Phenyliodine Diacetate-Mediated Intramolecular C(sp2)H Amidation for 1,2-Disubstituted Benzimidazole Synthesis under Metal-Free Conditions

Indole Synthesis Based On A Modified Koser Reagent

(2014) Laura Fra et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free Annulation of Arenes with 2-Aminopyridine Derivatives: The Methyl Group as a Traceless Non-Chelating Directing Group

(2014) Srimanta Manna et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Free Coupling Reactions

(2014) Chang-Liang Sun et al.   CHEMICAL REVIEWS

Copper catalysed Ullmann type chemistry: from mechanistic aspects to modern development

(2014) Carlo Sambiagio et al.   CHEMICAL SOCIETY REVIEWS

The Synthesis of Benzimidazoles and Quinoxalines from Aromatic Diamines and Alcohols by Iridium-Catalyzed Acceptorless Dehydrogenative Alkylation

(2014) Toni Hille et al.   CHEMISTRY-A EUROPEAN JOURNAL

Hypervalent Iodine(III) Promoted Direct Synthesis of Imidazo[1,2-a]pyrimidines

(2014) Guangyin Qian et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Au catalyzed synthesis of benzimidazoles from 2-nitroanilines and CO2/H2

(2014) Leiduan Hao et al.   GREEN CHEMISTRY

Substituent Electronic Effects Govern Direct Intramolecular C–N Cyclization of N-(Biphenyl)pyridin-2-amines Induced by Hypervalent Iodine(III) Reagents

(2014) Jean-Ho Chu et al.   JOURNAL OF ORGANIC CHEMISTRY

Molecular Iodine Promoted Divergent Synthesis of Benzimidazoles, Benzothiazoles, and 2-Benzyl-3-phenyl-3,4-dihydro-2H-benzo[e][1,2,4]thiadiazines

(2014) Gunaganti Naresh et al.   JOURNAL OF ORGANIC CHEMISTRY

Regioselective (Diacetoxyiodo)benzene-Promoted Halocyclization of Unfunctionalized Olefins

(2014) Gong-Qing Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Ligand-free MCR for linking quinoxaline framework with a benzimidazole nucleus: a new strategy for the identification of novel hybrid molecules as potential inducers of apoptosis

(2014) Rajnikanth Sunke et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Alkene Diamination Using Electron-Rich Amines: Hypervalent Iodine-Promoted Inter-/Intramolecular C–N Bond Formation

(2014) Ki Bum Hong et al.   ORGANIC LETTERS

Development of a Concise, Asymmetric Synthesis of a Smoothened Receptor (SMO) Inhibitor: Enzymatic Transamination of a 4-Piperidinone with Dynamic Kinetic Resolution

(2014) Zhihui Peng et al.   ORGANIC LETTERS

Convenient Synthesis of Benzothiazoles and Benzimidazoles through Brønsted Acid Catalyzed Cyclization of 2-Amino Thiophenols/Anilines with β-Diketones

(2014) Muhammad Shareef Mayo et al.   ORGANIC LETTERS

Solvent/Oxidant-Switchable Synthesis of Multisubstituted Quinazolines and Benzimidazoles via Metal-Free Selective Oxidative Annulation of Arylamidines

(2014) Jian-Ping Lin et al.   ORGANIC LETTERS

Iodoarene-catalyzed fluorination and aminofluorination by an Ar-I/HF·pyridine/mCPBA system

(2014) Satoru Suzuki et al.   Chemical Science

Hypervalent iodine(iii) catalyzed oxidative C–N bond formation in water: synthesis of benzimidazole-fused heterocycles

(2014) D. Nageswar Rao et al.   RSC Advances

IBX works efficiently under solvent free conditions in ball milling

(2014) Tapas Kumar Achar et al.   RSC Advances

Cascade Palladium Catalysis: A Predictable and Selectable Regiocontrolled Synthesis ofN-Arylbenzimidazoles

(2013) Nathan T. Jui et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Hypervalent iodine(iii)-induced oxidative [4+2] annulation of o-phenylenediamines and electron-deficient alkynes: direct synthesis of quinoxalines from alkyne substrates under metal-free conditions

(2013) Sota Okumura et al.   CHEMICAL COMMUNICATIONS

Oxidative C–H amination reactions

(2013) Marie-Laure Louillat et al.   CHEMICAL SOCIETY REVIEWS

Metal-Free OxidativeparaCross-Coupling of Phenols

(2013) Koji Morimoto et al.   CHEMISTRY-A EUROPEAN JOURNAL

Metal-Free Oxidative Carbon-Heteroatom Bond Formation Through C-H Bond Functionalization

(2013) Rajarshi Samanta et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Photocatalysis by 3,6-Disubstituted-s-Tetrazine: Visible-Light Driven Metal-Free Green Synthesis of 2-Substituted Benzimidazole and Benzothiazole

(2013) Suvendu Samanta et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodobenzene Catalyzed C–H Amination of N-Substituted Amidines Using m-Chloroperbenzoic Acid

(2013) Santhosh Kumar Alla et al.   ORGANIC LETTERS

Hypervalent Iodine Reagents as Powerful Electrophiles

(2013) Thomas Wirth et al.   SYNLETT

Transition metal-catalyzed N-arylations of amidines and guanidines

(2012) Tom R. M. Rauws et al.   CHEMICAL SOCIETY REVIEWS

Preparation of 2-Azido-1-Substituted-1 H-Benzo[d]imidazoles Using a Copper-Promoted Three-Component Reaction and Their Further Conversion into 2-Amino and 2-Triazolyl Derivatives

(2012) Tamminana Ramana et al.   CHEMISTRY-A EUROPEAN JOURNAL

“All-water” chemistry of tandem N-alkylation–reduction–condensation for synthesis of N-arylmethyl-2-substituted benzimidazoles

(2012) Damodara N. Kommi et al.   GREEN CHEMISTRY

Hydrogen-Bond-Driven Electrophilic Activation for Selectivity Control: Scope and Limitations of Fluorous Alcohol-Promoted Selective Formation of 1,2-Disubstituted Benzimidazoles and Mechanistic Insight for Rationale of Selectivity

(2012) Rajesh Chebolu et al.   JOURNAL OF ORGANIC CHEMISTRY

Oxidative ipso-Rearrangement Performed by a Hypervalent Iodine Reagent and Its Application

(2012) Guillaume Jacquemot et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of carbazolones and 3-acetylindoles via oxidative C–N bond formation through PIFA-mediated annulation of 2-aryl enaminones

(2012) Xu Ban et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalyzed Enantioselective Synthesis of Axially Chiral Allenes

(2012) Hailing Li et al.   ORGANIC LETTERS

Organocatalytic, Oxidative, Intermolecular Amination and Hydrazination of Simple Arenes at Ambient Temperature

(2012) Rajarshi Samanta et al.   ORGANIC LETTERS

Simple and Practical Method for Preparation of [(Diacetoxy)iodo]arenes with Iodoarenes and m-Chloroperoxybenzoic Acid

(2012) Hideo Togo et al.   SYNLETT

Palladium-catalyzed aerobic oxidative C–H amination: synthesis of 2-unsubstituted and 2-substituted N-aryl benzimidazoles

(2012) Rapolu Kiran Kumar et al.   RSC Advances

Palladium-Catalyzed Intramolecular Sulfonamidation/Oxidation of Imines: Access to Multifunctional Benzimidazoles

(2011) Shaomin Fu et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic C–H amination: the stereoselectivity issue

(2011) Florence Collet et al.   CHEMICAL SOCIETY REVIEWS

Developments Towards Regioselective Synthesis of 1,2-Disubstituted Benzimidazoles

(2011) Luísa C. R. Carvalho et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Catalyzed, One-Pot, Three-Component Synthesis of Benzimidazoles by Condensation and C–N Bond Formation

(2011) Yong Kim et al.   JOURNAL OF ORGANIC CHEMISTRY

Intermolecular Oxidative C–N Bond Formation under Metal-Free Conditions: Control of Chemoselectivity between Aryl sp2and Benzylic sp3C–H Bond Imidation

(2011) Hyun Jin Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed One-Pot Synthesis of Substituted Benzimidazoles

(2010) Hongwei Jin et al.   ADVANCED SYNTHESIS & CATALYSIS

Benzimidazole Derivatives as New Serotonin 5-HT6Receptor Antagonists. Molecular Mechanisms of Receptor Inactivation

(2010) Tania de la Fuente et al.   JOURNAL OF MEDICINAL CHEMISTRY

Metal-Free Highly Regioselective Aminotrifluoroacetoxylation of Alkenes

(2010) Helena M. Lovick et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic C–H amination: recent progress and future directions

(2009) Florence Collet et al.   CHEMICAL COMMUNICATIONS

Hypervalent iodine reagents as a new entrance to organocatalysts

(2009) Toshifumi Dohi et al.   CHEMICAL COMMUNICATIONS

Synthesis and Evaluation of a New Generation of Orally Efficacious Benzimidazole-Based Poly(ADP-ribose) Polymerase-1 (PARP-1) Inhibitors as Anticancer Agents

(2009) Yunsong Tong et al.   JOURNAL OF MEDICINAL CHEMISTRY

Chemistry of Polyvalent Iodine

(2008) Viktor V. Zhdankin et al.   CHEMICAL REVIEWS

Iron(II) Bromide-Catalyzed Synthesis of Benzimidazoles from Aryl Azides

(2008) Meihua Shen et al.   ORGANIC LETTERS