Palladium-Catalyzed One-Pot Synthesis of Pyrroloindolines from 2-Alkynyl Arylazides and Thioacetamides

From Reactive Oxygen Species to Reactive Brominating Species: Fenton Chemistry for Oxidative Bromination

(2021) Guodong Zhao et al.   ACS Sustainable Chemistry & Engineering

Synthesis of N-fused Seven-Membered Indoline-3-ones via Palladium-Catalyzed One-Pot Insertion Reaction from 2-Alkynyl Arylazides and Cyclic β-diketones

(2020) Ping Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Advancements in synthesis of pharmacologically active imidazolidin‐4‐ones and stereochemistry of their Reactions with some Reagents

(2020) Khaled F. Saied et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Electrochemical Dearomative Halocyclization of Tryptamine and Tryptophol Derivatives

(2020) Kun Liu et al.   CHINESE JOURNAL OF CHEMISTRY

Synthesis and biological profiling of half-calycanthaceous alkaloid analogues

(2020) Rui Zhu et al.   JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH

Synthesis of Polycylic Fused Indoline Scaffolds through a Substrates-Guided Reactivity Switch

(2020) Cecilia Ciccolini et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Dearomatizing Fluoroamidation of Indole Derivatives with Dianionic Phase-Transfer Catalyst

(2020) Hiromichi Egami et al.   ORGANIC LETTERS

Recent Developments in Photo‐Catalyzed/Promoted Synthesis of Indoles and Their Functionalization: Reactions and Mechanisms

(2020) Lvyin Zheng et al.   ADVANCED SYNTHESIS & CATALYSIS

Axially Chiral Cyclic Phosphoric Acid Enabled Enantioselective Sequential Additions

(2019) Xi Yuan et al.   ORGANIC LETTERS

Asymmetric Synthesis of C2-Quaternary Indolin-3-ones Enabled by N-Heterocyclic Carbene Catalysis

(2019) Shuaishuai Fang et al.   ORGANIC LETTERS

Gold-catalyzed N,O-functionalization of 1,4-diyn-3-ols with N-hydroxyanilines to form highly functionalized pyrrole derivatives

(2018) Yu-Chen Hsu et al.   CHEMICAL COMMUNICATIONS

Synthesis of functionalized pyrroloindolines via a visible-light-induced radical cascade reaction: rapid synthesis of (±)-flustraminol B

(2018) Kui Wu et al.   CHEMICAL COMMUNICATIONS

Gold-catalyzed [4+3]- and [4+2]-annulations of 3-en-1-ynamides with isoxazoles via novel 6π-electrocyclizations of 3-azahepta trienyl cations

(2018) Sovan Sundar Giri et al.   Chemical Science

Gold-Catalyzed Oxidative Cyclization of Tryptamine Derived Enynamides: A Stereoselective Approach to Tetracyclic Spiroindolines

(2018) Meijun Lin et al.   ADVANCED SYNTHESIS & CATALYSIS

Chiral phosphoric acid-catalyzed direct asymmetric mannich reaction of cyclic C-acylimines with simple ketones: facile access to C2-quaternary indolin-3-ones

(2018) Jin-Shan Li et al.   CHEMICAL COMMUNICATIONS

Pd-Catalyzed One-Pot Insertion Reaction of Cyclic C -Acylimines into Carbon-Carbon σ-Bonds for the Synthesis of Polyfunctional Indolin-3-ones from 2-Alkynyl Arylazides and Aryl Ketones

(2018) Ping Li et al.   ADVANCED SYNTHESIS & CATALYSIS

An environmentally friendly protocol for oxidative halocyclization of tryptamine and tryptophol derivatives

(2017) Jun Xu et al.   GREEN CHEMISTRY

Synthesis of 1H-indole-3-sulfonates via palladium-catalyzed tandem reactions of 2-alkynyl arylazides with sulfonic acids

(2017) Xiaoxiang Zhang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Preparation of 2-Amino-3-arylindoles via Pd-Catalyzed Coupling between 3-Diazoindolin-2-imines and Arylboronic Acids as well as Their Extension to 3-Aryl-3-fluoroindolin-2-imines

(2017) Hualong Ding et al.   ORGANIC LETTERS

Catalytic Asymmetric Mukaiyama–Mannich Reaction of Cyclic C-Acylimines with Difluoroenoxysilanes: Access to Difluoroalkylated Indolin-3-ones

(2017) Jin-Shan Li et al.   ORGANIC LETTERS

Visible-Light-Mediated Construction of Pyrroloindolines via an Amidyl Radical Cyclization/Carbon Radical Addition Cascade: Rapid Synthesis of (±)-Flustramide B

(2017) Kui Wu et al.   ORGANIC LETTERS

Fischer indole synthesis applied to the total synthesis of natural products

(2017) Majid M. Heravi et al.   RSC Advances

Organocatalytic Enantioselective Aza-Friedel-Crafts Reaction of Cyclic Ketimines with Pyrroles using Imidazolinephosphoric Acid Catalysts

(2016) Shuichi Nakamura et al.   CHEMISTRY-A EUROPEAN JOURNAL

Palladium-Catalyzed Synthesis of Indoles and Isoquinolines with in Situ Generated Phosphinimine

(2016) Qi Zhou et al.   JOURNAL OF ORGANIC CHEMISTRY

Access to the Pyrroloindoline Core via [3 + 2] Annulation as well as the Application in the Synthetic Approach to (±)-Minfiensine

(2016) Wenzhi Ji et al.   ORGANIC LETTERS

One-pot synthesis of polyhydropyrido[1,2- a ]indoles and tetracyclic quinazolinones from 2-arylindoles using copper-mediated oxidative tandem reactions

(2016) Mitsuaki Yamashita et al.   TETRAHEDRON

Pd(0)-Catalyzed Carbene Insertion into Si–Si and Sn–Sn Bonds

(2015) Zhenxing Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper(I)-Catalyzed Kinetic Resolution of N-Sulfonylaziridines with Indoles: Efficient Construction of Pyrroloindolines

(2015) Zhuo Chai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ligand-Controlled Product Selectivity in Gold-Catalyzed Double Cycloisomerization of 1,11-Dien-3,9-Diyne Benzoates

(2015) Weidong Rao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Dearomative Indole Cycloaddition Reactions of Aza-Oxyallyl Cationic Intermediates: Modular Access to Pyrroloindolines

(2015) Arjun Acharya et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Dearomative Indole (3 + 2) Reactions with Azaoxyallyl Cations – New Method for the Synthesis of Pyrroloindolines

(2015) Maria C. DiPoto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Total Synthesis of (−)-Lansai B and (+)-Nocardioazines A and B

(2014) Haoxuan Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

2-Aryl-3H-indol-3-ones: Synthesis, electrochemical behaviour and antiplasmodial activities

(2014) Ennaji Najahi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Catalytic Asymmetric Construction of Pyrroloindolines via an in Situ Generated Magnesium Catalyst

(2014) Linqing Wang et al.   ORGANIC LETTERS

Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (−)-Chimonanthine

(2013) Weiqing Xie et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Evolution of a Multicomponent System: Computational and Mechanistic Studies on the Chemo- and Stereoselectivity of a Divergent Process

(2013) Salomé Llabrés et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Developments in the Catalytic, Asymmetric Construction of Pyrroloindolines Bearing All-Carbon Quaternary Stereocenters

(2013) Lindsay M. Repka et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalytic Asymmetric Synthesis of Pyrroloindolines via a Rhodium(II)-Catalyzed Annulation of Indoles

(2013) Jillian E. Spangler et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Gold-Catalyzed Cycloisomerization of 1,6-Diyne Carbonates and Esters to 2,4a-Dihydro-1H-fluorenes

(2013) Weidong Rao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Michael Addition of Indoles to Isatylidene-3-acetaldehydes: Application to the Formal Total Synthesis of (−)-Chimonanthine

(2013) Renrong Liu et al.   ORGANIC LETTERS

Palladium-Catalyzed C–C Triple Bond Cleavage: Efficient Synthesis of 4H-Benzo[d][1,3]oxazin-4-ones

(2013) Qilun Liu et al.   ACS Catalysis

Catalytic Cascade Reactions Involving Metal Carbene Migratory Insertion

(2013) Ying Xia et al.   ACS Catalysis

Diazo Compounds and N-Tosylhydrazones: Novel Cross-Coupling Partners in Transition-Metal-Catalyzed Reactions

(2012) Qing Xiao et al.   ACCOUNTS OF CHEMICAL RESEARCH

Catalytic Asymmetric Total Synthesis of Chimonanthine, Folicanthine, and Calycanthine through Double Michael Reaction of Bisoxindole

(2012) Harunobu Mitsunuma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Exploration of Forbidden Povarov Processes as a Source of Unexpected Reactivity: A Multicomponent Mannich-Ritter Transformation

(2012) Sara Preciado et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective aza-Henry reactions of cyclic α-carbonyl ketimines under bifunctional catalysis

(2012) Alejandro Parra et al.   CHEMICAL COMMUNICATIONS

InCl3-Mediated Addition of Indole to Isatogens: An Expeditious Synthesis of 13-deoxy-Isatisine A

(2012) Chepuri V. Suneel Kumar et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric Brønsted Acid-Catalyzed Friedel-Crafts Reactions of Indoles with Cyclic Imines - Efficient Generation of Nitrogen-Substituted Quaternary Carbon Centers

(2011) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

Gold-Catalyzed Transformation of 2-Alkynyl Arylazides: Efficient Access to the Valuable Pseudoindoxyl and Indolyl Frameworks

(2011) Alexander Wetzel et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

N-Tosylhydrazones: versatile reagents for metal-catalyzed and metal-free cross-coupling reactions

(2011) Zhihui Shao et al.   CHEMICAL SOCIETY REVIEWS

Structure, Bioactivity and Synthesis of Natural Products with Hexahydropyrrolo[2,3-b]indole

(2011) Pau Ruiz-Sanchis et al.   CHEMISTRY-A EUROPEAN JOURNAL

The Palladium Catalyzed Asymmetric Addition of Oxindoles and Allenes: An Atom-Economical Versatile Method for the Construction of Chiral Indole Alkaloids

(2011) Barry M. Trost et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ethylene in Organic Synthesis: A New Route to Anticholenergic Pyrrolidinoindolines, and Other Molecules with All Carbon-Quaternary Centers via Asymmetric Hydrovinylation

(2011) Hwan Jung Lim et al.   ORGANIC LETTERS

Asymmetric Conjugate Addition of Oxindoles to 2-Chloroacrylonitrile: A Highly Effective Organocatalytic Strategy for Simultaneous Construction of 1,3-Nonadjacent Stereocenters Leading to Chiral Pyrroloindolines

(2010) Xin Li et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective Synthesis of Pyrroloindolines by a Formal [3 + 2] Cycloaddition Reaction

(2010) Lindsay M. Repka et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Exploration of the interrupted Fischer indolization reaction

(2010) Alex W. Schammel et al.   TETRAHEDRON

Phosphonium Salts as Chiral Phase-Transfer Catalysts: Asymmetric Michael and Mannich Reactions of 3-Aryloxindoles

(2009) Rongjun He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Thiourea-Catalyzed Highly Enantio- and Diastereoselective Additions of Oxindoles to Nitroolefins: Application to the Formal Synthesis of (+)-Physostigmine

(2009) Tommy Bui et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Interrupted Fischer Indolization Approach toward Fused Indoline-Containing Natural Products

(2009) Ben W. Boal et al.   ORGANIC LETTERS

Total Synthesis of (±)-Psychotrimine

(2008) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Intramolecular Arylcyanation of Alkenes Catalyzed by Nickel/AlMe2Cl

(2008) Yoshiaki Nakao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY