Regioselective Synthesis of 3‐Trifluoromethyl 4‐Subtituted Pyrazoles by [3+2] Cycloaddition of Trifluoroacetonitrile Imines and Nitroalkenes

Fluorinated Pyrazoles: From Synthesis to Applications

(2021) Pavel K. Mykhailiuk   CHEMICAL REVIEWS

Regioselective Synthesis of 5-Trifluoromethylpyrazoles by [3 + 2] Cycloaddition of Nitrile Imines and 2-Bromo-3,3,3-trifluoropropene

(2021) Hao Zeng et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Difluoromethylated Pyrazoles by the [3 + 2] Cycloaddition Reaction of Difluoroacetohydrazonoyl Bromides

(2021) Tongyu Han et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Evaluation of Halogenated 5-(2-Hydroxyphenyl)pyrazoles as Pseudilin Analogues Targeting the Enzyme IspD in the Methylerythritol Phosphate Pathway

(2020) Jili Wang et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Development of celecoxib-derived antifungals for crop protection

(2020) Yihui Ma et al.   BIOORGANIC CHEMISTRY

Contribution of Organofluorine Compounds to Pharmaceuticals

(2020) Munenori Inoue et al.   ACS Omega

Fluorine‐Containing Drugs Approved by the FDA in 2018

(2019) Haibo Mei et al.   CHEMISTRY-A EUROPEAN JOURNAL

[3 + 2] Cycloaddition of para-Quinone Methides with Nitrile Imines: Approach to Spiro-pyrazoline-cyclohexadienones

(2019) Yingpeng Su et al.   JOURNAL OF ORGANIC CHEMISTRY

1,1,1,4,4,4‐Hexafluorobut‐2‐yne (HFB) as a Versatile Dipolarophile for [3+2] Cycloaddition with 1,3‐Dipoles toward Azoles with Adjacent CF 3 Groups

(2019) Yurii L. Yagupolskii et al.   ChemistrySelect

An Integrated Continuous Flow Micro-Total Ultrafast Process System (μ-TUFPS) for the Synthesis of Celecoxib and Other Cyclooxygenase Inhibitors

(2019) Vinay Kumar Sthalam et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Enantioselective Friedel–Crafts Alkylation Reaction of Indoles with α-Trifluoromethylated β-Nitrostyrenes Catalyzed by Chiral BINOL Metal Phosphate

(2019) Ignacio Ibáñez et al.   ACS Catalysis

Mild and Regioselective Synthesis of 3-CF3 -Pyrazoles by the AgOTf-Catalysed Reaction of CF3 -Ynones with Hydrazines

(2018) Maxim A. Topchiy et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Polysubstituted 3-trifluoromethylpyrazoles: regioselective (3 + 2)-cycloaddition of trifluoroacetonitrile imines with enol ethers and functional group transformations

(2018) Greta Utecht et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

NHC-Catalyzed Dual Stetter Reaction: A Mild Cascade Annulation for the Syntheses of Naphthoquinones, Isoflavanones, and Sugar-Based Chiral Analogues

(2018) Rajendra N. Mitra et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective, Metal-Free Approach to 3- or 5-CF3-Pyrazoles: Solvent Switchable Reaction of CF3-Ynones with Hydrazines

(2017) Vasiliy M. Muzalevskiy et al.   JOURNAL OF ORGANIC CHEMISTRY

Fluorinated Oligomers and Polymers in Photopolymerization

(2015) Alessandra Vitale et al.   CHEMICAL REVIEWS

Synthesis of 3-(Trifluoromethyl)pyrazoles and Polysubstituted Pyrazoles by atBuOK-Mediated Intramolecular Cycli­zation

(2015) Jia-Jie Wen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Ir(III)-Based Phosphors with Bipyrazolate Ancillaries; Rational Design, Photophysics, and Applications in Organic Light-Emitting Diodes

(2015) Jia-Ling Liao et al.   INORGANIC CHEMISTRY

1,3-Dipolar Cycloadditions of Ethyl 2-Diazo-3,3,3-trifluoropropanoate to Alkynes and [1,5] Sigmatropic Rearrangements of the Resulting 3H-Pyrazoles: Synthesis of Mono-, Bis- and Tris(trifluoromethyl)-Substituted Pyrazoles

(2014) Daniel Gladow et al.   HELVETICA CHIMICA ACTA

Rings in Drugs

(2014) Richard D. Taylor et al.   JOURNAL OF MEDICINAL CHEMISTRY

Fluoroalkyl-substituted lithium 1,3-diketonates in reactions with hetarylhydrazines

(2014) N. S. Boltacheva et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Pyrazole containing natural products: Synthetic preview and biological significance

(2013) Vinod Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of 4-Fluoromethylsydnones and their Participation in Alkyne Cycloaddition Reactions

(2013) Robert S. Foster et al.   JOURNAL OF ORGANIC CHEMISTRY

A General and Regioselective Synthesis of 5-Trifluoromethyl-pyrazoles

(2012) Robert S. Foster et al.   ORGANIC LETTERS

Organic fluorine compounds: a great opportunity for enhanced materials properties

(2011) Ricarda Berger et al.   CHEMICAL SOCIETY REVIEWS