- Home
- Publications
- Publication Search
- Publication Details
Title
Recent Advances in Indole Synthesis and the Related Alkylation
Authors
Keywords
-
Journal
Asian Journal of Organic Chemistry
Volume 12, Issue 6, Pages -
Publisher
Wiley
Online
2023-05-02
DOI
10.1002/ajoc.202300092
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- A Metal-Free Reductive N-Alkylation of Indoles with Aldehydes
- (2021) Nicholas A. Clanton et al. ORGANIC LETTERS
- Domino C–N Bond Formation via a Palladacycle with Diaziridinone. An Approach to Indolo[3,2-b]indoles
- (2021) Sudarshan Debnath et al. ORGANIC LETTERS
- Diastereoselective Synthesis of Dihydro-quinolin-4-ones by a Borane-Catalyzed Redox-Neutral endo-1,7-Hydride Shift
- (2021) Garrit Wicker et al. ORGANIC LETTERS
- Electrocatalytic Dehydrogenative Cyclization of 2-Vinylanilides for the Synthesis of Indoles
- (2021) Yun-Tao Zheng et al. JOURNAL OF ORGANIC CHEMISTRY
- Synthesis of Dipeptide, Amide, and Ester without Racemization by Oxalyl Chloride and Catalytic Triphenylphosphine Oxide
- (2021) Ji-Wei Ren et al. ORGANIC LETTERS
- Copper-Catalyzed (4+1) Cascade Annulation of Terminal Alkynes with 2-(Tosylmethyl)anilines: Synthesis of 2,3-Disubstituted Indoles
- (2021) Xu Yan et al. ORGANIC LETTERS
- Palladium-Catalyzed Ligand-Free Double Cyclization Reactions for the Synthesis of 3-(1′-Indolyl)-phthalides
- (2020) Shuo Yuan et al. ORGANIC LETTERS
- B(C6F5)3-Catalyzed Direct C3 Alkylation of Indoles and Oxindoles
- (2020) Shyam Basak et al. ACS Catalysis
- Enantioselective Catalytic Synthesis of N-alkylated Indoles
- (2020) Dmitri Trubitsõn et al. Symmetry-Basel
- Nickel-Catalyzed Mizoroki–Heck/Amination Cascade Reactions of o-Dihaloarenes with Allylamines: Synthesis of Indoles
- (2020) Xu Chen et al. ORGANIC LETTERS
- Rhodium‐Catalyzed Chemodivergent Regio‐ and Enantioselective Allylic Alkylation of Indoles
- (2020) Minghe Sun et al. CHEMISTRY-A EUROPEAN JOURNAL
- Synthesis of N-Fused Polycyclic Indoles via Ligand-Free Palladium-Catalyzed Annulation/Acyl Migration Reaction
- (2019) Zhan Dong et al. ORGANIC LETTERS
- CuH-Catalyzed Enantioselective Alkylation of Indole Derivatives with Ligand-Controlled Regiodivergence
- (2019) Yuxuan Ye et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- One-Pot Synthesis of N-Imidoyl-(1H)-Indoles via Palladium-Catalyzed Oxidative Insertion Domino Reaction with Isocyanide and Arylboronic Acid
- (2019) Shou-wei Tao et al. JOURNAL OF ORGANIC CHEMISTRY
- Enantioselective N-Alkylation of Indoles via an Intermolecular Aza-Wacker-Type Reaction
- (2019) Jamie R. Allen et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Cu-Catalyzed Arylation/Acyl Migration Cascade Reaction of Enaminones: Access to N-Fused Polycyclic and 2,3-Disubstituted Indoles
- (2019) Weishuang Li et al. JOURNAL OF ORGANIC CHEMISTRY
- Rhenium-Catalyzed Intramolecular Carboalkoxylation and Carboamination of Alkynes for the Synthesis of C3-Substituted Benzofurans and Indoles
- (2019) Ming-Guang Rong et al. ORGANIC LETTERS
- Chemoselective N-Alkylation of Indoles in Aqueous Microdroplets
- (2019) Elumalai Gnanamani et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Brønsted Acids Enable Three Molecular Rearrangements of One 3-Alkylidene-2H-1,2-oxazine Molecule into Distinct Heterocyles
- (2018) Bhanudas Dattatray Mokar et al. ORGANIC LETTERS
- Metal and acid-free visible light-mediated Friedel-Crafts alkylation reactions of indole with anilines
- (2018) Xiao-Qiang Dai et al. TETRAHEDRON LETTERS
- “Back-to-Front” Indole Synthesis Using Silver(I) Catalysis: Unexpected C-3 Pyrrole Activation Mode Supported by DFT
- (2018) Aimee K. Clarke et al. ACS Catalysis
- Chiral phosphoric acid catalyzed enantioselective N-alkylation of indoles with in situ generated cyclic N-acyl ketimines
- (2018) Lvye Zhang et al. CHEMICAL COMMUNICATIONS
- Gold-catalyzed tandem reaction of 2-alkynylanilines followed by 1,6-conjugate addition to p-quinone methides: efficient access to unsymmetrical diarylindolylmethanes
- (2018) Raveendra Jillella et al. NEW JOURNAL OF CHEMISTRY
- Chemoselective N–H functionalization of indole derivatives via the Reissert-type reaction catalyzed by a chiral phosphoric acid
- (2018) Yue Cai et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- 3d-Metal Catalyzed N- and C-Alkylation Reactions via Borrowing Hydrogen or Hydrogen Autotransfer
- (2018) Torsten Irrgang et al. CHEMICAL REVIEWS
- Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen
- (2017) Giovanni Di Gregorio et al. JOURNAL OF ORGANIC CHEMISTRY
- Straight Access to Indoles from Anilines and Ethylene Glycol by Heterogeneous Acceptorless Dehydrogenative Condensation
- (2017) Pedro Juan Llabres-Campaner et al. JOURNAL OF ORGANIC CHEMISTRY
- Recent progress in transition-metal-catalyzed enantioselective indole functionalizations
- (2017) Jing-Biao Chen et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Dual visible-light photoredox and palladium(ii) catalysis for dehydrogenative C2-acylation of indoles at room temperature
- (2017) Manash Kumar Manna et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- trans-Aminoboration across Internal Alkynes Catalyzed by B(C6F5)3 for the Synthesis of Borylated Indoles
- (2017) Kang Yuan et al. ORGANIC LETTERS
- Gold/Copper-Co-catalyzed Tandem Reactions of 2-Alkynylanilines: A Synthetic Strategy for the C2-Quaternary Indolin-3-ones
- (2017) Yi-Jin Li et al. ORGANIC LETTERS
- Cs 2 CO 3 -catalyzed alkylation of indoles with trifluoromethyl ketones
- (2017) Xiao-Dong Liu et al. TETRAHEDRON
- Friedel-Crafts Reaction of Indoles with Isatin-Derived β,γ-Unsaturated α-Keto Esters Using a BINOL-Derived Bisoxazoline (BOX)/Copper(II) Complex as Catalyst
- (2016) Nai-Kai Li et al. ADVANCED SYNTHESIS & CATALYSIS
- Decarboxylative/decarbonylative C3-acylation of indoles via photocatalysis: a simple and efficient route to 3-acylindoles
- (2016) Qing Shi et al. GREEN CHEMISTRY
- Construction of 9H-Pyrrolo[1,2-a]indoles by a Copper-Catalyzed Friedel–Crafts Alkylation/Annulation Cascade Reaction
- (2016) Yongqing Sun et al. JOURNAL OF ORGANIC CHEMISTRY
- Ag(I)-Catalyzed Domino Cyclization–Addition Sequence with Simultaneous Carbonyl and Alkyne Activation as a Route to 2,2′-Disubstituted Bisindolylarylmethanes
- (2016) Swastik Karmakar et al. ORGANIC LETTERS
- Lewis Acid-Catalyzed or Base-Promoted Regioselective Cycloisomerization ofN-Imidoyl-o-alkynylanilines for Synthesis ofN-Imidoyl-(1 H)-indoles and 4-Alkylidene-3,4-dihydroquinazolines
- (2015) Takashi Otani et al. ADVANCED SYNTHESIS & CATALYSIS
- Facile Installation of 2-Reverse Prenyl Functionality into Indoles by a Tandem N-Alkylation-Aza-Cope Rearrangement Reaction and Its Application in Synthesis
- (2015) Xiaobei Chen et al. CHEMISTRY-A EUROPEAN JOURNAL
- Synthesis of N-vinylindoles through copper catalyzed cyclization reaction of N-(2-alkynylphenyl)imine
- (2015) Zhi-Qiang Wang et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Regio- and Enantioselective Synthesis ofN-Allylindoles by Iridium-Catalyzed Allylic Amination/Transition-Metal-Catalyzed Cyclization Reactions
- (2014) Ke-Yin Ye et al. CHEMISTRY-A EUROPEAN JOURNAL
- Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals
- (2014) Edon Vitaku et al. JOURNAL OF MEDICINAL CHEMISTRY
- Pd(ii)-catalyzed ligand controlled synthesis of methyl 1-benzyl-1H-indole-3-carboxylates and bis(1-benzyl-1H-indol-3-yl)methanones
- (2014) Rong Shen et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Copper-catalyzed decarboxylative C3-acylation of free (N–H) indoles with α-oxocarboxylic acids
- (2014) Cuiping Wang et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Brønsted Acid Catalyzed Cascade Reactions of 2-[(2-Aminophenyl)ethynyl]phenylamine Derivatives with Aldehydes: A New Approach to the Synthesis of 2,2′-Disubstituted 1H,1′H-3,3′-Biindoles
- (2014) Antonio Arcadi et al. ORGANIC LETTERS
- [Cp∗IrCl2]2-catalysed cyclization of 2-alkynylanilines into indoles
- (2014) Elumalai Kumaran et al. TETRAHEDRON LETTERS
- Choline chloride based eutectic solvents: direct C-3 alkenylation/alkylation of indoles with 1,3-dicarbonyl compounds
- (2014) Anita Kailas Sanap et al. RSC Advances
- Cycloisomerization of 2-Alkynylanilines to Indoles Catalyzed by Carbon-Supported Gold Nanoparticles and Subsequent Homocoupling to 3,3′-Biindoles
- (2013) Jesus E. Perea-Buceta et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Transition-Metal-Catalyzed Regioselective Alkylation of Indoles with Alcohols
- (2013) Anggi Eka Putra et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- A novel microwave-irradiated solvent-free 3-acylation of indoles on alumina
- (2013) Qiu Yu Lai et al. NEW JOURNAL OF CHEMISTRY
- Synthesis of indoles with a polyfluorinated benzene ring
- (2013) Larisa V. Politanskaya et al. TETRAHEDRON
- In(OTf)3 catalyzed C3-benzylation of indoles with benzyl alcohols in water
- (2013) Lin Wu et al. RSC Advances
- N-alkylation of indole via ring-closing metathesis/isomerization/Mannich cascade under ruthenium/chiral phosphoric acid sequential catalysis
- (2013) Yan-Chao Shi et al. Organic Chemistry Frontiers
- Cesium Carbonate-Promoted Hydroamidation of Alkynes: Enamides, Indoles and the Effect of Iron(III) Chloride
- (2012) María Teresa Herrero et al. ADVANCED SYNTHESIS & CATALYSIS
- AsymmetricN-Allylation of Indoles Through the Iridium-Catalyzed Allylic Alkylation/Oxidation of Indolines
- (2012) Wen-Bo Liu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Indoles in Multicomponent Processes (MCPs)
- (2012) Morteza Shiri CHEMICAL REVIEWS
- New strategies for the synthesis of N-alkylated indoles (Review)
- (2012) A. V. Karchava et al. Chemistry of Heterocyclic Compounds
- Domino Sonogashira Coupling/Cyclization Reaction Catalyzed by Copper and ppb Levels of Palladium: A Concise Route to Indoles and Benzo[b]furans
- (2011) Ruiping Wang et al. ADVANCED SYNTHESIS & CATALYSIS
- Efficient and convenient C-3 functionalization of indoles through Ce(OAc)3/TBHP-mediated oxidative C–H bond activation in the presence of β-cyclodextrin
- (2011) Yu Lin Hu et al. GREEN CHEMISTRY
- ZrCl4-Mediated Regio- and Chemoselective Friedel–Crafts Acylation of Indole
- (2011) Sankar K. Guchhait et al. JOURNAL OF ORGANIC CHEMISTRY
- Rh2(II)-Catalyzed Nitro-Group Migration Reactions: Selective Synthesis of 3-Nitroindoles from β-Nitro Styryl Azides
- (2011) Benjamin J. Stokes et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Palladium-Catalyzed Direct 2-Alkylation of Indoles by Norbornene-Mediated Regioselective Cascade C–H Activation
- (2011) Lei Jiao et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Ruthenium/TFA-catalyzed regioselective C-3-alkylation of indoles with terminal alkynes in water: efficient and unprecedented access to 3-(1-methylalkyl)-1H-indoles
- (2010) Victorio Cadierno et al. CHEMICAL COMMUNICATIONS
- Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety
- (2010) Anna J. Kochanowska-Karamyan et al. CHEMICAL REVIEWS
- Asymmetric Phase-Transfer-Catalyzed Intramolecular N-Alkylation of Indoles and Pyrroles: A Combined Experimental and Theoretical Investigation
- (2010) Marco Bandini et al. CHEMISTRY-A EUROPEAN JOURNAL
- Chiral Brønsted acid catalyzed asymmetric Friedel–Crafts alkylation reaction of indoles with α,β-unsaturated ketones: short access to optically active 2- and 3-substituted indole derivatives
- (2010) Tsubasa Sakamoto et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Copper-Catalyzed CC Bond Formation through CH Functionalization: Synthesis of Multisubstituted Indoles fromN-Aryl Enaminones
- (2009) Roberta Bernini et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Asymmetric Organocatalytic N-Alkylation of Indole-2-carbaldehydes with α,β-Unsaturated Aldehydes: One-Pot Synthesis of Chiral Pyrrolo[1,2-a]indole-2-carbaldehydes
- (2009) Liang Hong et al. CHEMISTRY-A EUROPEAN JOURNAL
- Efficient Regioselective Synthesis of IndoleN-Carboximidamides andN-Carboximidoates by a Sequential Aza-Wittig/Ag(I)-Catalyzed Cyclization
- (2009) Nian-Yu Huang et al. JOURNAL OF ORGANIC CHEMISTRY
- Stereoselective Double Friedel−Crafts Alkylation of Indoles with Divinyl Ketones
- (2009) Andrew C. Silvanus et al. ORGANIC LETTERS
- 3-Aroylindoles via Copper-Catalyzed Cyclization of N-(2-Iodoaryl)enaminones
- (2009) Sandro Cacchi et al. SYNLETT
- First example of FeCl3-catalyzed alkylation of indoles with pinenes
- (2009) J.S. Yadav et al. TETRAHEDRON LETTERS
- Catalytic Synthesis of Indoles from Alkynes
- (2008) Karolin Krüger (née Alex) et al. ADVANCED SYNTHESIS & CATALYSIS
- InBr3-Promoted Divergent Approach to Polysubstituted Indoles and Quinolines from 2-Ethynylanilines: Switch from an Intramolecular Cyclization to an Intermolecular Dimerization by a Type of Terminal Substituent Group
- (2008) Norio Sakai et al. JOURNAL OF ORGANIC CHEMISTRY
- One-Pot Multicomponent Synthesis of Indoles from 2-Iodobenzoic Acid
- (2007) Olivier Leogane et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- FeCl3-catalyzed alkylation of indoles with 1,3-dicarbonyl compounds: an expedient synthesis of 3-substituted indoles
- (2007) J.S. Yadav et al. TETRAHEDRON LETTERS
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreAdd your recorded webinar
Do you already have a recorded webinar? Grow your audience and get more views by easily listing your recording on Peeref.
Upload Now