Three-component synthesis of 2-heteroaryl-benzothiazoles under metal-free conditions

One-Pot Cascade Synthesis of Substituted Carbazoles from Indoles, Ketones, and Alkenes Using Oxygen as the Oxidant

(2017) Shanping Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

N-Iodosuccinimide involved one-pot metal-free synthesis of 2-heteroaromatic benzothiazole compounds

(2017) Xianglong Chu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition Metal-Free Carbazole Synthesis from Arylureas and Cyclohexanones

(2016) Jun Wu et al.   ADVANCED SYNTHESIS & CATALYSIS

Nickel Catalysis Enables Oxidative C(sp2 )-H/C(sp2 )-H Cross-Coupling Reactions between Two Heteroarenes

(2016) Yangyang Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient pyrido[1,2-a]benzimidazole formation from 2-aminopyridines and cyclohexanones under metal-free conditions

(2016) Yanjun Xie et al.   GREEN CHEMISTRY

Unparalleled Ease of Access to a Library of Biheteroaryl Fluorophores via Oxidative Cross-Coupling Reactions: Discovery of Photostable NIR Probe for Mitochondria

(2016) Yangyang Cheng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Three-Component Approach to 3,5-Diaryl-1,2,4-thiadiazoles under Transition-Metal-Free Conditions

(2016) Hao Xie et al.   ORGANIC LETTERS

Indole-to-Carbazole Strategy for the Synthesis of Substituted Carbazoles under Metal-Free Conditions

(2016) Shanping Chen et al.   ORGANIC LETTERS

Naphthothiazole-based highly selective and sensitive fluorescent and colorimetric chemosensor for detection of pollutant metal ions

(2016) Mohammad Zareh Jonaghani et al.   RSC Advances

Rhodium(III)-Catalyzedortho-Heteroarylation of Phenols through Internal Oxidative CH Activation: Rapid Screening of Single-Molecular White-Light-Emitting Materials

(2015) Bijin Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium(III)-CatalyzedorthoCH Heteroarylation of (Hetero)aromatic Carboxylic Acids: A Rapid and Concise Access to π-Conjugated Poly-heterocycles

(2015) Xurong Qin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-catalyzed oxidative C–H/C–H cross-coupling of benzamides and thiophenes

(2015) Sheng Zhao et al.   CHEMICAL COMMUNICATIONS

Oxidative Coupling between Two Hydrocarbons: An Update of Recent C–H Functionalizations

(2015) Chao Liu et al.   CHEMICAL REVIEWS

Unexpectedly Simple Synthesis of Benzazoles bytBuONa-Catalyzed Direct Aerobic Oxidative Cyclocondensation ofo-Thio/Hydroxy/Aminoanilines with Alcohols under Air

(2015) Xinkang Shi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synergism in semiconducting nanocomposites: visible light photocatalysis towards the formation of C–S and C–N bonds

(2015) Anil R. Wade et al.   GREEN CHEMISTRY

Efficient 4,5-dihydro-1H-imidazol-5-one formation from amidines and ketones under transition-metal free conditions

(2015) Yanjun Xie et al.   GREEN CHEMISTRY

External Oxidant-Free Oxidative Cross-Coupling: A Photoredox Cobalt-Catalyzed Aromatic C–H Thiolation for Constructing C–S Bonds

(2015) Guoting Zhang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Au-Catalyzed Cross-Coupling of Arenes via Double C–H Activation

(2015) Xacobe C. Cambeiro et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Four-Component Approach to N-Substituted Phenothiazines under Transition-Metal-Free Conditions

(2015) Jinjin Chen et al.   ORGANIC LETTERS

Use of the Wilkinson Catalyst for theortho-CH Heteroarylation of Aromatic Amines: Facile Access to Highly Extended π-Conjugated Heteroacenes for Organic Semiconductors

(2014) Yumin Huang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Mediated CH/CH Biaryl Coupling of Benzoic Acid Derivatives and 1,3-Azoles

(2013) Mayuko Nishino et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Evaluation of (4-aminobutyloxy)quinolines as a novel class of antifungal agents

(2013) Stéphanie Vandekerckhove et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cobalt-Catalyzed Oxidative Isocyanide Insertion to Amine-Based Bisnucleophiles: Diverse Synthesis of Substituted 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and 2-Aminobenzoxazoles

(2013) Tong-Hao Zhu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Novel Conjugated Quinoline–Indoles Compromise Plasmodium falciparum Mitochondrial Function and Show Promising Antimalarial Activity

(2013) Silvia C. Teguh et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Synthesis of Substituted Benzothiazoles via Condensation of 2-Aminobenzenethiols with Nitriles

(2013) Yadong Sun et al.   ORGANIC LETTERS

Pd-catalyzed oxidative cross-coupling between two electron rich heteroarenes

(2013) Chun-Yang He et al.   Chemical Science

Rhodium or Ruthenium-Catalyzed Oxidative CH/CH Cross-Coupling: Direct Access to Extended π-Conjugated Systems

(2012) Jiaxing Dong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Mediated and Copper-Catalyzed Cross-Coupling of Indoles and 1,3-Azoles: Double CH Activation

(2012) Mayuko Nishino et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selective Rhodium(III)-Catalyzed Cross-Dehydrogenative Coupling of Furan and Thiophene Derivatives

(2012) Nadine Kuhl et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper(II)-Mediated Dehydrogenative Cross-Coupling of Heteroarenes

(2012) Zhifeng Mao et al.   ORGANIC LETTERS

Efficient 2-Aryl Benzothiazole Formation from Aryl Ketones and 2-Aminobenzenethiols under Metal-Free Conditions

(2012) Yunfeng Liao et al.   ORGANIC LETTERS

Precursor-directed generation of amidine containing ammosamide analogs: ammosamides E–P

(2012) Ende Pan et al.   Chemical Science

Palladium-Catalyzed Dehydrogenative Cross-Couplings of Benzazoles with Azoles

(2011) Wei Han et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Oxidative CH/CH Cross-Coupling of Indoles and Pyrroles with Heteroarenes

(2011) Zhen Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Selective Dehydrogenative Cross-Couplings of Heteroarenes

(2011) Xavier Bugaut et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fe-catalysed oxidative C–H functionalization/C–S bond formation

(2011) Haibo Wang et al.   CHEMICAL COMMUNICATIONS

Metal Azolate Frameworks: From Crystal Engineering to Functional Materials

(2011) Jie-Peng Zhang et al.   CHEMICAL REVIEWS

Direct Arylation of Benzothiazoles and Benzoxazoles with Aryl Boronic Acids

(2011) Sadananda Ranjit et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Progress in Coupling of Two Heteroarenes

(2011) Dongbing Zhao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Antitumor Quinol PMX464 Is a Cytocidal Anti-trypanosomal Inhibitor Targeting Trypanothione Metabolism

(2011) Janine König et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Synthesis and Biological Evaluation of Analogues of AKT (Protein Kinase B) Inhibitor-IV

(2011) Qi Sun et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Mediated Intermolecular Direct Biaryl Coupling

(2011) Masanori Kitahara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Amyloid-binding compounds maintain protein homeostasis during ageing and extend lifespan

(2011) Silvestre Alavez et al.   NATURE

Aerobic Visible-Light Photoredox Radical C–H Functionalization: Catalytic Synthesis of 2-Substituted Benzothiazoles

(2011) Yannan Cheng et al.   ORGANIC LETTERS

Use of Molecular Oxygen as a Reoxidant in the Synthesis of 2-Substituted Benzothiazoles via Palladium-Catalyzed CH Functionalization/Intramolecular CS Bond Formation

(2010) Kiyofumi Inamoto et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

(2010) Thomas W. Lyons et al.   CHEMICAL REVIEWS

Quinolines and structurally related heterocycles as antimalarials

(2010) Kirandeep Kaur et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Palladium-Catalyzed C−H Functionalization of Heteroarenes with Aryl Bromides and Chlorides

(2010) Shunsuke Tamba et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium(II)-Catalyzed Oxidative C−H/C−H Cross-Coupling of Heteroarenes

(2010) Peihua Xi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds

(2009) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Efficient and Economical Access to Substituted Benzothiazoles: Copper-Catalyzed Coupling of 2-Haloanilides with Metal Sulfides and Subsequent Condensation

(2009) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(II)-Catalyzed CH Activation/CC Cross-Coupling Reactions: Versatility and Practicality

(2009) Xiao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The rhodium carbene route to oxazoles: a remarkable catalyst effect

(2009) Baolu Shi et al.   CHEMICAL COMMUNICATIONS

2-Arylbenzothiazole as a Privileged Scaffold in Drug Discovery

(2009) A. Weekes et al.   CURRENT MEDICINAL CHEMISTRY

Utilization of 2-benzo[b]furan carboxylic acid hydrazide in the synthesis of 1,3,4-oxadiazole derivatives

(2009) Yu-Xia Da et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Development of a Diversity-Oriented Approach to Oxazole-5-amide Libraries

(2009) Mark J. Thompson et al.   JOURNAL OF ORGANIC CHEMISTRY

Ligand-Free Copper-Catalyzed Synthesis of Substituted Benzimidazoles, 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and Benzoxazoles

(2009) Prasenjit Saha et al.   JOURNAL OF ORGANIC CHEMISTRY

Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed C−H Bond Activation

(2008) Jared C. Lewis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis and Biological Properties of Benzothiazole, Benzoxazole, and Chromen-4-one Analogues of the Potent Antitumor Agent 2-(3,4-Dimethoxyphenyl)-5-fluorobenzothiazole (PMX 610, NSC 721648)(1)

(2008) Stefania Aiello et al.   JOURNAL OF MEDICINAL CHEMISTRY

Palladium-Catalyzed Synthesis of 2-Substituted Benzothiazoles via a C−H Functionalization/Intramolecular C−S Bond Formation Process

(2008) Kiyofumi Inamoto et al.   ORGANIC LETTERS