Recent Developments in Photo‐Catalyzed/Promoted Synthesis of Indoles and Their Functionalization: Reactions and Mechanisms

Recent Advances in the Electrochemical Synthesis and Functionalization of Indole Derivatives

(2020) Keyin Ye et al.   ADVANCED SYNTHESIS & CATALYSIS

Visible Light-Catalyzed Cascade Radical Cyclization of N-Propargylindoles with Acyl Chlorides for the Synthesis of 2-Acyl-9H-pyrrolo[1,2-a]indoles

(2020) Yu Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Ynamide Smiles Rearrangement Triggered by Visible-Light-Mediated Regioselective Ketyl–Ynamide Coupling: Rapid Access to Functionalized Indoles and Isoquinolines

(2020) Ze-Shu Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

CF3SO2Na-Mediated, UV-Light-Induced Friedel–Crafts Alkylation of Indoles with Ketones/Aldehydes and Bioactivities of Products

(2020) Tianbao Yang et al.   ORGANIC LETTERS

Sequential Visible-Light and N-Heterocyclic Carbene Catalysis: Stereoselective Synthesis of Tetrahydropyrano[2,3-b]indoles

(2020) Chengyuan Wang et al.   ORGANIC LETTERS

Visible-Light-Driven Radical Multicomponent Reaction of 2-Vinylanilines, Sulfonyl Chlorides, and Sulfur Ylides for Synthesis of Indolines

(2020) Mukund M. D. Pramanik et al.   ORGANIC LETTERS

Gold-Catalyzed Reaction of Alkynes with Diazonium Salts under Photoirradiation Revisited: New Alkoxyarylation Variant Leading to Enol Ethers

(2020) Carlos Lázaro-Milla et al.   JOURNAL OF CATALYSIS

Heterogeneous Photocatalytic Organic Transformation Reactions Using Conjugated Polymers-Based Materials

(2020) Jie Xiao et al.   ACS Catalysis

Synthesis of Cyclobutane-Fused Angular Tetracyclic Spiroindolines via Visible-Light-Promoted Intramolecular Dearomatization of Indole Derivatives

(2019) Min Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Photocatalyzed Cascade Approach Toward the Tetracyclic Core of Akuammiline Alkaloids

(2019) Qile Wang et al.   ORGANIC LETTERS

Visible-Light-Promoted Three-Component Coupling Annulation: Synthesis of 2-Iminothiazolidin-4-ones via in Situ Formed Electron Donor–Acceptor Complexes

(2019) Wei Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Merging Visible-Light Photoredox and Chiral Phosphate Catalysis for Asymmetric Friedel–Crafts Reaction with in Situ Generation of N-Acyl Imines

(2019) Meng-Lan Shen et al.   ORGANIC LETTERS

Visible-Light-Mediated Ir(III)-Catalyzed Concomitant C3 Oxidation and C2 Amination of Indoles

(2019) Gaurav Shukla et al.   ORGANIC LETTERS

Visible-Light-Driven Organic Photochemical Reactions in the Absence of External Photocatalysts

(2019) Yi Wei et al.   SYNTHESIS-STUTTGART

Indole Alkaloid Synthesis Facilitated by Photoredox Catalytic Radical Cascade Reactions

(2019) Xiao-Yu Liu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Recent advances in asymmetric synthesis of 2-substituted indoline derivatives

(2019) Ting-Bi Hua et al.   CHINESE CHEMICAL LETTERS

Photodriven Photocatalyst/Metal-Free Direct C–C/C–N Bond Formation: Synthesis of Indoles via EDA Complexes

(2019) Wei Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible-Light-Catalyzed [3 + 1 + 2] Coupling Annulations for the Synthesis of Unsymmetrical Trisubstituted Amino-1,3,5-triazines

(2019) Wei Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible Light‐Mediated C2‐Quaternarization of N‐Alkyl Indoles through Oxidative Dearomatization using Ir(III) Catalyst

(2019) Gaurav Shukla et al.   Asian Journal of Organic Chemistry

Visible‐Light‐Mediated Dearomatisation of Indoles and Pyrroles to Pharmaceuticals and Pesticides

(2019) Waldemar Schilling et al.   CHEMISTRY-A EUROPEAN JOURNAL

Continuous Heterogeneous Photocatalysis in Serial Micro-Batch Reactors

(2018) Bartholomäus Pieber et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

An atmosphere and light tuned highly diastereoselective synthesis of cyclobuta/penta[b]indoles from aniline-tethered alkylidenecyclopropanes with alkynes

(2018) Bo Cao et al.   CHEMICAL COMMUNICATIONS

Synthesis of functionalized pyrroloindolines via a visible-light-induced radical cascade reaction: rapid synthesis of (±)-flustraminol B

(2018) Kui Wu et al.   CHEMICAL COMMUNICATIONS

Synthesis of indoles under the action of visible light (microreview)

(2018) Alexey A. Festa   Chemistry of Heterocyclic Compounds

Synthesis of gem -Difluorinated Spiro-γ-lactam Oxindoles by Visible-Light-Induced Consecutive Difluoromethylative Dearomatization, Hydroxylation, and Oxidation

(2018) Qiang Wang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Visible-Light Catalytic Photooxygenation of Monoterpene Indole Alkaloids: Access to Spirooxindole-1,3-oxazines

(2018) Thorsten von Drathen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic Asymmetric Cascade Aerobic Oxidation and Semipinacol Rearrangement Reaction: A Visible Light-Induced Approach to Access Chiral 2,2-Disubstituted Indolin-3-ones

(2018) Liwei Bu et al.   Chemistry-An Asian Journal

Visible-Light-Mediated Eosin Y Photoredox-Catalyzed Vicinal Thioamination of Alkynes: Radical Cascade Annulation Strategy for 2-Substituted-3-sulfenylindoles

(2018) Shrikant D. Tambe et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Visible-Light Organophotoredox-Catalyzed Synthesis of Precursors for Horner-Type Olefinations

(2018) Marco M. Nebe et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Visible light induced hydrodifluoromethylation of alkenes derived from oxindoles with (difluoromethyl)triphenylphosphonium bromide

(2018) Wei-Qiang Hu et al.   JOURNAL OF FLUORINE CHEMISTRY

Visible light and hydroxynaphthylbenzimidazoline promoted transition-metal-catalyst-free desulfonylation of N-sulfonylamides and N-sulfonylamines

(2018) Eietsu Hasegawa et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible Light-Promoted Three-Component Tandem Annulation for the Synthesis of 2-Iminothiazolidin-4-ones

(2018) Wei Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Photoredox Cyanomethylation of Indoles: Catalyst Modification and Mechanism

(2018) Connor J. O’Brien et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Synthesis of Pyrroloindolines via Noncovalent Stabilization of Indole Radical Cations and Applications to the Synthesis of Alkaloid Natural Products

(2018) Emily C. Gentry et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Eosin Y–Yb(OTf)3 catalyzed visible light mediated electrocyclization/indole ring opening towards the synthesis of heterobiaryl-pyrazolo[3,4-b]pyridines

(2018) Shikha Singh et al.   NEW JOURNAL OF CHEMISTRY

Rose Bengal catalysed photo-induced selenylation of indoles, imidazoles and arenes: a metal free approach

(2018) Sumbal Saba et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Autoxidation Photoredox Catalysis for the Synthesis of 2-Phosphinoylindoles

(2018) Chun-Hai Wang et al.   ORGANIC LETTERS

Temperature Controlled Selective C–S or C–C Bond Formation: Photocatalytic Sulfonylation versus Arylation of Unactivated Heterocycles Utilizing Aryl Sulfonyl Chlorides

(2018) Santosh K. Pagire et al.   ORGANIC LETTERS

Visible-Light-Promoted Cascade Alkene Trifluoromethylation and Dearomatization of Indole Derivatives via Intermolecular Charge Transfer

(2018) Min Zhu et al.   ORGANIC LETTERS

Metal and acid-free visible light-mediated Friedel-Crafts alkylation reactions of indole with anilines

(2018) Xiao-Qiang Dai et al.   TETRAHEDRON LETTERS

Redox and photocatalytic properties of a NiII complex with a macrocyclic biquinazoline (Mabiq) ligand

(2018) Michael Grübel et al.   Chemical Science

Visible Light-Driven C-3 Functionalization of Indoles over Conjugat-ed Microporous Polymers

(2018) Weijie Zhang et al.   ACS Catalysis

Visible-light-induced C(sp3)–H activation for a C–C bond forming reaction of 3,4-dihydroquinoxalin-2(1H)-one with nucleophiles using oxygen with a photoredox catalyst or under catalyst-free conditions

(2018) Pavan Sudheer Akula et al.   RSC Advances

Intramolecular radical cyclization approach to access highly substituted indolines and 2,3-dihydrobenzofurans under visible-light

(2018) Clarice A. D. Caiuby et al.   RSC Advances

Catalyst and Sensitizer-Free Visible-Light-Induced C(sp2 )−H Chalcogenation of Arenes/ Heteroarenes with Dichalcogenides

(2018) Gullapalli Kumaraswamy et al.   Asian Journal of Organic Chemistry

Photoredox-catalyzed direct aminoalkylation of isatins: diastereoselective access to 3-hydroxy-3-aminoalkylindolin-2-ones analogues

(2018) Chao-Ming Wang et al.   Organic Chemistry Frontiers

Synthesis of visible-light mediated tryptanthrin derivatives from isatin and isatoic anhydride under transition metal-free conditions

(2018) Hong Hou et al.   Organic Chemistry Frontiers

Visible light-induced aerobic oxidative cross-coupling of glycine derivatives with indoles: a facile access to 3,3′ bisindolylmethanes

(2018) Yuan Zhang et al.   Organic Chemistry Frontiers

Visible-Light-Mediated Dearomatization/Cyanation Cascade Reaction of Indoles: Access to Highly Functionalized Spiro-γ-lactam Indolines with Two Contiguous Sterically Congested Quaternary Carbon Stereocenters

(2018) Qiang Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Visible-Light-Induced Trifluoromethylation of Isonitrile-Substituted Indole Derivatives: Access to 1-(Trifluoromethyl)-4,9-dihydro-3H -pyrido[3,4-b]indole and β -Carboline Derivatives

(2018) Jiaxin Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Radical C−H-Amination of Heteroarenes using Dual Initiation by Visible Light and Iodine

(2018) Nicola Lucchetti et al.   ADVANCED SYNTHESIS & CATALYSIS

Visible-Light-Induced 3-Component Synthesis of Sulfonylated Oxindoles by Fixation of Sulfur Dioxide

(2018) Nai-Wei Liu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A methodology for the photocatalyzed radical trifluoromethylation of indoles: A combined experimental and computational study

(2018) Shelli A. Miller et al.   JOURNAL OF FLUORINE CHEMISTRY

Enantioselective Radical Cyclization of Tryptamines by Visible Light-Excited Nitroxides

(2018) Kangjiang Liang et al.   JOURNAL OF ORGANIC CHEMISTRY

Concurrent Asymmetric Reactions Combining Photocatalysis and Enzyme Catalysis: Direct Enantioselective Synthesis of 2,2-Disubstituted Indol-3-ones from 2-Arylindoles

(2018) Xuan Ding et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Bromo- or Methoxy-Group-Promoted Umpolung Electron Transfer Enabled, Visible-Light-Mediated Synthesis of 2-Substituted Indole-3-glyoxylates

(2018) Adiyala Vidyasagar et al.   ORGANIC LETTERS

9,10-Phenanthrenedione as Visible-Light Photoredox Catalyst: A Green Methodology for the Functionalization of 3,4-Dihydro-1,4-Benzoxazin-2-Ones through a Friedel-Crafts Reaction

(2018) Jaume Rostoll-Berenguer et al.   Catalysts

Photoredox-Induced Radical 6-exo -trig Cyclizations onto the Indole Nucleus: Aromative versus Dearomative Pathways

(2017) Dirk Alpers et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Tandem cyclisation of vinyl radicals: a sustainable approach to indolines utilizing visible-light photoredox catalysis

(2017) Santosh K. Pagire et al.   GREEN CHEMISTRY

Visible-light-mediated aerobic selenation of (hetero)arenes with diselenides

(2017) Qing-Bao Zhang et al.   GREEN CHEMISTRY

Visible-Light-Promoted Tandem Difluoroalkylation–Amidation: Access to Difluorooxindoles from Free Anilines

(2017) Ling-Chao Yu et al.   JOURNAL OF ORGANIC CHEMISTRY

Photoredox-Catalyzed Reductive Dimerization of Isatins and Isatin-Derived Ketimines: Diastereoselective Construction of 3,3′-Disubstituted Bisoxindoles

(2017) Chao-Ming Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Selenylation of Imidazo[1,2-a]pyridines with Selenium Powder via a Radical Pathway

(2017) Pengfei Sun et al.   JOURNAL OF ORGANIC CHEMISTRY

Transition-metal-free, visible-light-mediated cyclization of o-azidoarylalkynes with aryl diazonium salts

(2017) Cheng Jin et al.   NEW JOURNAL OF CHEMISTRY

Dual visible-light photoredox and palladium(ii) catalysis for dehydrogenative C2-acylation of indoles at room temperature

(2017) Manash Kumar Manna et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Visible-Light-Mediated Anti-Regioselective Nitrone 1,3-Dipolar Cycloaddition Reaction and Synthesis of Bisindolylmethanes

(2017) Lewei Zheng et al.   ORGANIC LETTERS

Visible Light Promoted Synthesis of Indoles by Single Photosensitizer under Aerobic Conditions

(2017) Wen-Qiang Liu et al.   ORGANIC LETTERS

A General Copper Catalyst for Photoredox Transformations of Organic Halides

(2017) Bastien Michelet et al.   ORGANIC LETTERS

Photoredox Catalysis Induced Bisindolylation of Ethers/Alcohols via Sequential C–H and C–O Bond Cleavage

(2017) Lu Ye et al.   ORGANIC LETTERS

Cross-Dehydrogenative C–H Amination of Indoles under Aerobic Photo-oxidative Conditions

(2017) Tomoaki Yamaguchi et al.   ORGANIC LETTERS

Visible-Light-Mediated Construction of Pyrroloindolines via an Amidyl Radical Cyclization/Carbon Radical Addition Cascade: Rapid Synthesis of (±)-Flustramide B

(2017) Kui Wu et al.   ORGANIC LETTERS

Visible-light promoted synthesis of 3-arylthioindoles from indoles and diaryl disulfides

(2017) Lin-miao Ye et al.   TETRAHEDRON LETTERS

Visible-light-induced oxidant and metal-free dehydrogenative cascade trifluoromethylation and oxidation of 1,6-enynes with water

(2017) Sadhan Jana et al.   Chemical Science

Regioselective Synthesis of 2-Substituted Indoles from Benzotriazoles and Alkynes by Photoinitiated Denitrogenation

(2017) Michael Teders et al.   ACS Catalysis

Photocatalytic Indole Diels–Alder Cycloadditions Mediated by Heterogeneous Platinum-Modified Titanium Dioxide

(2017) Spencer P. Pitre et al.   ACS Catalysis

Merger of Visible-Light Photoredox Catalysis and C–H Activation for the Room-Temperature C-2 Acylation of Indoles in Batch and Flow

(2017) Upendra K. Sharma et al.   ACS Catalysis

Photocatalytic direct C–S bond formation: facile access to 3-sulfenylindoles via metal-free C-3 sulfenylation of indoles with thiophenols

(2017) Wei Guo et al.   RSC Advances

Visible light-induced tandem oxidative cyclization of 2-alkynylanilines with disulfides (diselenides) to 3-sulfenyl- and 3-selenylindoles under transition metal-free and photocatalyst-free conditions

(2017) Qing Shi et al.   Organic Chemistry Frontiers

A Radical Cascade Enabling Collective Syntheses of Natural Products

(2017) Xiaobei Wang et al.   Chem

Synthetic Utilization of α-Aminoalkyl Radicals and Related Species in Visible Light Photoredox Catalysis

(2016) Kazunari Nakajima et al.   ACCOUNTS OF CHEMICAL RESEARCH

Rare Metal-Free Photo-Aerobic Intramolecular Dehydrogenative Cyclization Reaction towards Polycyclic Heteroarenes

(2016) Eiji Yamaguchi et al.   ADVANCED SYNTHESIS & CATALYSIS

Noble metal-based bimetallic nanoparticles: the effect of the structure on the optical, catalytic and photocatalytic properties

(2016) Adriana Zaleska-Medynska et al.   ADVANCES IN COLLOID AND INTERFACE SCIENCE

Multifunctional Antioxidants: Regenerable Radical-Trapping and Hydroperoxide-Decomposing Ebselenols

(2016) Shailesh Kumar et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Photosensitizer-Free Visible-Light-Mediated Gold-Catalyzed 1,2-Difunctionalization of Alkynes

(2016) Long Huang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Photoinduced Multicomponent Reactions

(2016) Silvia Garbarino et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible light-photocatalysed carbazole synthesis via a formal (4+2) cycloaddition of indole-derived bromides and alkynes

(2016) Zhi-Guang Yuan et al.   CHEMICAL COMMUNICATIONS

Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas

(2016) Yu Zhou et al.   CHEMICAL REVIEWS

Visible-Light-Driven Photocatalytic Activation of Inert Sulfur Ylides for 3-Acyl Oxindole Synthesis

(2016) Xu-Dong Xia et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of indol-3-yl aryl ketones through visible-light-mediated carbonylation

(2016) Hong-Tao Zhang et al.   CHINESE CHEMICAL LETTERS

Oxindole: A chemical prism carrying plethora of therapeutic benefits

(2016) Maninder Kaur et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Combining enzyme and photoredox catalysis for aminoalkylation of indoles via a relay catalysis strategy in one pot

(2016) Yan-Hong He et al.   GREEN CHEMISTRY

Synthesis of 3-Fluoroindoles via Photoredox Catalysis

(2016) Liubov I. Panferova et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible-Light-Promoted (Phenylsulfonyl)methylation of Electron-Rich Heteroarenes and N-Arylacrylamides

(2016) Fei Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Assembly of 3-Sulfenylbenzofurans and 3-Sulfenylindoles by Palladium-Catalyzed Cascade Annulation/Arylthiolation Reaction

(2016) Jianxiao Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Oxidative Sulfenylation of Indoles and Related Electron-Rich Heteroarenes with Aryl Boronic Acids and Elemental Sulfur

(2016) Jianxiao Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Photoredox Catalysis in Organic Chemistry

(2016) Megan H. Shaw et al.   JOURNAL OF ORGANIC CHEMISTRY

Radical Smiles Rearrangement: An Update

(2016) Ingrid Allart-Simon et al.   MOLECULES

Brønsted acid cocatalysis in photocatalytic intramolecular coupling of tertiary amines: efficient synthesis of 2-arylindols

(2016) Xiaoqian Yuan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Tryptanthrins by Organocatalytic and Substrate Co-catalyzed Photochemical Condensation of Indoles and Anthranilic Acids with Visible Light and O2

(2016) Xiangmin Li et al.   ORGANIC LETTERS

Intermolecular Photocatalytic C–H Functionalization of Electron-Rich Heterocycles with Tertiary Alkyl Halides

(2016) Corey Stephenson et al.   SYNLETT

Review of synthesis and various biological activities of spiro heterocyclic compounds comprising oxindole and pyrrolidine moities

(2016) Pankaj Saraswat et al.   SYNTHETIC COMMUNICATIONS

Visible light-induced carbonylation of indoles with arylsulfonyl chlorides and CO

(2016) Xiangguang Li et al.   TETRAHEDRON

Recent advances on the synthesis of acylindoles

(2016) Shun-Jiang Yao et al.   TETRAHEDRON LETTERS

Visible-light-induced aerobic thiocyanation of indoles using reusable TiO2/MoS2 nanocomposite photocatalyst

(2016) Liang Wang et al.   TETRAHEDRON LETTERS

Discovery and mechanistic study of a photocatalytic indoline dehydrogenation for the synthesis of elbasvir

(2016) Hatice G. Yayla et al.   Chemical Science

Organic Synthesis Enabled by Light-Irradiation of EDA Complexes: Theoretical Background and Synthetic Applications

(2016) Carolina G. S. Lima et al.   ACS Catalysis

An Oxidant-Free Strategy for Indole Synthesis via Intramolecular C–C Bond Construction under Visible Light Irradiation: Cross-Coupling Hydrogen Evolution Reaction

(2016) Cheng-Juan Wu et al.   ACS Catalysis

Visible Light Photocatalytic Aerobic Oxygenation of Indoles and pH as a Chemoselective Switch

(2016) Chenhao Zhang et al.   ACS Catalysis

Synthesis Of Biologically Active Bis(Indolyl)Methane Derivatives by Bisindole Alkylation of Tetrahydroisoquinolines with Visible-Light Induced Ring-Opening Fragmentation.

(2016) Chia-Chueng Chen et al.   Asian Journal of Organic Chemistry

Amine Functionalization via Oxidative Photoredox Catalysis: Methodology Development and Complex Molecule Synthesis

(2015) Joel W. Beatty et al.   ACCOUNTS OF CHEMICAL RESEARCH

Photoinduced Copper-Catalyzed Regioselective Synthesis of Indoles: Three-Component Coupling of Arylamines, Terminal Alkynes, and Quinones

(2015) Arunachalam Sagadevan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible light induced cyclopropanation of dibromomalonates with alkenes via double-SET by photoredox catalysis

(2015) Yanbin Zhang et al.   CHEMICAL COMMUNICATIONS

Visible-Light-Induced Direct Photocatalytic Carboxylation of Indoles with CBr4/MeOH

(2015) Qing-Qing Yang et al.   CHEMISTRY-A EUROPEAN JOURNAL

NickelN-Heterocyclic Carbene Catalyzed CC Bond Formation: A New Route to Aryl Ketones

(2015) Li-Jun Gu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Iridium(III) Photocatalysis: A Visible-Light-Induced Dearomatizative Tandem [4+2] Cyclization to Furnish Benzindolizidines

(2015) Sandra Mühmel et al.   CHEMISTRY-A EUROPEAN JOURNAL

Acylation of (Hetero)Arenes through CH Activation with Aroyl Surrogates

(2015) Xiao-Feng Wu   CHEMISTRY-A EUROPEAN JOURNAL

A review on recent developments of indole-containing antiviral agents

(2015) Ming-Zhi Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Applications of Fluorine in Medicinal Chemistry

(2015) Eric P. Gillis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Visible Light Mediated Organocatalytic Activation of Ethyl Bromofluoroacetate: Coupling with Indoles and Anilines

(2015) Santosh D. Jadhav et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Regioselective Indoline Synthesis under Nickel/Photoredox Dual Catalysis

(2015) Sarah Z. Tasker et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indole Alkaloids from Catharanthus roseus: Bioproduction and Their Effect on Human Health

(2015) Lorena Almagro et al.   MOLECULES

Ylide formal [4 + 1] annulation

(2015) Chunyin Zhu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Indole Functionalization via Photoredox Gold Catalysis

(2015) Sherif J. Kaldas et al.   ORGANIC LETTERS

Bis(indolyl)methane Alkaloids: Isolation, Bioactivity, and Syntheses

(2015) P. Parameswaran et al.   SYNTHESIS-STUTTGART

Photoredox catalyst-mediated direct regioselective phosphonylation of indoles

(2015) Zijian Zhao et al.   SYNTHETIC COMMUNICATIONS

Efficient synthetic route to bisaryl ketones via copper-catalyzed C–C triple bonds cleavage

(2015) Xiangguang Li et al.   TETRAHEDRON

Catalytic Methods for Aromatic C–H Amination: An Ideal Strategy for Nitrogen-Based Functional Molecules

(2015) Jiao Jiao et al.   ACS Catalysis

Electroluminescence and fluorescence response towards acid vapors depending on the structures of indole-fused phospholes

(2015) Peng Gong et al.   RSC Advances

Transition-Metal-Catalyzed Asymmetric Allylic Dearomatization Reactions

(2014) Chun-Xiang Zhuo et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of 2-Substituted Indoles through Visible Light-Induced Photocatalytic Cyclizations of Styryl Azides

(2014) Xu-Dong Xia et al.   ADVANCED SYNTHESIS & CATALYSIS

A Cascade Cross-Coupling andin SituHydrogenation Reaction by Visible Light Catalysis

(2014) Jian-Ji Zhong et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Bis(heteroaryl) Ketones by Removal of Benzylic CHR and CO Groups

(2014) Arun Maji et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Indoles Using Visible Light: Photoredox Catalysis for Palladium-Catalyzed CH Activation

(2014) Jochen Zoller et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

X-Ray Characterization of an Electron Donor-Acceptor Complex that Drives the Photochemical Alkylation of Indoles

(2014) Sandeep R. Kandukuri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Phototandem Catalysis: Efficient Synthesis of 3-Ester-3-hydroxy-2-oxindoles by a Visible Light-Induced Cyclization of Diazoamides through an Aerobic Oxidation Sequence

(2014) Xu-Dong Xia et al.   Chemistry-An Asian Journal

Optimization of Chemical Functionalities of Indole-2-carboxamides To Improve Allosteric Parameters for the Cannabinoid Receptor 1 (CB1)

(2014) Leepakshi Khurana et al.   JOURNAL OF MEDICINAL CHEMISTRY

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

Asymmetric Synthesis of Cyclic Indole Aminals via 1,3-Stereoinduction

(2014) Hongmei Li et al.   JOURNAL OF ORGANIC CHEMISTRY

In Situ Generation of Palladium Nanoparticles: Ligand-Free Palladium Catalyzed Pivalic Acid Assisted Carbonylative Suzuki Reactions at Ambient Conditions

(2014) Qing Zhou et al.   JOURNAL OF ORGANIC CHEMISTRY

A Visible-Light-Promoted Aerobic Metal-Free C-3 Thiocyanation of Indoles

(2014) Weigang Fan et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 3-Acylindoles by Visible-Light Induced Intramolecular Oxidative Cyclization of o-Alkynylated N,N-Dialkylamines

(2014) Ping Zhang et al.   ORGANIC LETTERS

Enantioselective Synthesis of an HCV NS5a Antagonist

(2014) Ian K. Mangion et al.   ORGANIC LETTERS

Cross-Coupling Hydrogen Evolution Reaction in Homogeneous Solution without Noble Metals

(2014) Jian-Ji Zhong et al.   ORGANIC LETTERS

Cytotoxic 7S-oxindole alkaloids from Gardneria multiflora

(2014) Xiu-Hong Zhong et al.   Phytochemistry Letters

Photocatalytic aerobic oxidation/semipinacol rearrangement sequence: a concise route to the core of pseudoindoxyl alkaloids

(2014) Wei Ding et al.   TETRAHEDRON LETTERS

Aerobic Transition-Metal-Free Visible-Light Photoredox Indole C-3 Formylation Reaction

(2014) Xiang Li et al.   ACS Catalysis

Antithyroid Drugs and Their Analogues: Synthesis, Structure, and Mechanism of Action

(2013) Debasish Manna et al.   ACCOUNTS OF CHEMICAL RESEARCH

Homogeneous Visible-Light Photoredox Catalysis

(2013) You-Quan Zou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A room temperature decarboxylation/C–H functionalization cascade by visible-light photoredox catalysis

(2013) Jin Xie et al.   CHEMICAL COMMUNICATIONS

Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

(2013) Jiang Wang et al.   CHEMICAL REVIEWS

A Highly Efficient and Selective Aerobic Cross-Dehydrogenative-Coupling Reaction Photocatalyzed by a Platinum(II) Terpyridyl Complex

(2013) Jian-Ji Zhong et al.   CHEMISTRY-A EUROPEAN JOURNAL

Visible-Light-Induced Trifluoromethylation ofN-Aryl Acrylamides: A Convenient and Effective Method To Synthesize CF3-Containing Oxindoles Bearing a Quaternary Carbon Center

(2013) Pan Xu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Low toxicity and unprecedented anti-osteoclast activity of a simple sulfur-containing gem-bisphosphonate: A comparative study

(2013) Donatella Granchi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of 3,3-Disubstituted Oxindoles by Visible-Light-Mediated Radical Reactions of Aryl Diazonium Salts with N-Arylacrylamides

(2013) Weijun Fu et al.   JOURNAL OF ORGANIC CHEMISTRY

Solvent-Controlled Halo-Selective Selenylation of Aryl Halides Catalyzed by Cu(II) Supported on Al2O3. A General Protocol for the Synthesis of Unsymmetrical Organo Mono- and Bis-Selenides

(2013) Tanmay Chatterjee et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent Developments in the Catalytic, Asymmetric Construction of Pyrroloindolines Bearing All-Carbon Quaternary Stereocenters

(2013) Lindsay M. Repka et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis of Ellipticine Quinones, Olivacine, and Calothrixin B

(2013) Nagarajan Ramkumar et al.   JOURNAL OF ORGANIC CHEMISTRY

The Akuammiline Alkaloids; Origin and Synthesis

(2013) Tanja Gaich et al.   SYNTHESIS-STUTTGART

Catalytic hydrotrifluoromethylation of styrenes and unactivated aliphatic alkenes via an organic photoredox system

(2013) Dale J. Wilger et al.   Chemical Science

A Visible-Light-Mediated Oxidative CN Bond Formation/Aromatization Cascade: Photocatalytic Preparation of N-Arylindoles

(2012) Soumitra Maity et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible-Light Photoredox Catalysis

(2012) Jun Xuan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible-Light-Induced Photocatalytic Reductive Transformations of Organohalides

(2012) Hyejin Kim et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible-Light Photoredox Catalysis in Flow

(2012) Joseph W. Tucker et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible light-induced 3-sulfenylation of N-methylindoles with arylsulfonyl chlorides

(2012) Min Chen et al.   CHEMICAL COMMUNICATIONS

Photoredox functionalization of C–H bonds adjacent to a nitrogen atom

(2012) Lei Shi et al.   CHEMICAL SOCIETY REVIEWS

Double Axially Chiral Bisphosphorylimides Catalyzed Highly Enantioselective and Efficient Friedel-Crafts Reaction of Indoles with Imines

(2012) Kun Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Total Synthesis and Evaluation of Vinblastine Analogues Containing Systematic Deep-Seated Modifications in the Vindoline Subunit Ring System: Core Redesign

(2012) Kristin D. Schleicher et al.   JOURNAL OF MEDICINAL CHEMISTRY

Friedel–Crafts Amidoalkylation via Thermolysis and Oxidative Photocatalysis

(2012) Chunhui Dai et al.   JOURNAL OF ORGANIC CHEMISTRY

Direct α-Arylation of α-Amino Carbonyl Compounds with Indoles Using Visible Light Photoredox Catalysis

(2012) Zhi-Qiang Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Pentanidium–Catalyzed Enantioselective α-Hydroxylation of Oxindoles Using Molecular Oxygen

(2012) Yuanyong Yang et al.   ORGANIC LETTERS

Transition-Metal-Catalyzed Synthesis of Aromatic Ketones via Direct C-H Bond Activation

(2012) Jiang Cheng et al.   SYNTHESIS-STUTTGART

Visible light induced intermolecular [2+2]-cycloaddition reactions of 3-ylideneoxindoles through energy transfer pathway

(2012) You-Quan Zou et al.   TETRAHEDRON

Trifluoromethylation of heterocycles via visible light photoredox catalysis

(2012) Naeem Iqbal et al.   TETRAHEDRON LETTERS

Radical-Mediated Enzymatic Methylation: A Tale of Two SAMS

(2011) Qi Zhang et al.   ACCOUNTS OF CHEMICAL RESEARCH

Trifluoromethylation of arenes and heteroarenes by means of photoredox catalysis

(2011) David A. Nagib et al.   NATURE

Indole synthesis: a review and proposed classification

(2011) Douglass F. Taber et al.   TETRAHEDRON

Divergent reactions of indoles with aminobenzaldehydes: indole ring-opening vs. annulation and facile synthesis of neocryptolepine

(2011) Matthew K. Vecchione et al.   Chemical Science

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Visible light photoredox catalysis: applications in organic synthesis

(2010) Jagan M. R. Narayanam et al.   CHEMICAL SOCIETY REVIEWS

Antimicrobial Activity of Tryptanthrins inEscherichia coli

(2010) Pooja P. Bandekar et al.   JOURNAL OF MEDICINAL CHEMISTRY

SPINOL-Derived Phosphoric Acids: Synthesis and Application in Enantioselective Friedel−Crafts Reaction of Indoles with Imines

(2010) Fangxi Xu et al.   JOURNAL OF ORGANIC CHEMISTRY

Memory of Axial Chirality in Aryl Radical Phosphanylations

(2010) Achim Bruch et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Visible light photocatalysis as a greener approach to photochemical synthesis

(2010) Tehshik P. Yoon et al.   Nature Chemistry

Visible Light-Mediated Intermolecular C−H Functionalization of Electron-Rich Heterocycles with Malonates

(2010) Laura Furst et al.   ORGANIC LETTERS

Hydrogen Evolution Catalyzed by Cobaloximes

(2009) Jillian L. Dempsey et al.   ACCOUNTS OF CHEMICAL RESEARCH

Stereoselective Palladium-Catalyzed Carboaminoxylations of Indoles with Arylboronic Acids and TEMPO

(2009) Sylvia Kirchberg et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Bis- and Trisindolylmethanes (BIMs and TIMs)†

(2009) Morteza Shiri et al.   CHEMICAL REVIEWS

Electron-Transfer Photoredox Catalysis: Development of a Tin-Free Reductive Dehalogenation Reaction

(2009) Jagan M. R. Narayanam et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Making Hydrogen from Water Using a Homogeneous System Without Noble Metals

(2009) Theodore Lazarides et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Simple indole alkaloids and those with a nonrearranged monoterpenoid unit

(2009) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

An Efficient One-Step Synthesis of Heterobiaryl Pyrazolo[3,4-b]pyridines via Indole Ring Opening

(2009) Sanghee Lee et al.   ORGANIC LETTERS

Electron Transfer Photoredox Catalysis: Intramolecular Radical Addition to Indoles and Pyrroles

(2009) Joseph W. Tucker et al.   ORGANIC LETTERS

Radicals in organic synthesis. Part 1

(2009) Gareth J. Rowlands   TETRAHEDRON

Ylide-Initiated Michael Addition−Cyclization Reactions beyond Cyclopropanes

(2008) Xiu-Li Sun et al.   ACCOUNTS OF CHEMICAL RESEARCH

Cross-Dehydrogenative Coupling (CDC): Exploring C−C Bond Formations beyond Functional Group Transformations

(2008) Chao-Jun Li   ACCOUNTS OF CHEMICAL RESEARCH

Chemodivergence in Enantioselective Desymmetrization of Diazabicycles: Ring-Opening versus Reductive Arylation

(2008) Frederic Menard et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organic Reactions of Ionic Intermediates Promoted by Atmospheric-Pressure Thermal Activation

(2008) Hao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A truce on the Smiles rearrangement: revisiting an old reaction—the Truce–Smiles rearrangement

(2008) Timothy J. Snape   CHEMICAL SOCIETY REVIEWS

Arbidol: A Broad-Spectrum Antiviral Compound that Blocks Viral Fusion

(2008) Y. Boriskin et al.   CURRENT MEDICINAL CHEMISTRY

Codrugs Linkingl-Dopa and Sulfur-Containing Antioxidants: New Pharmacological Tools against Parkinson’s Disease

(2008) Francesco Pinnen et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Homogeneous System for the Photogeneration of Hydrogen from Water Based on a Platinum(II) Terpyridyl Acetylide Chromophore and a Molecular Cobalt Catalyst

(2008) Pingwu Du et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Efficient Visible Light Photocatalysis of [2+2] Enone Cycloadditions

(2008) Michael A. Ischay et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Microwave-Assisted Palladium-Catalyzed Cross-Coupling of Aryl and Vinyl Halides with H-Phosphonate Diesters

(2008) Marcin Kalek et al.   ORGANIC LETTERS

Catalytic Asymmetric Hydroxylation of Oxindoles by Molecular Oxygen Using a Phase-Transfer Catalyst

(2008) Daisuke Sano et al.   ORGANIC LETTERS

Merging Photoredox Catalysis with Organocatalysis: The Direct Asymmetric Alkylation of Aldehydes

(2008) D. A. Nicewicz et al.   SCIENCE

Understanding organofluorine chemistry. An introduction to the C–F bond

(2007) David O'Hagan   CHEMICAL SOCIETY REVIEWS