Chiral Fused 1,2,3‐Triazoles: A Synthetic Overview

Enantioselective Access to Chiral Cyclic Sulfamidates Through Iridium-Catalyzed Asymmetric Hydrogenation

(2019) Yuanhua Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Bestmann-Ohira Reagent: A Convenient and Promising Reagent in the Chemical World

(2018) Manoj Dhameja et al.   Asian Journal of Organic Chemistry

Aziridine Ring Opening: An Overview of Sustainable Methods

(2018) Shekh Sabir et al.   ChemistrySelect

Recent advances in click chemistry reactions mediated by transition metal based systems

(2017) Aurel Tăbăcaru et al.   INORGANICA CHIMICA ACTA

A Dipolar Cycloaddition Reaction To Access 6-Methyl-4,5,6,7-tetrahydro-1H-[1,2,3]triazolo[4,5-c]pyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate

(2017) Christa C. Chrovian et al.   JOURNAL OF MEDICINAL CHEMISTRY

gem-Disubstituent Effect in Rate Acceleration of Intramolecular Alkyne-Azide Cycloaddition Reaction

(2017) Shrawan R. Chavan et al.   TETRAHEDRON

A single-step acid catalyzed reaction for rapid assembly of NH-1,2,3-triazoles

(2016) Joice Thomas et al.   CHEMICAL COMMUNICATIONS

A general metal-free route towards the synthesis of 1,2,3-triazoles from readily available primary amines and ketones

(2016) Joice Thomas et al.   CHEMICAL COMMUNICATIONS

Cu-Catalyzed Click Reaction in Carbohydrate Chemistry

(2016) Vinod K. Tiwari et al.   CHEMICAL REVIEWS

Metal-catalyzed azide-alkyne “click” reactions: Mechanistic overview and recent trends

(2016) Changlong Wang et al.   COORDINATION CHEMISTRY REVIEWS

A One-Pot Procedure for the Synthesis of “Click-Ready” Triazoles from Ketones

(2016) Sampad Jana et al.   JOURNAL OF ORGANIC CHEMISTRY

Advances of azide-alkyne cycloaddition-click chemistry over the recent decade

(2016) Maya Shankar Singh et al.   TETRAHEDRON

Triazole: A Promising Antitubercular Agent

(2015) Rangappa S. Keri et al.   Chemical Biology & Drug Design

New click-chemistry methods for 1,2,3-triazoles synthesis: recent advances and applications

(2015) Jane Totobenazara et al.   TETRAHEDRON LETTERS

Synthesis of triazole-fused tetracyclic glycosides in aqueous medium: application of nanodomain cubic cuprous oxide as reusable catalyst in one-pot domino Sonogashira-cyclization

(2015) Nivedita Chatterjee et al.   TETRAHEDRON LETTERS

Metal free synthesis of morpholine fused [5,1-c] triazolyl glycoconjugates via glycosyl azido alcohols

(2015) Kunj B. Mishra et al.   RSC Advances

Efficient Atropodiastereoselective Access to 5,5′-Bis-1,2,3-triazoles: Studies on 1-Glucosylated 5-Halogeno 1,2,3-Triazoles and Their 5-Substituted Derivatives as Glycogen Phosphorylase Inhibitors

(2014) David Goyard et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and Antiviral Properties of Spirocyclic [1,2,3]-Triazolooxazine Nucleosides

(2014) Antonio Dell'Isola et al.   CHEMISTRY-A EUROPEAN JOURNAL

Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?

(2014) Alberto Massarotti et al.   ChemMedChem

Stereoselective Synthesis of 1,2,3-Triazolooxazine and Fused 1,2,3-Triazolo-δ-Lactone Derivatives

(2014) Ayşegül Gümüş et al.   HELVETICA CHIMICA ACTA

Novel effective dye sorbents: synthesis and properties of 1,2,3-triazole-modified thiacalix[4]arene polymers based on click chemistry

(2014) Jianbin Lai et al.   IRANIAN POLYMER JOURNAL

Click Chemistry Inspired Synthesis of Morpholine-Fused Triazoles

(2014) Kunj B. Mishra et al.   JOURNAL OF ORGANIC CHEMISTRY

Design, synthesis and biological evaluation of bicyclic iminosugar hybrids: conformational constraint as an effective tool for tailoring the selectivity of α-glucosidase inhibitors

(2014) Inderpreet Arora et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Efficient synthesis of conformationally constrained, amino-triazoloazepinone-containing di- and tripeptides via a one-pot Ugi–Huisgen tandem reaction

(2014) T. M. A. Barlow et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of l-rhamnose derived chiral bicyclic triazoles as novel sodium-glucose transporter (SGLT) inhibitors

(2014) Siddamal Reddy Putapatri et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A rapid entry to amino acid derived diverse 3,4-dihydropyrazines and dihydro[1,2,3]triazolo[1,5-a]pyrazines through 1,3-dipolar cycloaddition

(2014) Saurav Bera et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

I2/TBPB Mediated Oxidative Reaction of N-Tosylhydrazones with Anilines: Practical Construction of 1,4-Disubstituted 1,2,3-Triazoles under Metal-Free and Azide-Free Conditions

(2014) Zhong-Jian Cai et al.   ORGANIC LETTERS

Applications of Allenylsilanes in Organic Synthesis

(2014) Sharada Swain   SYNLETT

Click chemistry route to tricyclic monosaccharide triazole hybrids: design and synthesis of substituted hexahydro-4H-pyrano[2,3-f][1,2,3]triazolo[5,1-c][1,4]oxazepines

(2014) Saidulu Konda et al.   RSC Advances

Synthesis of C-spiro-glycoconjugates from sugar lactones via zinc mediated Barbier reaction

(2014) Mallikharjuna Rao Lambu et al.   RSC Advances

1,2,3-Triazoles as Amide Bond Mimics: Triazole Scan Yields Protease-Resistant Peptidomimetics for Tumor Targeting

(2013) Ibai E. Valverde et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The “Click” Reaction Involving Metal Azides, Metal Alkynes, or Both: An Exploration into Multimetal Structures

(2013) Luis Casarrubios et al.   CHEMISTRY-A EUROPEAN JOURNAL

Traceless Tosylhydrazone-Based Triazole Formation: A Metal-Free Alternative to Strain-Promoted Azide-Alkyne Cycloaddition

(2012) Sander S. van Berkel et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design and Synthesis of 1,2,3-Triazole-Fused Chiral Medium-Ring Benzo-Heterocycles, Scaffolds Mimicking Benzolactams

(2012) Nirmal Das Adhikary et al.   JOURNAL OF ORGANIC CHEMISTRY

Fused ring aziridines as a facile entry into triazole fused tricyclic and bicyclic heterocycles

(2012) Fang Fang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A One-Pot–Three-Step Route to Triazolotriazepinoindazolones from Oxazolino-2H-indazoles

(2012) Wayne E. Conrad et al.   ORGANIC LETTERS

Intramolecular Huisgen [3+2] cycloaddition in water: synthesis of fused pyrrolidine–triazoles

(2012) Indresh Kumar et al.   TETRAHEDRON-ASYMMETRY

Synthesis of quinoline coupled [1,2,3]-triazoles as a promising class of anti-tuberculosis agents

(2011) K. Karthik Kumar et al.   CARBOHYDRATE RESEARCH

10 Years of Click Chemistry: Synthesis and Applications of Ferrocene-Derived Triazoles

(2011) Venkataraman Ganesh et al.   Chemistry-An Asian Journal

Click Chemistry: 1,2,3-Triazoles as Pharmacophores

(2011) Sandip G. Agalave et al.   Chemistry-An Asian Journal

Triphenylamine-based organic dyes containing a 1,2,3-triazole bridge for dye-sensitized solar cells via a ‘Click’ reaction

(2011) Tainan Duan et al.   DYES AND PIGMENTS

Ceric Ammonium Nitrate-Catalyzed Azidation of 1,2-Anhydro Sugars: Application in the Synthesis of Structurally Diverse Sugar-Derived Morpholine 1,2,3-Triazoles and 1,4-Oxazin-2-ones

(2011) Y. Suman Reddy et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Free Intramolecular Alkyne–Azide Cycloadditions Leading to Seven-Membered Heterocycles

(2011) Míriam Sau et al.   ORGANIC LETTERS

Amino Triazolo Diazepines (Ata) as Constrained Histidine Mimics

(2011) Koen Buysse et al.   ORGANIC LETTERS

Synthesis of 1,2,3-Triazole-Fused Heterocycles via Intramolecular Azide-Alkyne Cycloaddition Reactions

(2011) Krishna Majumdar et al.   SYNTHESIS-STUTTGART

Synthesis and antitumor activity of novel 2′,3′-diethanethio-2′,3′,5′-trideoxy-5′-triazolonucleoside analogues

(2010) Jin-Lan Yu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pharmacological significance of triazole scaffold

(2010) Rajeev Kharb et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Click chemistry and biocatalysis for the preparation of pancratistatin analogs

(2010) Victoria de la Sovera et al.   TETRAHEDRON LETTERS

Synthesis of hybrid 1,2,3-triazolo-δ-lactams/lactones using Huisgen [3+2] cycloaddition ‘click-chemistry’ in water

(2010) Indresh Kumar et al.   TETRAHEDRON-ASYMMETRY

Click chemistry based rapid one-pot synthesis and evaluation for protease inhibition of new tetracyclic triazole fused benzodiazepine derivatives

(2009) Debendra K. Mohapatra et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and antitumor activity of novel 2′,3′-dideoxy-2′,3′-diethanethionucleosides bearing 1,2,3-triazole residues

(2009) Jin-Lan Yu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

One pot synthesis and SAR of some novel 3-substituted 5,6-diphenyl-1,2,4-triazines as antifungal agents

(2009) Jaiprakash N. Sangshetti et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and antibacterial activity of novel 5-(4-methyl-1H-1,2,3-triazole) methyl oxazolidinones

(2009) Oludotun A. Phillips et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Facile Entry into Triazole Fused Heterocycles via Sulfamidate Derived Azido-alkynes

(2009) V. Sai Sudhir et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular azide-alkyne [3 + 2] cycloaddition: versatile route to new heterocyclic structural scaffolds

(2009) Rongti Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Regioselective Intramolecular Dipolar Cycloaddition of Azides and Unsymmetrical Alkynes

(2009) Ryan A. Brawn et al.   ORGANIC LETTERS

Preparation and reactions of sugar azides with alkynes: synthesis of sugar triazoles as antitubercular agents

(2008) Biswajit Kumar Singh et al.   CARBOHYDRATE RESEARCH

Condensed 1,2,3-triazoles (review)

(2008) E. A. Shafran et al.   Chemistry of Heterocyclic Compounds

Facile Entry to 4,5,6,7-Tetrahydro[1,2,3]triazolo[1,5-a]pyrazin-6-ones from Amines and Amino Acids

(2008) V. Sai Sudhir et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An efficient synthesis of triazolo-carbohydrate mimetics and their conformational analysis

(2008) Hikaru Yanai et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of 1,2,3-triazole and 1,2,3,4-tetrazole-fused glycosides and nucleosides by an intramolecular 1,3-dipolar cycloaddition reaction

(2008) Ramakrishna I. Anegundi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Intramolecular Azide−Alkyne Cycloaddition for the Fast Assembly of Structurally Diverse, Tricyclic 1,2,3-Triazoles

(2008) Ana I. Oliva et al.   ORGANIC LETTERS

Synthesis of novel oxazolidinone antimicrobial agents

(2007) David C. Ebner et al.   BIOORGANIC & MEDICINAL CHEMISTRY