Isatin thiazoles as antidiabetic: Synthesis, in vitro enzyme inhibitory activities, kinetics, and in silico studies

Synthesis of benzimidazole derivatives as potent inhibitors for α-amylase and their molecular docking study in management of type-II diabetes

(2021) Shafqat Hussain et al.   JOURNAL OF MOLECULAR STRUCTURE

Synthesis, α-amylase and α-glucosidase inhibition and molecular docking studies of indazole derivatives

(2021) Muhammad Nawaz et al.   JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS

Narrative review of the influence of diabetes mellitus and hyperglycemia on colorectal cancer risk and oncological outcomes

(2021) Hsiu-Chung Cheng et al.   Translational Oncology

Synthesis of indole derivatives as diabetics II inhibitors and enzymatic kinetics study of α-glucosidase and α-amylase along with their in-silico study

(2021) Muhammad Taha et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Synthesis, in vitro, and in silico evaluation of Indazole Schiff bases as potential α-glucosidase inhibitors

(2021) Bushra et al.   JOURNAL OF MOLECULAR STRUCTURE

Molecular docking of phenolic compounds and screening of antioxidant and antidiabetic potential of Olea europaea L. Ethanolic leaves extract

(2021) Sridevi Chigurupati et al.   Arabian Journal of Chemistry

Recent advances in isatin hybrids as potential anticancer agents

(2020) Zhen Ding et al.   ARCHIV DER PHARMAZIE

Synthesis and DNA binding of novel bioactive thiazole derivatives pendent to N-phenylmorpholine moiety

(2020) Thoraya A. Farghaly et al.   BIOORGANIC CHEMISTRY

Synthesis of azachalcones, their α-amylase, α-glucosidase inhibitory activities, kinetics, and molecular docking studies

(2020) Faiza Saleem et al.   BIOORGANIC CHEMISTRY

Synthesis of new indazole based dual inhibitors of α-glucosidase and α-amylase enzymes, their in vitro, in silico and kinetics studies

(2019) Rafaila Rafique et al.   BIOORGANIC CHEMISTRY

WITHDRAWN: Global and regional diabetes prevalence estimates for 2019 and projections for 2030 and 2045: results from the International Diabetes Federation Diabetes Atlas, 9th edition

(2019) Pouya Saeedi et al.   DIABETES RESEARCH AND CLINICAL PRACTICE

Synthesis of benzotriazoles derivatives and their dual potential as α-amylase and α-glucosidase inhibitors in vitro: Structure-activity relationship, molecular docking, and kinetic studies

(2019) Shehryar Hameed et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

1-[(4′-Chlorophenyl) carbonyl-4-(aryl) thiosemicarbazide derivatives as potent urease inhibitors: Synthesis, in vitro and in silico studies

(2018) Basharat Ali et al.   BIOORGANIC CHEMISTRY

Synthesis and biological evaluation of certain hydrazonoindolin-2-one derivatives as new potent anti-proliferative agents

(2018) Wagdy M. Eldehna et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis, in vitro $$\alpha $$α-glucosidase inhibitory activity, and in silico study of (E)-thiosemicarbazones and (E)-2-(2-(arylmethylene)hydrazinyl)-4-arylthiazole derivatives

(2018) Muhammad Ali et al.   MOLECULAR DIVERSITY

Insights into Structure-Activity Relationships of 3-Arylhydrazonoindolin-2-One Derivatives for Their Multitarget Activity on β-Amyloid Aggregation and Neurotoxicity

(2018) Rosa Purgatorio et al.   MOLECULES

2ʹ-Aryl and 4ʹ-arylidene substituted pyrazolones: As potential α-amylase inhibitors

(2018) Sahar Yousuf et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Biological Evaluation, and Molecular Docking Studies of Novel Isatin-Thiazole Derivatives as α-Glucosidase Inhibitors

(2017) et al.   MOLECULES

Structural Analysis of β-Fructofuranosidase fromXanthophyllomyces dendrorhousReveals Unique Features and the Crucial Role ofN-Glycosylation in Oligomerization and Activity

(2016) Mercedes Ramírez-Escudero et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Synthesis and anti-inflammatory activity evaluation of novel triazolyl-isatin hybrids

(2016) Pramod K. Sharma et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Clinical applications of amylase: Novel perspectives

(2016) Ernest Azzopardi et al.   SURGERY

Isatin based Schiff bases as inhibitors of α-glucosidase: Synthesis, characterization, in vitro evaluation and molecular docking studies

(2015) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Synthesis,In vitroand Docking Studies of New Flavone Ethers asα-Glucosidase Inhibitors

(2015) Syahrul Imran et al.   Chemical Biology & Drug Design

(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase

(2015) Rita Meleddu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design and synthesis of new antidiabetic α-glucosidase and α-amylase inhibitors based on pyrimidine-fused heterocycles

(2015) Sara Shahidpour et al.   MEDICINAL CHEMISTRY RESEARCH

A fluorescent chemosensor for sequential recognition of gallium and hydrogen sulfate ions based on a new phenylthiazole derivative

(2015) Bo-Yeon Kim et al.   SENSORS AND ACTUATORS B-CHEMICAL

One pot, multi-component synthesis of 3-[4-aryl-thiazol-2-yl)-hydrazono]-1,3-dihydro-indole-2-one

(2014) Tewodros Birhanu Aychiluhim et al.   CHEMICAL RESEARCH IN CHINESE UNIVERSITIES

Molecular Characterization of anrsmD-Like rRNA Methyltransferase from the Wolbachia Endosymbiont of Brugia malayi and Antifilarial Activity of Specific Inhibitors of the Enzyme

(2013) Ajay Kumar Rana et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Design and synthesis of 4-(1-(4-chlorobenzyl)-2,3-dioxoindolin-5-yl)-1-(4-substituted/unsubstituted benzylidene) semicarbazide: Novel agents with analgesic, anti-inflammatory and ulcerogenic properties

(2012) Chinnasamy Rajaram Prakash et al.   CHINESE CHEMICAL LETTERS

Synthesis and biological significances of 1,3,4-thiadiazolines and related heterocyclic compounds

(2011) Mohamad Yusuf et al.   Arabian Journal of Chemistry

Synthesis and Evaluation of Novel Indolylthiadiazinoazetidinones and Indolylthiadiazinothiazolidinones as Antimicrobial Agents

(2010) Vikas Kumar et al.   ARCHIV DER PHARMAZIE

Design and synthesis of anti-breast cancer agents from 4-piperazinylquinoline: A hybrid pharmacophore approach

(2010) V. Raja Solomon et al.   BIOORGANIC & MEDICINAL CHEMISTRY

N-Aroylated Isatins: Antiglycation Activity

(2010) Khalid Khan et al.   Letters in Drug Design & Discovery

New isatin derivatives with antioxidant activity

(2009) Aldo Andreani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY