Design, Synthesis and Cytotoxic Evaluation of Novel Chalcone Derivatives Bearing Triazolo[4,3-a]-quinoxaline Moieties as Potent Anticancer Agents with Dual EGFR Kinase and Tubulin Polymerization Inhibitory Effects

Design, synthesis, molecular docking of new lipophilic acetamide derivatives affording potential anticancer and antimicrobial agents

(2018) Hany E.A. Ahmed et al.   BIOORGANIC CHEMISTRY

Spectroscopic studies of the molecular organization of 4-([ 1,2,4 ] triazolo [ 4,3- a ] pyridin-3-yl)-6-methylbenzene-1,3-diol in selected solvents

(2018) Arkadiusz Matwijczuk et al.   JOURNAL OF LUMINESCENCE

Microwave-Assisted Facile Synthesis, Anticancer Evaluation and Docking Study of N-((5-(Substituted methylene amino)-1,3,4-thiadiazol-2-yl)methyl) Benzamide Derivatives

(2017) Shailee Tiwari et al.   MOLECULES

Zn(II)-selective and sensitive fluorescent chemosensor based on steric constrains and inhibition of ESIPT

(2017) Caixia Yuan et al.   SENSORS AND ACTUATORS B-CHEMICAL

Mechanisms underlying the antiproliferative effects of a series of quinoxaline-derived chalcones

(2017) Tânia R. Mielcke et al.   Scientific Reports

N-2-Aryl-1,2,3-Triazoles: A novel class of blue–green emitting fluorophores-synthesis, photophysical properties study and dft computations

(2015) Vikas S. Padalkar et al.   JOURNAL OF LUMINESCENCE

Synthesis of phenstatin/isocombretastatin–chalcone conjugates as potent tubulin polymerization inhibitors and mitochondrial apoptotic inducers

(2015) Ahmed Kamal et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Design, synthesis and biological evaluation of novel 1,2,4-triazolo and 1,2,4-triazino[4,3-a]quinoxalines as potential anticancer and antimicrobial agents

(2015) Doaa A. E. Issa et al.   MedChemComm

Chalcone based azacarboline analogues as novel antitubulin agents: Design, synthesis, biological evaluation and molecular modelling studies

(2014) Sahil Sharma et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Pharmacological Evaluation of 5-Pyrrolidinylquinoxalines as a Novel Class of Peripherally Restricted κ-Opioid Receptor Agonists

(2014) Christian Bourgeois et al.   JOURNAL OF MEDICINAL CHEMISTRY

Sulphonamido-quinoxalines: Search for anticancer agent

(2013) Rahul Ingle et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

New Challenges and Inspired Answers for Anticancer Drug Discovery and Development

(2013) T. Utsugi   JAPANESE JOURNAL OF CLINICAL ONCOLOGY

Synthesis and Pharmacological Evaluation of Novel Quinoxalines as Potential Nonulcerogenic Anti-inflammatory and Analgesic Agents

(2012) Magda Ismail et al.   ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH

Exploring Pharmacological Significance of Chalcone Scaffold: A Review

(2012) N. K. Sahu et al.   CURRENT MEDICINAL CHEMISTRY

Synthesis of Some Phenylpyrazolo Benzimidazolo Quinoxaline Derivatives as Potent Antihistaminic Agents

(2012) C. H. Sridevi et al.   E-Journal of Chemistry

An Overview of Tubulin Inhibitors That Interact with the Colchicine Binding Site

(2012) Yan Lu et al.   PHARMACEUTICAL RESEARCH

Synthesis, biological evaluation, and molecular modeling of cinnamic acyl sulfonamide derivatives as novel antitubulin agents

(2011) Yin Luo et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Inhibitors and promoters of tubulin polymerization: Synthesis and biological evaluation of chalcones and related dienones as potential anticancer agents

(2011) Christine Dyrager et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Activity of novel quinoxaline-derived chalcones on in vitro glioma cell proliferation

(2011) Tânia R. Mielcke et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pharmacological significance of triazole scaffold

(2010) Rajeev Kharb et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Evaluation of diffusion and dilution methods to determine the antibacterial activity of plant extracts

(2010) Anja Klančnik et al.   JOURNAL OF MICROBIOLOGICAL METHODS

Combretastatin-like chalcones as inhibitors of microtubule polymerization. Part 1: Synthesis and biological evaluation of antivascular activity

(2009) Sylvie Ducki et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A boronic acid chalcone analog of combretastatin A-4 as a potent anti-proliferation agent

(2009) Yali Kong et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of 2,3-dichloroquinoxalinesviaVilsmeier reagent chlorination

(2009) Duane R. Romer   JOURNAL OF HETEROCYCLIC CHEMISTRY

QSAR analysis for quinoxaline-2-carboxylate 1,4-di-N-oxides as anti-mycobacterial agents

(2009) Esther Vicente et al.   JOURNAL OF MOLECULAR GRAPHICS & MODELLING

Antimitotic and Antiproliferative Activities of Chalcones: Forward Structure–Activity Relationship

(2008) Ahcène Boumendjel et al.   JOURNAL OF MEDICINAL CHEMISTRY