Regio- and Enantioselective Synthesis ofN-Allylindoles by Iridium-Catalyzed Allylic Amination/Transition-Metal-Catalyzed Cyclization Reactions

Merging Synthesis and Enantioselective Functionalization of Indoles by a Gold-Catalyzed Asymmetric Cascade Reaction

(2013) Michel Chiarucci et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Combined Theoretical and Experimental Investigation into the Highly Stereoselective Migration of Spiroindolenines

(2013) Chao Zheng et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Functionalization of Indoles and Pyrroles via an in Situ-Formed Spiro Intermediate

(2013) Chun-Xiang Zhuo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Enantioselective Construction of Trifluoromethylated All-Carbon Quaternary Stereocenters via Nickel-Catalyzed Friedel–Crafts Alkylation Reaction

(2013) Jian-Rong Gao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Enantioselective Synthesis of Tetrahydrocarbolines via Iridium-Catalyzed Intramolecular Friedel–Crafts Type Allylic Alkylation Reactions

(2013) Qing-Long Xu et al.   ORGANIC LETTERS

Concise Asymmetric Synthesis of Orthogonally Protected syn- and anti-1,3-Aminoalcohols

(2013) Jae Seung Lee et al.   ORGANIC LETTERS

One-Pot Gold-Catalyzed Aminofluorination of Unprotected 2-Alkynylanilines

(2013) Antonio Arcadi et al.   ORGANIC LETTERS

Synthesis of 1 Z,4 E,6 E-Triene Derivatives by Chemo- and Regioselective Iridium-Catalyzed Dienylation ofortho-Aminostyrenes with Dienyl Carbonates

(2013) Ke-Yin Ye et al.   Asian Journal of Organic Chemistry

Enantioselective Synthesis of Spiro Cyclopentane-1,3′-indoles and 2,3,4,9-Tetrahydro-1H-carbazoles by Iridium-Catalyzed Allylic Dearomatization and Stereospecific Migration

(2012) Qing-Feng Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct, Enantioselective Iridium-Catalyzed Allylic Amination of Racemic Allylic Alcohols

(2012) Marc Lafrance et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

AsymmetricN-Allylation of Indoles Through the Iridium-Catalyzed Allylic Alkylation/Oxidation of Indolines

(2012) Wen-Bo Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Coupling ofortho-Alkynylanilines with Terminal Alkynes Under Aerobic Conditions: Efficient Synthesis of 2,3-Disubstituted 3-Alkynylindoles

(2012) Bo Yao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Progress in palladium-based catalytic systems for the sustainable synthesis of annulated heterocycles: a focus on indole backbones

(2012) Mélanie Platon et al.   CHEMICAL SOCIETY REVIEWS

New strategies for the synthesis of N-alkylated indoles (Review)

(2012) A. V. Karchava et al.   Chemistry of Heterocyclic Compounds

Highly Enantioselective Pictet-Spengler Reaction Catalyzed by SPINOL-Phosphoric Acids

(2012) Dan Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

A General Synthesis of Indole-3-carboxylic Esters by Palladium-Catalyzed Direct Oxidative Carbonylation of 2-Alkynylaniline Derivatives

(2012) Bartolo Gabriele et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iridium-Catalyzed Allylic Alkylation Reaction with N-Aryl Phosphoramidite Ligands: Scope and Mechanistic Studies

(2012) Wen-Bo Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Synthesis of Tryptophan Derivatives by a Tandem Friedel–Crafts Conjugate Addition/Asymmetric Protonation Reaction

(2012) Madeleine E. Kieffer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Thiourea-catalysed ring opening of episulfonium ions with indole derivatives by means of stabilizing non-covalent interactions

(2012) Song Lin et al.   Nature Chemistry

Recent advances and applications of iridium-catalysed asymmetric allylic substitution

(2012) Paolo Tosatti et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Diversity oriented synthesis of indole-based peri-annulated compounds via allylic alkylation reactions

(2012) Qing-Long Xu et al.   Chemical Science

Umpolung Reactivity of Indole through Gold Catalysis

(2011) Biao Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Binary Acid Catalysis: A Regioselectivity Switch between Enantioselective 1,2- and 1,4-Addition through Different Counteranions of InIII

(2011) Jian Lv et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iridium-Catalyzed Asymmetric Intramolecular Allylic Amidation: Enantioselective Synthesis of Chiral Tetrahydroisoquinolines and Saturated Nitrogen Heterocycles

(2011) Johannes F. Teichert et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Update 1 of: Synthesis and Functionalization of Indoles Through Palladium-Catalyzed Reactions

(2011) Sandro Cacchi et al.   CHEMICAL REVIEWS

Enantio- and Regioselective Iridium-Catalyzed Allylic Hydroxylation

(2011) Martin Gärtner et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iridium-Catalyzed Allylic Vinylation and Asymmetric Allylic Amination Reactions witho-Aminostyrenes

(2011) Ke-Yin Ye et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent advances in indole syntheses: New routes for a classic target

(2011) Rubén Vicente   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective Iridium-Catalyzed Allylic Substitutions with Hydroxamic Acid Derivatives as N-Nucleophiles

(2011) Martin Gärtner et al.   ORGANIC LETTERS

Asymmetric dearomatization of pyrrolesviaIr-catalyzed allylic substitution reaction: enantioselective synthesis of spiro-2H-pyrroles

(2011) Chun-Xiang Zhuo et al.   Chemical Science

Mechanistically Driven Development of Iridium Catalysts for Asymmetric Allylic Substitution

(2010) John F. Hartwig et al.   ACCOUNTS OF CHEMICAL RESEARCH

Enantioselective Synthesis of 2,3-Dihydro-1H-benzo[b]azepines: Iridium-Catalyzed Tandem Allylic Vinylation/Amination Reaction

(2010) Hu He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Intramolecular Aza-Michael Additions of Indoles Catalyzed by Chiral Phosphoric Acids

(2010) Quan Cai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Organocatalytic strategies for the asymmetric functionalization of indoles

(2010) Giuseppe Bartoli et al.   CHEMICAL SOCIETY REVIEWS

A General Synthesis of Alkenyl-Substituted Benzofurans, Indoles, and Isoquinolones by Cascade Palladium-Catalyzed Heterocyclization/Oxidative Heck Coupling

(2010) Rosana Álvarez et al.   CHEMISTRY-A EUROPEAN JOURNAL

Palladium-Catalyzed Dynamic Kinetic Asymmetric Transformations of Vinyl Aziridines with Nitrogen Heterocycles: Rapid Access to Biologically Active Pyrroles and Indoles

(2010) Barry M. Trost et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Platinum(II)-Catalyzed Generation and [3+2] Cycloaddition Reaction of α,β-Unsaturated Carbene Complex Intermediates for the Preparation of Polycyclic Compounds

(2010) Kodai Saito et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

2,3-Disubstituted Indoles via Palladium-Catalyzed Reaction of 2-Alkynyltrifluoroacetanilides with Arenediazonium Tetrafluoroborates

(2010) Sandro Cacchi et al.   ORGANIC LETTERS

Enantioselective Modular Synthesis of Cyclohexenones: Total Syntheses of (+)-Crypto- and (+)-Infectocaryone

(2010) Géraldine Franck et al.   ORGANIC LETTERS

Palladium-Catalyzed Annulation of 2-(1-Alkynyl)benzenamines with Disulfides: Synthesis of 3-Sulfenylindoles

(2009) Yan-Jin Guo et al.   ADVANCED SYNTHESIS & CATALYSIS

Chemoselective Asymmetric N-Allylic Alkylation of Indoles with Morita-Baylis-Hillman Carbonates

(2009) Hai-Lei Cui et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iridium-Catalyzed Regio- and Enantioselective N-Allylation of Indoles

(2009) Levi M. Stanley et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Asymmetric Organocatalytic N-Alkylation of Indole-2-carbaldehydes with α,β-Unsaturated Aldehydes: One-Pot Synthesis of Chiral Pyrrolo[1,2-a]indole-2-carbaldehydes

(2009) Liang Hong et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective, Iridium-Catalyzed Monoallylation of Ammonia

(2009) Mark J. Pouy et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Brønsted Acid-CatalyzedN-Acyliminium Cyclization Cascades

(2009) Michael E. Muratore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regio- and EnantioselectiveN-Allylations of Imidazole, Benzimidazole, and Purine Heterocycles Catalyzed by Single-Component Metallacyclic Iridium Complexes

(2009) Levi M. Stanley et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct, Intermolecular, Enantioselective, Iridium-Catalyzed Allylation of Carbamates to Form Carbamate-Protected, Branched Allylic Amines

(2009) Daniel J. Weix et al.   ORGANIC LETTERS

Catalytic Synthesis of Indoles from Alkynes

(2008) Karolin Krüger (née Alex) et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Phase-Transfer-Catalyzed Intramolecular Aza-Michael Reaction: Effective Route to Pyrazino-Indole Compounds

(2008) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Phosphoric Acid Catalyzed Enantioselective Friedel–Crafts Alkylation of Indoles with Nitroalkenes: Cooperative Effect of 3 Å Molecular Sieves

(2008) Junji Itoh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iridium-Catalyzed Asymmetric Allylic Substitutions-Very High Regioselectivity and Air Stability with a Catalyst Derived from Dibenzo[a,e]cyclooctatetraene and a Phosphoramidite

(2008) Stephanie Spiess et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Asymmetric Brønsted Acid Catalysis: Enantioselective Nucleophilic Substitutions and 1,4-Additions

(2007) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Platinum-Catalyzed Formation of Cyclic-Ketone-Fused Indoles fromN-(2-Alkynylphenyl)lactams

(2007) Guotao Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION