Synthesis, Biological Evaluation, and Molecular Docking Studies of Novel Isatin-Thiazole Derivatives as α-Glucosidase Inhibitors

Synthesis, in vitro evaluation and molecular docking studies of novel triazine-triazole derivatives as potential α-glucosidase inhibitors

(2017) Guangcheng Wang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, biological evaluation and molecular docking study of N -arylbenzo[ d ]oxazol-2-amines as potential α-glucosidase inhibitors

(2016) Guangcheng Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological evaluation of novel 2,4,5-triarylimidazole–1,2,3-triazole derivatives via click chemistry as α-glucosidase inhibitors

(2016) Guangcheng Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of novel 1,2,4-triazine derivatives bearing carbazole moiety as potent α-glucosidase inhibitors

(2016) Guangcheng Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, in vitro α-glucosidase inhibitory activity and molecular docking studies of new thiazole derivatives

(2016) Khalid Mohammed Khan et al.   BIOORGANIC CHEMISTRY

Synthesis,in vitroevaluation and molecular docking studies of novel coumarin-isatin derivatives as α-glucosidase inhibitors

(2016) Guangcheng Wang et al.   Chemical Biology & Drug Design

Inhibitory activity evaluation and mechanistic studies of tetracyclic oxindole derivatives as α-glucosidase inhibitors

(2016) Hua Sun et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Syntheses of new 3-thiazolyl coumarin derivatives, in vitro α -glucosidase inhibitory activity, and molecular modeling studies

(2016) Uzma Salar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Hybrid molecules: The privileged scaffolds for various pharmaceuticals

(2016) Shaveta et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

One-Pot and Three-Component Synthesis, Characterization and Biological Evaluation of Some New 1,2,4-Triazine-coumarins

(2016) Guang-cheng Wang et al.   HETEROCYCLES

Synthesis and anti-inflammatory activity evaluation of novel triazolyl-isatin hybrids

(2016) Pramod K. Sharma et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis, in vitro evaluation and molecular docking studies of thiazole derivatives as new inhibitors of α-glucosidase

(2015) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Isatin based Schiff bases as inhibitors of α-glucosidase: Synthesis, characterization, in vitro evaluation and molecular docking studies

(2015) Fazal Rahim et al.   BIOORGANIC CHEMISTRY

Synthesis of diethyl 4-substituted-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates as a new series of inhibitors against yeast α-glucosidase

(2015) Huma Niaz et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and evaluation of isatin-β-thiosemicarbazones as novel agents against antibiotic-resistant Gram-positive bacterial species

(2015) Xu-Meng Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of novel inhibitors of α-glucosidase based on the benzothiazole skeleton containing benzohydrazide moiety and their molecular docking studies

(2015) Muhammad Taha et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Therapeutic potential of α-glucosidase inhibitors in type 2 diabetes mellitus: an evidence-based review

(2015) Shashank R Joshi et al.   EXPERT OPINION ON PHARMACOTHERAPY

Advances in Pharmacology of Isatin and its Derivatives: A Review

(2015) Farhan A Khan et al.   TROPICAL JOURNAL OF PHARMACEUTICAL RESEARCH

Design, synthesis and biological evaluation of metronidazole–thiazole derivatives as antibacterial inhibitors

(2014) Ya-Juan Qin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Novel isatin-based hydroxamic acids as histone deacetylase inhibitors and antitumor agents

(2013) Nguyen-Hai Nam et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and pharmacological evaluation of some novel 2-(5-hydroxy-5-trifluoromethyl-4,5-dihydropyrazol-1-yl)-4-(coumarin-3-yl)thiazoles

(2013) Ranjana Aggarwal et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Structure-based design, synthesis, and anticonvulsant activity of isatin-1-N-phenylacetamide derivatives

(2013) Chao Xie et al.   MEDICINAL CHEMISTRY RESEARCH

2H-chromene derivatives bearing thiazolidine-2,4-dione, rhodanine or hydantoin moieties as potential anticancer agents

(2012) Mohammad Azizmohammadi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Triazole incorporated thiazoles as a new class of anticonvulsants: Design, synthesis and in vivo screening

(2010) Nadeem Siddiqui et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Crystal structures of isomaltase from Saccharomyces cerevisiae and in complex with its competitive inhibitor maltose

(2010) Keizo Yamamoto et al.   FEBS Journal

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

(2009) Garrett M. Morris et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY

Epidemiology of Diabetes and Diabetes-Related Complications

(2008) Anjali D Deshpande et al.   PHYSICAL THERAPY