Functionalization of Quinolines through Copper-Catalyzed Regioselective Halogenation Reaction

Copper-Catalyzed Regioselective C–H Sulfonylation of 8-Aminoquinolines

(2016) Jun Wei et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper(ii)-catalyzed C5 and C7 halogenation of quinolines using sodium halides under mild conditions

(2016) Jun Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Developing structure–activity relationships from an HTS hit for inhibition of the Cks1–Skp2 protein–protein interaction

(2015) Rajinder Singh et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Selective remote C–H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis

(2015) Hong-Wen Liang et al.   CHEMICAL COMMUNICATIONS

Metal-free synthesis of N-fused heterocyclic iodides via C–H functionalization mediated by tert-butylhydroperoxide

(2015) Krishna K. Sharma et al.   CHEMICAL COMMUNICATIONS

The regioselective iodination of quinolines, quinolones, pyridones, pyridines and uracil

(2015) Uttam Dutta et al.   CHEMICAL COMMUNICATIONS

Cobalt-Catalyzed C5-Selective C-H Functionalization of 4-Me-Quinolines with Styrenes: An Approach to 5,6-Dihydro-4H-benzo[de]quinolines

(2015) Shigeki Matsunaga et al.   HETEROCYCLES

Cp*Ir(III)-Catalyzed Mild and Broad C−H Arylation of Arenes and Alkenes with Aryldiazonium Salts Leading to the External Oxidant-Free Approach

(2015) Kwangmin Shin et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Multimetallic catalysed cross-coupling of aryl bromides with aryl triflates

(2015) Laura K. G. Ackerman et al.   NATURE

Nickel-catalyzed synthesis of diarylsulfides and sulfones via C–H bond functionalization of arylamides

(2015) Vutukuri Prakash Reddy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Regioselective, Molecular Iodine-Mediated C3 Iodination of Quinolines

(2015) Kai Sun et al.   ORGANIC LETTERS

Copper-Mediated Remote C–H Bond Chalcogenation of Quinolines on the C5 Position

(2015) Longzhi Zhu et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Sulfonylation of 8-Aminoquinoline Amides with Sulfonyl Chlorides in Air

(2015) Huijie Qiao et al.   ORGANIC LETTERS

Direct ortho-Thiolation of Arenes and Alkenes by Nickel Catalysis

(2015) Cong Lin et al.   ORGANIC LETTERS

Copper and palladium mediated C–H chlorination on 8-acylaminoquinoline scaffolds

(2015) Haili Guo et al.   TETRAHEDRON

Recent advances in the C–H-functionalization of the distal positions in pyridines and quinolines

(2015) David E. Stephens et al.   TETRAHEDRON

Transition-Metal-Catalyzed Site-Selective C–H Functionalization of Quinolines beyond C2 Selectivity

(2015) Tomohiro Iwai et al.   ACS Catalysis

Copper-catalyzed C–H alkylation of 8-aminoquinolines via 8-amide chelation assistance

(2015) Xiao-Feng Xia et al.   RSC Advances

Cobalt-Catalyzed C-4 Selective Alkylation of Quinolines

(2014) Shohei Yamamoto et al.   ADVANCED SYNTHESIS & CATALYSIS

Rh(III)-Catalyzed Traceless Coupling of Quinoline N-Oxides with Internal Diarylalkynes

(2014) Upendra Sharma et al.   JOURNAL OF ORGANIC CHEMISTRY

Regioselective Introduction of Heteroatoms at the C-8 Position of Quinoline N-Oxides: Remote C–H Activation Using N-Oxide as a Stepping Stone

(2014) Heejun Hwang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iron-Catalyzed, Chelation-Induced Remote C–H Allylation of Quinolines via 8-Amido Assistance

(2014) Xuefeng Cong et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Amination of Quinoline N-Oxides via C–H Bond Activation under Mild Conditions

(2014) Chongwei Zhu et al.   ORGANIC LETTERS

Palladium-Catalyzed C8-Selective C–H Arylation of Quinoline N-Oxides: Insights into the Electronic, Steric, and Solvation Effects on the Site Selectivity by Mechanistic and DFT Computational Studies

(2014) David E. Stephens et al.   ACS Catalysis

A novel pyrene-containing fluorescent organogel derived from a quinoline-based fluorescent porbe: synthesis, sensing properties, and its aggregation behavior

(2014) Chang-Bo Huang et al.   RSC Advances

Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups

(2013) Guy Rouquet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Site-Selective CH Borylation of Quinolines at the C8 Position Catalyzed by a Silica-Supported Phosphane-Iridium System

(2013) Shota Konishi et al.   Chemistry-An Asian Journal

Transition-Metal-Free BF3-Mediated Regioselective Direct Alkylation and Arylation of Functionalized Pyridines Using Grignard or Organozinc Reagents

(2013) Quan Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(III)-Catalyzed Oxidative Olefination of Pyridines and Quinolines: Multigram-Scale Synthesis of Naphthyridinones

(2013) Jun Zhou et al.   ORGANIC LETTERS

Palladium-Catalyzed C-2 Selective Arylation of Quinolines

(2013) Xiaoyu Ren et al.   ORGANIC LETTERS

Pd(ii)-catalyzed alkoxylation of unactivated C(sp3)–H and C(sp2)–H bonds using a removable directing group: efficient synthesis of alkyl ethers

(2013) Fa-Jie Chen et al.   Chemical Science

Ruthenium(II)-Catalyzed C–H Bond Activation and Functionalization

(2012) Percia Beatrice Arockiam et al.   CHEMICAL REVIEWS

Towards mild metal-catalyzed C–H bond activation

(2011) Joanna Wencel-Delord et al.   CHEMICAL SOCIETY REVIEWS

Recent developments in natural product synthesis using metal-catalysed C–H bond functionalisation

(2011) Lindsay McMurray et al.   CHEMICAL SOCIETY REVIEWS

Rh(NHC)-Catalyzed Direct and Selective Arylation of Quinolines at the 8-Position

(2011) Jaesung Kwak et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Nickel-catalyzed cross coupling of non-activated alkyl halides: a mechanistic perspective

(2011) Xile Hu   Chemical Science

Pd0/PR3-Catalyzed Arylation of Nicotinic and Isonicotinic Acid Derivatives

(2010) Masayuki Wasa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

(2010) Thomas W. Lyons et al.   CHEMICAL REVIEWS

A ratiometric fluorescent probe for oxalate based on alkyne-conjugated carboxamidoquinolines in aqueous solution and imaging in living cells

(2010) Chunsheng He et al.   DALTON TRANSACTIONS

Bimetallic Nickel Aluminun MediatedPara-Selective Alkenylation of Pyridine: Direct Observation of η2,η1-Pyridine Ni(0)−Al(III) Intermediates Prior to C−H Bond Activation

(2010) Chung-Chih Tsai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct C−H Arylation of Electron-Deficient Heterocycles with Arylboronic Acids

(2010) Ian B. Seiple et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Biological Activities of Quinoline Derivatives

(2010) Suresh Kumar et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds

(2009) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(II)-Catalyzed CH Activation/CC Cross-Coupling Reactions: Versatility and Practicality

(2009) Xiao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed Reaction of Arylzinc Reagents with N-Aromatic Heterocycles: A Straightforward Approach to C−H Bond Arylation of Electron-Deficient Heteroaromatic Compounds

(2009) Mamoru Tobisu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Organoboron Quinoline-8-thiolate and Quinoline-8-selenolate Complexes and Their Incorporation into the π-Conjugated Polymer Main-Chain

(2009) Yuichiro Tokoro et al.   MACROMOLECULES

Sc(OTf)3-Catalyzed Direct Alkylation of Quinolines and Pyridines with Alkanes

(2009) Guojun Deng et al.   ORGANIC LETTERS

Rh(I)-Catalyzed Direct Arylation of Pyridines and Quinolines

(2008) Ashley M. Berman et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS