A general method for the metal-free, regioselective, remote C–H halogenation of 8-substituted quinolines

Mild Aliphatic and Benzylic Hydrocarbon C–H Bond Chlorination Using Trichloroisocyanuric Acid

(2017) Sascha H. Combe et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed, ortho-Selective C–H Halogenation of Benzyl Nitriles, Aryl Weinreb Amides, and Anilides

(2017) Riki Das et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed, N-(2-Aminophenyl)acetamide-Assisted Ortho-Arylation of Substituted Benzamides: Application to the Synthesis of Urolithins B, M6, and M7

(2017) M. Damoder Reddy et al.   JOURNAL OF ORGANIC CHEMISTRY

Remote C(sp3)–H Oxygenation of Protonated Aliphatic Amines with Potassium Persulfate

(2017) Melissa Lee et al.   ORGANIC LETTERS

The regioselective C5 halogenation of quinolines using sodium halides under transition metal-free conditions

(2017) Jun-Ying Jiao et al.   TETRAHEDRON

Identification of monodentate oxazoline as a ligand for copper-promoted ortho-C–H hydroxylation and amination

(2017) Ming Shang et al.   Chemical Science

Metal-free C5-selective halogenation of quinolines under aqueous conditions

(2017) Jichao Chen et al.   Organic Chemistry Frontiers

Copper(i) and N-fluorobenzenesulfonimide-mediated direct regioselective halogenation of 8-amidoquinolines on the C5 position

(2017) Xin He et al.   Organic Chemistry Frontiers

Nickel-catalyzed selective C-5 fluorination of 8-aminoquinolines with NFSI

(2017) Junshuai Ding et al.   Organic Chemistry Frontiers

Regio-Selective C−H Halogenation of 8-Amido-Quinolines under Transition Metal Free Conditions

(2017) Chiranjit Sen et al.   ChemistrySelect

A First Example of Cobalt-Catalyzed Remote CH Functionalization of 8-Aminoquinolines Operating through a Single Electron Transfer Mechanism

(2016) Christopher J. Whiteoak et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed 8-Amido Chelation-Induced Remote C−H Amination of Quinolines

(2016) Harekrishna Sahoo et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Mediated Remote Highly Site-Selective C-H Bond Bromination and Chlorination of Quinolines at the C5 Position that is Geometrically Difficult to Access

(2016) Naidu Sambasiva Rao et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Transition-metal-free oxidative C5 C–H-halogenation of 8-aminoquinoline amides using sodium halides

(2016) Ying Wang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper(ii)-catalyzed C5 and C7 halogenation of quinolines using sodium halides under mild conditions

(2016) Jun Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

5-Position-selective C–H trifluoromethylation of 8-aminoquinoline derivatives

(2016) Yoichiro Kuninobu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Iron-Catalyzed Oxyfunctionalization of Aliphatic Amines at Remote Benzylic C–H Sites

(2016) Curren T. Mbofana et al.   ORGANIC LETTERS

Rh-Catalyzed, Regioselective, C–H Bond Functionalization: Access to Quinoline-Branched Amines and Dimers

(2016) M. Damoder Reddy et al.   ORGANIC LETTERS

Copper-Catalyzed Regioselective C–H Iodination of Aromatic Carboxamides

(2016) Qiaolin Wu et al.   SYNLETT

Directed evolution of RebH for catalyst-controlled halogenation of indole C–H bonds

(2016) Mary C. Andorfer et al.   Chemical Science

PhI(OAc)2 oxidative C5 halogenation of quinolines using copper halides under mild conditions

(2016) Xing-Xing Liu et al.   RSC Advances

Functionalization of Quinolines through Copper-Catalyzed Regioselective Halogenation Reaction

(2016) Harekrishna Sahoo et al.   ChemistrySelect

The Highly Regioselective Halogenation of N-(8-quinolinyl)amides on the C-5 Position with Cuprous Halides Under Mild Conditions

(2016) Junshuai Ding et al.   ChemistrySelect

Bidentate, Monoanionic Auxiliary-Directed Functionalization of Carbon–Hydrogen Bonds

(2015) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Developing structure–activity relationships from an HTS hit for inhibition of the Cks1–Skp2 protein–protein interaction

(2015) Rajinder Singh et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Selective remote C–H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis

(2015) Hong-Wen Liang et al.   CHEMICAL COMMUNICATIONS

Nickel Catalysts/N,N′-Bidentate Directing Groups: An Excellent Partnership in Directed C–H Activation Reactions

(2015) Luis C. Misal Castro et al.   CHEMISTRY LETTERS

Palladium-Catalyzed Direct Arylation of C(sp3)–H Bonds of α-Cyano Aliphatic Amides

(2015) M. Damoder Reddy et al.   JOURNAL OF ORGANIC CHEMISTRY

Identification of benzenesulfonamide quinoline derivatives as potent HIV-1 replication inhibitors targeting Rev protein

(2015) Fudi Zhong et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Mediated Remote C–H Bond Chalcogenation of Quinolines on the C5 Position

(2015) Longzhi Zhu et al.   ORGANIC LETTERS

Two-Photon “Caging” Groups: Effect of Position Isomery on the Photorelease Properties of Aminoquinoline-Derived Photolabile Protecting Groups

(2015) Christine Tran et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Sulfonylation of 8-Aminoquinoline Amides with Sulfonyl Chlorides in Air

(2015) Huijie Qiao et al.   ORGANIC LETTERS

Copper and palladium mediated C–H chlorination on 8-acylaminoquinoline scaffolds

(2015) Haili Guo et al.   TETRAHEDRON

Rh(iii)-catalyzed C–H olefination of N-pentafluoroaryl benzamides using air as the sole oxidant

(2015) Yi Lu et al.   Chemical Science

Transition-Metal-Catalyzed Site-Selective C–H Functionalization of Quinolines beyond C2 Selectivity

(2015) Tomohiro Iwai et al.   ACS Catalysis

Transition metal-catalyzed C–H bond functionalizations by the use of diverse directing groups

(2015) Zhengkai Chen et al.   Organic Chemistry Frontiers

Remote Meta-C–H Activation Using a Pyridine-Based Template: Achieving Site-Selectivity via the Recognition of Distance and Geometry

(2015) Ling Chu et al.   ACS Central Science

Discovery of quinoline small molecules with potent dispersal activity against methicillin-resistant Staphylococcus aureus and Staphylococcus epidermidis biofilms using a scaffold hopping strategy

(2014) Yasmeen Abouelhassan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Iron-Catalyzed, Chelation-Induced Remote C–H Allylation of Quinolines via 8-Amido Assistance

(2014) Xuefeng Cong et al.   ORGANIC LETTERS

Room-temperature enantioselective C–H iodination via kinetic resolution

(2014) Ling Chu et al.   SCIENCE

Pd-Catalyzed Enantioselective C–H Iodination: Asymmetric Synthesis of Chiral Diarylmethylamines

(2013) Ling Chu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A robust protocol for Pd(ii)-catalyzed C-3 arylation of (1H) indazoles and pyrazoles: total synthesis of nigellidine hydrobromide

(2013) Mengchun Ye et al.   Chemical Science

CH Activation: A Complementary Tool in the Total Synthesis of Complex Natural Products

(2012) David Y.-K. Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Effect of Postflood Quinclorac Applications on Commercial Rice Cultivars

(2012) Jason A. Bond et al.   WEED TECHNOLOGY

Palladium(II)-Catalyzed Selective Monofluorination of Benzoic Acids Using a Practical Auxiliary: A Weak-Coordination Approach

(2011) Kelvin S. L. Chan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

C–H Functionalization in organic synthesis

(2011) Huw M. L. Davies et al.   CHEMICAL SOCIETY REVIEWS

From Sensors to Silencers: Quinoline- and Benzimidazole-Sulfonamides as Inhibitors for Zinc Proteases

(2010) Matthieu Rouffet et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

PdII‐Catalyzed MonoselectiveorthoHalogenation of CH Bonds Assisted by Counter Cations: A Complementary Method to Directedortho Lithiation

(2008) Tian‐Sheng Mei et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ammosamides A and B Target Myosin

(2008) Chambers C. Hughes et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Ammosamides: Structures of Cell Cycle Modulators from a Marine-DerivedStreptomycesSpecies

(2008) Chambers C. Hughes et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Primaquine revisited six decades after its discovery

(2008) Nuno Vale et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Ammosamides A and B new cytotoxic alkaloids isolated from a marine Streptomyces sp

(2008) SP Gaudêncio et al.   PLANTA MEDICA

Remote C–H bond functionalization reveals the distance-dependent isotope effect

(2008) Jiao-Jie Li et al.   TETRAHEDRON