Recent developments in chemical reactivity of N,N-dimethylenamino ketones as synthons for various heterocycles

Lewis Acid-Catalyzed [3+2] Cycloaddition of Donor-Acceptor Cyclopropanes and Enamines: Enantioselective Synthesis of Nitrogen-Functionalized Cyclopentane Derivatives

(2016) Kamal Verma et al.   ADVANCED SYNTHESIS & CATALYSIS

Solvent-free synthesis of 6-unsubstituted dihydropyrimidinones using 2-pyrrolidonium bisulphate as efficient catalyst

(2016) Heshmatollah Alinezhad et al.   CHEMICAL PAPERS

Metal-free oxidative carbonylation on enaminone CC bond for the cascade synthesis of benzothiazole-containing vicinal diketones

(2016) Jie-Ping Wan et al.   GREEN CHEMISTRY

Promotion of 1,3-dipolar cycloaddition between azides and β-enaminones by deep eutectic solvents

(2016) Marcos Antonio Pinto Martins et al.   NEW JOURNAL OF CHEMISTRY

Base-Promoted Synthesis of N-Substituted 1,2,3-Triazoles via Enaminone–Azide Cycloaddition Involving Regitz Diazo Transfer

(2016) Jie-Ping Wan et al.   ORGANIC LETTERS

A simple one-pot synthesis of quinoline-4-carboxylic acids by the Pfitzinger reaction of isatin with enaminones in water

(2016) Ibrahim Elghamry et al.   TETRAHEDRON LETTERS

Cover Picture: Structurally Defined Molecular Hypervalent Iodine Catalysts for Intermolecular Enantioselective Reactions (Angew. Chem. Int. Ed. 1/2016)

(2015) Stefan Haubenreisser et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Novel 4-Heteroaryl-Antipyrines as DPP-IV Inhibitors

(2015) Sobhi M. Gomha et al.   Chemical Biology & Drug Design

Utility of 3-Acetyl-6-bromo-2H-chromen-2-one for the Synthesis of New Heterocycles as Potential Antiproliferative Agents

(2015) Sobhi Gomha et al.   MOLECULES

Enaminone-Based Three-Component Reactions for the Diastereoselective Synthesis of Fused Tetrahydropyridines

(2015) Jie-Ping Wan et al.   SYNTHESIS-STUTTGART

First examples of 2,6-diarylnicotinaldehydes prepared under conventional and microwave conditions

(2015) K. Shankaraiah et al.   TETRAHEDRON LETTERS

Correction: Novel pyrrole derivatives as selective CHK1 inhibitors: design, regioselective synthesis and molecular modeling

(2015) Taha M. A. Eldebss et al.   MedChemComm

Regioselective three-component reactions of enaminones, 2-aminopyridines and enals for the synthesis of 1,2-dihydropyridines

(2015) Shuo Cao et al.   RSC Advances

Discovery and structure–activity relationships study of novel thieno[2,3-b]pyridine analogues as hepatitis C virus inhibitors

(2014) Ning-Yu Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A Synthesis of Novel Pyrazolylthienopyrimidine Derivatives as IL-6/STAT3 Inhibitors

(2014) Sung Min Kim et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Diphenylpyrroles: Novel p53 activators

(2014) Sobhi M. Gomha et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Facile and General Approach to 3-((Trifluoromethyl)thio)-4H-chromen-4-one

(2014) Haoyue Xiang et al.   ORGANIC LETTERS

An efficient regioselective copper catalyzed multi-component synthesis of 1,3-disubstituted pyrazoles

(2014) Akula Raghunadh et al.   TETRAHEDRON LETTERS

Preparation of Polysubstituted Isochromanes by Addition of ortho-Lithiated Aryloxiranes to Enaminones

(2013) Antonio Salomone et al.   JOURNAL OF ORGANIC CHEMISTRY

Multicomponent reactions for synthesis of bioactive polyheterocyclic ring systems under controlled microwave irradiation

(2013) Eman M.H. Abbas et al.   Arabian Journal of Chemistry

Synthesis of 2-aminofurans and 2-unsubstituted furans via carbenoid-mediated [3 + 2] cycloaddition

(2012) Yaojia Jiang et al.   CHEMICAL COMMUNICATIONS

Enaminones as Building Blocks in Heterocyclic Preparations: Synthesis of Novel Pyrazoles, Pyrazolo[3,4-d]pyridazines, Pyrazolo[1,5-a]pyrimidines, Pyrido[2,3-d]pyrimidines Linked to Imidazo[2,1-b]thiazole System

(2012) Sobhi M. Gomha et al.   HETEROCYCLES

Mg–Al hydrotalcite as an efficient catalyst for microwave assisted regioselective 1,3-dipolar cycloaddition of nitrilimines with the enaminone derivatives: A green protocol

(2012) Tamer S. Saleh et al.   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Unexpected Behavior of Enaminones: Interesting New Routes to 1,6-Naphthyridines, 2-Oxopyrrolidines and Pyrano[4,3,2-de][1,6]naphthyridines

(2012) Moustafa Moustafa et al.   MOLECULES

A “Catch–React–Release” Method for the Flow Synthesis of 2-Aminopyrimidines and Preparation of the Imatinib Base

(2012) Richard J. Ingham et al.   ORGANIC LETTERS

Applications of 2-arylhydrazononitriles in synthesis: Preparation of new indole containing 1,2,3-triazole, pyrazole and pyrazolo[1,5-a]pyrimidine derivatives and evaluation of their antimicrobial activities

(2011) Haider Behbehani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Mg–Al hydrotalcites as efficient catalysts for aza-Michael addition reaction: A green protocol

(2011) Mohamed Mokhtar et al.   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Synthesis and Evaluation of the Anti-Microbial Activity of New Heterocycles Containing the 1,3,4-Thiadiazole Moiety

(2011) Thoraya A. Farghaly et al.   MOLECULES

Facile Diversity-Oriented Synthesis and Antitubercular Evaluation of Novel Aryl and Heteroaryl Tethered Pyridines and Dihydro-6H-quinolin-5-ones Derived via Variants of the Bohlmann–Rahtz Reaction

(2011) Srinivas Kantevari et al.   ACS Combinatorial Science

Chemo-/regioselective synthesis of 6-unsubstituted dihydropyrimidinones, 1,3-thiazines and chromones via novel variants of Biginelli reaction

(2009) Jie-Ping Wan et al.   CHEMICAL COMMUNICATIONS

Novel Regioselectivity: Three-Component Cascade Synthesis of Unsymmetrical 1,4- and 1,2-Dihydropyridines

(2009) Jie-Ping Wan et al.   JOURNAL OF ORGANIC CHEMISTRY

Toward Safer Processes for C−C Biaryl Bond Construction: Catalytic Direct C−H Arylation and Tin-Free Radical Coupling in the Synthesis of Pyrazolophenanthridines

(2009) Susana Hernández et al.   JOURNAL OF ORGANIC CHEMISTRY

5-CARBETHOXY- AND 5-ACETYLPYRAZOLES AS PRECURSORS FOR THE SYNTHESIS OF SOME NOVEL 1-p-CHLOROPHENYLPYRAZOLE-3-CARBONITRILES

(2009) Hatem M. Gaber   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

A Facile Total Synthesis of Imatinib Base and Its Analogues

(2008) Yi-Feng Liu et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Arylhydrazonals as the aldehyde component in Baylis–Hillman reactions

(2008) Nouria A. Al-Awadi et al.   TETRAHEDRON