Synthesis, in vitro $$\alpha $$α-glucosidase inhibitory activity, and in silico study of (E)-thiosemicarbazones and (E)-2-(2-(arylmethylene)hydrazinyl)-4-arylthiazole derivatives

Aryl thiosemicarbazones for the treatment of trypanosomatidic infections

(2018) Pasquale Linciano et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Biology-oriented drug synthesis (BIODS): In vitro β-glucuronidase inhibitory and in silico studies on 2-(2-methyl-5-nitro-1H-imidazol-1-yl)ethyl aryl carboxylate derivatives

(2017) Uzma Salar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Analogues of xanthones——Chalcones and bis-chalcones as α-glucosidase inhibitors and anti-diabetes candidates

(2017) Chao-Yun Cai et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies

(2017) Uzma Salar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Hydrazinyl arylthiazole based pyridine scaffolds: Synthesis, structural characterization, in vitro α -glucosidase inhibitory activity, and in silico studies

(2017) Farman Ali et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Constituent analysis of the ethanol extracts of Chimonanthus nitens Oliv. leaves and their inhibitory effect on α-glucosidase activity

(2017) Hui Chen et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Computational prediction integrating the inhibition kinetics of gallotannin on α-glucosidase

(2017) Li-Mei Yue et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

In vitro antioxidant, antiinflammatory and in silico molecular docking studies of thiosemicarbazones

(2017) G.R. Subhashree et al.   JOURNAL OF MOLECULAR STRUCTURE

Screening of enzyme inhibitors from traditional Chinese medicine by magnetic immobilized α-glucosidase coupled with capillary electrophoresis

(2017) Dong-Mei Liu et al.   TALANTA

Dihydropyrimidones: As novel class of β-glucuronidase inhibitors

(2016) Farman Ali et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Thiadiazole derivatives as New Class of β-glucuronidase inhibitors

(2016) Uzma Salar et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, in vitro α-glucosidase inhibitory activity and molecular docking studies of new thiazole derivatives

(2016) Khalid Mohammed Khan et al.   BIOORGANIC CHEMISTRY

Coordination chemistry of thiazoles, isothiazoles and thiadiazoles

(2016) Luís M.T. Frija et al.   COORDINATION CHEMISTRY REVIEWS

Syntheses of new 3-thiazolyl coumarin derivatives, in vitro α -glucosidase inhibitory activity, and molecular modeling studies

(2016) Uzma Salar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A small molecule mitigates hearing loss in a mouse model of Usher syndrome III

(2016) Kumar N Alagramam et al.   Nature Chemical Biology

Synthesis of 1,3-thiazolidin-4-ones; reactivity of the thiosemicarbazone function towards dimethyl acetylenedicarboxylate

(2016) Alaa A. Hassan et al.   JOURNAL OF CHEMICAL RESEARCH

Organocatalyzed solvent free an efficient novel synthesis of 2,4,5-trisubstituted imidazoles for α-glucosidase inhibition to treat diabetes

(2015) Muhammad Yar et al.   BIOORGANIC CHEMISTRY

Synthesis, in vitro evaluation and molecular docking studies of thiazole derivatives as new inhibitors of α-glucosidase

(2015) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Thiazole: A promising heterocycle for the development of potent CNS active agents

(2015) Chandra Bhushan Mishra et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Bioactive thiazole and benzothiazole derivatives

(2015) Abdul Rouf et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antiviral activity of some new bis-1,3-thiazole derivatives

(2015) Kamal M. Dawood et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Five-membered iminocyclitol α-glucosidase inhibitors: Synthetic, biological screening and in silico studies

(2013) Luis R. Guerreiro et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Highly Flexible π-Expanded Cyclooctatetraenes: Cyclic Thiazole Tetramers with Head-to-Tail Connection

(2012) Kazuhiro Mouri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Microwave-assisted synthesis and antioxidant properties of hydrazinyl thiazolyl coumarin derivatives

(2012) Hasnah Osman et al.   Chemistry Central Journal

Toward the Virtual Screening of α-Glucosidase Inhibitors with the Homology-Modeled Protein Structure

(2010)   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Pharmacology of α-glucosidase inhibition

(2010) H. BISCHOFF Bayer AG   EUROPEAN JOURNAL OF CLINICAL INVESTIGATION

α-Glucosidase inhibitors in diabetes: efficacy in NIDDM subjects

(2010) M. TOELLER   EUROPEAN JOURNAL OF CLINICAL INVESTIGATION

Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents

(2010) Franco Chimenti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Biological Activity, and Molecular Modeling Studies of 1H-1,2,3-Triazole Derivatives of Carbohydrates as α-Glucosidases Inhibitors

(2010) Sabrina B. Ferreira et al.   JOURNAL OF MEDICINAL CHEMISTRY