Efficient Atropodiastereoselective Access to 5,5′-Bis-1,2,3-triazoles: Studies on 1-Glucosylated 5-Halogeno 1,2,3-Triazoles and Their 5-Substituted Derivatives as Glycogen Phosphorylase Inhibitors

Click Chemistry for Drug Development and Diverse Chemical–Biology Applications

(2013) Prakasam Thirumurugan et al.   CHEMICAL REVIEWS

Direct Evidence of a Dinuclear Copper Intermediate in Cu(I)-Catalyzed Azide-Alkyne Cycloadditions

(2013) B. T. Worrell et al.   SCIENCE

Controllable synthesis of bis(1,2,3-triazole)s and 5-alkynyl-triazoles via temperature effect on copper-catalyzed Huisgen cycloaddition

(2013) Lingjun Li et al.   TETRAHEDRON

Synthesis of 5-halogenated 1,2,3-triazoles under stoichiometric Cu(I)-mediated azide–alkyne cycloaddition (CuAAC or ‘Click Chemistry’)

(2012) David Goyard et al.   CARBOHYDRATE RESEARCH

Synthesis of 1,2,3-triazoles from xylosyl and 5-thioxylosyl azides: evaluation of the xylose scaffold for the design of potential glycogen phosphorylase inhibitors

(2012) David Goyard et al.   CARBOHYDRATE RESEARCH

Copper-Catalyzed Huisgen and Oxidative Huisgen Coupling Reactions Controlled by Polysiloxane-Supported Amines (AFPs) for the Divergent Synthesis of Triazoles and Bistriazoles

(2012) Zhan-Jiang Zheng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Chemical Synthesis ofN-Aryl Glycosides

(2012) Marina Y. Fosso et al.   JOURNAL OF CARBOHYDRATE CHEMISTRY

A One-Pot Three-Component Radiochemical Reaction for Rapid Assembly of 125I-Labeled Molecular Probes

(2012) Ran Yan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Inhibition of Glycogen Phosphorylase in the Context of Type 2 Diabetes, with Focus on Recent Inhibitors Bound at the Active Site

(2012) J.-P. Praly et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

DNA glycoclusters and DNA-based carbohydrate microarrays: From design to applications

(2012) François Morvan et al.   RSC Advances

Reliable and Efficient Procedures for the Conjugation of Biomolecules through Huisgen Azide-Alkyne Cycloadditions

(2011) Enrique Lallana et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Facile synthesis of 1,2,3-triazole analogs of SGLT2 inhibitors by ‘click chemistry’

(2011) Lan-Tao Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent applications of thiol–ene coupling as a click process for glycoconjugation

(2011) Alessandro Dondoni et al.   CHEMICAL SOCIETY REVIEWS

Microwave-assisted construction of triazole-linked amino acid–glucoside conjugates as novel PTP1B inhibitors

(2011) Xiao-Peng He et al.   NEW JOURNAL OF CHEMISTRY

Assessing the whole range of CuAAC mechanisms by DFT calculations—on the intermediacy of copper acetylides

(2011) David Cantillo et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Fusing Triazoles: Toward Extending Aromaticity

(2011) Michal Juríček et al.   ORGANIC LETTERS

Synthesis of 5-Iodo-1,2,3-triazole-Containing Macrocycles Using Copper Flow Reactor Technology

(2011) Andrew R. Bogdan et al.   ORGANIC LETTERS

Effect of temperature on triazole and bistriazole formation through copper-catalyzed alkyne–azide cycloaddition

(2011) Jaime González et al.   TETRAHEDRON LETTERS

Mechanistic Insights into Copper(I)-Catalyzed Azide-Alkyne Cycloadditions using Continuous Flow Conditions

(2010) Michael Fuchs et al.   ADVANCED SYNTHESIS & CATALYSIS

Preparation of triazole-linked glycosylated α-ketocarboxylic acid derivatives as new PTP1B inhibitors

(2010) Zhuo Song et al.   CARBOHYDRATE RESEARCH

Alkynylcopper(i) polymers and their use in a mechanistic study of alkyne–azide click reactions

(2010) Benjamin R. Buckley et al.   CHEMICAL COMMUNICATIONS

Atroposelective Total Synthesis of Axially Chiral Biaryl Natural Products

(2010) Gerhard Bringmann et al.   CHEMICAL REVIEWS

Copper-catalyzed azide–alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(i) acetylides

(2010) Jason E. Hein et al.   CHEMICAL SOCIETY REVIEWS

Mechanistic Insights into Cu(I)-Catalyzed Azide−Alkyne “Click” Cycloaddition Monitored by Real Time Infrared Spectroscopy

(2010) Shengtong Sun et al.   JOURNAL OF PHYSICAL CHEMISTRY A

Tailored Ligand Acceleration of the Cu-Catalyzed Azide−Alkyne Cycloaddition Reaction: Practical and Mechanistic Implications

(2010) Stanislav I. Presolski et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Azide-Alkyne Cycloaddition: Regioselective Synthesis of 1,4,5-Trisubstituted 1,2,3-Triazoles

(2009) Christian Spiteri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes

(2009) Jason E. Hein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and structure–activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase

(2009) Marietta Tóth et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis of 1-(d-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors

(2009) Éva Bokor et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Base and concentration effects on the product distribution in copper-promoted alkyne–azide cycloaddition: additive-free route to 5-iodo-triazoles

(2009) Nicholas W. Smith et al.   TETRAHEDRON LETTERS

Amide-1,2,3-triazole bioisosterism: the glycogen phosphorylase case

(2009) Evangelia D. Chrysina et al.   TETRAHEDRON-ASYMMETRY

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Short cut to 1,2,3-triazole-based p38 MAP kinase inhibitorsvia [3+2]-cycloaddition chemistry

(2008) Peter Dinér et al.   NEW JOURNAL OF CHEMISTRY