Cesium Carbonate-Promoted Hydroamidation of Alkynes: Enamides, Indoles and the Effect of Iron(III) Chloride

Benzofurans from Benzophenones and Dimethylacetamide: Copper-Promoted Cascade Formation of Furan O1C2 and C2C3 Bonds Under Oxidative Conditions

(2012) María J. Moure et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Brønsted Acid-Promoted Sequential Hydroarylation- Hydroamidation of Arene-Tethered 1-(2-Alkynylphenyl)ureas: Direct Access to 4,4-Spiro-3,4-dihydro-2-(1H)-quinazolinones

(2011) Honggen Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Iron-Facilitated Iodine-Mediated Electrophilic Annulation of N,N-Dimethyl-2-alkynylanilines with Disulfides or Diselenides

(2011) Hui-Ai Du et al.   ADVANCED SYNTHESIS & CATALYSIS

Domino Sonogashira Coupling/Cyclization Reaction Catalyzed by Copper and ppb Levels of Palladium: A Concise Route to Indoles and Benzo[b]furans

(2011) Ruiping Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Control of 6-Exo and 7-Endo Cyclizations of Alkynylamides using Platinum and Bismuth Catalysts

(2011) Anne-Lise Girard et al.   Chemistry-An Asian Journal

Total Synthesis and Biological Evaluation of Pacidamycin D and Its 3′-Hydroxy Analogue

(2011) Kazuya Okamoto et al.   JOURNAL OF ORGANIC CHEMISTRY

Mechanistic Investigation of the Ru-Catalyzed Hydroamidation of Terminal Alkynes

(2011) Matthias Arndt et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An straightforward entry to new pyrazolo-fused dibenzo[1,4]diazepines

(2011) Susana Hernández et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Hydro-amination/-amidation of 1,3-diynes with indoles/azoles/amides under modified Ullmann conditions: stereo- and regio-selective synthesis of N-alkenynes via N–H bond activation

(2011) Sahaj Gupta et al.   TETRAHEDRON LETTERS

A Novel One-Pot, Two-Step Synthesis of Polycyclic Indoles via Tandem Intramolecular Hydroamidation/Palladium-Catalyzed Annulation

(2010) Jianxiu Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis and biological activities of novel indole derivatives as potent and selective PPARγ modulators

(2010) Yann Lamotte et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of 6-trifluoromethylindolo[1,2-c]quinazolines and related heterocycles using N-(2-iodophenyl)trifluoroacetimidoyl chlorides as starting material via C–H bond functionalization

(2010) Jiangtao Zhu et al.   CHEMICAL COMMUNICATIONS

Convenient Synthesis of Tetrahydro-γ-carbolines and Tetrahydroquinolines through a Chemo- and Regioselectivity Switch by a Brønsted Acid Catalyzed, One-Pot, Multicomponent Reaction

(2010) Hong-Gang Cheng et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Regioselective Synthesis of 3-Benzazepinones and Unexpected 5-Bromo-3-benzazepinones

(2010) Lei Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Z-Selective hydroamidation of terminal alkynes with secondary amides and imides catalyzed by a Ru/Yb-system

(2010) Annette E. Buba et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Highly Diastereoselective Zinc-Catalyzed Propargylation oftert-Butanesulfinyl Imines

(2010) Daniel R. Fandrick et al.   ORGANIC LETTERS

Cupric Halide-Mediated Intramolecular Halocyclization of N-Electron-Withdrawing Group-Substituted 2-Alkynylanilines for the Synthesis of 3-Haloindoles

(2009) Zengming Shen et al.   ADVANCED SYNTHESIS & CATALYSIS

Iron-Catalyzed Regioselective Hydroaryloxylation of CC Triple Bonds: An Efficient Synthesis of 2H-1-Benzopyran Derivatives

(2009) Xiaobing Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-CatalyzedN-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore

(2009) Lutz Ackermann et al.   ADVANCED SYNTHESIS & CATALYSIS

6-Substituted Indolo[1,2-c]quinazolines as New Antimicrobial Agents

(2009) Rondla Rohini et al.   ARCHIV DER PHARMAZIE

Dichotomous Control ofE/Z-Geometry in Intramolecular Cyclization ofo-Alkynylbenzamide Derivatives Catalyzed by Organic Superbase P4-tBu in the Presence/Absence of Water

(2009) Chikashi Kanazawa et al.   Chemistry-An Asian Journal

A General Route to Cyclopeptide Alkaloids: Total Syntheses and Biological Evaluation of Paliurines E and F, Ziziphines N and Q, Abyssenine A, Mucronine E, and Analogues

(2009) Mathieu Toumi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Enamide-Benzyne-[2 + 2] Cycloaddition: Stereoselective Tandem [2 + 2]−Pericyclic Ring-Opening−IntramolecularN-Tethered [4 + 2] Cycloadditions

(2009) John B. Feltenberger et al.   ORGANIC LETTERS

Radical-initiated cyclization as a key step for the synthesis of oxoprotoberberine alkaloids

(2009) Chih-Shone Lee et al.   TETRAHEDRON LETTERS

Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles†

(2008) Dawei Ma et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of Secondary Enamides by Ruthenium-Catalyzed Selective Addition of Amides to Terminal Alkynes

(2008) Lukas J. Gooßen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Mediated Coupling Reactions and Their Applications in Natural Products and Designed Biomolecules Synthesis

(2008) Gwilherm Evano et al.   CHEMICAL REVIEWS

Concise Synthesis of the CDE Ring System of Tetrahydroisoquinoline Alkaloids Using Carbophilic Lewis Acid-Catalyzed Hydroamidation and Oxidative Friedel−Crafts Cyclization

(2008) Shingo Obika et al.   JOURNAL OF ORGANIC CHEMISTRY

Enamides: valuable organic substrates

(2008) David R. Carbery   ORGANIC & BIOMOLECULAR CHEMISTRY

A rapid synthesis of 2-alkynylindoles and 2-alkynylbenzofurans

(2008) Vito Fiandanese et al.   TETRAHEDRON

Copper-promoted iodovinylation of amides: synthesis of β-functionalized enamides

(2008) Gabriel F. Sanapo et al.   TETRAHEDRON LETTERS

Preparation of Fully Substituted Anilines for the Synthesis of Functionalized Indoles

(2007) Armin H. Stoll et al.   ORGANIC LETTERS

Annulation of internal alkynes through a hydroamination/aza-Heck reaction sequence for the regioselective synthesis of indoles

(2007) Lutz Ackermann et al.   TETRAHEDRON