PhI(OAc)2 oxidative C5 halogenation of quinolines using copper halides under mild conditions

Remote C−H Activation of Quinolines through Copper-Catalyzed Radical Cross-Coupling

(2016) Jun Xu et al.   Chemistry-An Asian Journal

Copper(ii)-catalyzed C5 and C7 halogenation of quinolines using sodium halides under mild conditions

(2016) Jun Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalyzed Regioselective C–H Iodination of Aromatic Carboxamides

(2016) Qiaolin Wu et al.   SYNLETT

Oxidative Remote C−H Trifluoromethylation of Quinolineamides on the C5 Position with Iodobenzene Diacetate as the Oxidizing Agent

(2016) Zhaoyang Wu et al.   Asian Journal of Organic Chemistry

Ligand-Enabled Cross-Coupling of C(sp3)–H Bonds with Arylsilanes

(2015) Jian He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bifunctional Organocatalysts for the Enantioselective Synthesis of Axially Chiral Isoquinoline N-Oxides

(2015) Ryota Miyaji et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper and palladium mediated C–H chlorination on 8-acylaminoquinoline scaffolds

(2015) Haili Guo et al.   TETRAHEDRON

Ligand-Enabled Triple CH Activation Reactions: One-Pot Synthesis of Diverse 4-Aryl-2-quinolinones from Propionamides

(2014) Youqian Deng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of quinoline small molecules with potent dispersal activity against methicillin-resistant Staphylococcus aureus and Staphylococcus epidermidis biofilms using a scaffold hopping strategy

(2014) Yasmeen Abouelhassan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Coordination of Hydroxyquinolines to a Ruthenium Bis-dimethyl-phenanthroline Scaffold Radically Improves Potency for Potential as Antineoplastic Agents

(2014) David K. Heidary et al.   JOURNAL OF MEDICINAL CHEMISTRY

Evaluation of (4-aminobutyloxy)quinolines as a novel class of antifungal agents

(2013) Stéphanie Vandekerckhove et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The antitumor activity of zinc(II) and copper(II) complexes with 5,7-dihalo-substituted-8-quinolinoline

(2013) Yan-Cheng Liu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric chroman synthesis via an intramolecular oxy-Michael addition by bifunctional organocatalysts

(2013) Ryota Miyaji et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of 3-(1-alkyl/aminoalkyl-3-vinyl-piperidin-4-yl)-1-(quinolin-4-yl)-propan-1-ones and their 2-methylene derivatives as potential spermicidal and microbicidal agents

(2012) Rishi Ranjan Pandey et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and antiplasmodial evaluation of novel (4-aminobutyloxy)quinolines

(2012) Stéphanie Vandekerckhove et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Copper-Dependent Cytotoxicity of 8-Hydroxyquinoline Derivatives Correlates with Their Hydrophobicity and Does Not Require Caspase Activation

(2012) Saverio Tardito et al.   JOURNAL OF MEDICINAL CHEMISTRY

Substituted oxines inhibit endothelial cell proliferation and angiogenesis

(2012) Shridhar Bhat et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Ammosamide D, an Oxidatively Ring Opened Ammosamide Analog from a Marine-Derived Streptomyces variabilis

(2012) Ende Pan et al.   ORGANIC LETTERS

Precursor-directed generation of amidine containing ammosamide analogs: ammosamides E–P

(2012) Ende Pan et al.   Chemical Science

Nitroxoline (8-hydroxy-5-nitroquinoline) is more a potent anti-cancer agent than clioquinol (5-chloro-7-iodo-8-quinoline)

(2011) Hongchao Jiang et al.   CANCER LETTERS

Solvent-free aromatic C–H functionalisation/halogenation reactions

(2010) Robin B. Bedford et al.   DALTON TRANSACTIONS

Expedient Drug Synthesis and Diversification via ortho-C−H Iodination using Recyclable PdI2as the Precatalyst

(2010) Tian-Sheng Mei et al.   ORGANIC LETTERS

Regioselective copper-catalyzed chlorination and bromination of arenes with O2 as the oxidant

(2009) Lujuan Yang et al.   CHEMICAL COMMUNICATIONS

Copper-Catalyzed Oxybromination and Oxychlorination of Primary Aromatic Amines Using LiBr or LiCl and Molecular Oxygen

(2008) Luciano Menini et al.   ADVANCED SYNTHESIS & CATALYSIS

The Ammosamides: Structures of Cell Cycle Modulators from a Marine-DerivedStreptomycesSpecies

(2008) Chambers C. Hughes et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION