Best practices in current models mimicking drug permeability in the gastrointestinal tract - An UNGAP review
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Title
Best practices in current models mimicking drug permeability in the gastrointestinal tract - An UNGAP review
Authors
Keywords
Intestinal permeability, Oral absorption, In vitro models, In vivo models, In silico, models, oral biopharmaceutics
Journal
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
Volume 170, Issue -, Pages 106098
Publisher
Elsevier BV
Online
2021-12-23
DOI
10.1016/j.ejps.2021.106098
References
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- Oral Delivery of Lipophilic Drugs: The Tradeoff between Solubility Increase and Permeability Decrease When Using Cyclodextrin-Based Formulations
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- Accounting for the solubility–permeability interplay in oral formulation development for poor water solubility drugs: The effect of PEG-400 on carbamazepine absorption
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- The Developability Classification System: Application of Biopharmaceutics Concepts to Formulation Development
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