Synthesis of Benzimidazoles through Palladium-Catalyzed Amination of 2-Iodobenzimines with Diaziridinone

Palladium-Catalyzed C−H Silylation through Palladacycles Generated from Aryl Halides

(2018) Ailan Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Air-stable Ruthenium(II)-NNN Pincer Complexes for the Efficient Coupling of Aromatic Diamines and Alcohols to 1H -benzo[d ]imidazoles with the Liberation of H2

(2018) Lin Li et al.   ChemCatChem

Synthesis of 9,9-Disubstituted Fluorenes from 2-Iodobiphenyls and α-Diazoesters under Palladium Catalysis

(2018) Ding Ma et al.   JOURNAL OF ORGANIC CHEMISTRY

Aerobic Copper-Catalyzed Synthesis of Benzimidazoles from Diaryl- and Alkylamines via Tandem Triple C–H Aminations

(2018) Taoyuan Liang et al.   ACS Catalysis

Synthesis of Indoles through Palladium-Catalyzed Three-Component Reaction of Aryl Iodides, Alkynes, and Diaziridinone

(2018) Bo Zhou et al.   ORGANIC LETTERS

N-Doped Cationic PAHs by Rh(III)-Catalyzed Double C–H Activation and Annulation of 2-Arylbenzimidazoles with Alkynes

(2017) José M. Villar et al.   ORGANIC LETTERS

Palladium-Catalyzed Domino Heck/Aryne Carbopalladation/C–H Functionalization: Synthesis of Heterocycle-Fused 9,10-Dihydrophenanthrenes

(2017) Tuanli Yao et al.   ORGANIC LETTERS

Iridium(III)-Catalyzed Synthesis of Benzimidazoles via C–H Activation and Amidation of Aniline Derivatives

(2017) Jintao Xia et al.   ORGANIC LETTERS

Palladium(0)-catalyzed asymmetric C(sp3)–H arylation using a chiral binol-derived phosphate and an achiral ligand

(2017) Lei Yang et al.   Chemical Science

Direct Synthesis of Benzimidazoles by Dehydrogenative Coupling of Aromatic Diamines and Alcohols Catalyzed by Cobalt

(2017) Prosenjit Daw et al.   ACS Catalysis

Trapping σ-Alkyl-Palladium(II) Intermediates with Arynes Encompassing Intramolecular C−H Activation: Spirobiaryls through Pd-Catalyzed Cascade Reactions

(2016) Marta Pérez-Gómez et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Pd-Catalyzed C(sp3)–H Functionalization/Carbenoid Insertion: All-Carbon Quaternary Centers via Multiple C–C Bond Formation

(2016) Álvaro Gutiérrez-Bonet et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Borylation of Olefin C–H Bond via Aryl to Vinyl Palladium 1,4-Migration

(2016) Tian-Jiao Hu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Remote C−H alkylation and C−C bond cleavage enabled by an in situ generated palladacycle

(2016) Juntao Ye et al.   Nature Chemistry

Synthesis of Triphenylenes Starting from 2-Iodobiphenyls and Iodobenzenes via Palladium-Catalyzed Dual C–H Activation and Double C–C Bond Formation

(2016) Shulei Pan et al.   ORGANIC LETTERS

An Approach to Tetraphenylenes via Pd-Catalyzed C–H Functionalization

(2016) Hang Jiang et al.   ORGANIC LETTERS

Sequential Difunctionalization of 2-Iodobiphenyls by Exploiting the Reactivities of a Palladacycle and an Acyclic Arylpalladium Species

(2016) Dushen Chen et al.   ORGANIC LETTERS

Synthesis of Fluorenes Starting from 2-Iodobiphenyls and CH2Br2 through Palladium-Catalyzed Dual C–C Bond Formation

(2016) Guangfa Shi et al.   ORGANIC LETTERS

Pd-Catalyzed Spirocyclization via C–H Activation and Benzyne Insertion

(2016) Hyung Yoon et al.   ORGANIC LETTERS

Structure activity relationship (SAR) study of benzimidazole scaffold for different biological activities: A mini-review

(2015) Geeta Yadav et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pd-Catalyzed Intramolecular C–N Bond Cleavage, 1,4-Migration, sp3 C–H Activation, and Heck Reaction: Four Controllable Diverse Pathways Depending on the Judicious Choice of the Base and Ligand

(2015) Min Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Ketene-Surrogate Coupling: Catalytic Conversion of Aryl Iodides into Aryl Ketenes through Ynol Ethers

(2014) Wenhan Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(0)-Catalyzed Heck Reaction/CH Activation/Amination Sequence with Diaziridinone: A Facile Approach to Indolines

(2014) Huaiji Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed C–H Functionalization Reactions: Efficient Synthesis of Heterocycles

(2014) Xun-Xiang Guo et al.   CHEMICAL REVIEWS

Synthesis of 3,4-dihydro-2H-1,4-benzoxazines and their Oxo Derivatives: A Review

(2014) Malgorzata Smist et al.   CURRENT ORGANIC SYNTHESIS

Enantioselective Synthesis of Planar Chiral Ferrocenes via Pd(0)-Catalyzed Intramolecular Direct C–H Bond Arylation

(2014) De-Wei Gao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Intramolecular Asymmetric C–H Functionalization/Cyclization Reaction of Metallocenes: An Efficient Approach toward the Synthesis of Planar Chiral Metallocene Compounds

(2014) Ruixian Deng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Modular Synthesis of Benzimidazole-Fused Phenanthridines from 2-Arylbenzimidazoles and o-Dibromoarenes by a Palladium-Catalyzed Cascade Process

(2014) Chunxia Chen et al.   ORGANIC LETTERS

Roles of Bases in Transition-Metal Catalyzed Organic Reactions

(2013) Kunbing Ouyang et al.   ACTA CHIMICA SINICA

Palladium-Catalyzed Through-Space C(sp3)H and C(sp2)H Bond Activation by 1,4-Palladium Migration: Efficient Synthesis of [3,4]-Fused Oxindoles

(2013) Tiffany Piou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Pd(0)-Catalyzed Sequential C–N Bond Formation via Allylic and Aromatic C–H Amination of α-Methylstyrenes with Diaziridinone

(2013) Thomas A. Ramirez et al.   ORGANIC LETTERS

Transition-Metal-Free Synthesis of Benzimidazoles Mediated by KOH/DMSO

(2013) Hannah Baars et al.   ORGANIC LETTERS

Iodobenzene Catalyzed C–H Amination of N-Substituted Amidines Using m-Chloroperbenzoic Acid

(2013) Santhosh Kumar Alla et al.   ORGANIC LETTERS

Catalyst free approach to benzimidazoles using air as the oxidant at room temperature

(2012) Chun Zhang et al.   GREEN CHEMISTRY

Nucleophilic Addition of Benzimidazoles to Alkynyl Bromides/Palladium-Catalyzed Intramolecular C–H Vinylation: Synthesis of Benzo[4,5]imidazo[2,1-a]isoquinolines

(2012) Jinsong Peng et al.   JOURNAL OF ORGANIC CHEMISTRY

Functionalized Orthoesters as Powerful Building Blocks for the Efficient Preparation of Heteroaromatic Bicycles

(2012) Gulluzar Bastug et al.   ORGANIC LETTERS

Benzazoles from Aliphatic Amines and o-Amino/Mercaptan/Hydroxyanilines: Elemental Sulfur as a Highly Efficient and Traceless Oxidizing Agent

(2012) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Copper Catalyzed N-Arylation of Amidines with Aryl Boronic Acids and One-Pot Synthesis of Benzimidazoles by a Chan–Lam–Evans N-Arylation and C–H Activation/C–N Bond Forming Process

(2012) Jihui Li et al.   ORGANIC LETTERS

Developments Towards Regioselective Synthesis of 1,2-Disubstituted Benzimidazoles

(2011) Luísa C. R. Carvalho et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Mediated Synthesis of Substituted 2-Aryl-N-benzylbenzimidazoles and 2-Arylbenzoxazoles via C–H Functionalization/C–N/C–O Bond Formation

(2011) Murali Mohan Guru et al.   JOURNAL OF ORGANIC CHEMISTRY

Dibenzometallacyclopentadienes, boroles and selected transition metal and main group heterocyclopentadienes: Synthesis, catalytic and optical properties

(2010) Andreas Steffen et al.   COORDINATION CHEMISTRY REVIEWS

Synthesis and anticancer activity of some novel 2-substituted benzimidazole derivatives

(2010) Hanan M. Refaat   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Cobalt-catalyzed intramolecular C–N and C–O cross-coupling reactions: synthesis of benzimidazoles and benzoxazoles

(2010) Prasenjit Saha et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Direct Imidation to Construct 1H-Benzo[d]imidazole through PdII-Catalyzed CH Activation Promoted by Thiourea

(2009) Qing Xiao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Microwave assisted, one-pot synthesis of 5-nitro- 2-aryl substituted-1H-benzimidazole libraries: Screeningin vitrofor antimicrobial activity

(2009) Kallappa Mahadevappa Hosamani et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Ligand-Free Copper-Catalyzed Synthesis of Substituted Benzimidazoles, 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and Benzoxazoles

(2009) Prasenjit Saha et al.   JOURNAL OF ORGANIC CHEMISTRY

Hidden signatures: new reagents for developing latent fingerprints

(2009) M. John Plater et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

CH Functionalization/CN Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

(2008) Gordon Brasche et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient Aerobic Oxidative Synthesis of 2-Substituted Benzoxazoles, Benzothiazoles, and Benzimidazoles Catalyzed by 4-Methoxy-TEMPO

(2008) Yong-Xing Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of the Poly(ADP-ribose) Polymerase (PARP) Inhibitor 2-[(R)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide (ABT-888) for the Treatment of Cancer

(2008) Thomas D. Penning et al.   JOURNAL OF MEDICINAL CHEMISTRY