Double Cu‐Catalyzed Direct Csp 3 −H Azidation/CuAAC Reaction: A Direct Approach towards Demanding Triazole Conjugates

Recent advances in the synthesis and synthetic applications of 1,2,3-triazoles (microreview)

(2018) Shengjia Lin et al.   Chemistry of Heterocyclic Compounds

Novel Oxidative Ugi-Reaction for the Synthesis of Highly Active Visible Light Imide-Acridinium OrganoPhotocatalysts

(2018) Andrea Gini et al.   CHEMISTRY-A EUROPEAN JOURNAL

C(sp3)–H Azidation Reaction: A Protocol for Preparation of Aminals

(2018) Jianyang Dong et al.   JOURNAL OF ORGANIC CHEMISTRY

Triazole derivatives and their anti-tubercular activity

(2017) Shu Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Ir4(CO)12-Catalyzed Benzylic C(sp3)–H Silylation of 2-Alkylpyridines with Hydrosilanes Leading to 2-(1-Silylalkyl)pyridines

(2017) Yoshiya Fukumoto et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent progress in mild Csp3–H bond dehydrogenative or (mono-) oxidative functionalization

(2017) Andrea Gini et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of pyrrolo[1,2-a]quinoxalines via copper or iron-catalyzed aerobic oxidative carboamination of sp3C–H bonds

(2017) Chenshu Dai et al.   RSC Advances

Cyclic Hypervalent Iodine Reagents for Atom-Transfer Reactions: Beyond Trifluoromethylation

(2016) Yifan Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Click Chemistry Route to the Synthesis of Unusual Amino Acids, Peptides, Triazole-Fused Heterocycles and Pseudodisaccharides

(2016) Srinivasan Chandrasekaran et al.   CHEMICAL RECORD

Metal-Catalysed Azidation of Organic Molecules

(2016) Monalisa Goswami et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

1,2,3-Triazoles as Amide Bioisosteres: Discovery of a New Class of Potent HIV-1 Vif Antagonists

(2016) Idrees Mohammed et al.   JOURNAL OF MEDICINAL CHEMISTRY

Benzylic C–H Azidation Using the Zhdankin Reagent and a Copper Photoredox Catalyst

(2016) Pauline T. G. Rabet et al.   ORGANIC LETTERS

Mild Radical Oxidative sp3-Carbon–Hydrogen Functionalization: Innovative Construction of Isoxazoline and Dibenz[b,f]oxepine/azepine Derivatives

(2016) Olga Mancheño et al.   SYNLETT

Advances of azide-alkyne cycloaddition-click chemistry over the recent decade

(2016) Maya Shankar Singh et al.   TETRAHEDRON

A visible-light-promoted radical reaction system for azidation and halogenation of tertiary aliphatic C–H bonds

(2016) Yaxin Wang et al.   Chemical Science

Asymmetric Copper-Catalyzed Azide–Alkyne Cycloadditions

(2016) William D. G. Brittain et al.   ACS Catalysis

Multicomponent Syntheses based upon Copper-Catalyzed Alkyne-Azide Cycloaddition

(2015) Sidra Hassan et al.   ADVANCED SYNTHESIS & CATALYSIS

Cyclic Hypervalent Iodine Reagents and Iron Catalysts: The Winning Team for Late-Stage CH Azidation

(2015) Maria Victoria Vita et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Oxidative CH Bond Functionalization and Ring Expansion with TMSCHN2: A Copper(I)-Catalyzed Approach to Dibenzoxepines and Dibenzoazepines

(2015) Tobias Stopka et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Triazole: A Promising Antitubercular Agent

(2015) Rangappa S. Keri et al.   Chemical Biology & Drug Design

Cu-catalyzed selective cascade sp3 C–H bond oxidative functionalization towards isoxazoline derivatives

(2015) Gang-Wei Wang et al.   CHEMICAL COMMUNICATIONS

Oxidative Coupling between Two Hydrocarbons: An Update of Recent C–H Functionalizations

(2015) Chao Liu et al.   CHEMICAL REVIEWS

Metal-Free Oxidative CC Bond Formation through CH Bond Functionalization

(2015) Rishikesh Narayan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Metal-catalysed azidation of tertiary C–H bonds suitable for late-stage functionalization

(2015) Ankit Sharma et al.   NATURE

New click-chemistry methods for 1,2,3-triazoles synthesis: recent advances and applications

(2015) Jane Totobenazara et al.   TETRAHEDRON LETTERS

Taming Azide Radicals for Catalytic C–H Azidation

(2015) Xiongyi Huang et al.   ACS Catalysis

Cu-catalyzed sp3 C–H bond oxidative functionalization of alkylazaarenes and substituted ethanones: an efficient approach to isoxazoline derivatives

(2015) Gang-Wei Wang et al.   Organic Chemistry Frontiers

Copper-Catalyzed Oxidative α-Alkylation of α-Amino Carbonyl Compounds with EthersviaDual C(sp3)-H Oxidative Cross- Coupling

(2014) Wen-Ting Wei et al.   ADVANCED SYNTHESIS & CATALYSIS

1,2,3-Triazole in Heterocyclic Compounds, Endowed with Biological Activity, through 1,3-Dipolar Cycloadditions

(2014) Antonino Lauria et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Intermolecular Amidation and Imidation of Unactivated Alkanes

(2014) Ba L. Tran et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Cross-Dehydrogenative Coupling of C sp 3H Bonds: A Versatile Strategy for CC Bond Formations

(2013) Simon A. Girard et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, Synthesis and Biological Evaluation of Rose Bengal Analogues as SecA Inhibitors

(2013) Jianmei Cui et al.   ChemMedChem

Mechanistic Investigation of Oxidative Mannich Reaction with tert-Butyl Hydroperoxide. The Role of Transition Metal Salt

(2013) Maxim O. Ratnikov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct Evidence of a Dinuclear Copper Intermediate in Cu(I)-Catalyzed Azide-Alkyne Cycloadditions

(2013) B. T. Worrell et al.   SCIENCE

Hexachlorocyclohexa-2,5-dien-1-one

(2013) Zahra Tanbakouchian   SYNLETT

Expedient Synthesis of SMAMPs via Click Chemistry

(2013) Tsung-hao Fu et al.   ACS Medicinal Chemistry Letters

Copper-catalyzed ortho-acylation of phenols with aryl aldehydes and its application in one-step preparation of xanthones

(2012) Jun Hu et al.   CHEMICAL COMMUNICATIONS

Recent Researches in Triazole Compounds as Medicinal Drugs

(2012) C. -H. Zhou et al.   CURRENT MEDICINAL CHEMISTRY

A Comparative Mechanistic Study of Cu-Catalyzed Oxidative Coupling Reactions with N-Phenyltetrahydroisoquinoline

(2012) Esther Boess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chemoselective Sequential “Click” Ligation Using Unsymmetrical Bisazides

(2012) Zhao Yuan et al.   ORGANIC LETTERS

From Mechanism to Mouse: A Tale of Two Bioorthogonal Reactions

(2011) Ellen M. Sletten et al.   ACCOUNTS OF CHEMICAL RESEARCH

Click Dendrimers and Triazole-Related Aspects: Catalysts, Mechanism, Synthesis, and Functions. A Bridge between Dendritic Architectures and Nanomaterials

(2011) Didier Astruc et al.   ACCOUNTS OF CHEMICAL RESEARCH

If CH Bonds Could Talk: Selective CH Bond Oxidation

(2011) Timothy Newhouse et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design and synthesis of novel photoaffinity probes for study of the target proteins of oleanolic acid

(2011) Liying Zhang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of quinoline coupled [1,2,3]-triazoles as a promising class of anti-tuberculosis agents

(2011) K. Karthik Kumar et al.   CARBOHYDRATE RESEARCH

Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds

(2011) Charles S. Yeung et al.   CHEMICAL REVIEWS

Click Chemistry: 1,2,3-Triazoles as Pharmacophores

(2011) Sandip G. Agalave et al.   Chemistry-An Asian Journal

The copper(I)-catalyzed alkyne-azide cycloaddition (CuAAC) “click” reaction and its applications. An overview

(2011) Liyuan Liang et al.   COORDINATION CHEMISTRY REVIEWS

Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

(2011) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

Mechanistic Studies on a Cu-Catalyzed Aerobic Oxidative Coupling Reaction withN-Phenyl Tetrahydroisoquinoline: Structure of Intermediates and the Role of Methanol As a Solvent

(2011) Esther Boess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Gold-catalysed synthesis of amino acid-derived 2,5-disubstituted oxazoles

(2011) Christopher L. Paradise et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper(I) 1,2,3-Triazol-5-ylidene Complexes as Efficient Catalysts for Click Reactions of Azides with Alkynes

(2011) Tatsuhito Nakamura et al.   ORGANIC LETTERS

Synthesis of 1,2,3-Triazole-Fused Heterocycles via Intramolecular Azide-Alkyne Cycloaddition Reactions

(2011) Krishna Majumdar et al.   SYNTHESIS-STUTTGART

Well-defined copper(i) complexes for Click azide–alkyne cycloaddition reactions: one Click beyond

(2011) Silvia Díez-González   Catalysis Science & Technology

Autoxidative Carbon-Carbon Bond Formation from Carbon-Hydrogen Bonds

(2010) Áron Pintér et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One pot ‘click’ reactions: tandem enantioselective biocatalytic epoxide ring opening and [3+2] azide alkyne cycloaddition

(2010) Lachlan S. Campbell-Verduyn et al.   CHEMICAL COMMUNICATIONS

Copper-catalyzed azide–alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(i) acetylides

(2010) Jason E. Hein et al.   CHEMICAL SOCIETY REVIEWS

Copper-Catalyzed Cross Dehydrogenative Coupling Reactions of Tertiary Amines with Ketones or Indoles

(2010) Fei Yang et al.   ORGANIC LETTERS

Copper-in-Charcoal-Catalyzed, Tandem One-Pot Diazo Transfer-Click Reactions

(2009) Ching-Tien Lee et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed Azide-Alkyne Cycloaddition: Regioselective Synthesis of 1,4,5-Trisubstituted 1,2,3-Triazoles

(2009) Christian Spiteri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Cu(I)-promoted one-pot ‘SNAr–click reaction’ of fluoronitrobenzenes

(2009) Kulbhushan A. Dururgkar et al.   TETRAHEDRON

A Rational Approach towards the Nucleophilic Substitutions of Alcohols “on Water”

(2008) Pier Giorgio Cozzi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and antifungal activity of 1,2,3-triazole containing fluconazole analogues

(2008) Nilkanth G. Aher et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Copper-Catalyzed “Click” Reaction/Direct Arylation Sequence: Modular Syntheses of 1,2,3-Triazoles

(2008) Lutz Ackermann et al.   ORGANIC LETTERS

Synthesis of the Novel Chiral Catalysts by Click Chemistry and Their Application

(2008) Qian Li et al.   SYNTHETIC COMMUNICATIONS

Click chemistry reactions in medicinal chemistry: Applications of the 1,3-dipolar cycloaddition between azides and alkynes

(2007) Gian Cesare Tron et al.   MEDICINAL RESEARCH REVIEWS