Multicomponent Syntheses based upon Copper-Catalyzed Alkyne-Azide Cycloaddition

Fine-Tunable Tris(triazolyl)methane Ligands for Copper(I)- Catalyzed Azide-Alkyne Cycloaddition Reactions

(2014) Erhan Ozkal et al.   ADVANCED SYNTHESIS & CATALYSIS

Silver and gold-catalyzed multicomponent reactions

(2014) Giorgio Abbiati et al.   Beilstein Journal of Organic Chemistry

Syntheses and structure–activity relationships for some triazolyl p38α MAPK inhibitors

(2014) Jean-Paul G. Seerden et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Click chemistry approach: Regioselective one-pot synthesis of some new 8-trifluoromethylquinoline based 1,2,3-triazoles as potent antimicrobial agents

(2014) B. Garudachari et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Copper Immobilized on Nanosilica Triazine Dendrimer (Cu(II)-TD@nSiO2)-Catalyzed Regioselective Synthesis of 1,4-Disubstituted 1,2,3-Triazoles and Bis- and Tris-Triazoles via a One-Pot Multicomponent Click Reaction

(2014) Mahboobeh Nasr-Esfahani et al.   JOURNAL OF ORGANIC CHEMISTRY

One-step synthesis of poly(triazole-ether-quinoxaline)s using click reaction: preparation and properties of magnetic nanocomposites with modified Fe3O4 for metal ions removal

(2014) Mousa Ghaemy et al.   JOURNAL OF POLYMER RESEARCH

Combining a Click–Multicomponent Reaction: One-Pot Synthesis of 1,2,3-Triazol-4-ylmethyl 3-Amino-5,10-dihydro-5,10-dioxo-1H-pyrazolo[1,2-b]phthalazine-2-carboxylate Derivatives

(2014) Minoo Dabiri et al.   SYNTHETIC COMMUNICATIONS

Preparation of 1,4,5-Trisubstituted 5-Acyl-1,2,3-triazoles by Selective Acylation between Copper(I)-Carbon(sp) and Copper(I)-Carbon(sp2) Bonds with Acyl Chlorides

(2013) Bo Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper(I)-Catalyzed Cycloaddition of Bismuth(III) Acetylides with Organic Azides: Synthesis of Stable Triazole Anion Equivalents

(2013) Brady T. Worrell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Advancements in the mechanistic understanding of the copper-catalyzed azide–alkyne cycloaddition

(2013) Regina Berg et al.   Beilstein Journal of Organic Chemistry

One-pot synthesis of O-glycosyl triazoles by O-glycosylation–click reaction

(2013) Wadchara Mangsang et al.   CARBOHYDRATE RESEARCH

Coupling biocatalysis and click chemistry: one-pot two-step convergent synthesis of enantioenriched 1,2,3-triazole-derived diols

(2013) Aníbal Cuetos et al.   CHEMICAL COMMUNICATIONS

Chemicals from Alkynes with Palladium Catalysts

(2013) Rafael Chinchilla et al.   CHEMICAL REVIEWS

Facet-Dependent Catalytic Activity of Cu2O Nanocrystals in the One-Pot Synthesis of 1,2,3-Triazoles by Multicomponent Click Reactions

(2013) Kaushik Chanda et al.   CHEMISTRY-A EUROPEAN JOURNAL

Polymer anchored Cu(ii) complex: an efficient and recyclable catalytic system for the one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles starting from anilines in water

(2013) Susmita Roy et al.   GREEN CHEMISTRY

Tandem Reaction of 1-Copper(I) Alkynes for the Synthesis of 1,4,5-Trisubstituted 5-Chloro-1,2,3-triazoles

(2013) Bo Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Alkenes as Azido Precursors for the One-Pot Synthesis of 1,2,3-Triazoles Catalyzed by Copper Nanoparticles on Activated Carbon

(2013) Francisco Alonso et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of New 1,2,3-Triazole Derivatives of Uracil and Thymine with Potential Inhibitory Activity against Acidic Corrosion of Steels

(2013) Guillermo Negrón-Silva et al.   MOLECULES

Multicomponent Click Synthesis of New 1,2,3-Triazole Derivatives of Pyrimidine Nucleobases: Promising Acidic Corrosion Inhibitors for Steel

(2013) Rodrigo González-Olvera et al.   MOLECULES

One-Pot Synthesis of 3-Triazolyl-2-iminochromenes via a Catalytic Three Component Cascade Reaction

(2013) Wenyuan Qian et al.   ORGANIC LETTERS

Direct Evidence of a Dinuclear Copper Intermediate in Cu(I)-Catalyzed Azide-Alkyne Cycloadditions

(2013) B. T. Worrell et al.   SCIENCE

Efficient Multicomponent Synthesis of Mono-, Bis-, and Tris-1,2,3-triazoles Supported by Hydroxybenzene Scaffolds

(2013) Guillermo Negrón-Silva et al.   SYNTHESIS-STUTTGART

Synthesis of 5-Iodo-1,2,3-triazoles from Organic Azides and Terminal Alkynes­: Ligand Acceleration Effect, Substrate Scope, and Mechanistic Insights

(2013) Lei Zhu et al.   SYNTHESIS-STUTTGART

Simple, efficient one-pot method for synthesis of novel N-attached 1,2,3-triazole containing bisphosphonates

(2013) Xiaolan Chen et al.   TETRAHEDRON

Easy preparation of 1,4,5-trisubstituted 5-(2-alkoxy-1,2-dioxoethyl)-1,2,3-triazoles by chemoselective trapping of copper(I)–carbon bond with alkoxalyl chloride

(2013) Bo Wang et al.   TETRAHEDRON LETTERS

Three-component chemoenzymatic synthesis of amide ligated 1,2,3-triazoles

(2013) Sidra Hassan et al.   TETRAHEDRON LETTERS

One-pot esterification-click (CuAAC) and esterification–acetylene coupling (Glaser/Eglinton) for functionalization of Wang polystyrene resin

(2013) Sagi Eppel et al.   TETRAHEDRON LETTERS

One-pot three-component synthesis of indole-3-glyoxyl derivatives and indole-3-glyoxyl triazoles

(2013) Hélio A. Stefani et al.   TETRAHEDRON LETTERS

A facile one-pot five-component synthesis of glycoside annulated dihydropyrimidinone derivatives with 1,2,3-triazol linkage via transesterification/Biginelli/click reactions in aqueous medium

(2013) G.B. Dharma Rao et al.   TETRAHEDRON LETTERS

Copper-catalyzed one-pot synthesis of glycosylated iminocoumarins and 3-triazolyl-2-iminocoumarins

(2013) Pintu Kumar Mandal   RSC Advances

Macroporous polymer supported azide and nanocopper (I): efficient and reusable reagent and catalyst for multicomponent click synthesis of 1,4-disubstituted-1H-1,2,3-triazoles from benzyl halides

(2013) Mosadegh Keshavarz et al.   SpringerPlus

One-Pot Three-Component Click Reaction of Cyclic Sulfates and Cyclic Sulfamidates

(2012) Alicia Megia-Fernandez et al.   ADVANCED SYNTHESIS & CATALYSIS

High-affinity multivalent wheat germ agglutinin ligands by one-pot click reaction

(2012) Henning S G Beckmann et al.   Beilstein Journal of Organic Chemistry

Targeting heat shock factor 1 with a triazole nucleoside analog to elicit potent anticancer activity on drug-resistant pancreatic cancer

(2012) Yi Xia et al.   CANCER LETTERS

One-pot synthesis of chitosan-g-(PEO-PLLA-PEO) via “click” chemistry and “SET-NRC” reaction

(2012) Ke Zhang et al.   CARBOHYDRATE POLYMERS

Copper iodide nanoparticles on poly(4-vinyl pyridine): A new and efficient catalyst for multicomponent click synthesis of 1,4-disubstituted-1,2,3-triazoles in water

(2012) Jalal Albadi et al.   CATALYSIS COMMUNICATIONS

Multicomponent Synthesis of 1,2,3-Triazoles in Water Catalyzed by Silica-Immobilized NHC–Cu(I)

(2012) Li Wan et al.   CATALYSIS LETTERS

Stereo- and regio-selective one-pot synthesis of triazole-based unnatural amino acids and β-amino triazoles

(2012) R. B. Nasir Baig et al.   CHEMICAL COMMUNICATIONS

Advances in Copper-Catalyzed CC Coupling Reactions and Related Domino Reactions Based on Active Methylene Compounds

(2012) Yunyun Liu et al.   Chemistry-An Asian Journal

Copper iodide nanoparticles on poly(4-vinyl pyridine) as new and green catalyst for multicomponent click synthesis of 1,4-disubstituted-1,2,3-triazoles in water

(2012) Jalal Albadi et al.   CHINESE CHEMICAL LETTERS

(Iminophosphorane)copper(I) Complexes as Highly Efficient Catalysts for 1,3-Dipolar Cycloaddition of Azides with Terminal and 1-Iodoalkynes in Water: One-Pot Multi-Component Reaction from Alkynes and in situ Generated Azides

(2012) Joaquín García-Álvarez et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Solvent-free one-pot synthesis of 1,2,3-triazole derivatives by the ‘Click’ reaction of alkyl halides or aryl boronic acids, sodium azide and terminal alkynes over a Cu/Al2O3surface under ball-milling

(2012) Nirmalya Mukherjee et al.   GREEN CHEMISTRY

A One-Pot Tandem Ugi Multicomponent Reaction (MCR)/Click Reaction as an Efficient Protecting-Group-Free Route to 1H-1,2,3-Triazole-Modified α-Amino Acid Derivatives and Peptidomimetics

(2012) Teng-Fei Niu et al.   HELVETICA CHIMICA ACTA

Facile One-Pot Synthesis of Monosubstituted 1-Aryl-1H-1,2,3-triazoles from Arylboronic Acids and Prop-2-ynoic Acid (=Propiolic Acid) or Calcium Acetylide (=Calcium Carbide) as Acetylene Source

(2012) Qing Yang et al.   HELVETICA CHIMICA ACTA

Synthesis of 5-Iodo-1,4-disubstituted-1,2,3-triazoles Mediated by in Situ Generated Copper(I) Catalyst and Electrophilic Triiodide Ion

(2012) Wendy S. Brotherton et al.   JOURNAL OF ORGANIC CHEMISTRY

One-pot synthesis of 1,2,3-triazoles from boronic acids in water using Cu(ii)–β-cyclodextrin complex as a nanocatalyst

(2012) Babak Kaboudin et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalysed Multicomponent Click Synthesis of 5-Alkynyl 1,2,3-Triazoles under Ambient Conditions

(2012) Francisco Alonso et al.   SYNLETT

Copper-Catalyzed Synthesis of N-Heterocyclic Compounds

(2012) Hua Fu et al.   SYNTHESIS-STUTTGART

Multicomponent Synthesis of 1,2,3-Triazol-4-yl-methylthio-3-arylquinazolin-4(3H)-one Derivatives

(2012) Majid Koohshari et al.   SYNTHETIC COMMUNICATIONS

Concise synthesis of chiral 2(5H)-furanone derivatives possessing 1,2,3-triazole moiety via one-pot approach

(2012) Yue-He Tan et al.   TETRAHEDRON

Recyclable clay supported Cu (II) catalyzed tandem one-pot synthesis of 1-aryl-1,2,3-triazoles

(2012) Shabber Mohammed et al.   TETRAHEDRON

Copper-catalyzed click synthesis of functionalized 1,2,3-triazoles with 3,4-dihydropyrimidinone or amide group via a one-pot four-component reaction

(2012) Zheng-Jun Quan et al.   TETRAHEDRON

Magnetically separable CuFe2O4 nano particles catalyzed multicomponent synthesis of 1,4-disubstituted 1,2,3-triazoles in tap water using ‘click chemistry’

(2012) B.S.P. Anil Kumar et al.   TETRAHEDRON LETTERS

One-pot, efficient, and regioselective syntheses of 1,4-disubstituted 1,2,3-triazoles using aryldiazonium silica sulfates in water

(2012) Amin Zarei   TETRAHEDRON LETTERS

Click chemistry inspired structural modification of azole antifungal agents to synthesize novel ‘drug like’ molecules

(2012) Kasiviswanadharaju Pericherla et al.   TETRAHEDRON LETTERS

Ultrasound-assisted one-pot synthesis of anti-CML nucleosides featuring 1,2,3-triazole nucleobase under iron-copper catalysis

(2012) Mohsine Driowya et al.   ULTRASONICS SONOCHEMISTRY

One pot ‘click’ reaction: CuII–hydrotalcite catalyzed tandem synthesis of β-hydroxy triazoles via regioselective opening of epoxide followed by [3+2] cycloaddition

(2012) Avvari N. Prasad et al.   Catalysis Science & Technology

Novel Synthesis of Difluoromethyl-Containing 1,4-Disubstituted 1,2,3-Triazoles via a Click-Multicomponent Reaction and Desulfanylation Strategy

(2011) Jian Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Antiviral Breadth and Combination Potential of Peptide Triazole HIV-1 Entry Inhibitors

(2011) Karyn McFadden et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Transition-Metal-Catalyzed C−S, C−Se, and C−Te Bond Formation via Cross-Coupling and Atom-Economic Addition Reactions

(2011) Irina P. Beletskaya et al.   CHEMICAL REVIEWS

Recent advances in Sonogashira reactions

(2011) Rafael Chinchilla et al.   CHEMICAL SOCIETY REVIEWS

The copper(I)-catalyzed alkyne-azide cycloaddition (CuAAC) “click” reaction and its applications. An overview

(2011) Liyuan Liang et al.   COORDINATION CHEMISTRY REVIEWS

1,2,3-Triazoles in Peptidomimetic Chemistry

(2011) Daniel Sejer Pedersen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

An Efficient One-Pot, Four-Component Synthesis of {[(1H-1,2,3-Triazol-4-yl)methoxy]phenyl}-1H-pyrazolo[1,2-b]phthalazine-5,10-dione Derivatives

(2011) Laleh Torkian et al.   HELVETICA CHIMICA ACTA

Multicomponent Click Synthesis of Potentially Biologically Active Triazoles Catalysed by Copper Nanoparticles on Activated Carbon in Water

(2011) Miguel Yus et al.   HETEROCYCLES

Citrus Peel Additives for One-Pot Triazole Formation by Decarboxylation, Nucleophilic Substitution, and Azide–Alkyne Cycloaddition Reactions

(2011) Desiree E. Mendes et al.   JOURNAL OF CHEMICAL EDUCATION

[CuBr(PPh3)3] for Azide−Alkyne Cycloaddition Reactions under Strict Click Conditions

(2011) Steven Lal et al.   JOURNAL OF ORGANIC CHEMISTRY

Tandem Catalysis: From Alkynoic Acids and Aryl Iodides to 1,2,3-Triazoles in One Pot

(2011) Andrej Kolarovič et al.   JOURNAL OF ORGANIC CHEMISTRY

Sequential One-Pot Ruthenium-Catalyzed Azide−Alkyne Cycloaddition from Primary Alkyl Halides and Sodium Azide

(2011) Johan R. Johansson et al.   JOURNAL OF ORGANIC CHEMISTRY

Multicomponent Click Synthesis of 1,2,3-Triazoles from Epoxides in Water Catalyzed by Copper Nanoparticles on Activated Carbon

(2011) Francisco Alonso et al.   JOURNAL OF ORGANIC CHEMISTRY

One-Pot Synthesis of PS-b-PEO-b-PtBA Triblock Copolymers via Combination of SET-LRP and “Click” Chemistry Using Copper(0)/PMDETA as Catalyst System

(2011) Rongkuan Jing et al.   MACROMOLECULES

Combining click-multicomponent reaction: one-pot synthesis of triazolyl methoxy-phenyl indazolo[2,1-b]phthalazine-trione derivatives

(2011) Peyman Salehi et al.   MOLECULAR DIVERSITY

One-pot synthesis of 1,2,3-triazole linked dihydropyrimidinones via Huisgen 1,3-dipolar/Biginelli cycloaddition

(2011) Peyman Salehi et al.   MOLECULAR DIVERSITY

Assessing the whole range of CuAAC mechanisms by DFT calculations—on the intermediacy of copper acetylides

(2011) David Cantillo et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling–TMS-deprotection–CuAAC sequence

(2011) Eugen Merkul et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Click chemistry from organic halides, diazonium salts and anilines in water catalysed by copper nanoparticles on activated carbon

(2011) Francisco Alonso et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Three-Component Synthesis of Neoglycopeptides Using a Cu(II)-Triggered Aminolysis of Peptide Hydrazide Resin and an Azide–Alkyne Cycloaddition Sequence

(2011) Jean-Philippe Ebran et al.   ORGANIC LETTERS

A “Click and Activate” Approach in One-Pot Synthesis of a Triazolyl-Pyridazinone Library

(2011) Wenyuan Qian et al.   ORGANIC LETTERS

Synthesis of Unsymmetrical 1,1′-Disubstituted Bis(1,2,3-triazole)s Using Monosilylbutadiynes

(2011) Bradley C. Doak et al.   ORGANIC LETTERS

CuBr-NCS-Mediated Multicomponent Azide-Alkyne Cycloaddition: Mild and Efficient Synthesis of 5-Bromo-1,4-Disubstituted-1,2,3-Triazoles

(2011) Lingjun Li et al.   SYNLETT

Synthesis of Carbo- and Heterocycles via Coupling-Isomerization Reactions

(2011) Thomas Müller   SYNTHESIS-STUTTGART

Spiro-sulfamidate and sulfate nucleosides via 2′ and 3′-C-branched-chain sugars and nucleosides

(2011) Jérôme Lalot et al.   TETRAHEDRON

An efficient and high-yielding one-pot synthesis of 4-acyl-1,2,3-triazoles via triisopropylsilyl-protected ynones

(2011) Soonho Hwang et al.   TETRAHEDRON

Click reaction on in situ generated β-azidostyrenes from cinnamic acid using CAN–NaN3: synthesis of N-styryl triazoles

(2011) Mitta Kavitha et al.   TETRAHEDRON LETTERS

Fast dye salts provide fast access to azidoarene synthons in multi-step one-pot tandem click transformations

(2011) James T. Fletcher et al.   TETRAHEDRON LETTERS

Modular synthesis of mono, di, and tri-1,4-disubstituted-1,2,3-triazoles through copper-mediated alkyne–azide cycloaddition

(2011) Hélio A. Stefani et al.   TETRAHEDRON LETTERS

One-pot synthesis of [1,2,3]triazole-fused pyrazinopyridazindione tricycles by a ‘click and activate’ approach

(2011) Wenyuan Qian et al.   TETRAHEDRON LETTERS

Triazole-Containing Isothiazolidine 1,1-Dioxide Library Synthesis: One-Pot, Multi-Component Protocols for Small Molecular Probe Discovery

(2011) Alan Rolfe et al.   ACS Combinatorial Science

Covalently immobilized tris(triazolyl)methanol–Cu(i) complexes: highly active and recyclable catalysts for CuAAC reactions

(2011) Erhan Ozkal et al.   Catalysis Science & Technology

Multicomponent Synthesis of 1,2,3-Triazoles in Water Catalyzed by Copper Nanoparticles on Activated Carbon

(2010) Francisco Alonso et al.   ADVANCED SYNTHESIS & CATALYSIS

Direct Synthesis of 1,4-Disubstituted-5-alumino-1,2,3-triazoles: Copper-Catalyzed Cycloaddition of Organic Azides and Mixed Aluminum Acetylides

(2010) Yuhan Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of new azaindole-based PI3Kα inhibitors: Apoptotic and antiangiogenic effect on cancer cells

(2010) Seunghee Hong et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A novel arylethynyltriazole acyclonucleoside inhibits proliferation of drug-resistant pancreatic cancer cells

(2010) Menghua Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Click chemistry inspired one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles and their Src kinase inhibitory activity

(2010) Dalip Kumar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

One pot ‘click’ reactions: tandem enantioselective biocatalytic epoxide ring opening and [3+2] azide alkyne cycloaddition

(2010) Lachlan S. Campbell-Verduyn et al.   CHEMICAL COMMUNICATIONS

In situ click chemistry: probing the binding landscapes of biological molecules

(2010) Sreeman K. Mamidyala et al.   CHEMICAL SOCIETY REVIEWS

Copper-catalyzed azide–alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(i) acetylides

(2010) Jason E. Hein et al.   CHEMICAL SOCIETY REVIEWS

Zeo-Click Chemistry: Copper(I)-Zeolite-Catalyzed Cascade Reaction; One-Pot Epoxide Ring-Opening and Cycloaddition

(2010) Thirupathi Boningari et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Solvent-free synthesis of 1,4-disubstituted 1,2,3-triazoles using a low amount of Cu(PPh3)2NO3 complex

(2010) Dong Wang et al.   GREEN CHEMISTRY

One-Pot, Three-Component Synthesis of 1-(2-Hydroxyethyl)-1H-1,2,3-triazole Derivatives by Copper-Catalyzed 1,3-Dipolar Cycloaddition of 2-Azido Alcohols and Terminal Alkynes under Mild Conditions in Water

(2010) Hashem Sharghi et al.   HELVETICA CHIMICA ACTA

2-Anthryltriazolyl-Containing Multidentate Ligands: Zinc-Coordination Mediated Photophysical Processes and Potential in Live-Cell Imaging Applications

(2010) Heather A. Michaels et al.   INORGANIC CHEMISTRY

Synthesis of Diheterocyclic Compounds Based on Triazolyl Methoxy Phenylquinazolines via a One-Pot Four-Component-Click Reaction

(2010) Minoo Dabiri et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Multicomponent Cascade Transformation ofd-Glucal to Furan-Appended Triazole Glycoconjugates

(2010) Syed Khalid Yousuf et al.   JOURNAL OF ORGANIC CHEMISTRY

Mechanistic Insights into Cu(I)-Catalyzed Azide−Alkyne “Click” Cycloaddition Monitored by Real Time Infrared Spectroscopy

(2010) Shengtong Sun et al.   JOURNAL OF PHYSICAL CHEMISTRY A

“One-pot” dispersion ATRP and alkyne-azide Huisgen's 1,3-dipolar cycloaddition in supercritical carbon dioxide: Towards the formation of functional microspheres

(2010) Bruno Grignard et al.   JOURNAL OF SUPERCRITICAL FLUIDS

One-Pot Syntheses of Amphiphilic Centipede-like Brush Copolymers via Combination of Ring-Opening Polymerization and “Click” Chemistry

(2010) You-Yong Yuan et al.   MACROMOLECULES

Virtual screening: an endless staircase?

(2010) Gisbert Schneider   NATURE REVIEWS DRUG DISCOVERY

One-Pot Three-Step Synthesis of 1,2,3-Triazoles by Copper-Catalyzed Cycloaddition of Azides with Alkynes formed by a Sonogashira Cross-Coupling and Desilylation

(2010) Frédéric Friscourt et al.   ORGANIC LETTERS

“Clicktophycin-52”: A Bioactive Cryptophycin-52 Triazole Analogue

(2010) Markus Nahrwold et al.   ORGANIC LETTERS

Control of peptide secondary structure on star shape polypeptides tethered to polyhedral oligomeric silsesquioxane nanoparticle through click chemistry

(2010) Shiao-Wei Kuo et al.   POLYMER

An Efficient, One-Pot, Regioselective Synthesis of 1,4-Diaryl-1H-1,2,3-triazoles Using Click Chemistry

(2010) Dalip Kumar et al.   SYNTHESIS-STUTTGART

Zeo-click synthesis: CuI-zeolite-catalyzed one-pot two-step synthesis of triazoles from halides and related compounds

(2010) Valérie Bénéteau et al.   TETRAHEDRON LETTERS

One-pot syntheses of 1,2,3-triazoles containing a pentafluorosulfanylalkyl group via click chemistry

(2010) Yangen Huang et al.   TETRAHEDRON LETTERS

One-Pot Tandem Copper-Catalyzed Library Synthesis of 1-Thiazolyl-1,2,3-triazoles as Anticancer Agents

(2010) Wen-Tai Li et al.   ACS Combinatorial Science

Immobilization of Porphyrinatocopper Nanoparticles onto Activated Multi-Walled Carbon Nanotubes and a Study of its Catalytic Activity as an Efficient Heterogeneous Catalyst for a Click Approach to the Three-Component Synthesis of 1,2,3-Triazoles in Water

(2009) Hashem Sharghi et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-in-Charcoal-Catalyzed, Tandem One-Pot Diazo Transfer-Click Reactions

(2009) Ching-Tien Lee et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper Nanoparticles on Charcoal for Multicomponent Catalytic Synthesis of 1,2,3-Triazole Derivatives from Benzyl Halides or Alkyl Halides, Terminal Alkynes and Sodium Azide in Water as a “Green” Solvent

(2009) Hashem Sharghi et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal-Free, Regioselective Triazole Ligations that Deliver LockedcisPeptide Mimetics

(2009) Ahsanullah et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic CC, CN, and CO Ullmann-Type Coupling Reactions

(2009) Florian Monnier et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Exploration of click reaction for the synthesis of modified nucleosides as chitin synthase inhibitors

(2009) Preeti M. Chaudhary et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of orally bioavailable serum and glucocorticoid-regulated kinase 1 (SGK1) inhibitors

(2009) Marlys Hammond et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The application of CuAAC ‘click’ chemistry to catenane and rotaxane synthesis

(2009) Kevin D. Hänni et al.   CHEMICAL SOCIETY REVIEWS

Marrying click chemistry with polymerization: expanding the scope of polymeric materials

(2009) Patricia L. Golas et al.   CHEMICAL SOCIETY REVIEWS

Click chemistry under non-classical reaction conditions

(2009) C. Oliver Kappe et al.   CHEMICAL SOCIETY REVIEWS

Highly active copper-catalysts for azide-alkynecycloaddition

(2009) Zsombor Gonda et al.   DALTON TRANSACTIONS

A multicomponent CuAAC “click” approach to a library of hybrid polydentate 2-pyridyl-1,2,3-triazole ligands: new building blocks for the generation of metallosupramolecular architectures

(2009) James D. Crowley et al.   DALTON TRANSACTIONS

Facile Entry into Triazole Fused Heterocycles via Sulfamidate Derived Azido-alkynes

(2009) V. Sai Sudhir et al.   JOURNAL OF ORGANIC CHEMISTRY

Macromolecular Engineering through Click Chemistry and Other Efficient Transformations

(2009) Brent S. Sumerlin et al.   MACROMOLECULES

A One-Pot Approach to Neoglycopeptides using Orthogonal Native Chemical Ligation and Click Chemistry

(2009) Dong Jun Lee et al.   ORGANIC LETTERS

Facile One-Pot Synthesis of 4,5-Disubstituted 1,2,3-(NH)-Triazoles through Sonogashira Coupling/1,3-Dipolar Cycloaddition of Acid Chlorides, Terminal Acetylenes, and Sodium Azide

(2009) Jihui Li et al.   ORGANIC LETTERS

A Highly Active Catalyst for Huisgen 1,3-Dipolar Cycloadditions Based on the Tris(triazolyl)methanol−Cu(I) Structure

(2009) Salih Özçubukçu et al.   ORGANIC LETTERS

Copper(II)/Copper(I)-Catalyzed Aza-Michael Addition/Click Reaction of in Situ Generated α-Azidohydrazones: Synthesis of Novel Pyrazolone−Triazole Framework

(2009) Orazio A. Attanasi et al.   ORGANIC LETTERS

Synthesis of an Antibacterial Compound Containing a 1,4-Substituted 1H-1,2,3-Triazole: A Scaleable Alternative to the “Click” Reaction

(2009) Roger Hanselmann et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

A one pot multi-component CuAAC “click” approach to bidentate and tridentate pyridyl-1,2,3-triazole ligands: Synthesis, X-ray structures and copper(II) and silver(I) complexes

(2009) James D. Crowley et al.   POLYHEDRON

Greener and Expeditious Synthesis of 1,4-Disubstituted 1,2,3-Triazoles from Terminal Acetylenes and in situ Generated α-Azido Ketones

(2009) Dalip Kumar et al.   SYNLETT

Facile Deprotection of Bulky (Trialkylsilyl)acetylenes with Silver Fluoride

(2009) Sanghee Kim et al.   SYNTHESIS-STUTTGART

A Cu(I)-promoted one-pot ‘SNAr–click reaction’ of fluoronitrobenzenes

(2009) Kulbhushan A. Dururgkar et al.   TETRAHEDRON

Cu(OTf)2/Cu-catalyzed four-component reaction: a facile synthesis of α-alkoxytriazoles via click chemistry

(2009) J.S. Yadav et al.   TETRAHEDRON LETTERS

A facile and regioselective synthesis of 1,4-disubstituted 1,2,3-triazoles using click chemistry

(2009) Dalip Kumar et al.   TETRAHEDRON LETTERS

Base and concentration effects on the product distribution in copper-promoted alkyne–azide cycloaddition: additive-free route to 5-iodo-triazoles

(2009) Nicholas W. Smith et al.   TETRAHEDRON LETTERS

Synthesis and antimicrobial activity of β-lactam–bile acid conjugates linked via triazole

(2008) Namdev S. Vatmurge et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Metal-Catalyzed One-Step Synthesis: Towards Direct Alternatives to Multistep Heterocycle and Amino Acid Derivative Formation

(2008) Bruce A. Arndtsen   CHEMISTRY-A EUROPEAN JOURNAL

Chemistry strategies in early drug discovery: an overview of recent trends

(2008) Matteo Colombo et al.   DRUG DISCOVERY TODAY

Stereoselective Synthesis of Novel Cyclic γ-Amino Acids and Triazole Derivatives

(2008) Verónica F. V. Prazeres et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Convenient Preparation of 5-Iodo-1,4-disubstituted-1,2,3-triazole: Multicomponent One-Pot Reaction of Azide and Alkyne Mediated by CuI−NBS

(2008) Lingjun Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Conformational Analysis of a Cyclic Peptide Obtained viaitoi+4 Intramolecular Side-Chain to Side-Chain Azide−Alkyne 1,3-Dipolar Cycloaddition

(2008) Sonia Cantel et al.   JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Click Assisted One‐Pot Multi‐Step Reactions in Polymer Science: Accelerated Synthetic Protocols

(2008) Pontus Lundberg et al.   MACROMOLECULAR RAPID COMMUNICATIONS

Polymer “Clicking” by CuAAC Reactions

(2008) Morten Meldal   MACROMOLECULAR RAPID COMMUNICATIONS

Construction of Linear Polymers, Dendrimers, Networks, and Other Polymeric Architectures by Copper‐Catalyzed Azide‐Alkyne Cycloaddition “Click” Chemistry

(2008) Jeremiah A. Johnson et al.   MACROMOLECULAR RAPID COMMUNICATIONS

Synthesis and biological evaluation of bile acid dimers linked with 1,2,3-triazole and bis-β-lactam

(2008) Namdev S. Vatmurge et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

N-Myristoyl transferase-mediated protein labelling in vivo

(2008) William P. Heal et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Domino Transformation ofd-Glucal to Racemic α-Substituted α-Hydroxymethyl Furfuryl Derivatives

(2008) Debaraj Mukherjee et al.   ORGANIC LETTERS

Copper-Catalyzed “Click” Reaction/Direct Arylation Sequence: Modular Syntheses of 1,2,3-Triazoles

(2008) Lutz Ackermann et al.   ORGANIC LETTERS

Multidentate 1,2,3-Triazole-Containing Chelators from Tandem Deprotection/Click Reactions of (Trimethylsilyl)alkynes and Comparison of Their Ruthenium(II) Complexes

(2008) James T. Fletcher et al.   ORGANOMETALLICS

Construction of Heterocycles by the Strategic Use of Alkyne π-Activation in Catalyzed Cascade Reactions

(2008) Stefan Kirsch   SYNTHESIS-STUTTGART

Diastereodivergence and appendage diversity in the multicomponent synthesis of aryl-pyrrolo-tetrahydrocarbazoles

(2008) Daniel Royer et al.   TETRAHEDRON

A tandem Ferrier and Click reaction: a facile synthesis of triazolyl-2,3-dideoxypyranosides

(2008) J.S. Yadav et al.   TETRAHEDRON LETTERS

Rapid in situ synthesis of [11C]methyl azide and its application in 11C click-chemistry

(2008) Ralf Schirrmacher et al.   TETRAHEDRON LETTERS

Synthesis and antibiotic activity of a small molecules library of 1,2,3-triazole derivatives

(2007) Marie Aufort et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Click chemistry reactions in medicinal chemistry: Applications of the 1,3-dipolar cycloaddition between azides and alkynes

(2007) Gian Cesare Tron et al.   MEDICINAL RESEARCH REVIEWS