Synthesis and biological evaluation of phloroglucinol derivatives possessing α-glycosidase, acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase inhibitory activity

Recent progress in the identification of selective butyrylcholinesterase inhibitors for Alzheimer's disease

(2017) Qi Li et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A spectroscopic study on the absorption of carbonic anhydrase onto the nanoporous silica nanoparticle

(2017) Hannaneh Pourjabbari Khameneh et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors

(2017) Fevzi Topal et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Assessment of the inhibitory effects and molecular docking of some sulfonamides on human serum paraoxonase 1

(2017) Zuhal Alim et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Antidiabetic potential: in vitro inhibition effects of some natural phenolic compounds on α-glycosidase and α-amylase enzymes

(2017) Parham Taslimi et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Synephrine and phenylephrine act as α-amylase, α-glycosidase, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase enzymes inhibitors

(2017) Parham Taslimi et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Synthesis and bioactivity of several new hetaryl sulfonamides

(2017) Parham Taslimi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities

(2017) Halise I. Gul et al.   Letters in Drug Design & Discovery

Secondary Sulfonamides as Effective Lactoperoxidase Inhibitors

(2017) Zeynep Köksal et al.   MOLECULES

Effect of mutation in active site residue Trp209 to Val, Leu, Ile and Pro on the catalytic activity and affinity for some benzenesulfonamides of human carbonic anhydrase II

(2017) Deryanur KILIÇ et al.   TURKISH JOURNAL OF BIOLOGY

Biophenols of mints: Antioxidant, acetylcholinesterase, butyrylcholinesterase and histone deacetylase inhibition activities targeting Alzheimer’s disease treatment

(2017) Doaa M. Hanafy et al.   Journal of Functional Foods

Carbonic anhydrase inhibitory properties of phenolic sulfonamides derived from dopamine related compounds

(2017) Hulya Göcer et al.   Arabian Journal of Chemistry

Synthesis and Carbonic Anhydrase Inhibition of Novel 2-(4-(Aryl)thiazole-2-yl)-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-dione Derivatives

(2016) Umit M. Kocyigit et al.   ARCHIV DER PHARMAZIE

Antioxidant Activity, Acetylcholinesterase, and Carbonic Anhydrase Inhibitory Properties of Novel Ureas Derived from Phenethylamines

(2016) Kadir Aksu et al.   ARCHIV DER PHARMAZIE

Structure and function of carbonic anhydrases

(2016) C. T. Supuran   BIOCHEMICAL JOURNAL

Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds

(2016) Bünyamin Özgeriş et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase activators: Activation of the β-carbonic anhydrase from Malassezia globosa with amines and amino acids

(2016) Daniela Vullo et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Purification and characterization of the carbonic anhydrase enzyme from Black Sea trout (Salmo trutta Labrax Coruhensis) kidney and inhibition effects of some metal ions on enzyme activity

(2016) Murat Kucuk et al.   ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY

Synthesis, carbonic anhydrase I and II isoenzymes inhibition properties, and antibacterial activities of novel tetralone-based 1,4-benzothiazepine derivatives

(2016) Mustafa Ceylan et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Synthesis of two phloroglucinol derivatives with cinnamyl moieties as inhibitors of the carbonic anhydrase isozymes I and II: an in vitro study

(2016) Serdar Burmaoğlu et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and inhibitory properties of some carbamates on carbonic anhydrase and acetylcholine esterase

(2016) Süleyman Yılmaz et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles

(2016) Burhanettin Turan et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of diaryl ethers with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions

(2016) Fadime Özbey et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of 4,5-disubstituted-2-thioxo-1,2,3,4-tetrahydropyrimidines and investigation of their acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase I/II inhibitory and antioxidant activities

(2016) Emin Garibov et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The Use of Multiscale Molecular Simulations in Understanding a Relationship between the Structure and Function of Biological Systems of the Brain: The Application to Monoamine Oxidase Enzymes

(2016) Robert Vianello et al.   Frontiers in Neuroscience

Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune

(2015) Daniela Vullo et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of potent carbonic anhydrase and acetylcholine esterase inhibitors: Novel sulfamoylcarbamates and sulfamides derived from acetophenones

(2015) Akın Akıncıoğlu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II

(2015) Alper Yıldırım et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Antioxidant and acetylcholinesterase inhibition properties of novel bromophenol derivatives

(2015) Necla Öztaşkın et al.   BIOORGANIC CHEMISTRY

Metabolomic and chemometric study of Achras sapota L. fruit extracts for identification of metabolites contributing to the inhibition of α-amylase and α-glucosidase

(2015) Susmita Das et al.   EUROPEAN FOOD RESEARCH AND TECHNOLOGY

LC–MS/MS analysis, antioxidant and anticholinergic properties of galanga (Alpinia officinarum Hance) rhizomes

(2015) Leyla Polat Köse et al.   INDUSTRIAL CROPS AND PRODUCTS

Purification and Characterization of Polyphenol Oxidase from Hemşin Apple (Malus communisL.)

(2015) Bahar Aydin et al.   INTERNATIONAL JOURNAL OF FOOD PROPERTIES

The effect of caffeic acid phenethyl ester (CAPE) on metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, lactoperoxidase, and carbonic anhydrase isoenzymes I, II, IX, and XII

(2015) İlhami Gülçin et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Inhibitory effects of some phenolic compounds on the activities of carbonic anhydrase: from in vivo to ex vivo

(2015) Zübeyir Huyut et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII)

(2015) Andrea Scozzafava et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of Some Novel Norbornene-Fused Pyridazines as Potent Inhibitors of Carbonic Anhydrase and Acetylcholinesterase

(2015) Ramazan Kocak et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Protozoan Parasite Growth Inhibitors Discovered by Cross-Screening Yield Potent Scaffolds for Lead Discovery

(2015) William Devine et al.   JOURNAL OF MEDICINAL CHEMISTRY

The Chemistry of Neurodegeneration: Kinetic Data and Their Implications

(2015) Matic Pavlin et al.   MOLECULAR NEUROBIOLOGY

Dialkylzinc-mediated allylic polyfluoroarylation reaction

(2015) Daisuke Kurauchi et al.   TETRAHEDRON

Novel anticancer activity of phloroglucinol against breast cancer stem-like cells

(2015) Rae-Kwon Kim et al.   TOXICOLOGY AND APPLIED PHARMACOLOGY

Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties

(2014) Murat Boztaş et al.   JOURNAL OF MEDICINAL CHEMISTRY

An Isothiourea-Catalyzed Asymmetric [2,3]-Rearrangement of Allylic Ammonium Ylides

(2014) Thomas H. West et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Capsaicin: A Potent Inhibitor of Carbonic Anhydrase Isoenzymes

(2014) Betul Arabaci et al.   MOLECULES

α-Ketophosphonates as Ester Surrogates: Isothiourea-Catalyzed Asymmetric Diester and Lactone Synthesis

(2014) Siobhan R. Smith et al.   ORGANIC LETTERS

The Role of Phenolic Compounds in the Fight against Cancer – A Review

(2013) Márcio Carocho et al.   Anti-Cancer Agents in Medicinal Chemistry

Novel sulfamides as potential carbonic anhydrase isoenzymes inhibitors

(2013) Akın Akıncıoğlu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine

(2013) Kadir Aksu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Inhibitor Design for Monoamine Oxidases

(2013) Rona R. Ramsay   CURRENT PHARMACEUTICAL DESIGN

Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments

(2013) G. Madhavi Sastry et al.   JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN

Structures of Human Acetylcholinesterase Bound to Dihydrotanshinone I and Territrem B Show Peripheral Site Flexibility

(2013) Jonah Cheung et al.   ACS Medicinal Chemistry Letters

Rapid screening and identification ofα-glucosidase inhibitors from mulberry leaves using enzyme-immobilized magnetic beads coupled with HPLC/MS and NMR

(2012) Yi Tao et al.   BIOMEDICAL CHROMATOGRAPHY

One-step purification of lactoperoxidase from bovine milk by affinity chromatography

(2012) Ali Atasever et al.   FOOD CHEMISTRY

Synthesis of Arylnaphthalene Lignan Scaffold by Gold-Catalyzed Intramolecular Sequential Electrophilic Addition and Benzannulation

(2011) Vanajakshi Gudla et al.   JOURNAL OF ORGANIC CHEMISTRY

Crystal structures of isomaltase from Saccharomyces cerevisiae and in complex with its competitive inhibitor maltose

(2010) Keizo Yamamoto et al.   FEBS Journal

Synthesis and antioxidant properties of diphenylmethane derivative bromophenols including a natural product

(2010) Halis Türker Balaydın et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Isosorbide-2-benzyl Carbamate-5-salicylate, A Peripheral Anionic Site Binding Subnanomolar Selective Butyrylcholinesterase Inhibitor

(2010) Ciaran G. Carolan et al.   JOURNAL OF MEDICINAL CHEMISTRY

α-Amylase and Lipase Inhibitory Activity and Structural Characterization of Acacia Bark Proanthocyanidins

(2010) Rie Kusano et al.   JOURNAL OF NATURAL PRODUCTS

Phloroglucinol compounds of natural origin: Synthetic aspects

(2010) Inder Pal Singh et al.   NATURAL PRODUCT REPORTS

Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols

(2009) Murat Şentürk et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of Two Alnustone-Like Natural Diarylheptanoids via 4 + 3 Strategy

(2009) Serdar Burmaoğlu et al.   SYNTHETIC COMMUNICATIONS

Preparation and characterisation of a quinone-functionalised polythiophene film on a modified electrode. Application to the potentiometric determination of glutathione and cysteine concentrations

(2008) Stéphanie Étienne et al.   TETRAHEDRON