Journal
TETRAHEDRON LETTERS
Volume 56, Issue 22, Pages 2853-2859Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2015.03.136
Keywords
1,2,3-Triazoles; Click-chemistry; Metal-free cycloaddition; Regioselectivity; Amide isosters
Categories
Funding
- INMOLFARM-Molecular Innovation and Drug Discovery from FEDER-INALENTEJO program [ALENT-57-2011-20, ALENT-07-0224-FEDER-001743]
- Fundacao para a Ciencia e Tecnologia (FCT) [PEst-OE/QUI/UI0619/2014]
- Fundação para a Ciência e a Tecnologia [PEst-OE/QUI/UI0619/2014] Funding Source: FCT
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1,2,3-Triazoles find applications in several major technological areas, and especially in drug discovery. The click-chemistry approaches based on Huisgen's cycloaddition reaction are particularly attractive and have received enormous attention over the last decade and a half, due to their utility in preparing compounds with diverse applications, from drugs to linkers for bioconjugation. (C) 2015 Elsevier Ltd. All rights reserved.
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