Selenourea and thiourea derivatives of chiral and achiral enetetramines: Synthesis, characterization and enzyme inhibitory properties

PEPPSI type Pd(II)NHC Complexes Bearing Chloro-/Fluorobenzyl Group: Synthesis, Characterization, Crystal Structures, α-Glycosidase and Acetylcholinesterase Inhibitory Properties

(2021) Selma Bal et al.   POLYHEDRON

Potent Acetylcholinesterase Inhibitors: Potential Drugs for Alzheimer’s Disease

(2020) Hulya Akıncıoğlu et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

A Novel Ag-N-heterocyclic Carbene Complex Bearing the Hydroxyethyl Ligand: Synthesis, Characterization, Crystal and Spectral Structures and Bioactivity Properties

(2020) Aydin Aktas et al.   Crystals

Cholinesterases, α-glycosidase, and carbonic anhydrase inhibition properties of 1H-pyrazolo[1,2-b]phthalazine-5,10-dione derivatives: Synthetic analogues for the treatment of Alzheimer's disease and diabetes mellitus

(2020) Parham Taslimi et al.   BIOORGANIC CHEMISTRY

Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds – Determination of their carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibition properties

(2020) İlhami Gülçin et al.   BIOORGANIC CHEMISTRY

Design, synthesis, characterization, enzymatic inhibition evaluations, and docking study of novel quinazolinone derivatives

(2020) Keyvan Pedrood et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Synthesis, crystal structure, and biological evaluation of optically active 2-amino-4-aryl-7,7-dimethyl-5-oxo-5,6,7,8-tetrahydro-4H -chromen-3-carbonitriles: Antiepileptic, antidiabetic, and anticholinergics potentials

(2019) Abel Maharramov et al.   ARCHIV DER PHARMAZIE

Aminopyrazole-substituted metallophthalocyanines: Preparation, aggregation behavior, and investigation of metabolic enzymes inhibition properties

(2019) Emre Güzel et al.   ARCHIV DER PHARMAZIE

Phytochemical content, antioxidant activity, and enzyme inhibition effect of Salvia eriophora Boiss. & Kotschy against acetylcholinesterase, α-amylase, butyrylcholinesterase, and α-glycosidase enzymes

(2019) Ercan Bursal et al.   JOURNAL OF FOOD BIOCHEMISTRY

Synthesis, characterization, molecular docking and biological activities of novel pyrazoline derivatives

(2019) Fikret Turkan et al.   ARCHIV DER PHARMAZIE

Synthesis, biological evaluation and molecular docking of novel pyrazole derivatives as potent carbonic anhydrase and acetylcholinesterase inhibitors

(2019) Fikret Turkan et al.   BIOORGANIC CHEMISTRY

Synthesis and biological evaluation of novel tris-chalcones as potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibitors

(2019) Serdar Burmaoglu et al.   BIOORGANIC CHEMISTRY

Novel C-2 Symmetric Molecules as α-Glucosidase and α-Amylase Inhibitors: Design, Synthesis, Kinetic Evaluation, Molecular Docking and Pharmacokinetics

(2019) Danish Shahzad et al.   MOLECULES

Synthesis, characterization and biological applications of selenoureas having ferrocene and substituted benzoyl functionalities

(2019) Raja Azadar Hussain et al.   POLYHEDRON

Synthesis of novel tris-chalcones and determination of their inhibition profiles against some metabolic enzymes

(2019) Serdar Burmaoglu et al.   ARCHIVES OF PHYSIOLOGY AND BIOCHEMISTRY

Novel 2-aminopyridine liganded Pd(II) N-heterocyclic carbene complexes: Synthesis, characterization, crystal structure and bioactivity properties

(2019) Fatoş Erdemir et al.   BIOORGANIC CHEMISTRY

Treatment strategies against diabetes: Success so far and challenges ahead

(2019) Rubiya Khursheed et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Spectral and computational studies on regioselective synthesis of 4-oxo-6-phenyl-2-selenoxo-1,2,3,4-tetrahydropyrimidine-5-carbonitrile

(2019) Ibrahim A. Shaaban et al.   JOURNAL OF MOLECULAR STRUCTURE

Chemical Composition, Enantiomeric Distribution, and Sensory Evaluation of the Essential Oils Distilled from the Ecuadorian Species Myrcianthes myrsinoides (Kunth) Grifo and Myrcia mollis (Kunth) DC. (Myrtaceae)

(2019) Montalván et al.   Plants-Basel

Novel tribenzylaminobenzolsulphonylimine based on their pyrazine and pyridazines: Synthesis, characterization, antidiabetic, anticancer, anticholinergic, and molecular docking studies

(2019) Gulnar Mamedova et al.   BIOORGANIC CHEMISTRY

Synthesis and biological evaluation of phloroglucinol derivatives possessing α-glycosidase, acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase inhibitory activity

(2018) Serdar Burmaoglu et al.   ARCHIV DER PHARMAZIE

meta -Cyanobenzyl substituted benzimidazolium salts: Synthesis, characterization, crystal structure and carbonic anhydrase, α-glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties

(2018) Ferhat Türker et al.   ARCHIV DER PHARMAZIE

Recent Advances for the Synthesis of Selenium-containing Small Molecules as Potent Antitumor Agents

(2018) Qi Miao et al.   CURRENT MEDICINAL CHEMISTRY

Novel pyrimidinic selenourea induces DNA damage, cell cycle arrest, and apoptosis in human breast carcinoma

(2018) Flavio A.R. Barbosa et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Antioxidant and anticholinergic properties of olivetol

(2018) Parham Taslimi et al.   JOURNAL OF FOOD BIOCHEMISTRY

2-Hydroxyethyl substituted NHC precursors: Synthesis, characterization, crystal structure and carbonic anhydrase, α-glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties

(2018) Fatoş Erdemir et al.   JOURNAL OF MOLECULAR STRUCTURE

Novel thymol bearing oxypropanolamine derivatives as potent some metabolic enzyme inhibitors – Their antidiabetic, anticholinergic and antibacterial potentials

(2018) Mustafa Zengin et al.   BIOORGANIC CHEMISTRY

Antidiabetic and antiparasitic potentials: Inhibition effects of some natural antioxidant compounds on α-glycosidase, α-amylase and human glutathione S-transferase enzymes

(2018) İlhami Gulçin et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Synthesis, characterization, crystal structure, electrochemical studies and biological evaluation of metal complexes with thiosemicarbazone of glyoxylic acid

(2018) Mansura Huseynova et al.   POLYHEDRON

Screening the in vitro antioxidant, antimicrobial, anticholinesterase, antidiabetic activities of endemic Achillea cucullata (Asteraceae) ethanol extract

(2018) N. Eruygur et al.   SOUTH AFRICAN JOURNAL OF BOTANY

Current developments in chemistry, coordination, structure and biological aspects of 1-(acyl/aroyl)-3- (substituted)thioureas: advances Continue …

(2018) Aamer Saeed et al.   Journal of Sulfur Chemistry

Synthesis, characterization, crystal structure of novel bis-thiomethylcyclohexanone derivatives and their inhibitory properties against some metabolic enzymes

(2018) Abdullah Biçer et al.   BIOORGANIC CHEMISTRY

The first synthesis, carbonic anhydrase inhibition and anticholinergic activities of some bromophenol derivatives with S including natural products

(2018) Cetin Bayrak et al.   BIOORGANIC CHEMISTRY

The impact of some natural phenolic compounds on carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase, and α-glycosidase enzymes: An antidiabetic, anticholinergic, and antiepileptic study

(2017) Parham Taslimi et al.   JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY

Rb2 inhibits α-glucosidase and regulates glucose metabolism by activating AMPK pathways in HepG2 cells

(2017) Hui Teng et al.   Journal of Functional Foods

Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds

(2016) Bünyamin Özgeriş et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Benzimidazole derivatives as new α-glucosidase inhibitors and in silico studies

(2016) Nik Khairunissa Nik Abdullah Zawawi et al.   BIOORGANIC CHEMISTRY

Purification and characterization of the carbonic anhydrase enzyme from Black Sea trout (Salmo trutta Labrax Coruhensis) kidney and inhibition effects of some metal ions on enzyme activity

(2016) Murat Kucuk et al.   ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY

Selenoureido-iminosugars: A new family of multitarget drugs

(2016) Jacob Ingemar Olsen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Inhibitory effects of isatin Mannich bases on carbonic anhydrases, acetylcholinesterase, and butyrylcholinesterase

(2016) Dilan Ozmen Ozgun et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of diaryl ethers with acetylcholinesterase, butyrylcholinesterase and carbonic anhydrase inhibitory actions

(2016) Fadime Özbey et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis of 4,5-disubstituted-2-thioxo-1,2,3,4-tetrahydropyrimidines and investigation of their acetylcholinesterase, butyrylcholinesterase, carbonic anhydrase I/II inhibitory and antioxidant activities

(2016) Emin Garibov et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis and bioactivity studies on new 4-(3-(4-Substitutedphenyl)-3a,4-dihydro-3H-indeno[1,2-c]pyrazol-2-yl) benzenesulfonamides

(2016) Halise Inci Gul et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Chemical Constituents of Muehlenbeckia tamnifolia (Kunth) Meisn (Polygonaceae) and Its In Vitro α-Amilase and α-Glucosidase Inhibitory Activities

(2016) María Torres-Naranjo et al.   MOLECULES

The effect of caffeic acid phenethyl ester (CAPE) on metabolic enzymes including acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, lactoperoxidase, and carbonic anhydrase isoenzymes I, II, IX, and XII

(2015) İlhami Gülçin et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

SHELXT– Integrated space-group and crystal-structure determination

(2015) George M. Sheldrick   Acta Crystallographica A-Foundation and Advances

3-Acetyl-2-fluoro-6H-benzo[c]chromen-6-one

(2014) Yoshinobu Ishikawa et al.   ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE

Antithyroid Drugs and Their Analogues: Synthesis, Structure, and Mechanism of Action

(2013) Debasish Manna et al.   ACCOUNTS OF CHEMICAL RESEARCH

Novel Sulphamides and Sulphonamides Incorporating the Tetralin Scaffold as Carbonic Anhydrase and Acetylcholine Esterase Inhibitors

(2013) Akın Akıncıoğlu et al.   ARCHIV DER PHARMAZIE

Structurally Diversified Heterocycles and Related Privileged Scaffolds as Potential Urease Inhibitors: A Brief Overview

(2013) Aliya Ibrar et al.   ARCHIV DER PHARMAZIE

Inhibition of Lactoperoxidase-Catalyzed Oxidation by Imidazole-Based Thiones and Selones: A Mechanistic Study

(2013) Gouriprasanna Roy et al.   Chemistry-An Asian Journal

Acetylcholinesterase Inhibitors: Pharmacology and Toxicology

(2013) Mirjana B. Colovic et al.   Current Neuropharmacology

Synthesis, chemical characterization, DNA binding and antioxidant studies of ferrocene incorporated selenoure

(2013) Raja Azadar Hussain et al.   JOURNAL OF MOLECULAR STRUCTURE

Synthesis of novel planar chiral Ag and Rh N-heterocyclic carbene complexes derived from [2.2]paracyclophane and their application in ultrasound assisted asymmetric addition reactions of organoboronic acids to aldehydes

(2013) Wenzeng Duan et al.   TETRAHEDRON-ASYMMETRY

Rapid screening and identification ofα-glucosidase inhibitors from mulberry leaves using enzyme-immobilized magnetic beads coupled with HPLC/MS and NMR

(2012) Yi Tao et al.   BIOMEDICAL CHROMATOGRAPHY

(3,4-Dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and its derivatives as carbonic anhydrase isoenzymes inhibitors

(2012) Meryem Nar et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis, structural and vibrational properties of 1-(adamantane-1-carbonyl)-3-halophenyl thioureas

(2012) Aamer Saeed et al.   SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY

Steric tuning of C2-symmetric chiral N-heterocyclic carbene in gold-catalyzed asymmetric cyclization of 1,6-enynes

(2012) Ken-ichi Yamada et al.   TETRAHEDRON

(E)-2-Cyano-3-(2,3-dimethoxyphenyl)acrylic acid

(2011) Aliakbar Dehno Khalaji et al.   ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE

Synthesis, structural and vibrational properties of 1-(4-Fluorobenzoyl)-3-(isomeric fluorophenyl)thioureas

(2011) Aamer Saeed et al.   JOURNAL OF MOLECULAR STRUCTURE

Inhibition of peroxynitrite- and peroxidase-mediated protein tyrosine nitration by imidazole-based thiourea and selenourea derivatives

(2011) Krishna P. Bhabak et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

New Chiral N-Heterocyclic Carbene Ligands in Palladium-Catalyzed α-Arylations of Amides: Conformational Locking through Allylic Strain as a Device for Stereocontrol

(2010) Yi-Xia Jia et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Concise Synthesis of Substituted Thiourea Derivatives in Aqueous Medium

(2010) Mahagundappa R. Maddani et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of rhodium(I) and iridium(I) complexes of chiral N-heterocyclic carbenes and their application to asymmetric transfer hydrogenation

(2009) Gavin Dyson et al.   DALTON TRANSACTIONS

OLEX2: a complete structure solution, refinement and analysis program

(2009) Oleg V. Dolomanov et al.   JOURNAL OF APPLIED CRYSTALLOGRAPHY

Antioxidative effects of novel synthetic organoselenium compound in rat lung and kidney

(2008) Zeliha Selamoglu Talas et al.   ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY

Purification and Characterization of Peroxidase from Cauliflower (Brassica oleracea L. var. botrytis) Buds

(2008) Ekrem Koksal et al.   PROTEIN AND PEPTIDE LETTERS