Developments Towards Regioselective Synthesis of 1,2-Disubstituted Benzimidazoles

Optimization of a novel class of benzimidazole-based farnesoid X receptor (FXR) agonists to improve physicochemical and ADME properties

(2011) Hans G.F. Richter et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A Protocol to 2-Aminobenzimidazoles via Copper-Catalyzed Cascade Addition and Cyclization ofo-Haloanilines and Carbodiimides

(2011) Fei Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and SAR studies of benzimidazole derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Focus to detune hERG inhibition

(2011) Pradip K. Sasmal et al.   MedChemComm

Copper(II) Acetate/Oxygen-Mediated Nucleophilic Addition and Intramolecular CH Activation/CN or CC Bond Formation: One-Pot Synthesis of Benzimidazoles or Quinazolines

(2010) Hua-Feng He et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed One-Pot Synthesis of Substituted Benzimidazoles

(2010) Hongwei Jin et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Benzoxazole and Benzimidazole Derivatives via Ligand-Free Copper(I)-Catalyzed Cross-Coupling Reaction of o-Halophenols or o-Haloanilines with Carbodiimides

(2010) Guodong Shen et al.   ADVANCED SYNTHESIS & CATALYSIS

Angiotensin II receptor type 1 (AT1) selective nonpeptidic antagonists—A perspective

(2010) Prashant Naik et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Novel N-substituted benzimidazole CXCR4 antagonists as potential anti-HIV agents

(2010) John F. Miller et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Ruthenium-Catalyzed Synthesis of Benzimidazoles from N-Alkyl-1,2-diaminobenzenes via Alkyl Group Transfer

(2010)   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Proton-conducting membranes based on benzimidazole polymers for high-temperature PEM fuel cells. A chemical quest

(2010) Juan Antonio Asensio et al.   CHEMICAL SOCIETY REVIEWS

Microwave supported synthesis of some novel 1,3-Diarylpyrazino[1,2-a]benzimidazole derivatives and investigation of their anticancer activities

(2010) Seref Demirayak et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Direct, Regioselective Palladium-Catalyzed Synthesis of N-Substituted Benzimidazoles and Imidazopyridines

(2010) Jorge Alonso et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 1,2-disubstituted benzimidazoles, 2-substituted benzimidazoles and 2-substituted benzothiazoles in SDS micelles

(2010) Kiumars Bahrami et al.   GREEN CHEMISTRY

Multidisciplinary Synthetic Approach for Rapid Combinatorial Library Synthesis of Triaza-Fluorenes

(2010) Ya-Shan Hsiao et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Fructose-1,6-bisphosphatase Inhibitors. 2. Design, Synthesis, and Structure−Activity Relationship of a Series of Phosphonic Acid Containing Benzimidazoles that Function as 5′-Adenosinemonophosphate (AMP) Mimics

(2010) Qun Dang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Intramolecular C−N Bond Formation: A Straightforward Synthesis of Benzimidazole Derivatives in Water

(2010) Jinsong Peng et al.   JOURNAL OF ORGANIC CHEMISTRY

Substituted Benzimidazole Derivatives as Angiotensin II -AT1 Receptor Antagonist: A Review

(2010) V. K. Vyas et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Cobalt-catalyzed intramolecular C–N and C–O cross-coupling reactions: synthesis of benzimidazoles and benzoxazoles

(2010) Prasenjit Saha et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient and Green Synthesis of 1,2-Disubstituted Benzimidazoles and Quinoxalines Using Br⊘nsted Acid Ionic Liquid, [(CH2)4SO3HMIM][HSO4], in Water at Room Temperature

(2010) Yahya S. Beheshtiha et al.   SYNTHETIC COMMUNICATIONS

A novel and practical synthesis of substituted 2-ethoxy benzimidazole: candesartan cilexetil

(2010) Ping Wang et al.   TETRAHEDRON

One-pot synthesis of benzimidazoles from gem-dibromomethylarenes using o-diaminoarenes

(2010) Chandrappa Siddappa et al.   TETRAHEDRON LETTERS

Structure–activity relationships of benzimidazole derivatives as antiparasitic agents: Dual activity-difference (DAD) maps

(2010) Jaime Pérez-Villanueva et al.   MedChemComm

Synthesis of Aminoboronic Acids and Their Applications in Bifunctional Catalysis

(2009) Irene Georgiou et al.   ACCOUNTS OF CHEMICAL RESEARCH

Catalytic CC, CN, and CO Ullmann-Type Coupling Reactions

(2009) Florian Monnier et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Brain-penetrating 2-aminobenzimidazole H1-antihistamines for the treatment of insomnia

(2009) Timothy Coon et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of 2-fluoroalkylbenzimidazoles via copper(i)-catalyzed tandem reactions

(2009) Jiangtao Zhu et al.   CHEMICAL COMMUNICATIONS

Reactivity-Controlled Regioselectivity: A Regiospecific Synthesis of 1,2-Disubstituted Benzimidazoles

(2009) Xiaohu Deng et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Water mediated chemoselective synthesis of 1,2-disubstituted benzimidazoles using o-phenylenediamine and the extended synthesis of quinoxalines

(2009) Jie-Ping Wan et al.   GREEN CHEMISTRY

Copper(I)-Catalyzed Synthesis of Substituted 2-Mercapto Benzimidazoles

(2009) Siva Murru et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Synthesis of 2-Unsubstituted,N-Substituted Benzimidazoles

(2009) Keiichi Hirano et al.   JOURNAL OF ORGANIC CHEMISTRY

Ligand-Free Copper-Catalyzed Synthesis of Substituted Benzimidazoles, 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and Benzoxazoles

(2009) Prasenjit Saha et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Cascade Addition/Cyclization: An Efficient and Versatile Synthesis ofN-Substituted 2-Heterobenzimidazoles

(2009) Xin Lv et al.   JOURNAL OF ORGANIC CHEMISTRY

The application of poly(N, N′-dibromo-N-ethyl-benzene-1,3-disulfonamide) and N, N, N′, N′-tetrabromobenzene-1,3-disulfonamide as catalysts for one-pot synthesis of 2-aryl-1-arylmethyl-1H-1,3-benzimidazoles and 1,5-benzodiazepines, and new reagents for synthesis of benzimidazoles

(2009) Ramin Ghorbani-Vaghei et al.   MOLECULAR DIVERSITY

Hidden signatures: new reagents for developing latent fingerprints

(2009) M. John Plater et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Mutations in a β-Tubulin Confer Resistance of Gibberella zeae to Benzimidazole Fungicides

(2009) Chang-Jun Chen et al.   PHYTOPATHOLOGY

An ionic liquid mediated one-pot synthesis of substituted thiazolidinones and benzimidazoles

(2009) Ashok K. Yadav et al.   TETRAHEDRON LETTERS

Synthesis of 1,2-disubstitued benzimidazoles using SiO2/ZnCl2

(2009) Raquel G. Jacob et al.   TETRAHEDRON LETTERS

CH Functionalization/CN Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

(2008) Gordon Brasche et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Biaryl Phosphane Ligands in Palladium-Catalyzed Amination

(2008) David S. Surry et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Solid-Phase Synthesis of Biologically Active Benzoannelated Nitrogen Heterocycles: An Update

(2008) Carmen Gil et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Copper-Catalyzed Synthesis of Benzimidazoles via Cascade Reactions ofo-Haloacetanilide Derivatives with Amidine Hydrochlorides

(2008) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 6,7,8-Trisubstituted Purines via a Copper-Catalyzed Amidation Reaction

(2008) Nada Ibrahim et al.   JOURNAL OF ORGANIC CHEMISTRY

Iron(II) Bromide-Catalyzed Synthesis of Benzimidazoles from Aryl Azides

(2008) Meihua Shen et al.   ORGANIC LETTERS

M(HSO4)n-Promoted Synthesis of 2-Aryl-1-arylmethyl-1H-1,3-benzimidazole Derivatives

(2008) Khodabakhsh Niknam et al.   SYNTHETIC COMMUNICATIONS

Water-Accelerated Selective Synthesis of 1,2-Disubstituted Benzimidazoles at Room Temperature Catalyzed by Br⊘nsted Acidic Ionic Liquid

(2008) Minoo Dabiri et al.   SYNTHETIC COMMUNICATIONS

Synthesis of benzimidazoles from 1,1-dibromoethenes

(2008) Wang Shen et al.   TETRAHEDRON LETTERS