Triazole: A Promising Antitubercular Agent

Design, synthesis and evaluation of 1,2,3-triazole-adamantylacetamide hybrids as potent inhibitors of Mycobacterium tuberculosis

(2014) Dinesh Addla et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of novel 1,2,3-triazole derivatives of isoniazid and their in vitro and in vivo antimycobacterial activity evaluation

(2014) Deepak Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Sulfur rich 2-mercaptobenzothiazole and 1,2,3-triazole conjugates as novel antitubercular agents

(2014) Fauzia Mir et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis and 3D-QSAR studies of new diphenylamine containing 1,2,4-triazoles as potential antitubercular agents

(2014) K. Mohan Krishna et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Anti-tubercular agents. Part 8: Synthesis, antibacterial and antitubercular activity of 5-nitrofuran based 1,2,3-triazoles

(2013) Ahmed Kamal et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Rational design, synthesis and antitubercular evaluation of novel 2-(trifluoromethyl)phenothiazine-[1,2,3]triazole hybrids

(2013) Dinesh Addla et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and Biological Applications of Triazole Derivatives – A Review

(2013) S. Sathish Kumar et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Design and synthesis of 1H-1,2,3-triazoles derived from econazole as antitubercular agents

(2012) Suhyun Kim et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Click Chemistry Approach for Bis-Chromenyl Triazole Hybrids and Their Antitubercular Activity

(2012) Reshma J. Naik et al.   Chemical Biology & Drug Design

Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents

(2012) Christophe Menendez et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, Synthesis, and Structure–Activity Correlations of Novel Dibenzo[b,d]furan, Dibenzo[b,d]thiophene, and N-Methylcarbazole Clubbed 1,2,3-Triazoles as Potent Inhibitors of Mycobacterium tuberculosis

(2012) Santhosh Reddy Patpi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Novel 4H-1,2,4-triazol-3-yl cycloalkanols as potent antitubercular agents

(2012) Nutan H. Palsule Desai et al.   MEDICINAL CHEMISTRY RESEARCH

Tuberculosis Pathogenesis and Immunity

(2011) Jennifer A. Philips et al.   Annual Review of Pathology-Mechanisms of Disease

Synthesis, antitubercular activity, and SAR study of N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides

(2011) Alessandro K. Jordão et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Efficient synthesis and in vitro antitubercular activity of 1,2,3-triazoles as inhibitors of Mycobacterium tuberculosis

(2011) Poovan Shanmugavelan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and preliminary biological evaluation of novel N-(3-aryl-1,2,4-triazol-5-yl) cinnamamide derivatives as potential antimycobacterial agents: An operational Topliss Tree approach

(2011) Manoj D. Kakwani et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of quinoline coupled [1,2,3]-triazoles as a promising class of anti-tuberculosis agents

(2011) K. Karthik Kumar et al.   CARBOHYDRATE RESEARCH

Mycobacterium tuberculosis and the intimate discourse of a chronic infection

(2011) David G. Russell   IMMUNOLOGICAL REVIEWS

Novel 1,2,3-Triazole Derivatives for Use againstMycobacterium tuberculosisH37Rv (ATCC 27294) Strain

(2011) Nubia Boechat et al.   JOURNAL OF MEDICINAL CHEMISTRY

Tuberculosis

(2011) Stephen D Lawn et al.   LANCET

Syntheses and biological evaluation of new triazole-spirochromone conjugates as inhibitors of Mycobacterium tuberculosis

(2011) M. Muthukrishnan et al.   TETRAHEDRON LETTERS

Antimycobacterial and antimicrobial study of new 1,2,4-triazoles with benzothiazoles

(2010) Navin B. Patel et al.   ARCHIV DER PHARMAZIE

Rip Van Winkle Wakes Up: Development of Tuberculosis Treatment in the 21st Century

(2010) William J. Burman   CLINICAL INFECTIOUS DISEASES

Pharmacological evaluation and characterizations of newly synthesized 1,2,4-triazoles

(2010) Navin B. Patel et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of some novel 2-substituted-5-[isopropylthiazole] clubbed 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents

(2010) G.V. Suresh Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pharmacological significance of triazole scaffold

(2010) Rajeev Kharb et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

The Population Dynamics and Control of Tuberculosis

(2010) C. Dye et al.   SCIENCE

NH-1,2,3-Triazole Inhibitors of the VIM-2 Metallo-β-Lactamase

(2010) Timo Weide et al.   ACS Medicinal Chemistry Letters

Identification of arylamine N-acetyltransferase inhibitors as an approach towards novel anti-tuberculars

(2010) Isaac M. Westwood et al.   Protein & Cell

The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophore

(2009) Brian A. Johns et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis

(2009) Daniele Castagnolo et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Extensively drug-resistant tuberculosis

(2009) Philip LoBue   CURRENT OPINION IN INFECTIOUS DISEASES

Identification of a Metabolically Stable Triazolopyrimidine-Based Dihydroorotate Dehydrogenase Inhibitor with Antimalarial Activity in Mice

(2009) Ramesh Gujjar et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and evaluation of analgesic, anti-inflammatory and ulcerogenic activities of some triazolo- and 2-pyrazolyl-pyrido[2,3-d]-pyrimidines

(2008) Hend Hafez et al.   ACTA PHARMACEUTICA

Preparation and reactions of sugar azides with alkynes: synthesis of sugar triazoles as antitubercular agents

(2008) Biswajit Kumar Singh et al.   CARBOHYDRATE RESEARCH

SAR study of clubbed [1,2,4]-triazolyl with fluorobenzimidazoles as antimicrobial and antituberculosis agents

(2008) Ganesh Rajaram Jadhav et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY