Synthesis and biological evaluation of phloroglucinol derivatives possessing α-glycosidase, acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase inhibitory activity
出版年份 2018 全文链接
标题
Synthesis and biological evaluation of phloroglucinol derivatives possessing α-glycosidase, acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase inhibitory activity
作者
关键词
-
出版物
ARCHIV DER PHARMAZIE
Volume 351, Issue 2, Pages 1700314
出版商
Wiley
发表日期
2018-01-11
DOI
10.1002/ardp.201700314
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注意：仅列出部分参考文献，下载原文获取全部文献信息。- Recent progress in the identification of selective butyrylcholinesterase inhibitors for Alzheimer's disease
- (2017) Qi Li et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- A spectroscopic study on the absorption of carbonic anhydrase onto the nanoporous silica nanoparticle
- (2017) Hannaneh Pourjabbari Khameneh et al. INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES
- Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors
- (2017) Fevzi Topal et al. INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES
- Assessment of the inhibitory effects and molecular docking of some sulfonamides on human serum paraoxonase 1
- (2017) Zuhal Alim et al. JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY
- Antidiabetic potential: in vitro inhibition effects of some natural phenolic compounds on α-glycosidase and α-amylase enzymes
- (2017) Parham Taslimi et al. JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY
- Synephrine and phenylephrine act as α-amylase, α-glycosidase, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase enzymes inhibitors
- (2017) Parham Taslimi et al. JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY
- Synthesis and bioactivity of several new hetaryl sulfonamides
- (2017) Parham Taslimi et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities
- (2017) Halise I. Gul et al. Letters in Drug Design & Discovery
- Secondary Sulfonamides as Effective Lactoperoxidase Inhibitors
- (2017) Zeynep Köksal et al. MOLECULES
- Effect of mutation in active site residue Trp209 to Val, Leu, Ile and Pro on the catalytic activity and affinity for some benzenesulfonamides of human carbonic anhydrase II
- (2017) Deryanur KILIÇ et al. TURKISH JOURNAL OF BIOLOGY
- Biophenols of mints: Antioxidant, acetylcholinesterase, butyrylcholinesterase and histone deacetylase inhibition activities targeting Alzheimer’s disease treatment
- (2017) Doaa M. Hanafy et al. Journal of Functional Foods
- Carbonic anhydrase inhibitory properties of phenolic sulfonamides derived from dopamine related compounds
- (2017) Hulya Göcer et al. Arabian Journal of Chemistry
- Synthesis and Carbonic Anhydrase Inhibition of Novel 2-(4-(Aryl)thiazole-2-yl)-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-dione Derivatives
- (2016) Umit M. Kocyigit et al. ARCHIV DER PHARMAZIE
- Antioxidant Activity, Acetylcholinesterase, and Carbonic Anhydrase Inhibitory Properties of Novel Ureas Derived from Phenethylamines
- (2016) Kadir Aksu et al. ARCHIV DER PHARMAZIE
- Structure and function of carbonic anhydrases
- (2016) C. T. Supuran BIOCHEMICAL JOURNAL
- Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds
- (2016) Bünyamin Özgeriş et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Carbonic anhydrase activators: Activation of the β-carbonic anhydrase from Malassezia globosa with amines and amino acids
- (2016) Daniela Vullo et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Purification and characterization of the carbonic anhydrase enzyme from Black Sea trout (Salmo trutta Labrax Coruhensis) kidney and inhibition effects of some metal ions on enzyme activity
- (2016) Murat Kucuk et al. ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY
- Synthesis, carbonic anhydrase I and II isoenzymes inhibition properties, and antibacterial activities of novel tetralone-based 1,4-benzothiazepine derivatives
- (2016) Mustafa Ceylan et al. JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY
- Synthesis of two phloroglucinol derivatives with cinnamyl moieties as inhibitors of the carbonic anhydrase isozymes I and II: an in vitro study
- (2016) Serdar Burmaoğlu et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis and inhibitory properties of some carbamates on carbonic anhydrase and acetylcholine esterase
- (2016) Süleyman Yılmaz et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles
- (2016) Burhanettin Turan et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis of diaryl ethers with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions
- (2016) Fadime Özbey et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis of 4,5-disubstituted-2-thioxo-1,2,3,4-tetrahydropyrimidines and investigation of their acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase I/II inhibitory and antioxidant activities
- (2016) Emin Garibov et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- The Use of Multiscale Molecular Simulations in Understanding a Relationship between the Structure and Function of Biological Systems of the Brain: The Application to Monoamine Oxidase Enzymes
- (2016) Robert Vianello et al. Frontiers in Neuroscience
- Sulfonamide inhibition studies of the γ-carbonic anhydrase from the Antarctic cyanobacterium Nostoc commune
- (2015) Daniela Vullo et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Discovery of potent carbonic anhydrase and acetylcholine esterase inhibitors: Novel sulfamoylcarbamates and sulfamides derived from acetophenones
- (2015) Akın Akıncıoğlu et al. BIOORGANIC & MEDICINAL CHEMISTRY
- N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II
- (2015) Alper Yıldırım et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Antioxidant and acetylcholinesterase inhibition properties of novel bromophenol derivatives
- (2015) Necla Öztaşkın et al. BIOORGANIC CHEMISTRY
- Metabolomic and chemometric study of Achras sapota L. fruit extracts for identification of metabolites contributing to the inhibition of α-amylase and α-glucosidase
- (2015) Susmita Das et al. EUROPEAN FOOD RESEARCH AND TECHNOLOGY
- LC–MS/MS analysis, antioxidant and anticholinergic properties of galanga (Alpinia officinarum Hance) rhizomes
- (2015) Leyla Polat Köse et al. INDUSTRIAL CROPS AND PRODUCTS
- Purification and Characterization of Polyphenol Oxidase from Hemşin Apple (Malus communisL.)
- (2015) Bahar Aydin et al. INTERNATIONAL JOURNAL OF FOOD PROPERTIES
- The effect of caffeic acid phenethyl ester (CAPE) on metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, lactoperoxidase, and carbonic anhydrase isoenzymes I, II, IX, and XII
- (2015) İlhami Gülçin et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Inhibitory effects of some phenolic compounds on the activities of carbonic anhydrase: from in vivo to ex vivo
- (2015) Zübeyir Huyut et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- The impact of hydroquinone on acetylcholine esterase and certain human carbonic anhydrase isoenzymes (hCA I, II, IX, and XII)
- (2015) Andrea Scozzafava et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis of Some Novel Norbornene-Fused Pyridazines as Potent Inhibitors of Carbonic Anhydrase and Acetylcholinesterase
- (2015) Ramazan Kocak et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- Protozoan Parasite Growth Inhibitors Discovered by Cross-Screening Yield Potent Scaffolds for Lead Discovery
- (2015) William Devine et al. JOURNAL OF MEDICINAL CHEMISTRY
- The Chemistry of Neurodegeneration: Kinetic Data and Their Implications
- (2015) Matic Pavlin et al. MOLECULAR NEUROBIOLOGY
- Dialkylzinc-mediated allylic polyfluoroarylation reaction
- (2015) Daisuke Kurauchi et al. TETRAHEDRON
- Novel anticancer activity of phloroglucinol against breast cancer stem-like cells
- (2015) Rae-Kwon Kim et al. TOXICOLOGY AND APPLIED PHARMACOLOGY
- Synthesis and Carbonic Anhydrase Isoenzymes I, II, IX, and XII Inhibitory Effects of Dimethoxybromophenol Derivatives Incorporating Cyclopropane Moieties
- (2014) Murat Boztaş et al. JOURNAL OF MEDICINAL CHEMISTRY
- An Isothiourea-Catalyzed Asymmetric [2,3]-Rearrangement of Allylic Ammonium Ylides
- (2014) Thomas H. West et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Capsaicin: A Potent Inhibitor of Carbonic Anhydrase Isoenzymes
- (2014) Betul Arabaci et al. MOLECULES
- α-Ketophosphonates as Ester Surrogates: Isothiourea-Catalyzed Asymmetric Diester and Lactone Synthesis
- (2014) Siobhan R. Smith et al. ORGANIC LETTERS
- The Role of Phenolic Compounds in the Fight against Cancer – A Review
- (2013) Márcio Carocho et al. Anti-Cancer Agents in Medicinal Chemistry
- Novel sulfamides as potential carbonic anhydrase isoenzymes inhibitors
- (2013) Akın Akıncıoğlu et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine
- (2013) Kadir Aksu et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Inhibitor Design for Monoamine Oxidases
- (2013) Rona R. Ramsay CURRENT PHARMACEUTICAL DESIGN
- Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments
- (2013) G. Madhavi Sastry et al. JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN
- Structures of Human Acetylcholinesterase Bound to Dihydrotanshinone I and Territrem B Show Peripheral Site Flexibility
- (2013) Jonah Cheung et al. ACS Medicinal Chemistry Letters
- Rapid screening and identification ofα-glucosidase inhibitors from mulberry leaves using enzyme-immobilized magnetic beads coupled with HPLC/MS and NMR
- (2012) Yi Tao et al. BIOMEDICAL CHROMATOGRAPHY
- One-step purification of lactoperoxidase from bovine milk by affinity chromatography
- (2012) Ali Atasever et al. FOOD CHEMISTRY
- Synthesis of Arylnaphthalene Lignan Scaffold by Gold-Catalyzed Intramolecular Sequential Electrophilic Addition and Benzannulation
- (2011) Vanajakshi Gudla et al. JOURNAL OF ORGANIC CHEMISTRY
- Crystal structures of isomaltase from Saccharomyces cerevisiae and in complex with its competitive inhibitor maltose
- (2010) Keizo Yamamoto et al. FEBS Journal
- Synthesis and antioxidant properties of diphenylmethane derivative bromophenols including a natural product
- (2010) Halis Türker Balaydın et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Isosorbide-2-benzyl Carbamate-5-salicylate, A Peripheral Anionic Site Binding Subnanomolar Selective Butyrylcholinesterase Inhibitor
- (2010) Ciaran G. Carolan et al. JOURNAL OF MEDICINAL CHEMISTRY
- α-Amylase and Lipase Inhibitory Activity and Structural Characterization of Acacia Bark Proanthocyanidins
- (2010) Rie Kusano et al. JOURNAL OF NATURAL PRODUCTS
- Phloroglucinol compounds of natural origin: Synthetic aspects
- (2010) Inder Pal Singh et al. NATURAL PRODUCT REPORTS
- Carbonic anhydrase inhibitors. Inhibition of human erythrocyte isozymes I and II with a series of antioxidant phenols
- (2009) Murat Şentürk et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of Two Alnustone-Like Natural Diarylheptanoids via 4 + 3 Strategy
- (2009) Serdar Burmaoğlu et al. SYNTHETIC COMMUNICATIONS
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