Mild and Regioselective Synthesis of 3-CF3 -Pyrazoles by the AgOTf-Catalysed Reaction of CF3 -Ynones with Hydrazines

Selective, Metal-Free Approach to 3- or 5-CF3-Pyrazoles: Solvent Switchable Reaction of CF3-Ynones with Hydrazines

(2017) Vasiliy M. Muzalevskiy et al.   JOURNAL OF ORGANIC CHEMISTRY

Hydrohydrazination of Arylalkynes Catalyzed by an Expanded Ring N-Heterocyclic Carbene (er-NHC) Gold Complex Under Solvent-Free Conditions

(2016) Oleg S. Morozov et al.   ADVANCED SYNTHESIS & CATALYSIS

Trifluoromethyl nitrogen heterocycles: synthetic aspects and potential biological targets

(2016) F. Meyer   CHEMICAL COMMUNICATIONS

Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas

(2016) Yu Zhou et al.   CHEMICAL REVIEWS

Synthesis of fluazolate via the application of regioselective [3+2] cyclocondensation and nucleophilic substitution-cyclization strategies

(2016) Min-Tsang Hsieh et al.   TETRAHEDRON

Corrigendum: Solvent- and Transition Metal Catalyst-Dependent Regioselectivity in the [3+2] Cyclocondensation of Trifluoromethyl-α,β-ynones with Hydrazines: Switchable Access to 3- and 5-Trifluoromethylpyrazoles

(2015) Min-Tsang Hsieh et al.   ADVANCED SYNTHESIS & CATALYSIS

Solvent- and Transition Metal Catalyst-Dependent Regioselectivity in the [3+2] Cyclocondensation of Trifluoromethyl-α,β-ynones with Hydrazines: Switchable Access to 3- and 5-Trifluoromethylpyrazoles

(2015) Min-Tsang Hsieh et al.   ADVANCED SYNTHESIS & CATALYSIS

Recent Progress on Pyrazole Scaffold-Based Antimycobacterial Agents

(2015) Rangappa S. Keri et al.   ARCHIV DER PHARMAZIE

Gold(I)-Catalyzed Activation of Alkynes for the Construction of Molecular Complexity

(2015) Ruth Dorel et al.   CHEMICAL REVIEWS

Trifluoromethylpyrazoles as anti-inflammatory and antibacterial agents: A review

(2015) Kamalneet Kaur et al.   JOURNAL OF FLUORINE CHEMISTRY

Synthesis of 3-trifluoromethylpyrazoles via trifluoromethylation/cyclization of α,β-alkynic hydrazones using a hypervalent iodine reagent

(2014) Guojing Ji et al.   CHEMICAL COMMUNICATIONS

Expanded-RingN-Heterocyclic Carbenes Efficiently Stabilize Gold(I) Cations, Leading to High Activity in π-Acid-Catalyzed Cyclizations

(2014) Oleg S. Morozov et al.   CHEMISTRY-A EUROPEAN JOURNAL

A concise approach to CF3-containing furan-3-ones, (bis)pyrazoles from novel fluorinated building blocks based on 2,3-butanedione

(2014) Denis N. Bazhin et al.   TETRAHEDRON LETTERS

Comparative Study of the Regioselectivity and Reaction Media for the Synthesis of 1-tert-Butyl-3(5)-trifluoromethyl-1H-pyrazoles

(2012) Marcos A. P. Martins et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synergic Effects of Ionic Liquid and Microwave Irradiation in Promoting Trifluoromethylpyrazole Synthesis

(2011) Lilian Buriol et al.   CATALYSIS LETTERS

From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles

(2011) Santos Fustero et al.   CHEMICAL REVIEWS

Synthesis of Pyrazoles via CuI-Mediated Electrophilic Cyclizations of α,β-Alkynic Hydrazones

(2011) Metin Zora et al.   JOURNAL OF ORGANIC CHEMISTRY

A Novel Synthesis of Fluorinated Pyrazoles via Gold(I)-Catalyzed Tandem Aminofluorination of Alkynes in the Presence of Selectfluor

(2011) Jianqiang Qian et al.   ORGANIC LETTERS

A general strategy for the synthesis of difluoromethyl-containing pyrazoles, pyridines and pyrimidines

(2011) Viktor O. Iaroshenko et al.   TETRAHEDRON

Highly Convenient Regioselective Intermolecular Hydroamination of Alkynes Yielding Ketimines Catalyzed by Gold(I) Complexes of 1,2,4-triazole Based N-heterocyclic Carbenes

(2010) Chandrakanta Dash et al.   INORGANIC CHEMISTRY

NMR Chemical Shifts of Trace Impurities: Common Laboratory Solvents, Organics, and Gases in Deuterated Solvents Relevant to the Organometallic Chemist

(2010) Gregory R. Fulmer et al.   ORGANOMETALLICS

Reusable Gold(I) Catalysts with Unique Regioselectivity for Intermolecular Hydroamination of Alkynes

(2009) Antonio Leyva et al.   ADVANCED SYNTHESIS & CATALYSIS

A Cationic Gold(I) Complex as a General Catalyst for the Intermolecular Hydroamination of Alkynes: Application to the One-Pot Synthesis of Allenes from Two Alkynes and a Sacrificial Amine

(2009) Xiaoming Zeng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Reaction of Hydrazines and Hydroxylamine with Trifluoromethyl-β-diketones: Synthesis of Trifluoromethylpyrazole and Isoxazole Derivatives

(2009) Shiv P. Singh et al.   HETEROCYCLES

Improved Regioselectivity in Pyrazole Formation through the Use of Fluorinated Alcohols as Solvents: Synthesis and Biological Activity of Fluorinated Tebufenpyrad Analogs

(2008) Santos Fustero et al.   JOURNAL OF ORGANIC CHEMISTRY