Cu‐Catalyzed Coupling Reactions of Sulfonamides with (Hetero)Aryl Chlorides/Bromides

Room Temperature Cu-Catalyzed N-Arylation of Oxazolidinones and Amides with (Hetero)Aryl Iodides

(2022) Subhajit Bhunia et al.   ORGANIC LETTERS

Cu-Mediated Ullmann-Type Cross-Coupling and Industrial Applications in Route Design, Process Development, and Scale-up of Pharmaceutical and Agrochemical Processes

(2022) Qiang Yang et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Modular Two‐Step Access to π‐Extended Naphthyridine Systems—Potent Building Blocks for Organic Electronics

(2021) Fabian Stuck et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Methoxylation of Aryl Bromides with 9-BBN−OMe

(2021) Jing-Ru Wang et al.   ORGANIC LETTERS

Copper-Catalyzed Ullmann-Type Coupling and Decarboxylation Cascade of Arylhalides with Malonates to Access α-Aryl Esters

(2021) Fei Cheng et al.   ORGANIC LETTERS

Nickel‐Catalyzed Cross‐Coupling of Sulfonamides With (Hetero)aryl Chlorides

(2020) Ryan T. McGuire et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Oxalohydrazide Ligands for Copper‐Catalyzed C−O Coupling Reactions with High Turnover Numbers

(2020) Ritwika Ray et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Assembly of α‐(Hetero)aryl Nitriles via Cu‐Catalyzed Coupling Reactions with (Hetero)aryl Chlorides and Bromides

(2020) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Oxalic Diamides and tert-Butoxide: Two Types of Ligands Enabling Practical Access to Alkyl Aryl Ethers via Cu-Catalyzed Coupling Reaction

(2019) Zhixiang Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cu-Catalyzed Couplings of Heteroaryl Primary Amines and (Hetero)aryl Bromides with 6-Hydroxypicolinamide Ligands

(2019) David J. Bernhardson et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Cu/N,N′-Dibenzyloxalamide-Catalyzed N-Arylation of Heteroanilines

(2019) Zhixiang Chen et al.   ORGANIC LETTERS

Reductive Cleavage of Secondary Sulfonamides: Converting Terminal Functional Groups into Versatile Synthetic Handles

(2019) Patrick S. Fier et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

High-Throughput Discovery and Evaluation of a General Catalytic Method for N-Arylation of Weakly Nucleophilic Sulfonamides

(2019) Joseph Becica et al.   ORGANIC LETTERS

Pd-Catalyzed Cross-Coupling Reactions Promoted by Biaryl Phosphorinane Ligands

(2019) Summer D. Laffoon et al.   ACS Catalysis

Sulfonamidation of Aryl and Heteroaryl Halides through Photosensitized Nickel Catalysis

(2018) Taehoon Kim et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent Development of Sulfonyl or Sulfonamide Hybrids as Potential Anticancer Agents: A Key Review

(2018) K. P. Rakesh et al.   Anti-Cancer Agents in Medicinal Chemistry

A Class of Amide Ligands Enable Cu-Catalyzed Coupling of (Hetero)aryl Halides with Sulfinic Acid Salts under Mild Conditions

(2018) Jinlong Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

Analysis of US FDA-Approved Drugs Containing Sulfur Atoms

(2018) Kevin A. Scott et al.   Topics in Current Chemistry

Mechanistic Insight Enables Practical, Scalable, Room Temperature Chan–Lam N-Arylation of N-Aryl Sulfonamides

(2018) Julien C. Vantourout et al.   ACS Catalysis

Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review

(2018) Chuang Zhao et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Survey of the Structures of US FDA Approved Combination Drugs

(2018) Pradipta Das et al.   JOURNAL OF MEDICINAL CHEMISTRY

The Journey of HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTIs) from Lab to Clinic

(2018) Vigneshwaran Namasivayam et al.   JOURNAL OF MEDICINAL CHEMISTRY

Convergent Synthesis of the NS5B Inhibitor GSK8175 Enabled by Transition Metal Catalysis

(2018) Kenneth Arrington et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Diaryl Ether Formation from (Hetero)aryl Halides at Low Catalytic Loadings

(2017) Yuntong Zhai et al.   JOURNAL OF ORGANIC CHEMISTRY

N,N′-Bisoxalamides Enhance the Catalytic Activity in Cu-Catalyzed Coupling of (Hetero)Aryl Bromides with Anilines and Secondary Amines

(2017) Subhajit Bhunia et al.   JOURNAL OF ORGANIC CHEMISTRY

Reagent Design and Ligand Evolution for the Development of a Mild Copper-Catalyzed Hydroxylation Reaction

(2017) Patrick S. Fier et al.   ORGANIC LETTERS

Discovery of N-(Naphthalen-1-yl)-N′-alkyl Oxalamide Ligands Enables Cu-Catalyzed Aryl Amination with High Turnovers

(2017) Jie Gao et al.   ORGANIC LETTERS

Copper-Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amides

(2017) Subhadip De et al.   ORGANIC LETTERS

Sulfur-Containing Agrochemicals

(2017) Ponnam Devendar et al.   Topics in Current Chemistry

CuI/Oxalamide Catalyzed Couplings of (Hetero)aryl Chlorides and Phenols for Diaryl Ether Formation

(2016) Mengyang Fan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Hydroxylation of (Hetero)aryl Halides under Mild Conditions

(2016) Shanghua Xia et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

CuI/Oxalic Diamide Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amines

(2015) Wei Zhou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Assembly of Primary (Hetero)Arylamines via CuI/Oxalic Diamide-Catalyzed Coupling of Aryl Chlorides and Ammonia

(2015) Mengyang Fan et al.   ORGANIC LETTERS

Copper-catalyzed direct N-arylation of N-arylsulfonamides using diaryliodonium salts in water

(2014) Xu Geng et al.   TETRAHEDRON LETTERS

BippyPhos: A Single Ligand With Unprecedented Scope in the Buchwald-Hartwig Amination of (Hetero)aryl Chlorides

(2013) Sarah M. Crawford et al.   CHEMISTRY-A EUROPEAN JOURNAL

Discovery of Dabrafenib: A Selective Inhibitor of Raf Kinases with Antitumor Activity against B-Raf-Driven Tumors

(2013) Tara R. Rheault et al.   ACS Medicinal Chemistry Letters

Stereocontrolled Synthesis of Vicinal Diamines by Organocatalytic Asymmetric Mannich Reaction of N-Protected Aminoacetaldehydes: Formal Synthesis of (−)-Agelastatin A

(2012) Taichi Kano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Divergent C–H Functionalizations Directed by Sulfonamide Pharmacophores: Late-Stage Diversification as a Tool for Drug Discovery

(2011) Hui-Xiong Dai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mild Pd-CatalyzedN-Arylation of Methanesulfonamide and Related Nucleophiles: Avoiding Potentially Genotoxic Reagents and Byproducts

(2011) Brandon R. Rosen et al.   ORGANIC LETTERS

Copper-MediatedN-Heteroarylation of Primary Sulfonamides: Synthesis of Mono-N-heteroaryl Sulfonamides

(2010) Jonathan Baffoe et al.   ORGANIC LETTERS

Genotoxic Impurities: From Structural Alerts to Qualification

(2010) David J. Snodin   ORGANIC PROCESS RESEARCH & DEVELOPMENT

A Designer Axially Chiral Amino Sulfonamide as an Efficient Organocatalyst for Direct Asymmetric Mannich Reactions of N-Boc-Protected Imines

(2009) Taichi Kano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Molecular Cloning, Characterization, and Inhibition Studies of the Rv1284 β-Carbonic Anhydrase fromMycobacterium tuberculosiswith Sulfonamides and a Sulfamate

(2009) Tomoko Minakuchi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Toolbox Approach to the Search for Effective Ligands for Catalytic Asymmetric Cr-Mediated Coupling Reactions

(2009) Haibing Guo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd-Catalyzed N-Arylation of Secondary Acyclic Amides: Catalyst Development, Scope, and Computational Study

(2009) Jacqueline D. Hicks et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cross coupling of 3-bromopyridine and sulfonamides (R1NHSO2R2·R1=H, Me, alkyl; R2=alkyl and aryl) catalyzed by CuI/1,3-di(pyridin-2-yl)propane-1,3-dione

(2009) Xiaojun Han   TETRAHEDRON LETTERS

Approaches to Assessment, Testing Decisions, and Analytical Determination of Genotoxic Impurities in Drug Substances

(2008) Duane A. Pierson et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

2-(Trimethylsilyl)ethanesulfonyl amide as a new ammonia equivalent for palladium-catalyzed amination of aryl halides

(2008) Prakash Anjanappa et al.   TETRAHEDRON LETTERS