Metal-free C5-selective halogenation of quinolines under aqueous conditions

Copper-catalyzed C5-selective thio/selenocyanation of 8-aminoquinolines

(2017) Jichao Chen et al.   Organic Chemistry Frontiers

Copper-Catalyzed Remote C−H Functionalization of 8-Aminoquinolines with Sodium and Lithium Sulfinates

(2016) Shuai Liang et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed Three-Component One-Pot Synthesis of Aryl Sulfides with Sulfur Powder under Aqueous Conditions

(2016) Fuhong Xiao et al.   ADVANCED SYNTHESIS & CATALYSIS

A First Example of Cobalt-Catalyzed Remote CH Functionalization of 8-Aminoquinolines Operating through a Single Electron Transfer Mechanism

(2016) Christopher J. Whiteoak et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed 8-Amido Chelation-Induced Remote C−H Amination of Quinolines

(2016) Harekrishna Sahoo et al.   CHEMISTRY-A EUROPEAN JOURNAL

Remote C−H Activation of Quinolines through Copper-Catalyzed Radical Cross-Coupling

(2016) Jun Xu et al.   Chemistry-An Asian Journal

Remote C-H Selenylation of 8-Amidoquinolines via Copper-Catalyzed Radical Cross-Coupling

(2016) Harekrishna Sahoo et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Chemoselective cross-coupling reaction of sodium sulfinates with phenols under aqueous conditions

(2016) Fuhong Xiao et al.   GREEN CHEMISTRY

Copper-Catalyzed Regioselective C–H Sulfonylation of 8-Aminoquinolines

(2016) Jun Wei et al.   JOURNAL OF ORGANIC CHEMISTRY

4-Position-Selective C–H Perfluoroalkylation and Perfluoroarylation of Six-Membered Heteroaromatic Compounds

(2016) Masahiro Nagase et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transition-metal-free oxidative C5 C–H-halogenation of 8-aminoquinoline amides using sodium halides

(2016) Ying Wang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper(ii)-catalyzed C5 and C7 halogenation of quinolines using sodium halides under mild conditions

(2016) Jun Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

5-Position-selective C–H trifluoromethylation of 8-aminoquinoline derivatives

(2016) Yoichiro Kuninobu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Nickel-Catalyzed Site-Selective C–H Bond Difluoroalkylation of 8-Aminoquinolines on the C5-Position

(2016) Hao Chen et al.   ORGANIC LETTERS

Rh-Catalyzed, Regioselective, C–H Bond Functionalization: Access to Quinoline-Branched Amines and Dimers

(2016) M. Damoder Reddy et al.   ORGANIC LETTERS

Regio- and Chemoselective Mono- and Bisnitration of 8-Amino quinoline Amides with Fe(NO3)3·9H2O as Promoter and Nitro Source

(2016) Yan He et al.   ORGANIC LETTERS

Copper-Catalyzed Regioselective C–H Iodination of Aromatic Carboxamides

(2016) Qiaolin Wu et al.   SYNLETT

PhI(OAc)2 oxidative C5 halogenation of quinolines using copper halides under mild conditions

(2016) Xing-Xing Liu et al.   RSC Advances

Copper(ii)-catalyzed remote sulfonylation of aminoquinolines with sodium sulfinates via radical coupling

(2016) Chengcai Xia et al.   RSC Advances

Silver(i)-promoted C5–H phosphonation of 8-aminoquinoline amides with H-phosphonates

(2016) Mengmeng Sun et al.   Organic Chemistry Frontiers

Selective remote C–H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis

(2015) Hong-Wen Liang et al.   CHEMICAL COMMUNICATIONS

Copper-Mediated Remote C–H Bond Chalcogenation of Quinolines on the C5 Position

(2015) Longzhi Zhu et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Sulfonylation of 8-Aminoquinoline Amides with Sulfonyl Chlorides in Air

(2015) Huijie Qiao et al.   ORGANIC LETTERS

Copper and palladium mediated C–H chlorination on 8-acylaminoquinoline scaffolds

(2015) Haili Guo et al.   TETRAHEDRON

Cobalt-Catalyzed C-4 Selective Alkylation of Quinolines

(2014) Shohei Yamamoto et al.   ADVANCED SYNTHESIS & CATALYSIS

Discovery of quinoline small molecules with potent dispersal activity against methicillin-resistant Staphylococcus aureus and Staphylococcus epidermidis biofilms using a scaffold hopping strategy

(2014) Yasmeen Abouelhassan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Transition-metal-free C–C bond forming reactions of aryl, alkenyl and alkynylboronic acids and their derivatives

(2014) S. Roscales et al.   CHEMICAL SOCIETY REVIEWS

Coordination of Hydroxyquinolines to a Ruthenium Bis-dimethyl-phenanthroline Scaffold Radically Improves Potency for Potential as Antineoplastic Agents

(2014) David K. Heidary et al.   JOURNAL OF MEDICINAL CHEMISTRY

Syntheses, Radiolabelings, and in Vitro Evaluations of Fluorinated PET Radioligands of 5-HT6 Serotoninergic Receptors

(2014) Julie Colomb et al.   JOURNAL OF MEDICINAL CHEMISTRY

Rh(III)-Catalyzed Traceless Coupling of Quinoline N-Oxides with Internal Diarylalkynes

(2014) Upendra Sharma et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-Catalyzed Site-Selective Alkylation of Unactivated C(sp3)–H Bonds

(2014) Xuesong Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regioselective Introduction of Heteroatoms at the C-8 Position of Quinoline N-Oxides: Remote C–H Activation Using N-Oxide as a Stepping Stone

(2014) Heejun Hwang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iron-Catalyzed, Chelation-Induced Remote C–H Allylation of Quinolines via 8-Amido Assistance

(2014) Xuefeng Cong et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Amination of Quinoline N-Oxides via C–H Bond Activation under Mild Conditions

(2014) Chongwei Zhu et al.   ORGANIC LETTERS

Palladium-Catalyzed C8-Selective C–H Arylation of Quinoline N-Oxides: Insights into the Electronic, Steric, and Solvation Effects on the Site Selectivity by Mechanistic and DFT Computational Studies

(2014) David E. Stephens et al.   ACS Catalysis

8-Aminoquinoline: A Powerful Directing Group in Metal-Catalyzed Direct Functionalization of CH Bonds

(2013) Matthieu Corbet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups

(2013) Guy Rouquet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A tandem Friedel–Crafts based method for the construction of a tricyclic pyrroloquinoline skeleton and its application in the synthesis of ammosamide B

(2013) Yohei Takayama et al.   CHEMICAL COMMUNICATIONS

Benign by design: catalyst-free in-water, on-water green chemical methodologies in organic synthesis

(2013) Manoj B. Gawande et al.   CHEMICAL SOCIETY REVIEWS

Design, synthesis and biological evaluation of 2-substituted quinolines as potential antileishmanial agents

(2013) Vadiraj S. Gopinath et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The antitumor activity of zinc(II) and copper(II) complexes with 5,7-dihalo-substituted-8-quinolinoline

(2013) Yan-Cheng Liu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Transition-Metal-Free BF3-Mediated Regioselective Direct Alkylation and Arylation of Functionalized Pyridines Using Grignard or Organozinc Reagents

(2013) Quan Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed C-2 Selective Arylation of Quinolines

(2013) Xiaoyu Ren et al.   ORGANIC LETTERS

Recent advances in transition-metal-free carbon–carbon and carbon–heteroatom bond-forming reactions using arynes

(2012) Anup Bhunia et al.   CHEMICAL SOCIETY REVIEWS

Copper-Dependent Cytotoxicity of 8-Hydroxyquinoline Derivatives Correlates with Their Hydrophobicity and Does Not Require Caspase Activation

(2012) Saverio Tardito et al.   JOURNAL OF MEDICINAL CHEMISTRY

Substituted oxines inhibit endothelial cell proliferation and angiogenesis

(2012) Shridhar Bhat et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Ammosamide D, an Oxidatively Ring Opened Ammosamide Analog from a Marine-Derived Streptomyces variabilis

(2012) Ende Pan et al.   ORGANIC LETTERS

Precursor-directed generation of amidine containing ammosamide analogs: ammosamides E–P

(2012) Ende Pan et al.   Chemical Science

Green chemistry oriented organic synthesis in water

(2011) Marc-Olivier Simon et al.   CHEMICAL SOCIETY REVIEWS

Rh(NHC)-Catalyzed Direct and Selective Arylation of Quinolines at the 8-Position

(2011) Jaesung Kwak et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd0/PR3-Catalyzed Arylation of Nicotinic and Isonicotinic Acid Derivatives

(2010) Masayuki Wasa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and structure–activity relationships of antimalarial 4-oxo-3-carboxyl quinolones

(2010) Yiqun Zhang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Quinolines and structurally related heterocycles as antimalarials

(2010) Kirandeep Kaur et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Bimetallic Nickel Aluminun MediatedPara-Selective Alkenylation of Pyridine: Direct Observation of η2,η1-Pyridine Ni(0)−Al(III) Intermediates Prior to C−H Bond Activation

(2010) Chung-Chih Tsai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of the Ammosamides

(2010) Chambers C. Hughes et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct C−H Arylation of Electron-Deficient Heterocycles with Arylboronic Acids

(2010) Ian B. Seiple et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A3Receptor

(2009) Laura H. Heitman et al.   JOURNAL OF MEDICINAL CHEMISTRY

Sc(OTf)3-Catalyzed Direct Alkylation of Quinolines and Pyridines with Alkanes

(2009) Guojun Deng et al.   ORGANIC LETTERS

The Ammosamides: Structures of Cell Cycle Modulators from a Marine-DerivedStreptomycesSpecies

(2008) Chambers C. Hughes et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rh(I)-Catalyzed Direct Arylation of Pyridines and Quinolines

(2008) Ashley M. Berman et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS