Elemental Sulfur and Dimethyl Sulfoxide‐Promoted Oxidative Cyclization of Trifluoroacetimidohydrazides with Methylhetarenes for the Synthesis of 3‐Hetaryl ‐5‐trifluoromethyl‐1,2,4‐triazoles

Silver-Mediated [3 + 2] Cycloaddition of Azomethine Ylides with Trifluoroacetimidoyl Chlorides for the Synthesis of 5-(Trifluoromethyl)imidazoles

(2021) Hefei Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 5‐Trifluoromethyl‐1,2,4‐Triazoles via Metal‐Free Annulation of Trifluoroacetimidohydrazides and Methyl Ketones

(2021) Jiajun Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Four-Component Carbonylative Cyclization Reaction of Trifluoroacetimidoyl Chlorides, Propargyl Amines, and Diaryliodonium Salts: Access to Trifluoromethyl-Containing Trisubstituted Imidazoles

(2020) Zhengkai Chen et al.   ORGANIC LETTERS

Recent Advances in the Synthesis of Heterocycles via Reactions Involving Elemental Sulfur

(2020) Thanh Binh Nguyen   ADVANCED SYNTHESIS & CATALYSIS

FeCl3-Mediated Synthesis of 2-(Trifluoromethyl)quinazolin-4(3H)-ones from Isatins and Trifluoroacetimidoyl Chlorides

(2020) Le-Cheng Wang et al.   ORGANIC LETTERS

A Convenient FeCl 3 ‐Mediated Synthesis of 5‐Trifluoromethyl‐1,2,4‐triazoles from Trifluoroacetimidoyl Chlorides and Hydrazides

(2020) Shiying Du et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium‐Catalyzed Cascade Carbonylative Cyclization Reaction of Trifluoroacetimidoyl Chlorides and 2‐Iodoanilines: Toward 2‐(Trifluoromethyl)quinazolin‐4(3H)‐ones Synthesis

(2020) Hefei Yang et al.   ChemistrySelect

Elemental Sulfur/DMSO‐Promoted Multicomponent One‐pot Synthesis of Malonic Acid Derivatives from Maleic Anhydride and Amines

(2019) Le Anh Nguyen et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal‐Free Synthesis of 5‐Trifluoromethyl‐1,2,4‐Triazoles from Iodine‐Mediated Annulation of Trifluoroacetimidoyl Chlorides and Hydrazones

(2019) Sipei Hu et al.   ADVANCED SYNTHESIS & CATALYSIS

DMSO: yesterday’s solvent, today’s reagent

(2019) Zahra Tashrifi et al.   ADVANCED SYNTHESIS & CATALYSIS

Iodine Promoted Domino Oxidative Cyclization for One‐Pot Synthesis of Novel Fused Four‐ring Quinoxaline Fluorophore via sp³ C‐H Functionalization

(2019) Yong Zhang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Three-Component Cascade Bis-heteroannulation of Aryl or Vinyl Methylketoxime Acetates toward Thieno[3,2-c]isoquinolines

(2019) Zhenhua Xu et al.   ORGANIC LETTERS

Homo- and Heteroannulation of sp3 C–H Bonds in Acetophenones for Divergent Synthesis of Thienothiazoles

(2019) Phuc H. Pham et al.   ORGANIC LETTERS

Access to 2-Aroylthienothiazoles via C–H/N–O Bond Functionalization of Oximes

(2019) Peiqi Zhou et al.   ORGANIC LETTERS

Selective Construction of 2-Substituted Benzothiazoles from o-Iodoaniline Derivatives S8 and N-Tosylhydrazones

(2018) Yubing Huang et al.   JOURNAL OF ORGANIC CHEMISTRY

Thiophene-Fused Heteroaromatic Systems Enabled by Internal Oxidant-Induced Cascade Bis-Heteroannulation

(2018) Huawen Huang et al.   ORGANIC LETTERS

Tri-Functional Elemental Sulfur Enabling Bis-Heteroannulation of Methyl Ketoximes with Methyl N -Heteroarenes

(2018) Huawen Huang et al.   ADVANCED SYNTHESIS & CATALYSIS

Elemental sulfur as a polyvalent reagent in redox condensation with o-chloronitrobenzenes and benzaldehydes: three-component access to 2-arylbenzothiazoles

(2017) Le Anh Nguyen et al.   GREEN CHEMISTRY

Three-component synthesis of 2-heteroaryl-benzothiazoles under metal-free conditions

(2017) Guozheng Li et al.   GREEN CHEMISTRY

Solvent-controlled highly regio-selective thieno[2,3-b]indole formation under metal-free conditions

(2017) Penghui Ni et al.   GREEN CHEMISTRY

Copper-Catalyzed Tandem Aerobic Oxidative Cyclization for the Synthesis of Polysubstituted Quinolines via C(sp3)/C(sp2)–H Bond Functionalization

(2017) Xiaobo Pang et al.   JOURNAL OF ORGANIC CHEMISTRY

Elemental Sulfur-Promoted Oxidative Rearranging Coupling between o-Aminophenols and Ketones: A Synthesis of 2-Alkyl benzoxazoles under Mild Conditions

(2017) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Redox-Neutral Access to Sultams from 2-Nitrochalcones and Sulfur with Complete Atom Economy

(2017) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Trifluoromethyl nitrogen heterocycles: synthetic aspects and potential biological targets

(2016) F. Meyer   CHEMICAL COMMUNICATIONS

Aerobic Copper-Catalyzed Halocyclization of Methyl N-Heteroaromatics with Aliphatic Amines: Access to Functionalized Imidazo-Fused N-Heterocycles

(2016) Zhenda Tan et al.   JOURNAL OF ORGANIC CHEMISTRY

Direct and metal-free oxidative amination of sp3 C–H bonds for the construction of 2-hetarylquinazolin-4(3H)-ones

(2016) Huanhuan Liu et al.   Organic Chemistry Frontiers

Applications of Fluorine in Medicinal Chemistry

(2015) Eric P. Gillis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Aerobic Oxidative Amination of sp3C–H Bonds: Efficient Synthesis of 2-Hetarylquinazolin-4(3H)-ones

(2014) Qiang Li et al.   ORGANIC LETTERS

Catalysis for fluorination and trifluoromethylation

(2011) Takeru Furuya et al.   NATURE

Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4H-1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors

(2010) Takashi Sugane et al.   JOURNAL OF MEDICINAL CHEMISTRY