Site-Selectivity of the Reaction of 3-Amino-4-Cyano-5-Phenyl-1H-Pyrrole-2-Carboxylic Acid Amide with α-Halocarbonyl Compounds. Antimicrobial Activity and Docking Study for COVID-19 of the Products

Advances in the development of therapeutic strategies against COVID-19 and perspectives in the drug design for emerging SARS-CoV-2 variants

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Novel sulfonyl thiazolyl-hydrazone derivatives as EGFR inhibitors: Design, synthesis, biological evaluation and molecular docking studies

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Pyrazoles and fused pyrimidines: Synthesis, structure elucidation, antitubercular activity and molecular docking study

(2021) Amerah M. Al-Soliemy et al.   Medicinal Chemistry

Synthesis, molecular docking, and in silico ADMET studies of 4-benzyl-1-(2,4,6-trimethyl-benzyl)-piperidine: Potential Inhibitor of SARS-CoV2

(2021) R. Nandini Asha et al.   BIOORGANIC CHEMISTRY

Drug repurposing against coronavirus disease 2019 (COVID-19): A review

(2021) Lianxiang Luo et al.   Journal of Pharmaceutical Analysis

Synthesis of a new series of pyrazolo[1,5-a]pyrimidines as CDK2 inhibitors and anti-leukemia

(2021) Samar J. Almehmadi et al.   BIOORGANIC CHEMISTRY

Microwaves assisted synthesis of antitumor agents of novel azoles, azines, and azoloazines pendant to phenyl sulfone moiety and molecular docking for VEGFR-2 kinase

(2021) Mohamed R. Shaaban et al.   JOURNAL OF MOLECULAR STRUCTURE

VEGFR2 and hepatocellular carcinoma inhibitory activities of trisubstituted triazole derivatives

(2021) Amani M.R. Alsaedi et al.   JOURNAL OF MOLECULAR STRUCTURE

Mono- and bimetallic complexes of pyrazolone based ligand: Synthesis, characterization, antitumor and molecular docking studies

(2021) Mona A. Alhasani et al.   JOURNAL OF MOLECULAR STRUCTURE

Nano-sized formazan analogues: Synthesis, structure elucidation, antimicrobial activity and docking study for COVID-19

(2020) Huda K. Mahmoud et al.   BIOORGANIC CHEMISTRY

Synthesis, molecular docking, and in silico ADME/Tox profiling studies of new 1-aryl-5-(3-azidopropyl)indol-4-ones: Potential inhibitors of SARS CoV-2 main protease

(2020) Francisco Xavier Domínguez-Villa et al.   BIOORGANIC CHEMISTRY

Design, Synthesis, and Biological Evaluation of Novel Pyrrolo[1,2-a]pyrazine Derivatives

(2019) Jinwoo Kim et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and Antimicrobial Evaluation of Novel Pyrazolopyrimidines Incorporated with Mono- and Diphenylsulfonyl Groups

(2019) Alsaedi et al.   MOLECULES

Benzosuberone as Precursor for Synthesis of Antimicrobial Agents: Synthesis, Antimicrobial Activity, and Molecular Docking

(2019) Ismail Althagafi et al.   POLYCYCLIC AROMATIC COMPOUNDS

Synthesis of Thiazole Linked Imidazo[2,1-b]Thiazoles as Anticancer Agents

(2019) Huda K. Mahmoud et al.   POLYCYCLIC AROMATIC COMPOUNDS

An antibiotic agent pyrrolo[1,2-a]pyrazine-1,4-dione,hexahydro isolated from a marine bacteria Bacillus tequilensis MSI45 effectively controls multi-drug resistant Staphylococcus aureus

(2018) George Seghal Kiran et al.   RSC Advances

Synthesis and biological evaluation of 1,2-dithiol-3-thiones and pyrrolo[1,2-a]pyrazines as novel hypoxia inducible factor-1 (HIF-1) inhibitor

(2016) Young Hun Lee et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and reactivity of novel pyrrolo[1,2-a]pyrazine derivatives

(2015) Maxim Voievudskyi et al.   MONATSHEFTE FUR CHEMIE

Synthesis, Tautomeric Structures, and Antitumor Activity of New Perimidines

(2013) Thoraya A. Farghaly et al.   ARCHIV DER PHARMAZIE

Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 1: Perhydropyrrole[1,2-a]pyrazines

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Pyrrolo[1,2-a]pyrazine and pyrazolo[1,5-a]pyrazine: Novel, potent, and selective series of Vasopressin1b receptor antagonists

(2010) Roberto Arban et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS