Structure-based discovery of 1-(3-fluoro-5-(5-(3-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-b]pyridin-3-yl)phenyl)-3-(pyrimidin-5-yl)urea as a potent and selective nanomolar type-II PLK4 inhibitor
出版年份 2022 全文链接
标题
Structure-based discovery of 1-(3-fluoro-5-(5-(3-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-b]pyridin-3-yl)phenyl)-3-(pyrimidin-5-yl)urea as a potent and selective nanomolar type-II PLK4 inhibitor
作者
关键词
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出版物
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 243, Issue -, Pages 114714
出版商
Elsevier BV
发表日期
2022-08-30
DOI
10.1016/j.ejmech.2022.114714
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