponent reaction using tetrabutylammonium tribromide (TBATB)

(2010) Abu T. Khan et al.   TETRAHEDRON LETTERS

1,3-Dicarbonyl compounds in stereoselective domino and multicomponent reactions

(2010) Damien Bonne et al.   TETRAHEDRON-ASYMMETRY

Organocatalytic Activity of N-Heterocyclic Carbenes in the Michael Addition of 1,3-Dicarbonyl Compounds: Application to a Stereoselective Spirocyclization Sequence

(2009) Thomas Boddaert et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly Enantioselective Biginelli Reaction Promoted by Chiral Bifunctional Primary Amine-Thiourea Catalysts: Asymmetric Synthesis of Dihydropyrimidines

(2009) Yangyun Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Redox Economy in Organic Synthesis

(2009) Noah Z. Burns et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Microwave-Assisted Ruthenium-Catalyzed Reactions

(2009) François Nicks et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

Bond formations by intermolecular and intramolecular trappings of acylketenes and their applications in natural product synthesis

(2009) Keith P. Reber et al.   CHEMICAL SOCIETY REVIEWS

The economies of synthesis

(2009) Timothy Newhouse et al.   CHEMICAL SOCIETY REVIEWS

Microwave-assisted cross-metathesis of acrylonitrile

(2009) Thomas Boddaert et al.   COMPTES RENDUS CHIMIE

Diastereoselective Synthesis oftrans-2,3-Dihydrofurans with Pyridinium Ylide Assisted Tandem Reaction

(2009) Qi-Fang Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Enantioselective Organocatalytic Biginelli and Biginelli-Like Condensations: Reversal of the Stereochemistry by Tuning the 3,3′-Disubstituents of Phosphoric Acids

(2009) Nan Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Protecting-group-free synthesis as an opportunity for invention

(2009) Ian S. Young et al.   Nature Chemistry

User-friendly stereoselective one-pot access to 1,4-diazepane derivatives by a cyclodehydrative three-component reaction with 1,3-dicarbonyls

(2009) Enrique Sotoca et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Dihydropyridine C-glycoconjugates by organocatalytic Hantzsch cyclocondensation. Stereoselective synthesis of α-threofuranose C-nucleoside enantiomers

(2009) Diogo R. B. Ducatti et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective Organocatalytic Hantzsch Synthesis of Polyhydroquinolines

(2009) Christopher G. Evans et al.   ORGANIC LETTERS

Microwave-Assisted Domino and Multicomponent Reactions with Cyclic Acylketenes: Expeditious Syntheses of Oxazinones and Oxazindiones

(2009) Marc Presset et al.   ORGANIC LETTERS

Asymmetric Syntheses of Oxindole and Indole Spirocyclic Alkaloid Natural Products

(2009) Barry Trost et al.   SYNTHESIS-STUTTGART

Organocatalytic Asymmetric Three-Component Cyclization of Cinnamaldehydes and Primary Amines with 1,3-Dicarbonyl Compounds: Straightforward Access to Enantiomerically Enriched Dihydropyridines

(2008) Jun Jiang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Alkaloid Synthesis: A One-Pot Organocatalytic Reaction to Quinolizidine Derivatives

(2008) Johan Franzén et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The MARDi Cascade: A Michael-Initiated Domino-Multicomponent Approach for the Stereoselective Synthesis of Seven-Membered Rings

(2008) Yoann Coquerel et al.   CHEMISTRY-A EUROPEAN JOURNAL

An Enantioselective Biginelli Reaction Catalyzed by a Simple Chiral Secondary Amine and Achiral Brønsted Acid by a Dual-Activation Route

(2008) Junguo Xin et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthetic Studies towards Guaianolide Sesquiterpene Lactones

(2008) Isabelle Reboul et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Synthesis of SNAP-7941: Chiral Dihydropyrimidone Inhibitor of MCH1-R

(2008) Jennifer M. Goss et al.   JOURNAL OF ORGANIC CHEMISTRY

Effects of Substituents in the β-Position of 1,3-Dicarbonyl Compounds in Bromodimethylsulfonium Bromide-Catalyzed Multicomponent Reactions: A Facile Access to Functionalized Piperidines

(2008) Abu T. Khan et al.   JOURNAL OF ORGANIC CHEMISTRY

Microwave-Assisted Wolff Rearrangement of Cyclic 2-Diazo-1,3-Diketones: An Eco-compatible Route to α-Carbonylated Cycloalkanones

(2008) Marc Presset et al.   JOURNAL OF ORGANIC CHEMISTRY

Two-Step Stereocontrolled Synthesis of Densely Functionalized Cyclic β-Aminoesters Containing Four Stereocenters, Based on a New Cerium(IV) Ammonium Nitrate Catalyzed Sequential Three-Component Reaction

(2008) Vellaisamy Sridharan et al.   ORGANIC LETTERS

One-pot three-component reaction providing 1,5-benzodiazepine derivatives

(2008) Kenichi Murai et al.   TETRAHEDRON

Synthesis of novel annulated uracils via domino Knoevenagel-hetero-Diels–Alder reaction in aqueous media

(2008) Malihe Javan Khoshkholgh et al.   TETRAHEDRON LETTERS

Function-Oriented Synthesis, Step Economy, and Drug Design

(2007) Paul A. Wender et al.   ACCOUNTS OF CHEMICAL RESEARCH

Organocatalytic Enantioselective One-Pot Synthesis and Application of Substituted 1,4-Dihydropyridines-Hantzsch Ester Analogues

(2007) Patrick T. Franke et al.   Chemistry-An Asian Journal

Microwave-Assisted Olefin Metathesis

(2007) Yoann Coquerel et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY